bay-k-8644 and oxadiazoles

bay-k-8644 has been researched along with oxadiazoles in 51 studies

Research

Studies (51)

TimeframeStudies, this research(%)All Research%
pre-199028 (54.90)18.7374
1990's19 (37.25)18.2507
2000's3 (5.88)29.6817
2010's1 (1.96)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Henderson, G; Kennedy, C1
Hammond, C; Henderson, G; Mason, WT; Morton, AJ1
Little, HJ; Littleton, JM; Whittington, MA1
Battaini, F; Bergamaschi, S; Govoni, S; Meucci, O; Parenti, M; Schettini, G; Trabucchi, M1
Creazzo, TL1
Bolger, GT; Campbell, N; Crowley, M; McKay, DW; O'Neill, SK; Triggle, CR1
Fraser, S; Kenny, BA; Kilpatrick, AT; Spedding, M1
Finch, DM; Fisher, RS; Jackson, MB1
Naitoh, T; Sugimoto, T; Toyo-Oka, T1
Abraham, C; Aptel, H; Lombet, A; Nagel, N; Peglion, JL; Randle, JC; Renaud, JF1
Lory, P; Schultz, D; Schwartz, A; Varadi, G; Varadi, M1
Henstenberg, JD; Sharp, GW; Stafford, GA; Weiland, GA; Yaney, GC1
Collins, F; Guthrie, PB; Kater, SB; Schmidt, MF1
Drimal, J1
Glossmann, H; Goll, A; Moosburger, K; Striessnig, J1
Cognard, C; Fosset, M; Galizzi, JP; Lazdunski, M; Romey, G1
Carpenter, CL; Greenberg, DA; Messing, RO1
Kendall, DA1
Luchowski, EM; Rutledge, A; Su, CM; Triggle, DJ; Wei, XY1
Hosey, MM; Maan, AC; Ptasienski, J1
Nahorski, SR; Rooney, TA1
Barhanin, J; Borsotto, M; Fosset, M; Galizzi, JP; Lazdunski, M; Renaud, JF; Romey, G; Schmid, A1
Brown, AM; Brush, K; Hamilton, SL; Schwartz, A; Yatani, A1
Baik, YH; Koch, WJ; Schwartz, A; Williams, JS1
Lee, RT; Marsh, JD; Smith, TW1
DeRoth, L; Godfraind, T; Wibo, M1
Brown, AM; Kunze, DL; Yatani, A1
Lamb, GD; Walsh, T1
Laterre, EC; Maloteaux, JM; Octave, JN1
Massieu, L; Tapia, R1
Dunn, SM2
Brisac, AM; Lacolley, P; Laurent, S; Legrand, M; Schmitt, H; Tsoucaris-Kupfer, D1
Barhanin, J; Frelin, C; Lazdunski, M; Schmid-Alliana, A; Van Renterghem, C; Vigne, P1
Faivre-Bauman, A; Loudes, C; Patte, C; Tixier-Vidal, A1
Borges, R; Cárdenas, AM; Esteban, C; García, AG; Montiel, C1
Allen, PD; Marsh, JD1
Boarder, MR; Owen, PJ; Plevin, R1
Carpenter, CL; Greenberg, DA; Marks, SS; Messing, RO; Watson, DL1
Poder, T; Rampe, D; Schilling, WP; Zhao, ZY1
Akbarali, H; Gilbert, R; Hall, J; Moody-Corbett, F1
Buisson, N; Gourdji, D; Laverrière, JN; Martial, JA; Richard, JL; Tixier-Vidal, A1
Dakshinamurti, K; Lal, KJ1
Bolger, GT; O'Neill, SK; Triggle, CR1
Ehrenstein, G; Fitzpatrick, LA; Pocotte, SL1
Glossmann, H; Hering, S; Strübing, C1
Bieger, D; Martin-Caraballo, M; Triggle, CR1
Kan, E; Kelly, JE; Lokuta, AJ; Nishio, M; Sagawa, K; Sagawa, T; Tsai, J; Wasserstrom, JA1
Gonzalez, A; Sarna, SK1
Anderson, U; Keef, KD; O'Driscoll, K; Sanders, KM; Ward, SM1
Gajdus, M; Grzesk, G; Malinowski, B; Szadujkis-Szadurska, K; Szadujkis-Szadurski, L; Wicinski, M1

Other Studies

51 other study(ies) available for bay-k-8644 and oxadiazoles

ArticleYear
Chronic exposure to morphine does not induce dependence at the level of the calcium channel current in human SH-SY5Y cells.
    Neuroscience, 1992, Volume: 49, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium Channel Blockers; Calcium Channels; Cell Line; Drug Tolerance; Humans; Kinetics; Membrane Potentials; Models, Biological; Mollusk Venoms; Morphine; Naloxone; Nicotinic Acids; omega-Conotoxin GVIA; Oxadiazoles; Peptides, Cyclic; Time Factors

1992
Characterisation of the L- and N-type calcium channels in differentiated SH-SY5Y neuroblastoma cells: calcium imaging and single channel recording.
    Brain research. Molecular brain research, 1992, Volume: 13, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Cadmium; Cadmium Chloride; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Differentiation; Cell Line; Cell Membrane; Chlorides; Evoked Potentials; Fura-2; Humans; Kinetics; Microscopy, Fluorescence; Neuroblastoma; Nicotinic Acids; Nifedipine; omega-Conotoxins; Oxadiazoles; Peptides, Cyclic; Potassium; Tretinoin

1992
Effects of dihydropyridine calcium channel antagonists in ethanol withdrawal; doses required, stereospecificity and actions of Bay K 8644.
    Psychopharmacology, 1990, Volume: 100, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; Ethanol; Isradipine; Male; Mice; Nimodipine; Nitrendipine; Oxadiazoles; Stereoisomerism; Substance Withdrawal Syndrome; Time Factors

1990
Modulation of dihydropyridine-sensitive calcium channels: a role for G proteins.
    European neurology, 1990, Volume: 30 Suppl 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Dihydropyridines; GTP-Binding Proteins; Guanosine Triphosphate; Isradipine; Neurons; Nitrendipine; Oxadiazoles; Rats; Tumor Cells, Cultured

1990
Reduced L-type calcium current in the embryonic chick heart with persistent truncus arteriosus.
    Circulation research, 1990, Volume: 66, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Chick Embryo; Electrophysiology; Heart; Isradipine; Myocardium; Oxadiazoles; Receptors, Nicotinic; Truncus Arteriosus, Persistent

1990
Comparative behavioral, neurochemical and pharmacological activities of dihydropyridine calcium channel activating drugs.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain; Calcium Channel Agonists; Catecholamines; Chromatography, High Pressure Liquid; Dihydropyridines; Guinea Pigs; Injections, Intraperitoneal; Male; Mice; Motor Activity; Muscle Contraction; Muscle, Smooth; Nicotinic Acids; Nifedipine; Oxadiazoles; Pyridines; Stereoisomerism; Structure-Activity Relationship

1990
Selective antagonism of calcium channel activators by fluspirilene.
    British journal of pharmacology, 1990, Volume: 100, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding Sites; Binding, Competitive; Calcium Channel Agonists; Calcium Channel Blockers; Cecum; Cerebral Cortex; Female; Fluspirilene; Guinea Pigs; In Vitro Techniques; Isradipine; Kinetics; Muscle, Smooth; Oxadiazoles; Potassium; Pyridines; Radioligand Assay; Spiro Compounds

1990
Miniature excitatory synaptic currents in cultured hippocampal neurons.
    Brain research, 1990, Jun-04, Volume: 518, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Aspartic Acid; Calcium Channel Blockers; Cells, Cultured; Dipeptides; Electrophysiology; Fetus; Hippocampus; Kinetics; Membrane Potentials; Mice; N-Methylaspartate; Neurons; Oxadiazoles; Potassium; Quisqualic Acid; Synapses; Tetrodotoxin

1990
An endogenous Ca2+ channel agonist, endothelin-1, does not directly activate partially purified dihydropyridine-sensitive Ca2+ channel from cardiac muscle in a reconstituted system.
    Biochemical and biophysical research communications, 1990, Sep-28, Volume: 171, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Diltiazem; Endothelins; Heart; Isradipine; Kinetics; Liposomes; Microsomes; Oxadiazoles; Proteolipids; Sarcolemma; Swine; Verapamil

1990
Ca2+ channel inhibition by a new dihydropyridine derivative, S11568, and its enantiomers S12967 and S12968.
    European journal of pharmacology, 1990, Nov-06, Volume: 190, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding, Competitive; Calcium Channel Blockers; Calcium Radioisotopes; Cell Line; Dihydropyridines; Electrophysiology; Guinea Pigs; Heart; In Vitro Techniques; Inosine Triphosphate; Isradipine; Male; Muscle, Smooth, Vascular; Myocardium; Oxadiazoles; Rats; Ryanodine; Stereoisomerism

1990
Acceleration of activation and inactivation by the beta subunit of the skeletal muscle calcium channel.
    Nature, 1991, Jul-11, Volume: 352, Issue:6331

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Binding Sites; Calcium Channels; Cell Line; Cell Membrane; Dihydropyridines; DNA; Electric Conductivity; Gene Expression; Ion Channel Gating; Isradipine; Kinetics; L Cells; Macromolecular Substances; Muscles; Oxadiazoles; Rabbits; Receptors, Nicotinic; Transfection

1991
Binding of the dihydropyridine calcium channel blocker (+)-[3H] isopropyl-4-(2,1,3-benzoxadiazol-4-yl)-1,4-dihydro-5-methoxycarbonyl-2, 6-dimethyl-3-pyridinecarboxylate (PN200-110) to RINm5F membranes and cells: characterization and functional significanc
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Line; Cell Membrane; Insulin; Insulin Secretion; Islets of Langerhans; Isradipine; Membrane Potentials; Oxadiazoles; Potassium Chloride

1991
Sustained increase in intracellular calcium promotes neuronal survival.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1991, Volume: 11, Issue:8

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Cell Survival; Chick Embryo; Extracellular Space; Intracellular Membranes; Isradipine; Neurons; Osmolar Concentration; Oxadiazoles; Potassium

1991
Regulation of 1,4-dihydropyridine and beta-adrenergic receptor sites in coronary artery smooth muscle membranes.
    Cellular signalling, 1991, Volume: 3, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Coronary Vessels; Dogs; Isradipine; Male; Muscle, Smooth, Vascular; Oxadiazoles; Receptors, Adrenergic, beta; Receptors, Nicotinic; Temperature

1991
Purified calcium channels have three allosterically coupled drug receptors.
    FEBS letters, 1986, Mar-03, Volume: 197, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Allosteric Regulation; Amines; Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; Diltiazem; Guinea Pigs; Ion Channels; Isradipine; Muscles; Nifedipine; Oxadiazoles; Pyridines; Receptors, Drug; Verapamil

1986
Dihydropyridine-sensitive Ca2+ channels in mammalian skeletal muscle cells in culture: electrophysiological properties and interactions with Ca2+ channel activator (Bay K8644) and inhibitor (PN 200-110).
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Cells, Cultured; Electric Conductivity; Ion Channels; Isradipine; Membrane Potentials; Muscles; Nifedipine; Oxadiazoles; Rats

1986
Depolarization-dependent binding of the calcium channel antagonist, (+)-[3H]PN200-110, to intact cultured PC12 cells.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium; Calcium Channel Blockers; Cells, Cultured; Isradipine; Kinetics; Membrane Potentials; Nifedipine; Nitrendipine; Onium Compounds; Organophosphorus Compounds; Oxadiazoles; Potassium; Pyridines; Tritium

1986
Cyclic GMP formation and inositol phosphate accumulation do not share common origins in rat brain slices.
    Journal of neurochemistry, 1986, Volume: 47, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain; Cell Compartmentation; Cyclic GMP; Inositol Phosphates; Isradipine; Male; Oxadiazoles; Potassium; Rats; Rats, Inbred Strains; Sugar Phosphates; Type C Phospholipases

1986
Pharmacologic and radioligand binding analysis of the actions of 1,4-dihydropyridine activator-antagonist pairs in smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding, Competitive; Calcium; Drug Synergism; Guinea Pigs; Ion Channels; Muscle Contraction; Muscle, Smooth, Vascular; Nicotinic Acids; Nitrendipine; Oxadiazoles; Potassium Chloride; Rats; Stereoisomerism

1986
Influence of Mg++ on the effect of diltiazem to increase dihydropyridine binding to receptors on Ca++-channels in chick cardiac and skeletal muscle membranes.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Chickens; Diltiazem; Dose-Response Relationship, Drug; Ion Channels; Isradipine; Magnesium; Membranes; Muscles; Myocardium; Nitrendipine; Oxadiazoles; Receptors, Nicotinic

1986
Regional characterization of agonist and depolarization-induced phosphoinositide hydrolysis in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atropine; Brain; Calcium Channel Blockers; Carbachol; Hydrolysis; Isradipine; Male; Norepinephrine; Oxadiazoles; Phosphatidylinositols; Physostigmine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Muscarinic; Tissue Distribution

1986
Dihydropyridine-sensitive Ca2+ channels: molecular properties of interaction with Ca2+ channel blockers, purification, subunit structure, and differentiation.
    Journal of cardiovascular pharmacology, 1986, Volume: 8 Suppl 8

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Affinity Labels; Animals; Bepridil; Binding, Competitive; Calcium; Calcium Channel Blockers; Calcium Channels; Chick Embryo; Cholic Acids; Diltiazem; Ion Channels; Isradipine; Kinetics; Macromolecular Substances; Molecular Weight; Muscles; Myocardial Contraction; Oxadiazoles; Pyridines; Pyrrolidines; Receptors, Nicotinic; Verapamil

1986
A comparison between the binding and electrophysiological effects of dihydropyridines on cardiac membranes.
    Molecular pharmacology, 1987, Volume: 31, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; Guinea Pigs; Heart; Ion Channels; Isradipine; Kinetics; Membrane Potentials; Membranes; Myocardium; Nicotinic Acids; Nimodipine; Nitrendipine; Oxadiazoles; Pyridines; Stereoisomerism; Structure-Activity Relationship

1987
A possible role for the endothelium in porcine coronary smooth muscle responses to dihydropyridine calcium channel modulators.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Endothelium; Histamine; Isomerism; Isosorbide Dinitrate; Muscle, Smooth, Vascular; Nicotinic Acids; Oxadiazoles; Swine; Vasoconstriction; Vasodilation

1987
Evidence for distinct calcium channel agonist and antagonist binding sites in intact cultured embryonic chick ventricular cells.
    Circulation research, 1987, Volume: 60, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding Sites; Calcium; Calcium Channel Blockers; Cells, Cultured; Chick Embryo; Heart Ventricles; Isradipine; Kinetics; Myocardial Contraction; Myocardium; Oxadiazoles; Radioligand Assay

1987
Pharmacologic relevance of dihydropyridine binding sites in membranes from rat aorta: kinetic and equilibrium studies.
    Circulation research, 1988, Volume: 62, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Binding, Competitive; Calcium; Calcium Channels; Ion Channels; Isradipine; Kinetics; Muscle, Smooth, Vascular; Nifedipine; Nisoldipine; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, Nicotinic; Stereoisomerism

1988
Effects of dihydropyridine calcium channel modulators on cardiac sodium channels.
    The American journal of physiology, 1988, Volume: 254, Issue:1 Pt 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Heart; Ion Channels; Isradipine; Myocardium; Nitrendipine; Oxadiazoles; Rats; Receptors, Nicotinic; Sodium; Stereoisomerism

1988
Calcium currents, charge movement and dihydropyridine binding in fast- and slow-twitch muscles of rat and rabbit.
    The Journal of physiology, 1987, Volume: 393

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; In Vitro Techniques; Ion Channels; Isradipine; Muscles; Nifedipine; Oxadiazoles; Rabbits; Rats; Time Factors

1987
Functional dihydropyridine binding site associated with slow calcium channel in rat cultured neurones.
    Neuroscience letters, 1988, Apr-22, Volume: 87, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding Sites; Binding, Competitive; Calcium; Calcium Channels; Cells, Cultured; Frontal Lobe; Ion Channels; Isradipine; Oxadiazoles; Potassium; Rats; Rats, Inbred Strains; Receptors, Nicotinic

1988
Relationship of dihydropyridine binding sites with calcium-dependent neurotransmitter release in synaptosomes.
    Journal of neurochemistry, 1988, Volume: 51, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Aminopyridines; Animals; Brain; Calcium; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; gamma-Aminobutyric Acid; Ion Channels; Isradipine; Lanthanum; Male; Mice; Neurotransmitter Agents; Nifedipine; Nitrendipine; Oxadiazoles; Potassium; Receptors, Nicotinic; Ruthenium Red; Synaptosomes

1988
Multiple calcium channels in synaptosomes: voltage dependence of 1,4-dihydropyridine binding and effects on function.
    Biochemistry, 1988, Jul-12, Volume: 27, Issue:14

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Dihydropyridines; Ion Channels; Isradipine; Kinetics; Male; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Spectrometry, Fluorescence; Synaptosomes; Verapamil

1988
Central modulation of baroreceptor reflex response to phenylephrine by dihydropyridines in rats.
    Hypertension (Dallas, Tex. : 1979), 1988, Volume: 12, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atropine Derivatives; Blood Pressure; Brain; Calcium Channel Agonists; Calcium Channel Blockers; Dihydropyridines; Isradipine; Male; Muscarine; Oxadiazoles; Phenylephrine; Pressoreceptors; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Reflex

1988
Molecular mechanism of action of the vasoconstrictor peptide endothelin.
    Biochemical and biophysical research communications, 1988, Dec-30, Volume: 157, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Angiotensin II; Animals; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Electrophysiology; Endothelins; Endothelium, Vascular; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Isradipine; Oxadiazoles; Peptides; Phosphatidylinositols; Rats; Rats, Inbred Strains; Vasoconstriction; Vasopressins

1988
Involvement of DHP voltage-sensitive calcium channels and protein kinase C in thyroliberin (TRH) release by developing hypothalamic neurons in culture.
    Brain research, 1988, Jul-26, Volume: 456, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Cells, Cultured; Hypothalamus; Ion Channels; Isradipine; Mice; Mollusk Venoms; Neurons; omega-Conotoxins; Oxadiazoles; Phorbol Esters; Potassium; Reference Values; Thyrotropin-Releasing Hormone

1988
Secretion from adrenaline- and noradrenaline-storing adrenomedullary cells is regulated by a common dihydropyridine-sensitive calcium channel.
    Brain research, 1988, Jul-26, Volume: 456, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Calcium; Calcium Channel Blockers; Cats; Dihydropyridines; Dimethylphenylpiperazinium Iodide; Epinephrine; In Vitro Techniques; Ion Channels; Isradipine; Norepinephrine; Oxadiazoles; Potassium; Reference Values

1988
Developmental regulation of cardiac calcium channels and contractile sensitivity to [Ca]o.
    The American journal of physiology, 1989, Volume: 256, Issue:1 Pt 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding Sites; Calcium Channels; Chick Embryo; Isradipine; Kinetics; Myocardial Contraction; Oxadiazoles

1989
Characterization of bradykinin-stimulated release of noradrenaline from cultured bovine adrenal chromaffin cells.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bradykinin; Calcium; Cattle; Cells, Cultured; Chromaffin Granules; Chromaffin System; Dose-Response Relationship, Drug; In Vitro Techniques; Inositol Phosphates; Nicotinic Acids; Nitrendipine; Norepinephrine; Oxadiazoles; Potassium

1989
Comparative effects of chronic exposure to ethanol and calcium channel antagonists on calcium channel antagonist receptors in cultured neural (PC12) cells.
    Journal of neurochemistry, 1989, Volume: 53, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Gland Neoplasms; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Ethanol; Isradipine; Nerve Tissue; Oxadiazoles; Pheochromocytoma; Rats; Receptors, Nicotinic; Stereoisomerism; Time Factors; Tumor Cells, Cultured

1989
Calcium channel agonist and antagonist binding in a highly enriched sarcolemma preparation obtained from canine ventricle.
    Journal of cardiovascular pharmacology, 1989, Volume: 13, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding, Competitive; Calcium Channel Blockers; Calcium Channels; Diltiazem; Dogs; Dose-Response Relationship, Drug; Heart Ventricles; Imines; In Vitro Techniques; Isradipine; Oxadiazoles; Sarcolemma

1989
Voltage-dependent calcium channels in skeletal muscle transverse tubules. Measurements of calcium efflux in membrane vesicles.
    The Journal of biological chemistry, 1989, Jul-05, Volume: 264, Issue:19

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Benzothiazoles; Calcium Channel Blockers; Calcium Channels; Calcium Radioisotopes; Carbocyanines; Cell Membrane; Dihydropyridines; Edetic Acid; Fluorescent Dyes; Isradipine; Lanthanum; Membrane Potentials; Muscles; Nitrendipine; Oxadiazoles; Potassium; Rabbits; Verapamil

1989
Calcium current in embryonic Xenopus muscle cells in culture.
    Canadian journal of physiology and pharmacology, 1989, Volume: 67, Issue:10

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Calcium Chloride; Cells, Cultured; Embryo, Nonmammalian; Isradipine; Muscles; Nifedipine; Oxadiazoles; Xenopus

1989
Thyroliberin and dihydropyridines modulate prolactin gene expression through interacting pathways in GH3 cells.
    Neuroendocrinology, 1989, Volume: 50, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Gene Expression; Isradipine; Kinetics; Oxadiazoles; Pituitary Neoplasms; Prolactin; Rats; RNA, Messenger; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone; Tumor Cells, Cultured

1989
Calcium channels in vitamin B6 deficiency-induced hypertension.
    Journal of hypertension, 1993, Volume: 11, Issue:12

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Blood Pressure; Calcium Channel Blockers; Calcium Channels; Diltiazem; Hypertension; Male; Nicotinic Acids; Nifedipine; Oxadiazoles; Rats; Rats, Sprague-Dawley; Verapamil; Vitamin B 6 Deficiency

1993
Competitive binding experiments reveal differential interactions for dihydropyridine calcium channel activators and antagonists at dihydropyridine receptors on mouse brain membranes.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:7

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding, Competitive; Brain; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; In Vitro Techniques; Male; Membranes; Mice; Muscle Proteins; Nicotinic Acids; Nitrendipine; Oxadiazoles; Stereoisomerism; Thermodynamics

1994
Role of calcium channels in parathyroid hormone secretion.
    Bone, 1995, Volume: 16, Issue:4 Suppl

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cattle; Cyclic AMP; Electrophoresis, Polyacrylamide Gel; Ionomycin; Isotope Labeling; Nicotinic Acids; Nifedipine; Oxadiazoles; Parathyroid Glands; Parathyroid Hormone; Pertussis Toxin; Phosphorylation; Potassium; Radioimmunoassay; Stereoisomerism; Verapamil; Virulence Factors, Bordetella

1995
Evidence for an external location of the dihydropyridine agonist receptor site on smooth muscle and skeletal muscle calcium channels.
    British journal of pharmacology, 1993, Volume: 108, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Calcium Channel Blockers; Calcium Channels; Cell Line; Diffusion; Electrophysiology; Ion Channels; Mice; Muscle, Smooth; Muscles; Nicotinic Acids; Oxadiazoles; Potassium Channels; Spectrometry, Fluorescence

1993
Photosensitization of oesophageal smooth muscle by 3-NO2-1, 4-dihydropyridines: evidence for two cyclic GMP-dependent effector pathways.
    British journal of pharmacology, 1995, Volume: 116, Issue:8

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 3',5'-Cyclic-GMP Phosphodiesterases; Aminoquinolines; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium-Transporting ATPases; Chelating Agents; Egtazic Acid; Esophagus; Guanylate Cyclase; In Vitro Techniques; Indoles; Marine Toxins; Muscle, Smooth; Nicotinic Acids; Nitric Oxide; Oxadiazoles; Oxazoles; Phosphoprotein Phosphatases; Photosensitizing Agents; Purinones; Rats; Rats, Sprague-Dawley; Ryanodine

1995
Activation of purified cardiac ryanodine receptors by dihydropyridine agonists.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 280, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Dihydropyridines; Dogs; Membrane Potentials; Myocardium; Nicotinic Acids; Nifedipine; Oxadiazoles; Ryanodine Receptor Calcium Release Channel; Sarcoplasmic Reticulum; Stereoisomerism

2001
Neural regulation of in vitro giant contractions in the rat colon.
    American journal of physiology. Gastrointestinal and liver physiology, 2001, Volume: 281, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Antineoplastic Agents; Benzazepines; Calcium Channel Agonists; Calcium Channel Blockers; Colon; Cyclic GMP; Dopamine Antagonists; Enzyme Inhibitors; Hexamethonium; Imines; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nicotinic Antagonists; Nitric Oxide; Nitroarginine; omega-Conotoxins; Oxadiazoles; Peristalsis; Quinoxalines; Rats; Rats, Sprague-Dawley; Suramin; Tetrodotoxin

2001
Electrical activity induced by nitric oxide in canine colonic circular muscle.
    American journal of physiology. Gastrointestinal and liver physiology, 2002, Volume: 282, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Colon; Dogs; Electric Conductivity; Enteric Nervous System; Enzyme Inhibitors; Female; Gastrointestinal Motility; In Vitro Techniques; Indoles; Male; Membrane Potentials; Mitochondria; Muscle, Smooth; Nickel; Nifedipine; Nitric Oxide; Nitric Oxide Donors; Nitroarginine; Nitroprusside; Oxadiazoles; Potassium; Quinoxalines; Uncoupling Agents

2002
Role of endothelium, acetylocholine and calcium ions in Bay K8644- and KCl-induced contraction.
    Molecular medicine reports, 2013, Volume: 8, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Arteries; Calcium; Calcium Channel Agonists; Calcium Channels; Endothelium, Vascular; Guanylate Cyclase; Ions; Male; Muscle Contraction; Nitric Oxide Synthase; Nitroarginine; Oxadiazoles; Potassium Chloride; Quinoxalines; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Soluble Guanylyl Cyclase

2013