Page last updated: 2024-08-17

benzimidazole and pyrazolone

benzimidazole has been researched along with pyrazolone in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Filipek, S; Stepniewski, TM1
Carter, DM; Gohlke, U; Heinemann, U; Nazaré, M; Neuenschwander, M; Przygodda, J; Specker, E; von Kries, JP1

Other Studies

2 other study(ies) available for benzimidazole and pyrazolone

ArticleYear
Non-peptide ligand binding to the formyl peptide receptor FPR2--A comparison to peptide ligand binding modes.
    Bioorganic & medicinal chemistry, 2015, Jul-15, Volume: 23, Issue:14

    Topics: Benzimidazoles; Binding Sites; Hydrophobic and Hydrophilic Interactions; Ligands; Models, Molecular; Molecular Docking Simulation; Phenylurea Compounds; Protein Conformation; Pyrazolones; Pyridazines; Quinazolinones; Receptors, Formyl Peptide; Receptors, Lipoxin; Structure-Activity Relationship

2015
Identification of a Novel Benzimidazole Pyrazolone Scaffold That Inhibits KDM4 Lysine Demethylases and Reduces Proliferation of Prostate Cancer Cells.
    SLAS discovery : advancing life sciences R & D, 2017, Volume: 22, Issue:7

    Topics: Benzimidazoles; Cell Line, Tumor; Cell Proliferation; Demethylation; Enzyme Inhibitors; Histone Demethylases; Histones; Humans; Hydroxyquinolines; Jumonji Domain-Containing Histone Demethylases; Lysine; Male; PC-3 Cells; Prostatic Neoplasms; Pyrazolones; Receptors, Androgen; Transcription, Genetic

2017