bay-k-8644 has been researched along with histamine in 39 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 13 (33.33) | 18.7374 |
1990's | 18 (46.15) | 18.2507 |
2000's | 4 (10.26) | 29.6817 |
2010's | 4 (10.26) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
Babycos, CR; Hood, JS; Ibrahim, IN; Kadowitz, PJ; McMahon, TJ; Nossaman, BD; Ragheb, MS | 1 |
Bhattacharya, J; Bhattacharya, S | 1 |
Rembold, CM | 1 |
Krielaart, MJ; van Buuren, KJ; Veenstra, DM | 1 |
Chambers, TJ; Gilgenkrantz, JL; Hall, TJ | 1 |
Casteels, R; Droogmans, G; Himpens, B | 1 |
Adeagbo, AS; Triggle, CR | 1 |
Chang, KJ; Collins, MA; Xu, SF | 1 |
Allen, SL; Foster, RW; Small, RC; Towart, R | 1 |
Advenier, C; Naline, E; Renier, A | 1 |
Hattori, Y; Kanno, M; Nakaya, H; Tohse, N | 1 |
Armour, CL; Black, JL; Johnson, PR; Marthan, R | 2 |
Godfraind, T; Hardy, JP; Morel, N | 1 |
Baik, YH; Koch, WJ; Schwartz, A; Williams, JS | 1 |
Kennedy, RH; Perlmutter, B; Seifen, E; Soulsby, M | 1 |
Rasmussen, H; Takuwa, Y | 1 |
Armour, C; Black, J; Johnson, P; Marthan, R | 1 |
Hai, CM; Murphy, RA; Ratz, PH | 1 |
Bevan, JA; Dowd, AL; Germann, P; Laher, I | 1 |
Goto, K; Ishikawa, T; Kasuya, Y; Kimura, S; Masaki, T; Yanagisawa, M | 1 |
Bevan, JA; Xiao, XH | 1 |
Ishimura, Y; Katoh, I; Masuda, Y; Oka, M; Yoshizumi, M | 1 |
Egashira, K; Fukai, T; Ito, A; Nakaike, R; Sakata, M; Shimokawa, H; Takayanagi, T; Takeshita, A | 1 |
Borges, R | 1 |
Egashira, K; Fukumoto, Y; Ito, A; Kadokami, T; Shimokawa, H; Takayanagi, T; Takeshita, A | 1 |
Dessy, C; Godfraind, T | 1 |
Bufler, J; Choi, GC; Franke, C; Prinz, C; Schepp, W | 1 |
Marley, PD; O'Farrell, M | 1 |
Athmann, C; Kang, T; Sachs, G; Walsh, JH; Zeng, N | 1 |
Horio, S; Moritoki, H; Nagare, T | 1 |
Koizumi, N; Masui, H; Siogawa, K; Wakabayashi, I | 1 |
Arias-Montaño, JA; García, L; Guerrero-Hernández, A; Rueda, A; Soria-Jasso, LE | 1 |
Bernsand, M; Björkqvist, M; Eliasson, L; Håkanson, R; Lindström, E | 1 |
Morris, CE; Skalak, TC | 1 |
Aboulafia, J; da Silva, BA; Ferreira, AT; Martins, IR; Nouailhetas, VL; Paredes-Gamero, EJ; Rigoni, VL; Santos, RF; Silva, MS; Tavares, JF; Travassos, RA | 1 |
Di, F; Huang, J; Li, P; Zhai, H | 1 |
Cavalcante, Fde A; Correia, AC; da Silva, BA; de Souza, IL; Paredes-Gamero, EJ; Santos, BV; Silva, Mda C; Vasconcelos, LH | 1 |
39 other study(ies) available for bay-k-8644 and histamine
Article | Year |
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Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
Blockade of thromboxane/endoperoxide receptor-mediated responses in the pulmonary vascular bed of the cat by sulotroban.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Angiotensin II; Animals; Arachidonic Acid; Blood Pressure; Cats; Endothelins; Female; Histamine; Lung; Male; Norepinephrine; Platelet Activating Factor; Prostaglandin Endoperoxides, Synthetic; Prostaglandins; Receptors, Prostaglandin; Receptors, Thromboxane; Serotonin; Sulfonamides | 1992 |
Segmental vascular responses to voltage-gated calcium channel potentiation in rat lung.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arginine; Blood Pressure; Calcium; Calcium Channels; Histamine; In Vitro Techniques; Indomethacin; Ion Channel Gating; Lung; omega-N-Methylarginine; Potassium; Rats; Rats, Sprague-Dawley; Vasoconstriction | 1992 |
Modulation of the [Ca2+] sensitivity of myosin phosphorylation in intact swine arterial smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Endothelins; Histamine; Isometric Contraction; Muscle, Smooth, Vascular; Phosphorylation; Potassium Chloride; Sodium Fluoride; Swine | 1990 |
Mechanism of action of H2-antagonists on histamine- or dimaprit-stimulated H2-receptors of spontaneously beating guinea-pig atrium.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cimetidine; Dimaprit; Famotidine; Female; Guinea Pigs; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Radioligand Assay; Ranitidine; Receptors, Histamine H2; Thiourea | 1990 |
Regulation of calcitonin release from the 6.23 rat C-cell line by cyclic nucleotide analogues and pharmacological mediators.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcitonin; Carcinoma; Dibutyryl Cyclic GMP; Dinoprostone; Histamine; Isoproterenol; Rats; Thyroid Neoplasms; Tumor Cells, Cultured | 1991 |
Carbachol-induced nonspecific desensitization in guinea-pig ileum.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atropine; Biological Transport, Active; Calcium; Carbachol; Cyclic AMP; Female; Guinea Pigs; Histamine; Ileum; Male; Muscle Contraction; Muscle, Smooth; Ouabain; Potassium; Prostaglandins; Sodium; Substance P; Temperature; Virulence Factors, Bordetella | 1991 |
Effects of some inorganic divalent cations and protein kinase C inhibitors on endothelium-dependent relaxation in rat isolated aorta and mesenteric arteries.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Alkaloids; Animals; Aorta, Thoracic; Calcium; Cations, Divalent; Endothelium, Vascular; Histamine; In Vitro Techniques; Isoquinolines; Male; Mesenteric Arteries; Muscle Relaxation; Muscle, Smooth, Vascular; Nitrendipine; Nitroprusside; Norepinephrine; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Staurosporine | 1991 |
Phorbol esters induce oscillatory contractions of intestinal smooth muscles.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atropine; Bradykinin; Calcium; Calcium Channel Blockers; Dihydropyridines; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Depolarizing Agents; Parasympatholytics; Parasympathomimetics; Phorbol Esters; Potassium Chloride; Protein Kinase C | 1991 |
The effects of the dihydropyridine Bay K 8644 in guinea-pig isolated trachealis.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium Channel Blockers; Calcium Chloride; Electrophysiology; Female; Guinea Pigs; Histamine; In Vitro Techniques; Lanthanum; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Potassium Chloride; Tetraethylammonium; Tetraethylammonium Compounds; Trachea | 1985 |
Effects of Bay K 8644 on contraction of the human isolated bronchus and guinea-pig isolated trachea.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Bronchi; Calcium; Calcium Channel Blockers; Guinea Pigs; Histamine; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nicardipine; Nifedipine; Potassium Chloride; Trachea; Verapamil | 1986 |
Voltage-dependent effects of YC-170, a dihydropyridine calcium channel modulator, in cardiovascular tissues.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Cardiovascular System; Female; Guinea Pigs; Heart; Histamine; In Vitro Techniques; Ion Channels; Isoproterenol; Male; Muscle, Smooth; Nifedipine; Potassium; Rabbits; Sinoatrial Node; Tetraethylammonium Compounds | 1986 |
The calcium channel agonist BAY K8644 enhances the responsiveness of human airway muscle to KCl and histamine but not to carbachol.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aged; Calcium; Calcium Channel Blockers; Carbachol; Drug Synergism; Histamine; Humans; In Vitro Techniques; Ion Channels; Lung; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Potassium Chloride | 1987 |
Histamine-operated calcium channels in intestinal smooth muscle of the guinea-pig.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Electrophysiology; Guinea Pigs; Histamine; In Vitro Techniques; Intestinal Mucosa; Intestines; Ion Channels; Muscle, Smooth, Vascular; Nifedipine | 1987 |
A possible role for the endothelium in porcine coronary smooth muscle responses to dihydropyridine calcium channel modulators.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Endothelium; Histamine; Isomerism; Isosorbide Dinitrate; Muscle, Smooth, Vascular; Nicotinic Acids; Oxadiazoles; Swine; Vasoconstriction; Vasodilation | 1987 |
Effects of norepinephrine on BAY K-8644-induced contraction in porcine coronary artery.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Coronary Vessels; Histamine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Swine | 1987 |
Measurement of cytoplasmic free Ca2+ concentration in rabbit aorta using the photoprotein, aequorin. Effect of atrial natriuretic peptide on agonist-induced Ca2+ signal generation.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aequorin; Angiotensin II; Animals; Aorta, Thoracic; Atrial Natriuretic Factor; Caffeine; Calcium; Histamine; Kinetics; Luminescent Proteins; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Rabbits | 1987 |
Is airway hyperresponsiveness a smooth muscle abnormality?
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Bronchi; Bronchial Spasm; Calcium; Carbachol; Histamine; Humans; Immunization; In Vitro Techniques; Ion Channels; Muscle Contraction; Muscle, Smooth | 1988 |
Dependence of stress on cross-bridge phosphorylation in vascular smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Ethers; Histamine; Ionomycin; Kinetics; Muscle Contraction; Muscle, Smooth, Vascular; Myosins; Phorbol 12,13-Dibutyrate; Phosphoproteins; Potassium; Swine | 1989 |
Sensitization alters contractile responses and calcium influx in human airway smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aged; Bronchi; Calcium; Carbachol; Female; Histamine; Humans; Immunization; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Potassium Chloride | 1989 |
The selective potentiation of noradrenaline-induced tone by Bay K 8644 in the rabbit basilar artery.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Basilar Artery; Drug Synergism; Histamine; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Rabbits | 1989 |
Mechanism of contraction to endothelin in isolated porcine coronary artery.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium; Calcium Channels; Coronary Vessels; Dinoprost; Endothelins; Endothelium, Vascular; Histamine; In Vitro Techniques; Kinetics; Membrane Potentials; Muscle, Smooth, Vascular; Nicardipine; Peptides; Potassium Chloride; Receptors, Nicotinic; Swine; Vasoconstriction | 1989 |
Pharmacological evidence that flow- and potassium-induced contraction of rabbit facial vein may involve the same calcium entry pathway.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Face; Histamine; In Vitro Techniques; Male; Potassium; Rabbits; Regional Blood Flow; Vasoconstriction; Veins | 1994 |
Effects of the potassium channel openers cromakalim and pinacidil on catecholamine secretion and calcium mobilization in cultured bovine adrenal chromaffin cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Barium; Benzopyrans; Bradykinin; Calcimycin; Calcium; Carbachol; Catecholamines; Cattle; Cells, Cultured; Cromakalim; Guanidines; Histamine; Pinacidil; Potassium; Potassium Channels; Pyrroles; Rubidium Radioisotopes | 1994 |
Role of protein kinase C-mediated pathway in the pathogenesis of coronary artery spasm in a swine model.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Calcium; Coronary Vasospasm; Disease Models, Animal; Histamine; Male; Phorbol 12,13-Dibutyrate; Protein Kinase C; Serotonin; Staurosporine; Swine; Swine, Miniature | 1994 |
Ionic mechanisms involved in the secretory effects of histamine in the rat adrenal medulla.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Calcium; Catecholamines; Female; Histamine; In Vitro Techniques; Nitrendipine; Rats; Rats, Sprague-Dawley; Sodium | 1993 |
Coronary artery spasm does not depend on the intracellular calcium store but is substantially mediated by the protein kinase C-mediated pathway in a swine model with interleukin-1 beta in vivo.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium-Transporting ATPases; Coronary Vasospasm; Cytosol; Enzyme Activation; Histamine; Interleukin-1; Male; Muscle, Smooth, Vascular; Nifedipine; Phorbol 12,13-Dibutyrate; Protein Kinase C; Ryanodine; Sarcoplasmic Reticulum; Serotonin; Sphingosine; Staurosporine; Swine; Terpenes; Thapsigargin | 1996 |
The effect of L-type calcium channel modulators on the mobilization of intracellular calcium stores in guinea-pig intestinal smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Diazoxide; Fura-2; Guinea Pigs; Histamine; Ileum; Isometric Contraction; Muscle, Smooth; Nimodipine; Ryanodine; Thapsigargin | 1996 |
Voltage-gated Ca2+ currents in rat gastric enterochromaffin-like cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Enterochromaffin-like Cells; Female; Gastric Fundus; Gastric Mucosa; Histamine; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Verapamil | 1998 |
Different contributions of voltage-sensitive Ca2+ channels to histamine-induced catecholamine release and tyrosine hydroxylase activation in bovine adrenal chromaffin cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Glands; Animals; Calcium Channel Blockers; Calcium Channels; Catecholamines; Cattle; Chromaffin Cells; Dose-Response Relationship, Drug; GTP-Binding Proteins; Histamine; Nitrendipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; Peptides; Spider Venoms; Tetrodotoxin; Tyrosine 3-Monooxygenase | 1999 |
Role of neuropeptide-sensitive L-type Ca(2+) channels in histamine release in gastric enterochromaffin-like cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylate Cyclase Toxin; Animals; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Dihydropyridines; DNA Primers; Enterochromaffin-like Cells; Galanin; Gastric Acid; Gastric Mucosa; Gastrins; Gene Expression; GTP-Binding Proteins; Histamine; Histamine Release; Membrane Potentials; Neuropeptides; Neurotransmitter Agents; omega-Conotoxin GVIA; Peptide YY; Pertussis Toxin; Pituitary Adenylate Cyclase-Activating Polypeptide; Potassium; Rabbits; Rats; Receptors, Histamine H2; Somatostatin; Stomach; Tetraethylammonium; Virulence Factors, Bordetella | 1999 |
Enhancement of acetylcholine-induced desensitization of guinea-pig ileal longitudinal muscle in Ca2+-free conditions.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium; Calcium Channel Agonists; Desensitization, Immunologic; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Histamine; Ileum; Ion Channel Gating; Male; Muscle, Smooth; Protein Kinase C; Vasodilator Agents | 1999 |
Diminished inibitory action of ethanol on the contraction of gallbladder isolated from chronically ethanol-fed Guinea pigs.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Body Weight; Calcium Channel Agonists; Dose-Response Relationship, Drug; Ethanol; Gallbladder; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Phorbol 12,13-Dibutyrate; Potassium Chloride; Verapamil | 2002 |
The initial inositol 1,4,5-trisphosphate response induced by histamine is strongly amplified by Ca(2+) release from internal stores in smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Androstadienes; Animals; Calcium; Carbachol; Cimetidine; Extracellular Space; Guinea Pigs; Histamine; Histamine Agonists; Inositol 1,4,5-Trisphosphate; Kinetics; Lithium; Muscle, Smooth; Pyrilamine; Ryanodine; Thapsigargin; Type C Phospholipases; Urinary Bladder; Wortmannin | 2002 |
Somatostatin, misoprostol and galanin inhibit gastrin- and PACAP-stimulated secretion of histamine and pancreastatin from ECL cells by blocking specific Ca2+ channels.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Ulcer Agents; Calcium; Calcium Channels; Cells, Cultured; Chromogranin A; Dose-Response Relationship, Drug; Enterochromaffin-like Cells; Exocytosis; Galanin; Gastrins; Histamine; Hormones; Male; Microscopy, Video; Misoprostol; Models, Biological; Nifedipine; Pancreatic Hormones; Peptides, Cyclic; Rats; Rats, Sprague-Dawley; Somatostatin; Time Factors | 2005 |
Acute exposure to a moderate strength static magnetic field reduces edema formation in rats.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arginine; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Carrageenan; Disease Models, Animal; Dose-Response Relationship, Radiation; Edema; Electromagnetic Fields; Histamine; Inflammation; Male; Muscle, Smooth, Vascular; Nitric Oxide; Nitric Oxide Synthase; Rats; Rats, Sprague-Dawley; Severity of Illness Index; Signal Transduction; Time Factors | 2008 |
Ent-7α-acetoxytrachyloban-18-oic acid and ent-7α-hydroxytrachyloban-18-oic acid from Xylopia langsdorfiana A. St-Hil. & Tul. modulate K(+) and Ca(2+) channels to reduce cytosolic calcium concentration on guinea pig ileum.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Calcium Chloride; Cells, Cultured; Cytosol; Diterpenes; Dose-Response Relationship, Drug; Drug Interactions; Female; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Parasympatholytics; Potassium Channels; Xylopia | 2012 |
Effects of dehydroeffusol on spasmogen-induced contractile responses of rat intestinal smooth muscles.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Histamine; Jejunum; Magnoliopsida; Male; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Phenanthrenes; Pilocarpine; Plant Extracts; Potassium Chloride; Rats, Sprague-Dawley | 2014 |
Flavonoid galetin 3,6-dimethyl ether attenuates guinea pig ileum contraction through K(+) channel activation and decrease in cytosolic calcium concentration.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Apamin; Calcium; Calcium Chloride; Carbachol; Cell Survival; Cesium; Chlorides; Flavonoids; Glyburide; Guinea Pigs; Histamine; Histamine Antagonists; Ileum; Muscle Cells; Muscle Contraction; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Tetraethylammonium | 2015 |