Page last updated: 2024-09-03

benidipine hydrochloride and nicardipine

benidipine hydrochloride has been researched along with nicardipine in 6 studies

Compound Research Comparison

Studies
(benidipine hydrochloride)
Trials
(benidipine hydrochloride)
Recent Studies (post-2010)
(benidipine hydrochloride)
Studies
(nicardipine)
Trials
(nicardipine)
Recent Studies (post-2010) (nicardipine)
541162,646444312

Protein Interaction Comparison

ProteinTaxonomybenidipine hydrochloride (IC50)nicardipine (IC50)
Bile salt export pumpHomo sapiens (human)8.314
ATP-dependent translocase ABCB1Mus musculus (house mouse)8
ATP-dependent translocase ABCB1Homo sapiens (human)4.2992
Cytochrome P450 3A4Homo sapiens (human)0.42
Cytochrome P450 2C9 Homo sapiens (human)1.69
ATP-dependent translocase ABCB1Mus musculus (house mouse)2.5
Cytochrome P450 2J2Homo sapiens (human)1.69
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)4.925
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)4.8

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19905 (83.33)18.7374
1990's1 (16.67)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Karasawa, A; Kubo, K; Nakamizo, N; Oka, T; Shuto, K2
Ishii, A; Nakamizo, N; Nishida, K; Oka, T1
Karasawa, A; Kubo, K; Nakamizo, N; Oka, T1
Ikeda, J; Karasawa, A; Kubo, K; Nakamizo, N; Oka, T; Yamada, K1
Deguchi, T; Hara, T; Hattori, O; Kato, Y; Saijyo, T; Suzuki, K; Tanaka, H1

Other Studies

6 other study(ies) available for benidipine hydrochloride and nicardipine

ArticleYear
Antihypertensive effects of the new calcium antagonist benidipine hydrochloride in rats.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:11A

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Calcium Channel Blockers; Chemical Phenomena; Chemistry; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Heart Rate; Hydralazine; Hypertension; Male; Nicardipine; Nifedipine; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Renin; Urination

1988
Slow dissociation of the new slow-onset and long-acting calcium antagonist benidipine hydrochloride from 3H-nitrendipine binding sites.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:11A

    Topics: Animals; Binding Sites; Binding, Competitive; Calcium Channel Blockers; Male; Nicardipine; Nifedipine; Nisoldipine; Nitrendipine; Rats; Rats, Inbred Strains

1988
Antihypertensive effects of intravenous administration of benidipine hydrochloride and some other calcium antagonists in conscious, spontaneously hypertensive rats.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:11A

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Injections, Intravenous; Male; Nicardipine; Nifedipine; Nisoldipine; Nitrendipine; Rats; Rats, Inbred SHR; Verapamil

1988
Antihypertensive effects of the new calcium antagonist benidipine hydrochloride in conscious, renal-hypertensive dogs.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:11A

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Calcium Channel Blockers; Chemical Phenomena; Chemistry; Dogs; Female; Heart Rate; Hypertension, Renal; Male; Nicardipine; Nifedipine; Nitrendipine; Propranolol

1988
Vasodilating effects of the new calcium antagonist benidipine hydrochloride in anesthetized dogs and cats.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:11A

    Topics: Animals; Blood Flow Velocity; Blood Pressure; Calcium Channel Blockers; Cats; Cerebral Cortex; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Injections, Intra-Arterial; Injections, Intravenous; Male; Nicardipine; Nifedipine; Papaverine; Vasodilation; Vasodilator Agents

1988
Effect of the new calcium antagonist (+/-)-(R*)-3-[(R*)-1-benzyl-3- piperidyl] methyl 1,4-dihydro-2,6-dimethyl-4-(m-nitrophenyl)-3,5- pyridinedicarboxylate hydrochloride (KW-3049) on cardiac hypertrophy in spontaneously hypertensive rats.
    The Journal of toxicological sciences, 1993, Volume: 18 Suppl 3

    Topics: Aldosterone; Animals; Antihypertensive Agents; Blood Pressure; Calcium Channel Blockers; Cardiomegaly; DNA; Heart Rate; Hypertension; Male; Myocardium; Nicardipine; Nifedipine; Organ Size; Propranolol; Rats; Rats, Inbred SHR; Renin; RNA

1993