Page last updated: 2024-08-23

be 2254 and prazosin

be 2254 has been researched along with prazosin in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-199014 (63.64)18.7374
1990's6 (27.27)18.2507
2000's2 (9.09)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Mante, S; Minneman, KP1
Martin, WH; Saffitz, JE; Tolley, TK1
Minneman, KP; Wilson, KM1
Gross, G; Hanft, G1
Gross, G; Hanft, G; Mehdorn, HM1
Rugevics, CU; Schümann, HJ1
Hoffman, BB; Tsujimoto, G1
Moulds, RF; Stevens, MJ1
Hoffman, BB; Timmins, PV; Tsujimoto, G1
Grady, R; Klein, DC; Mefford, IN; Namboodiri, MA; Pierce, JE; Sugden, D1
Caron, MG; Cotecchia, S; Hagen, PO; Leeb-Lundberg, LM; Lefkowitz, RJ1
Hicks, PE1
Corr, PB; Lee, BI; Saffitz, JE; Sharma, AD; Sobel, BE1
Digges, KG; Summers, RJ1
Coupar, IM; McPherson, GA; Taylor, DA1
Doell, G; Ferry, DR; Glossmann, H; Lübbecke, F; Sattler, EL1
Bristow, MR; Hoffman, BB; Tsujimoto, G1
Kuo, JS; Lee, FY; Liao, JF; Lin, HC; Yang, MC; Yu, PC1
Brown, F; Gaivin, R; Graham, RM; Hwa, J; Mathur, M; Perez, DM1
Hatano, A; Lepor, H; Tang, R; Walden, PD1
Cotecchia, S; Goepel, M; Hein, P; Michel, MC1
Minneman, KP; Pupo, AS; Uberti, MA1

Other Studies

22 other study(ies) available for be 2254 and prazosin

ArticleYear
The alkylating prazosin analog SZL 49 inactivates both alpha 1A- and alpha 1B-adrenoceptors.
    European journal of pharmacology, 1991, Oct-14, Volume: 208, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Drug Synergism; Hippocampus; Liver; Male; Membranes; Phenethylamines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones

1991
Autoradiographic delineation of skeletal muscle alpha 1-adrenergic receptor distribution.
    The American journal of physiology, 1990, Volume: 259, Issue:5 Pt 2

    Topics: Adrenergic alpha-Antagonists; Animals; Arterioles; Autoradiography; Muscles; Phenethylamines; Phentolamine; Prazosin; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Tissue Distribution; Vascular Resistance

1990
Pertussis toxin inhibits norepinephrine-stimulated inositol phosphate formation in primary brain cell cultures.
    Molecular pharmacology, 1990, Volume: 38, Issue:2

    Topics: Animals; Brain; Calcium; Carbachol; Cells, Cultured; Clonidine; Cyclic AMP; Dioxanes; GTP-Binding Proteins; Inositol Phosphates; Norepinephrine; Pertussis Toxin; Phenethylamines; Prazosin; Rats; Receptors, Adrenergic, alpha; Tetralones; Virulence Factors, Bordetella; Yohimbine

1990
Subclassification of alpha 1-adrenoceptor recognition sites by urapidil derivatives and other selective antagonists.
    British journal of pharmacology, 1989, Volume: 97, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Dioxanes; Heart; In Vitro Techniques; Male; Myocardium; Phenethylamines; Phentolamine; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Yohimbine

1989
Demonstration of alpha 1A- and alpha 1B-adrenoceptor binding sites in human brain tissue.
    European journal of pharmacology, 1989, Oct-10, Volume: 169, Issue:2-3

    Topics: Adrenergic alpha-Antagonists; Brain Chemistry; Calcium Channel Blockers; Cerebral Cortex; Dihydropyridines; Humans; In Vitro Techniques; Phenethylamines; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Tetralones

1989
Alpha 1-adrenoceptors in guinea-pig heart ventricles. [3H]prazosin and [125I]IBE 2254 are bound specifically to a receptor population with high affinity and low density.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 289, Issue:2

    Topics: Animals; Binding, Competitive; Guinea Pigs; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Male; Myocardium; Phenethylamines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Tetralones; Tritium

1987
Direct measurement of vascular alpha 1-adrenoceptors.
    Clinical science (London, England : 1979), 1985, Volume: 68 Suppl 10

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Cell Membrane; Female; Muscle, Smooth, Vascular; Phenethylamines; Phentolamine; Prazosin; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha; Tetralones; Yohimbine

1985
Neuronally released norepinephrine does not preferentially activate postjunctional alpha 1-adrenoceptors in human blood vessels in vitro.
    Circulation research, 1985, Volume: 57, Issue:3

    Topics: Adrenergic alpha-Antagonists; Blood Vessels; Humans; In Vitro Techniques; Norepinephrine; Phenethylamines; Prazosin; Receptors, Adrenergic, alpha; Tetralones; Yohimbine

1985
Alpha adrenergic receptors in the rabbit bladder base smooth muscle: alpha-1 adrenergic receptors mediate contractile responses.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Iodine Radioisotopes; Muscle Contraction; Phenethylamines; Prazosin; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha; Tetralones; Urinary Bladder; Yohimbine

1986
Ovine pineal alpha 1-adrenoceptors: characterization and evidence for a functional role in the regulation of serum melatonin.
    Endocrinology, 1985, Volume: 116, Issue:5

    Topics: Acetyltransferases; Animals; Binding, Competitive; Circadian Rhythm; In Vitro Techniques; Melatonin; Phenethylamines; Pineal Gland; Prazosin; Propranolol; Receptors, Adrenergic, alpha; Sheep; Tetralones

1985
Phorbol ester effects on alpha 1-adrenoceptor binding and phosphatidylinositol metabolism in cultured vascular smooth muscle cells.
    Life sciences, 1985, Dec-23, Volume: 37, Issue:25

    Topics: Animals; Aorta, Thoracic; Cells, Cultured; Muscle, Smooth, Vascular; Norepinephrine; Phenethylamines; Phorbol Esters; Phosphatidic Acids; Phosphatidylinositols; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Tetradecanoylphorbol Acetate; Tetralones

1985
Antagonism of pre and postsynaptic alpha-adrenoreceptors by BE 2254 (HEAT) and prazosin.
    Journal of autonomic pharmacology, 1981, Volume: 1, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Phenethylamines; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Synapses; Tetrahydronaphthalenes; Tetralones

1981
Alpha adrenergic-mediated accumulation of calcium in reperfused myocardium.
    The Journal of clinical investigation, 1983, Volume: 72, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Cats; Coronary Disease; Extracellular Space; Myocardium; Perfusion; Phenethylamines; Phentolamine; Prazosin; Tetralones

1983
Characterization of postsynaptic alpha-adrenoceptors in rat aortic strips and portal veins.
    British journal of pharmacology, 1983, Volume: 79, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta; Clonidine; Female; Male; Muscle, Smooth, Vascular; Nordefrin; Oxymetazoline; Phenethylamines; Portal Vein; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Yohimbine

1983
Competitive antagonism of alpha 1-adrenoceptor mediated pressor responses in the rat mesenteric artery.
    The Journal of pharmacy and pharmacology, 1984, Volume: 36, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Blood Pressure; Female; Kinetics; Mesenteric Arteries; Norepinephrine; Phenethylamines; Phentolamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Yohimbine

1984
Radiation inactivation of alpha 1-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 323, Issue:2

    Topics: Animals; Cerebral Cortex; Flunitrazepam; Phenethylamines; Prazosin; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Tetralones; Tritium

1983
Identification of alpha 1 adrenergic receptors in rabbit aorta with [125I] BE2254.
    Life sciences, 1984, Feb-13, Volume: 34, Issue:7

    Topics: Animals; Aorta, Abdominal; Aorta, Thoracic; Binding Sites; Binding, Competitive; Epinephrine; Female; Isoproterenol; Norepinephrine; Phenethylamines; Phentolamine; Prazosin; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha; Tetralones; Yohimbine

1984
Study on the vascular reactivity and alpha 1-adrenoceptors of portal hypertensive rats.
    British journal of pharmacology, 1994, Volume: 111, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Hypertension, Portal; Male; Membranes; Muscle Contraction; Muscle, Smooth, Vascular; Neurotransmitter Uptake Inhibitors; Norepinephrine; Phenethylamines; Portal Vein; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Tetralones

1994
Constitutive activation of a single effector pathway: evidence for multiple activation states of a G protein-coupled receptor.
    Molecular pharmacology, 1996, Volume: 49, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Arachidonic Acid; Base Sequence; Cell Line; DNA Primers; GTP-Binding Proteins; Inositol 1,4,5-Trisphosphate; Iodine Radioisotopes; Molecular Sequence Data; Mutagenesis, Site-Directed; Phenethylamines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1; Signal Transduction; Tetralones; Tritium; Virulence Factors, Bordetella

1996
The alpha-adrenoceptor antagonist properties of the enantiomers of doxazosin in the human prostate.
    European journal of pharmacology, 1996, Oct-10, Volume: 313, Issue:1-2

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Binding Sites; Binding, Competitive; Cell Line; Dose-Response Relationship, Drug; Doxazosin; Humans; Male; Phenethylamines; Prazosin; Prostate; Radioligand Assay; Receptors, Adrenergic, alpha; Stereoisomerism; Tetralones

1996
A quantitative analysis of antagonism and inverse agonism at wild-type and constitutively active hamster alpha1B-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 363, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Cell Line; Chromones; Cricetinae; Dose-Response Relationship, Drug; Doxazosin; Fibroblasts; Inositol Phosphates; Phenethylamines; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Tetralones; Tritium

2001
N-terminal truncation of human alpha1D-adrenoceptors increases expression of binding sites but not protein.
    European journal of pharmacology, 2003, Feb-21, Volume: 462, Issue:1-3

    Topics: Amino Acid Sequence; Azides; Binding Sites; Binding, Competitive; Calcium; Cell Line; Glycosylation; Humans; Iodine Radioisotopes; Kinetics; Molecular Sequence Data; Norepinephrine; Oligopeptides; Peptides; Phenethylamines; Photoaffinity Labels; Prazosin; Precipitin Tests; Radioligand Assay; Receptors, Adrenergic, alpha-1; Sequence Deletion; Tetralones; Transfection; Uridine Triphosphate

2003