Compounds > bay x 1005
Page last updated: 2024-09-03

bay x 1005 and pyrilamine

bay x 1005 has been researched along with pyrilamine in 4 studies

Compound Research Comparison

Studies
(bay x 1005)		Trials
(bay x 1005)		Recent Studies (post-2010)
(bay x 1005)		Studies
(pyrilamine)		Trials
(pyrilamine)		Recent Studies (post-2010) (pyrilamine)
58681,86026116

Protein Interaction Comparison

ProteinTaxonomybay x 1005 (IC50)pyrilamine (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.13
Alpha-2A adrenergic receptorHomo sapiens (human)2.976
Cytochrome P450 2D6Homo sapiens (human)0.3
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.997
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.13
Histamine H1 receptorCavia porcellus (domestic guinea pig)0.0015
Histamine H1 receptorRattus norvegicus (Norway rat)0.0126
Sodium-dependent serotonin transporterHomo sapiens (human)0.047
Histamine H1 receptorHomo sapiens (human)0.0166
5-hydroxytryptamine receptor 2BHomo sapiens (human)2.788
Sodium-dependent dopamine transporter Homo sapiens (human)0.879
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.1
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.558

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dahlén, SE; Jonsson, EW1
Amann, R; Donnerer, J; Peskar, BA; Schuligoi, R1
Burchardt, ER; Müller-Peddinghaus, R1
Dahlén, SE; Larsson, L; Sydbom, A1

Other Studies

4 other study(ies) available for bay x 1005 and pyrilamine

ArticleYear
Leukotrienes and other mediators of the Schultz-Dale reaction in guinea-pig lung parenchyma.
    Advances in prostaglandin, thromboxane, and leukotriene research, 1995, Volume: 23

    Topics: Animals; Guinea Pigs; Inflammation; Leukotriene B4; Leukotrienes; Lung; Male; Metiamide; Ovalbumin; Pyrilamine; Quinolines

1995
Release of calcitonin gene-related peptide in cardiac anaphylaxis.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:2

    Topics: 6-Ketoprostaglandin F1 alpha; Anaphylaxis; Animals; Calcitonin Gene-Related Peptide; Cimetidine; Coronary Circulation; Cyclooxygenase Inhibitors; Guinea Pigs; Heart; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Indomethacin; Leukotriene C4; Lipoxygenase Inhibitors; Myocardium; Ovalbumin; Pyrilamine; Quinolines; Thromboxane B2

1997
Antiedematous effects of combination therapies with the leukotriene synthesis inhibitor BAY X 1005 in the archidonic acid-induced mouse ear inflammation test.
    Prostaglandins, leukotrienes, and essential fatty acids, 1997, Volume: 56, Issue:4

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acid; Disease Models, Animal; Drug Therapy, Combination; Ear; Edema; Female; Histamine H1 Antagonists; Indomethacin; Inflammation; Lipoxygenase Inhibitors; Methysergide; Mice; Mice, Inbred Strains; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Pyrilamine; Quinolines; Serotonin Antagonists

1997
Selective effects of antileukotrienes on leukotriene and histamine release in human dispersed lung cells.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1999, Volume: 48 Suppl 1

    Topics: Histamine H1 Antagonists; Histamine Release; Humans; Hydroxyurea; Indazoles; Leukotriene Antagonists; Leukotrienes; Lipoxygenase Inhibitors; Lung; Lung Neoplasms; Pyrilamine; Quinolines

1999