Page last updated: 2024-09-03

bay x 1005 and aa 861

bay x 1005 has been researched along with aa 861 in 2 studies

Compound Research Comparison

Studies
(bay x 1005)
Trials
(bay x 1005)
Recent Studies (post-2010)
(bay x 1005)
Studies
(aa 861)
Trials
(aa 861)
Recent Studies (post-2010) (aa 861)
5868290234

Protein Interaction Comparison

ProteinTaxonomybay x 1005 (IC50)aa 861 (IC50)
Polyunsaturated fatty acid 5-lipoxygenaseHomo sapiens (human)1.7
Polyunsaturated fatty acid 5-lipoxygenaseRattus norvegicus (Norway rat)1.045
Polyunsaturated fatty acid 5-lipoxygenaseMus musculus (house mouse)0.032
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomeraseCavia porcellus (domestic guinea pig)1.7
M17 leucyl aminopeptidasePlasmodium falciparum 3D753.45

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carpenter, TG; Cuthbert, NJ; Fitzgerald, MF; Francis, HP; Gardiner, PJ; Mohrs, K; Müller-Peddinghaus, R; Newton, BB; Patel, UP; Thompson, AM1
Arroyo, V; Carrió, A; Clària, J; Jiménez, W; López-Parra, M; Miquel, R; Párrizas, M; Planagumà, A; Rivera, F; Rodés, J; Titos, E; Villamor, N1

Other Studies

2 other study(ies) available for bay x 1005 and aa 861

ArticleYear
Inhibition of antigen-induced contraction of guinea-pig airways by a leukotriene synthesis inhibitor, BAY x1005.
    European journal of pharmacology, 1994, Jun-02, Volume: 258, Issue:1-2

    Topics: 5-Lipoxygenase-Activating Proteins; Administration, Oral; Animals; Benzoquinones; Bronchoconstriction; Carrier Proteins; Guinea Pigs; Hydroxyurea; In Vitro Techniques; Indoles; Injections, Intravenous; Leukotriene Antagonists; Lipoxygenase Inhibitors; Male; Membrane Proteins; Ovalbumin; Pyrans; Quinolines; Quinolones; Trachea

1994
Inhibition of 5-lipoxygenase induces cell growth arrest and apoptosis in rat Kupffer cells: implications for liver fibrosis.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2003, Volume: 17, Issue:12

    Topics: Animals; Apoptosis; Benzoquinones; Cell Division; Cells, Cultured; Kupffer Cells; Lipoxygenase Inhibitors; Liver Cirrhosis, Experimental; Models, Biological; Quinolines; Rats

2003