Page last updated: 2024-08-17

benzimidazole and piperidines

benzimidazole has been researched along with piperidines in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (60.00)29.6817
2010's1 (20.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Alsasua, A; Benhamú, B; Girón, R; López-Rodríguez, ML; Martín, MI; Pascual, D1
Cox, JM; Edmondson, SD; Eiermann, GJ; He, H; Lyons, KA; Mastracchio, A; Patel, RA; Patel, SB; Petrov, A; Roy, RS; Scapin, G; Thornberry, NA; Weber, AE; Wu, JK; Xu, S; Zhu, B1
Able, SL; Clarke, TL; Duckworth, JM; Fish, RL; Ivarsson, M; Katugampola, SD; McCourt, C; Napier, C1
Armstrong, SR; Beattie, DT; Fatheree, PR; Long, DD; Marquess, DG; McKinnell, RM; Shaw, JP; Vickery, RG1
Lee, YT; Mancera, RL; Oon, CE; Tan, YJ1

Other Studies

5 other study(ies) available for benzimidazole and piperidines

ArticleYear
New benzimidazole derivatives: selective and orally active 5-HT3 receptor antagonists.
    European journal of pharmacology, 2003, Feb-21, Volume: 462, Issue:1-3

    Topics: 5-Hydroxytryptophan; Administration, Oral; Animals; Aza Compounds; Behavior, Animal; Benzimidazoles; Carbachol; Diarrhea; Dose-Response Relationship, Drug; Gastric Emptying; Gastrointestinal Motility; In Vitro Techniques; Injections, Intraperitoneal; Injections, Intravenous; Male; Mice; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ondansetron; Piperidines; Propane; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Reflex; Serotonin; Serotonin Antagonists

2003
Aminopiperidine-fused imidazoles as dipeptidyl peptidase-IV inhibitors.
    Bioorganic & medicinal chemistry letters, 2009, Aug-01, Volume: 19, Issue:15

    Topics: Animals; Benzimidazoles; Chemistry, Pharmaceutical; Crystallography, X-Ray; Dipeptidyl-Peptidase IV Inhibitors; Dogs; Drug Design; Glucagon-Like Peptide 1; Humans; Hydrolysis; Imidazoles; Inhibitory Concentration 50; Macaca mulatta; Mice; Piperidines; Pyrazines; Pyridines; Rats; Sitagliptin Phosphate; Triazoles

2009
Localisation of melanin-concentrating hormone receptor 1 in rat brain and evidence that sleep parameters are not altered despite high central receptor occupancy.
    European journal of pharmacology, 2009, Aug-15, Volume: 616, Issue:1-3

    Topics: Animals; Autoradiography; Benzimidazoles; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Electroencephalography; In Vitro Techniques; Male; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Somatostatin; Sleep; Substrate Specificity

2009
Discovery of TD-8954, a clinical stage 5-HT(4) receptor agonist with gastrointestinal prokinetic properties.
    Bioorganic & medicinal chemistry letters, 2013, Jul-15, Volume: 23, Issue:14

    Topics: Animals; Benzimidazoles; Crystallography, X-Ray; Dogs; Drug Evaluation, Preclinical; Guinea Pigs; Half-Life; Intestinal Mucosa; Male; Molecular Conformation; Piperidines; Protein Isoforms; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists

2013
BZD9L1 sirtuin inhibitor: Identification of key molecular targets and their biological functions in HCT 116 colorectal cancer cells.
    Life sciences, 2021, Nov-01, Volume: 284

    Topics: Apoptosis; Benzimidazoles; Cell Adhesion; Cell Polarity; Colorectal Neoplasms; Gene Expression Regulation, Neoplastic; Gene Ontology; HCT116 Cells; Humans; Neurites; Piperidines; Protein Interaction Maps; Reactive Oxygen Species; Signal Transduction; Sirtuins; Spheroids, Cellular

2021