Page last updated: 2024-09-03

bdf 9148 and ouabain

bdf 9148 has been researched along with ouabain in 10 studies

Compound Research Comparison

Studies
(bdf 9148)
Trials
(bdf 9148)
Recent Studies (post-2010)
(bdf 9148)
Studies
(ouabain)
Trials
(ouabain)
Recent Studies (post-2010) (ouabain)
390116,35772747

Protein Interaction Comparison

ProteinTaxonomybdf 9148 (IC50)ouabain (IC50)
STAT3, partialHomo sapiens (human)1.154
Kruppel-like factor 5Homo sapiens (human)0.0832
Sodium/potassium-transporting ATPase subunit alpha-1 Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit beta-1Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit alpha-1 Rattus norvegicus (Norway rat)4.3
Sodium/potassium-transporting ATPase subunit alpha-2Rattus norvegicus (Norway rat)0.17
Sodium/potassium-transporting ATPase subunit alpha-3 Rattus norvegicus (Norway rat)0.031
Sodium/potassium-transporting ATPase subunit beta-1 Rattus norvegicus (Norway rat)1.1263
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)0.1646
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 20.097
Sodium/potassium-transporting ATPase subunit alpha-3Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit beta-2Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit alpha-2Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit beta-3Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit gammaHomo sapiens (human)6
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.8
Sodium/potassium-transporting ATPase subunit alpha-4Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit beta-3Rattus norvegicus (Norway rat)0.0018
Sodium/potassium-transporting ATPase subunit alpha-4Rattus norvegicus (Norway rat)0.0031

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (80.00)18.2507
2000's2 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Böhm, M; Erdmann, E; La Rosée, K; Schmidt, U; Schulz, C; Schwinger, RH1
Böhm, M; Erdmann, E; La Rosée, K; Mittmann, C; Schwinger, RH1
Böhm, M; Eissner, HJ; Kreuzer, E; Müller-Ehmsen, J; Reichart, B; Schmidt, U; Schwinger, RH; Stäblein, A; Uberfuhr, P; Uhlmann, R1
Erdmann, E; Frank, K; Martin-Vasallo, P; McDonough, AA; Müller-Ehmsen, J; Pressley, TA; Schwinger, RH; Wang, J; Xiang, A1
Bavendiek, U; Brixius, K; Erdmann, E; Frank, K; Gross, A; Müller-Ehmsen, J; Pietsch, M; Reuter, H; Schwinger, RH1
Brixius, K; Frank, K; Müller-Ehmsen, J; Schwinger, RH1
Bavendiek, U; Brixius, K; Müller-Ehmsen, J; Münch, G; Schwinger, RH; Zobel, C1
Müller-Ehmsen, J; Näbauer, M; Schwinger, RH1
Böhm, M; Flesch, M; Häuseler, C; Hellige, G; Pfahlberg, A; Schiffmann, H1
Hackmann, F; Hellige, G; Hoebel, D; Luers, F; Pfahlberg, A; Rizouli, V; Schiffmann, H1

Other Studies

10 other study(ies) available for bdf 9148 and ouabain

ArticleYear
Na(+)-channel activators increase cardiac glycoside sensitivity in failing human myocardium.
    Journal of cardiovascular pharmacology, 1992, Volume: 19, Issue:4

    Topics: Adult; Azetidines; Cardiomyopathy, Dilated; Cardiotonic Agents; Drug Interactions; Female; Heart Transplantation; Humans; In Vitro Techniques; Male; Middle Aged; Myocardial Contraction; Myocardium; Ouabain; Papillary Muscles; Sodium Channels

1992
Evidence for a sustained effectiveness of sodium-channel activators in failing human myocardium.
    Journal of molecular and cellular cardiology, 1991, Volume: 23, Issue:4

    Topics: Adult; Azetidines; Cardiomyopathy, Dilated; Cardiotonic Agents; Cell Membrane; Dose-Response Relationship, Drug; Female; Heart; Humans; In Vitro Techniques; Isoproterenol; Kinetics; Male; Middle Aged; Molecular Structure; Myocardial Contraction; Myocardium; Ouabain; Piperazines; Sodium Channels

1991
Effect of inotropic stimulation on the negative force-frequency relationship in the failing human heart.
    Circulation, 1993, Volume: 88, Issue:5 Pt 1

    Topics: Adult; Azetidines; Calcium; Cardiac Output, Low; Cardiotonic Agents; Cyclic AMP; Electric Stimulation; Female; Heart; Humans; Isometric Contraction; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Ouabain

1993
Regional expression of sodium pump subunits isoforms and Na+-Ca++ exchanger in the human heart.
    The Journal of clinical investigation, 1996, Oct-01, Volume: 98, Issue:7

    Topics: Adult; Azetidines; Biological Transport; Calcium; Carrier Proteins; Female; Heart Atria; Heart Septum; Heart Ventricles; Humans; Immunoblotting; Isoenzymes; Male; Middle Aged; Myocardium; Ouabain; Potassium; Sodium; Sodium-Calcium Exchanger; Sodium-Potassium-Exchanging ATPase; Tissue Distribution; Tissue Donors

1996
Altered inotropism in the failing human myocardium.
    Basic research in cardiology, 1996, Volume: 91 Suppl 2

    Topics: Adrenergic beta-Agonists; Azetidines; Calcium; Calcium-Binding Proteins; Calcium-Transporting ATPases; Cardiotonic Agents; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Heart Failure; Humans; In Vitro Techniques; Indoles; Isoproterenol; Myocardial Contraction; Myocardium; Ouabain; Sarcoplasmic Reticulum; Sodium

1996
Increase in force of contraction by activation of the Na+/Ca(2+)-exchanger in human myocardium.
    British journal of clinical pharmacology, 1997, Volume: 43, Issue:4

    Topics: Adrenergic beta-Agonists; Antiporters; Azetidines; Calcium; Cardiotonic Agents; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Heart Failure; Heart Transplantation; Humans; Isoproterenol; Muscle Contraction; Muscle Fibers, Skeletal; Muscle, Smooth, Vascular; Myocardial Contraction; Ouabain; Papillary Muscles; Sodium; Sodium-Calcium Exchanger; Sodium-Potassium-Exchanging ATPase

1997
Effect of inotropic interventions on the force-frequency relation in the human heart.
    Basic research in cardiology, 1998, Volume: 93 Suppl 1

    Topics: Adrenergic beta-Agonists; Azetidines; Biomechanical Phenomena; Cardiac Output, Low; Cardiotonic Agents; Cyclic AMP; Drug Evaluation, Preclinical; Heart Rate; Humans; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Ouabain; Papillary Muscles

1998
Na+-channel modulating effect of the inotropic compound S(-)BDF 9196 in human myocardium.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:1

    Topics: Azetidines; Cardiotonic Agents; Cyclic AMP; Enzyme Inhibitors; Heart; Humans; In Vitro Techniques; Myocardial Contraction; Myocardium; Ouabain; Papillary Muscles; Sodium Channels; Sodium-Potassium-Exchanging ATPase; Stereoisomerism; Ventricular Function, Left

1999
Effects of different inotropic interventions on myocardial function in the developing rabbit heart.
    Basic research in cardiology, 2002, Volume: 97, Issue:1

    Topics: Adrenergic beta-Agonists; Aging; Animals; Animals, Newborn; Azetidines; Calcium; Calcium-Transporting ATPases; Cardiotonic Agents; Enzyme Inhibitors; Female; Gene Expression; Heart; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Ouabain; Rabbits; Sarcoplasmic Reticulum; Sodium-Calcium Exchanger; Ventricular Pressure

2002
Na(+)-channel modulation, a new principle of inotropic intervention: effects on hemodynamic and myocardial energetics in the immature rabbit heart.
    Pediatric research, 2003, Volume: 54, Issue:6

    Topics: Age Factors; Animals; Animals, Newborn; Azetidines; Cardiotonic Agents; Coronary Circulation; Cyclic AMP; Enoximone; Female; Isoproterenol; Models, Cardiovascular; Myocardial Contraction; Myocardium; Ouabain; Oxygen Consumption; Pregnancy; Rabbits; Sodium Channels

2003