be 2254 has been researched along with prazosin in 22 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 14 (63.64) | 18.7374 |
1990's | 6 (27.27) | 18.2507 |
2000's | 2 (9.09) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Mante, S; Minneman, KP | 1 |
Martin, WH; Saffitz, JE; Tolley, TK | 1 |
Minneman, KP; Wilson, KM | 1 |
Gross, G; Hanft, G | 1 |
Gross, G; Hanft, G; Mehdorn, HM | 1 |
Rugevics, CU; Schümann, HJ | 1 |
Hoffman, BB; Tsujimoto, G | 1 |
Moulds, RF; Stevens, MJ | 1 |
Hoffman, BB; Timmins, PV; Tsujimoto, G | 1 |
Grady, R; Klein, DC; Mefford, IN; Namboodiri, MA; Pierce, JE; Sugden, D | 1 |
Caron, MG; Cotecchia, S; Hagen, PO; Leeb-Lundberg, LM; Lefkowitz, RJ | 1 |
Hicks, PE | 1 |
Corr, PB; Lee, BI; Saffitz, JE; Sharma, AD; Sobel, BE | 1 |
Digges, KG; Summers, RJ | 1 |
Coupar, IM; McPherson, GA; Taylor, DA | 1 |
Doell, G; Ferry, DR; Glossmann, H; Lübbecke, F; Sattler, EL | 1 |
Bristow, MR; Hoffman, BB; Tsujimoto, G | 1 |
Kuo, JS; Lee, FY; Liao, JF; Lin, HC; Yang, MC; Yu, PC | 1 |
Brown, F; Gaivin, R; Graham, RM; Hwa, J; Mathur, M; Perez, DM | 1 |
Hatano, A; Lepor, H; Tang, R; Walden, PD | 1 |
Cotecchia, S; Goepel, M; Hein, P; Michel, MC | 1 |
Minneman, KP; Pupo, AS; Uberti, MA | 1 |
22 other study(ies) available for be 2254 and prazosin
Article | Year |
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The alkylating prazosin analog SZL 49 inactivates both alpha 1A- and alpha 1B-adrenoceptors.
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Drug Synergism; Hippocampus; Liver; Male; Membranes; Phenethylamines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones | 1991 |
Autoradiographic delineation of skeletal muscle alpha 1-adrenergic receptor distribution.
Topics: Adrenergic alpha-Antagonists; Animals; Arterioles; Autoradiography; Muscles; Phenethylamines; Phentolamine; Prazosin; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Tissue Distribution; Vascular Resistance | 1990 |
Pertussis toxin inhibits norepinephrine-stimulated inositol phosphate formation in primary brain cell cultures.
Topics: Animals; Brain; Calcium; Carbachol; Cells, Cultured; Clonidine; Cyclic AMP; Dioxanes; GTP-Binding Proteins; Inositol Phosphates; Norepinephrine; Pertussis Toxin; Phenethylamines; Prazosin; Rats; Receptors, Adrenergic, alpha; Tetralones; Virulence Factors, Bordetella; Yohimbine | 1990 |
Subclassification of alpha 1-adrenoceptor recognition sites by urapidil derivatives and other selective antagonists.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Dioxanes; Heart; In Vitro Techniques; Male; Myocardium; Phenethylamines; Phentolamine; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Yohimbine | 1989 |
Demonstration of alpha 1A- and alpha 1B-adrenoceptor binding sites in human brain tissue.
Topics: Adrenergic alpha-Antagonists; Brain Chemistry; Calcium Channel Blockers; Cerebral Cortex; Dihydropyridines; Humans; In Vitro Techniques; Phenethylamines; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Tetralones | 1989 |
Alpha 1-adrenoceptors in guinea-pig heart ventricles. [3H]prazosin and [125I]IBE 2254 are bound specifically to a receptor population with high affinity and low density.
Topics: Animals; Binding, Competitive; Guinea Pigs; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Male; Myocardium; Phenethylamines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Tetralones; Tritium | 1987 |
Direct measurement of vascular alpha 1-adrenoceptors.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Cell Membrane; Female; Muscle, Smooth, Vascular; Phenethylamines; Phentolamine; Prazosin; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha; Tetralones; Yohimbine | 1985 |
Neuronally released norepinephrine does not preferentially activate postjunctional alpha 1-adrenoceptors in human blood vessels in vitro.
Topics: Adrenergic alpha-Antagonists; Blood Vessels; Humans; In Vitro Techniques; Norepinephrine; Phenethylamines; Prazosin; Receptors, Adrenergic, alpha; Tetralones; Yohimbine | 1985 |
Alpha adrenergic receptors in the rabbit bladder base smooth muscle: alpha-1 adrenergic receptors mediate contractile responses.
Topics: Adrenergic alpha-Agonists; Animals; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Iodine Radioisotopes; Muscle Contraction; Phenethylamines; Prazosin; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha; Tetralones; Urinary Bladder; Yohimbine | 1986 |
Ovine pineal alpha 1-adrenoceptors: characterization and evidence for a functional role in the regulation of serum melatonin.
Topics: Acetyltransferases; Animals; Binding, Competitive; Circadian Rhythm; In Vitro Techniques; Melatonin; Phenethylamines; Pineal Gland; Prazosin; Propranolol; Receptors, Adrenergic, alpha; Sheep; Tetralones | 1985 |
Phorbol ester effects on alpha 1-adrenoceptor binding and phosphatidylinositol metabolism in cultured vascular smooth muscle cells.
Topics: Animals; Aorta, Thoracic; Cells, Cultured; Muscle, Smooth, Vascular; Norepinephrine; Phenethylamines; Phorbol Esters; Phosphatidic Acids; Phosphatidylinositols; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Tetradecanoylphorbol Acetate; Tetralones | 1985 |
Antagonism of pre and postsynaptic alpha-adrenoreceptors by BE 2254 (HEAT) and prazosin.
Topics: Adrenergic alpha-Antagonists; Animals; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Phenethylamines; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Synapses; Tetrahydronaphthalenes; Tetralones | 1981 |
Alpha adrenergic-mediated accumulation of calcium in reperfused myocardium.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Cats; Coronary Disease; Extracellular Space; Myocardium; Perfusion; Phenethylamines; Phentolamine; Prazosin; Tetralones | 1983 |
Characterization of postsynaptic alpha-adrenoceptors in rat aortic strips and portal veins.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta; Clonidine; Female; Male; Muscle, Smooth, Vascular; Nordefrin; Oxymetazoline; Phenethylamines; Portal Vein; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Yohimbine | 1983 |
Competitive antagonism of alpha 1-adrenoceptor mediated pressor responses in the rat mesenteric artery.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Blood Pressure; Female; Kinetics; Mesenteric Arteries; Norepinephrine; Phenethylamines; Phentolamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Yohimbine | 1984 |
Radiation inactivation of alpha 1-adrenoceptors.
Topics: Animals; Cerebral Cortex; Flunitrazepam; Phenethylamines; Prazosin; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Tetralones; Tritium | 1983 |
Identification of alpha 1 adrenergic receptors in rabbit aorta with [125I] BE2254.
Topics: Animals; Aorta, Abdominal; Aorta, Thoracic; Binding Sites; Binding, Competitive; Epinephrine; Female; Isoproterenol; Norepinephrine; Phenethylamines; Phentolamine; Prazosin; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha; Tetralones; Yohimbine | 1984 |
Study on the vascular reactivity and alpha 1-adrenoceptors of portal hypertensive rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Hypertension, Portal; Male; Membranes; Muscle Contraction; Muscle, Smooth, Vascular; Neurotransmitter Uptake Inhibitors; Norepinephrine; Phenethylamines; Portal Vein; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Tetralones | 1994 |
Constitutive activation of a single effector pathway: evidence for multiple activation states of a G protein-coupled receptor.
Topics: Adrenergic alpha-Antagonists; Animals; Arachidonic Acid; Base Sequence; Cell Line; DNA Primers; GTP-Binding Proteins; Inositol 1,4,5-Trisphosphate; Iodine Radioisotopes; Molecular Sequence Data; Mutagenesis, Site-Directed; Phenethylamines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1; Signal Transduction; Tetralones; Tritium; Virulence Factors, Bordetella | 1996 |
The alpha-adrenoceptor antagonist properties of the enantiomers of doxazosin in the human prostate.
Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Binding Sites; Binding, Competitive; Cell Line; Dose-Response Relationship, Drug; Doxazosin; Humans; Male; Phenethylamines; Prazosin; Prostate; Radioligand Assay; Receptors, Adrenergic, alpha; Stereoisomerism; Tetralones | 1996 |
A quantitative analysis of antagonism and inverse agonism at wild-type and constitutively active hamster alpha1B-adrenoceptors.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Cell Line; Chromones; Cricetinae; Dose-Response Relationship, Drug; Doxazosin; Fibroblasts; Inositol Phosphates; Phenethylamines; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Tetralones; Tritium | 2001 |
N-terminal truncation of human alpha1D-adrenoceptors increases expression of binding sites but not protein.
Topics: Amino Acid Sequence; Azides; Binding Sites; Binding, Competitive; Calcium; Cell Line; Glycosylation; Humans; Iodine Radioisotopes; Kinetics; Molecular Sequence Data; Norepinephrine; Oligopeptides; Peptides; Phenethylamines; Photoaffinity Labels; Prazosin; Precipitin Tests; Radioligand Assay; Receptors, Adrenergic, alpha-1; Sequence Deletion; Tetralones; Transfection; Uridine Triphosphate | 2003 |