Page last updated: 2024-09-03

bd 1008 and cocaine

bd 1008 has been researched along with cocaine in 7 studies

Compound Research Comparison

Studies
(bd 1008)
Trials
(bd 1008)
Recent Studies (post-2010)
(bd 1008)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
280432,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomybd 1008 (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (14.29)18.2507
2000's5 (71.43)29.6817
2010's1 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bowen, WD; Matsumoto, RR; McCracken, KA1
Bowen, WD; De Costa, BR; Matsumoto, RR; McCracken, KA; Miller, J; Pouw, B; Williams, W1
Bowen, WD; De Costa, BR; Friedman, MJ; Matsumoto, RR; McCracken, KA; Pouw, B1
Bowen, WD; Cao, JJ; Hewett, KL; Husbands, SM; Matsumoto, RR; Newman, AH; Pouw, B1
Bowen, WD; Matsumoto, RR; McCracken, KA; Pouw, B; Zhang, Y1
Bowen, WD; Coop, A; Gilmore, DL; Kausar, A; Matsumoto, RR; Pouw, B; Williams, W1
Garcés-Ramírez, L; Green, JL; Hiranita, T; Katz, JL; Kopajtic, TA; McCurdy, CR; Mereu, M; Mesangeau, C; Narayanan, S; Tanda, G; Thomas, AM1

Other Studies

7 other study(ies) available for bd 1008 and cocaine

ArticleYear
Novel sigma receptor ligands attenuate the locomotor stimulatory effects of cocaine.
    European journal of pharmacology, 1999, Jan-15, Volume: 365, Issue:1

    Topics: Animals; Binding, Competitive; Cocaine; Dopamine Uptake Inhibitors; Ethylamines; Guinea Pigs; Male; Mice; Motor Activity; Piperazines; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Receptors, Dopamine D2; Receptors, Opioid; Receptors, Phencyclidine; Receptors, Serotonin; Receptors, sigma

1999
N-alkyl substituted analogs of the sigma receptor ligand BD1008 and traditional sigma receptor ligands affect cocaine-induced convulsions and lethality in mice.
    European journal of pharmacology, 2001, Jan-12, Volume: 411, Issue:3

    Topics: Alkylation; Animals; Behavior, Animal; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Ethylamines; Guinea Pigs; In Vitro Techniques; Injections, Intraventricular; Ligands; Male; Mice; Microinjections; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Red Nucleus; Seizures

2001
Conformationally restricted analogs of BD1008 and an antisense oligodeoxynucleotide targeting sigma1 receptors produce anti-cocaine effects in mice.
    European journal of pharmacology, 2001, May-11, Volume: 419, Issue:2-3

    Topics: Analysis of Variance; Animals; Binding, Competitive; Cocaine; Ethylamines; Locomotion; Male; Mice; Motor Activity; Oligodeoxyribonucleotides, Antisense; Piperazines; Pyrrolidines; Receptors, sigma; Seizures; Structure-Activity Relationship

2001
Rimcazole analogs attenuate the convulsive effects of cocaine: correlation with binding to sigma receptors rather than dopamine transporters.
    Neuropharmacology, 2001, Volume: 41, Issue:7

    Topics: Animals; Anticonvulsants; Binding Sites; Carbazoles; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Ethylamines; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Pyrrolidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Seizures

2001
Involvement of sigma receptors in the behavioral effects of cocaine: evidence from novel ligands and antisense oligodeoxynucleotides.
    Neuropharmacology, 2002, Volume: 42, Issue:8

    Topics: Animals; Cocaine; Dose-Response Relationship, Drug; Ethylamines; Guinea Pigs; Ligands; Male; Mice; Motor Activity; Oligodeoxyribonucleotides, Antisense; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Seizures

2002
Novel analogs of the sigma receptor ligand BD1008 attenuate cocaine-induced toxicity in mice.
    European journal of pharmacology, 2004, May-10, Volume: 492, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Cocaine; Ethylamines; Guinea Pigs; Ligands; Male; Mice; Mice, Inbred Strains; Molecular Structure; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Seizures

2004
Sigma receptor agonists: receptor binding and effects on mesolimbic dopamine neurotransmission assessed by microdialysis.
    Biological psychiatry, 2011, Feb-01, Volume: 69, Issue:3

    Topics: Animals; Benzoxazoles; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Drug Interactions; Ethylamines; Ethylenediamines; Guanidines; Male; Microdialysis; Morpholines; Nucleus Accumbens; Piperazines; Pyrrolidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Synaptic Transmission

2011