bay-k-8644 and naloxone

bay-k-8644 has been researched along with naloxone in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19905 (26.32)18.7374
1990's11 (57.89)18.2507
2000's2 (10.53)29.6817
2010's1 (5.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Henderson, G; Kennedy, C1
Morrone, LA; Pimpinella, G; Romanelli, L; Valeri, P1
Martinelli, B; Morrone, LA; Severini, C; Valeri, P1
Baeyens, JM; Barrios, M2
Pillai, NP; Ross, DH1
Kavaliers, M1
Kavaliers, M; Ossenkopp, KP1
Bacciottini, L; Carlà, V; Moroni, F; Pellegrini-Giampietro, DE1
Hirota, K; Matsuki, A; Rabito, SF; Zsigmond, EK1
Alfaro, MJ; Colado, MI; Del Val, V; Lopez, F; Martin, MI1
Bélisle, S; Bellabarba, D; Gallo-Payet, N; Lehoux, JG; Petit, A1
Dierssen, M; Flórez, J; Hurlé, MA; Ruiz, F1
Hirota, K; Matsuki, A; Rabito, SF; Sato, T; Zsigmond, EK1
Moises, HC; Rusin, KI1
Carabelli, V; Carbone, E; Carra, I1
Hagiwara, K; Iijima, T; Miyoshi, I; Murakami, M; Murata, A; Nakagawasai, O; Tadano, T; Tan-No, K; Yamadera, F; Yanagisawa, T1
Kim, OM; Lim, DY; Lim, GH1
Chen, CH; Hsu, K; Huang, CJ; Jan, WC; Tsai, PS1

Other Studies

19 other study(ies) available for bay-k-8644 and naloxone

ArticleYear
Chronic exposure to morphine does not induce dependence at the level of the calcium channel current in human SH-SY5Y cells.
    Neuroscience, 1992, Volume: 49, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium Channel Blockers; Calcium Channels; Cell Line; Drug Tolerance; Humans; Kinetics; Membrane Potentials; Models, Biological; Mollusk Venoms; Morphine; Naloxone; Nicotinic Acids; omega-Conotoxin GVIA; Oxadiazoles; Peptides, Cyclic; Time Factors

1992
Some pharmacological characteristics of the guinea pig ileum opioid system activated by cholecystokinin.
    Neuropharmacology, 1990, Volume: 29, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atropine; Cholecystokinin; Clonidine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Nifedipine; Receptors, Opioid; Yohimbine

1990
Reproducible withdrawal contractions of isolated guinea-pig ileum after brief morphine exposure: effects of clonidine and nifedipine.
    The Journal of pharmacy and pharmacology, 1990, Volume: 42, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Clonidine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Nifedipine; Substance Withdrawal Syndrome; Yohimbine

1990
Differential effects of L-type calcium channel blockers and stimulants on naloxone-precipitated withdrawal in mice acutely dependent on morphine.
    Psychopharmacology, 1991, Volume: 104, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Female; Mice; Morphine Dependence; Naloxone; Nicardipine; Postural Balance; Substance Withdrawal Syndrome; Verapamil

1991
Opiate receptor mediated hyperthermic responses in rat following Ca++ channel antagonists.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Biological Transport, Active; Body Temperature Regulation; Brain; Ca(2+) Mg(2+)-ATPase; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Fever; Male; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid

1986
Stimulatory influences of calcium channel antagonists on stress-induced opioid analgesia and locomotor activity.
    Brain research, 1987, Apr-07, Volume: 408, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Diltiazem; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Immobilization; Mice; Mice, Inbred C57BL; Motor Activity; Naloxone; Nifedipine; Pain; Reaction Time; Stress, Physiological; Verapamil

1987
Magnetic fields inhibit opioid-mediated 'analgesic' behaviours of the terrestrial snail, Cepaea nemoralis.
    Journal of comparative physiology. A, Sensory, neural, and behavioral physiology, 1988, Volume: 162, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Calcium; Diltiazem; Ion Channels; Magnetics; Morphine; Naloxone; Nifedipine; Nociceptors; Pyrrolidines; Snails; Temperature; Verapamil

1988
Morphine withdrawal in cortical slices: suppression by Ca2+-channel inhibitors of abstinence-induced [3H]-noradrenaline release.
    British journal of pharmacology, 1988, Volume: 93, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Cerebral Cortex; Dihydropyridines; Disease Models, Animal; In Vitro Techniques; Ion Channels; Morphine; Naloxone; Nimodipine; Norepinephrine; Rats; Substance Withdrawal Syndrome; Tritium

1988
Differential effects of calcium channel blockers and stimulants on morphine withdrawal in vitro.
    European journal of pharmacology, 1988, Jul-26, Volume: 152, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Diltiazem; Ethanol; Female; In Vitro Techniques; Morphine; Muscle Contraction; Muscle, Smooth, Vascular; Naloxone; Rats; Rats, Inbred Strains; Stereoisomerism; Substance Withdrawal Syndrome; Verapamil

1988
Ketamine inhibits contractile responses of intestinal smooth muscle by decreasing the influx of calcium through the L-type calcium channel.
    Acta anaesthesiologica Scandinavica, 1995, Volume: 39, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcimycin; Calcium; Calcium Channels; Dose-Response Relationship, Drug; Female; Guinea Pigs; Ileum; In Vitro Techniques; Inflammation Mediators; Ionophores; Ketamine; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naloxone; Parasympatholytics

1995
Effect of nimodipine, diltiazem and BAY K 8644 on the behavioural and neurochemical changes associated with naloxone-precipitated withdrawal in the rat. A comparison with clonidine.
    General pharmacology, 1993, Volume: 24, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Behavior, Animal; Brain Chemistry; Clonidine; Diltiazem; Hydroxyindoleacetic Acid; Male; Morphine Dependence; Naloxone; Nimodipine; Rats; Rats, Sprague-Dawley; Serotonin; Spinal Cord; Substance Withdrawal Syndrome

1993
The modulation of placental lactogen release by opioids: a role for extracellular calcium.
    Molecular and cellular endocrinology, 1993, Volume: 90, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylate Cyclase Toxin; Analgesics; Calcium; Cells, Cultured; Dopamine; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Gene Expression Regulation; Humans; Ionomycin; Naloxone; Naltrexone; Narcotics; Pertussis Toxin; Placental Lactogen; Pyrrolidines; Time Factors; Trophoblasts; Virulence Factors, Bordetella

1993
The Ca2+ channel agonist Bay K 8644 induces central respiratory depression in cats, an effect blocked by naloxone.
    European journal of pharmacology, 1993, Aug-24, Volume: 240, Issue:2-3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analysis of Variance; Animals; Calcium Channels; Cats; Drug Interactions; Female; Male; Naloxone; Nimodipine; Respiration; Stereoisomerism

1993
Relaxant effect of ketamine and its isomers on histamine-induced contraction of tracheal smooth muscle.
    British journal of anaesthesia, 1996, Volume: 76, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Anesthetics, Dissociative; Animals; Calcium; Culture Techniques; Dose-Response Relationship, Drug; Drug Synergism; Epinephrine; Female; Guinea Pigs; Histamine Antagonists; Ketamine; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naloxone; Trachea

1996
Mu-opioid and GABA(B) receptors modulate different types of Ca2+ currents in rat nodose ganglion neurons.
    Neuroscience, 1998, Volume: 85, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analgesics, Opioid; Animals; Baclofen; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Calcium Channels, N-Type; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA Agonists; GABA Antagonists; Naloxone; Narcotic Antagonists; Nerve Tissue Proteins; Neurons; Nifedipine; Nodose Ganglion; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Patch-Clamp Techniques; Peptides; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Spider Venoms

1998
Localized secretion of ATP and opioids revealed through single Ca2+ channel modulation in bovine chromaffin cells.
    Neuron, 1998, Volume: 20, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Triphosphate; Analgesics; Analgesics, Opioid; Animals; Antineoplastic Agents; Autocrine Communication; Barium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Calcium Channels, N-Type; Cattle; Chromaffin Cells; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Exocytosis; Ion Channel Gating; Naloxone; Narcotic Antagonists; Neurotransmitter Agents; Nifedipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; Opioid Peptides; Patch-Clamp Techniques; Peptides; Receptors, Opioid; Receptors, Purinergic; Spider Venoms; Suramin; Virulence Factors, Bordetella

1998
Analgesic action of loperamide, an opioid agonist, and its blocking action on voltage-dependent Ca2+ channels.
    Neuroscience research, 2003, Volume: 46, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analgesia; Analgesics; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; Fluorescent Dyes; Fura-2; Loperamide; Mice; Naloxone; Narcotic Antagonists; Pain; Pain Measurement; Posterior Horn Cells; Potassium Chloride

2003
Influence of naloxone on catecholamine release evoked by nicotinic receptor stimulation in the isolated rat adrenal gland.
    Archives of pharmacal research, 2005, Volume: 28, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenal Glands; Animals; Catecholamines; Dimethylphenylpiperazinium Iodide; Dose-Response Relationship, Drug; Enkephalin, Methionine; Indoles; Male; Naloxone; Perfusion; Potassium; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Stimulation, Chemical; Time Factors

2005
L-type calcium channels and μ-opioid receptors are involved in mediating the anti-inflammatory effects of naloxone.
    The Journal of surgical research, 2011, May-15, Volume: 167, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Inflammatory Agents; Calcium Channels, L-Type; Cell Line; Chemokine CXCL2; Fentanyl; Inflammation; Interleukin-1beta; Interleukin-6; Lipopolysaccharides; Macrophages; Mice; Models, Animal; Morphine; Naloxone; NF-kappa B; Receptors, Opioid, mu

2011