Page last updated: 2024-09-04

bazedoxifene and entacapone

bazedoxifene has been researched along with entacapone in 1 studies

Compound Research Comparison

Studies
(bazedoxifene)
Trials
(bazedoxifene)
Recent Studies (post-2010)
(bazedoxifene)
Studies
(entacapone)
Trials
(entacapone)
Recent Studies (post-2010) (entacapone)
30769249503112173

Protein Interaction Comparison

ProteinTaxonomybazedoxifene (IC50)entacapone (IC50)
Multidrug resistance-associated protein 4Homo sapiens (human)6.8
Catechol O-methyltransferaseHomo sapiens (human)0.223
Catechol O-methyltransferaseRattus norvegicus (Norway rat)1.275
Adenosine receptor A2aHomo sapiens (human)2.32
Alpha-ketoglutarate-dependent dioxygenase FTOHomo sapiens (human)3

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Furukawa, T; Hosoya, K; Kadono, K; Moriguchi, H; Nakamori, F; Naritomi, Y; Teramura, T; Terashita, S; Tetsuka, K; Yamano, K1

Other Studies

1 other study(ies) available for bazedoxifene and entacapone

ArticleYear
Quantitative prediction of human intestinal glucuronidation effects on intestinal availability of UDP-glucuronosyltransferase substrates using in vitro data.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:9

    Topics: Administration, Oral; Biotransformation; Cell Membrane Permeability; Cytochrome P-450 Enzyme System; Glucuronides; Glucuronosyltransferase; Humans; Intestinal Absorption; Intestines; Isoenzymes; Kinetics; Metabolic Clearance Rate; Microsomes; Models, Biological; Pharmaceutical Preparations; Recombinant Proteins; Substrate Specificity

2012