bay-k-8644 and histamine

bay-k-8644 has been researched along with histamine in 39 studies

Research

Studies (39)

TimeframeStudies, this research(%)All Research%
pre-199013 (33.33)18.7374
1990's18 (46.15)18.2507
2000's4 (10.26)29.6817
2010's4 (10.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Babycos, CR; Hood, JS; Ibrahim, IN; Kadowitz, PJ; McMahon, TJ; Nossaman, BD; Ragheb, MS1
Bhattacharya, J; Bhattacharya, S1
Rembold, CM1
Krielaart, MJ; van Buuren, KJ; Veenstra, DM1
Chambers, TJ; Gilgenkrantz, JL; Hall, TJ1
Casteels, R; Droogmans, G; Himpens, B1
Adeagbo, AS; Triggle, CR1
Chang, KJ; Collins, MA; Xu, SF1
Allen, SL; Foster, RW; Small, RC; Towart, R1
Advenier, C; Naline, E; Renier, A1
Hattori, Y; Kanno, M; Nakaya, H; Tohse, N1
Armour, CL; Black, JL; Johnson, PR; Marthan, R2
Godfraind, T; Hardy, JP; Morel, N1
Baik, YH; Koch, WJ; Schwartz, A; Williams, JS1
Kennedy, RH; Perlmutter, B; Seifen, E; Soulsby, M1
Rasmussen, H; Takuwa, Y1
Armour, C; Black, J; Johnson, P; Marthan, R1
Hai, CM; Murphy, RA; Ratz, PH1
Bevan, JA; Dowd, AL; Germann, P; Laher, I1
Goto, K; Ishikawa, T; Kasuya, Y; Kimura, S; Masaki, T; Yanagisawa, M1
Bevan, JA; Xiao, XH1
Ishimura, Y; Katoh, I; Masuda, Y; Oka, M; Yoshizumi, M1
Egashira, K; Fukai, T; Ito, A; Nakaike, R; Sakata, M; Shimokawa, H; Takayanagi, T; Takeshita, A1
Borges, R1
Egashira, K; Fukumoto, Y; Ito, A; Kadokami, T; Shimokawa, H; Takayanagi, T; Takeshita, A1
Dessy, C; Godfraind, T1
Bufler, J; Choi, GC; Franke, C; Prinz, C; Schepp, W1
Marley, PD; O'Farrell, M1
Athmann, C; Kang, T; Sachs, G; Walsh, JH; Zeng, N1
Horio, S; Moritoki, H; Nagare, T1
Koizumi, N; Masui, H; Siogawa, K; Wakabayashi, I1
Arias-Montaño, JA; García, L; Guerrero-Hernández, A; Rueda, A; Soria-Jasso, LE1
Bernsand, M; Björkqvist, M; Eliasson, L; Håkanson, R; Lindström, E1
Morris, CE; Skalak, TC1
Aboulafia, J; da Silva, BA; Ferreira, AT; Martins, IR; Nouailhetas, VL; Paredes-Gamero, EJ; Rigoni, VL; Santos, RF; Silva, MS; Tavares, JF; Travassos, RA1
Di, F; Huang, J; Li, P; Zhai, H1
Cavalcante, Fde A; Correia, AC; da Silva, BA; de Souza, IL; Paredes-Gamero, EJ; Santos, BV; Silva, Mda C; Vasconcelos, LH1

Other Studies

39 other study(ies) available for bay-k-8644 and histamine

ArticleYear
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Blockade of thromboxane/endoperoxide receptor-mediated responses in the pulmonary vascular bed of the cat by sulotroban.
    European journal of pharmacology, 1992, Mar-17, Volume: 213, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Angiotensin II; Animals; Arachidonic Acid; Blood Pressure; Cats; Endothelins; Female; Histamine; Lung; Male; Norepinephrine; Platelet Activating Factor; Prostaglandin Endoperoxides, Synthetic; Prostaglandins; Receptors, Prostaglandin; Receptors, Thromboxane; Serotonin; Sulfonamides

1992
Segmental vascular responses to voltage-gated calcium channel potentiation in rat lung.
    Journal of applied physiology (Bethesda, Md. : 1985), 1992, Volume: 73, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arginine; Blood Pressure; Calcium; Calcium Channels; Histamine; In Vitro Techniques; Indomethacin; Ion Channel Gating; Lung; omega-N-Methylarginine; Potassium; Rats; Rats, Sprague-Dawley; Vasoconstriction

1992
Modulation of the [Ca2+] sensitivity of myosin phosphorylation in intact swine arterial smooth muscle.
    The Journal of physiology, 1990, Volume: 429

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Endothelins; Histamine; Isometric Contraction; Muscle, Smooth, Vascular; Phosphorylation; Potassium Chloride; Sodium Fluoride; Swine

1990
Mechanism of action of H2-antagonists on histamine- or dimaprit-stimulated H2-receptors of spontaneously beating guinea-pig atrium.
    Agents and actions, 1990, Volume: 31, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cimetidine; Dimaprit; Famotidine; Female; Guinea Pigs; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Radioligand Assay; Ranitidine; Receptors, Histamine H2; Thiourea

1990
Regulation of calcitonin release from the 6.23 rat C-cell line by cyclic nucleotide analogues and pharmacological mediators.
    Experientia, 1991, Oct-15, Volume: 47, Issue:10

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcitonin; Carcinoma; Dibutyryl Cyclic GMP; Dinoprostone; Histamine; Isoproterenol; Rats; Thyroid Neoplasms; Tumor Cells, Cultured

1991
Carbachol-induced nonspecific desensitization in guinea-pig ileum.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atropine; Biological Transport, Active; Calcium; Carbachol; Cyclic AMP; Female; Guinea Pigs; Histamine; Ileum; Male; Muscle Contraction; Muscle, Smooth; Ouabain; Potassium; Prostaglandins; Sodium; Substance P; Temperature; Virulence Factors, Bordetella

1991
Effects of some inorganic divalent cations and protein kinase C inhibitors on endothelium-dependent relaxation in rat isolated aorta and mesenteric arteries.
    Journal of cardiovascular pharmacology, 1991, Volume: 18, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Alkaloids; Animals; Aorta, Thoracic; Calcium; Cations, Divalent; Endothelium, Vascular; Histamine; In Vitro Techniques; Isoquinolines; Male; Mesenteric Arteries; Muscle Relaxation; Muscle, Smooth, Vascular; Nitrendipine; Nitroprusside; Norepinephrine; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Staurosporine

1991
Phorbol esters induce oscillatory contractions of intestinal smooth muscles.
    European journal of pharmacology, 1991, Aug-29, Volume: 201, Issue:2-3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atropine; Bradykinin; Calcium; Calcium Channel Blockers; Dihydropyridines; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Depolarizing Agents; Parasympatholytics; Parasympathomimetics; Phorbol Esters; Potassium Chloride; Protein Kinase C

1991
The effects of the dihydropyridine Bay K 8644 in guinea-pig isolated trachealis.
    British journal of pharmacology, 1985, Volume: 86, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium Channel Blockers; Calcium Chloride; Electrophysiology; Female; Guinea Pigs; Histamine; In Vitro Techniques; Lanthanum; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Potassium Chloride; Tetraethylammonium; Tetraethylammonium Compounds; Trachea

1985
Effects of Bay K 8644 on contraction of the human isolated bronchus and guinea-pig isolated trachea.
    British journal of pharmacology, 1986, Volume: 88, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Bronchi; Calcium; Calcium Channel Blockers; Guinea Pigs; Histamine; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nicardipine; Nifedipine; Potassium Chloride; Trachea; Verapamil

1986
Voltage-dependent effects of YC-170, a dihydropyridine calcium channel modulator, in cardiovascular tissues.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Cardiovascular System; Female; Guinea Pigs; Heart; Histamine; In Vitro Techniques; Ion Channels; Isoproterenol; Male; Muscle, Smooth; Nifedipine; Potassium; Rabbits; Sinoatrial Node; Tetraethylammonium Compounds

1986
The calcium channel agonist BAY K8644 enhances the responsiveness of human airway muscle to KCl and histamine but not to carbachol.
    The American review of respiratory disease, 1987, Volume: 135, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aged; Calcium; Calcium Channel Blockers; Carbachol; Drug Synergism; Histamine; Humans; In Vitro Techniques; Ion Channels; Lung; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Potassium Chloride

1987
Histamine-operated calcium channels in intestinal smooth muscle of the guinea-pig.
    European journal of pharmacology, 1987, Mar-03, Volume: 135, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Electrophysiology; Guinea Pigs; Histamine; In Vitro Techniques; Intestinal Mucosa; Intestines; Ion Channels; Muscle, Smooth, Vascular; Nifedipine

1987
A possible role for the endothelium in porcine coronary smooth muscle responses to dihydropyridine calcium channel modulators.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Endothelium; Histamine; Isomerism; Isosorbide Dinitrate; Muscle, Smooth, Vascular; Nicotinic Acids; Oxadiazoles; Swine; Vasoconstriction; Vasodilation

1987
Effects of norepinephrine on BAY K-8644-induced contraction in porcine coronary artery.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 285, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Coronary Vessels; Histamine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Swine

1987
Measurement of cytoplasmic free Ca2+ concentration in rabbit aorta using the photoprotein, aequorin. Effect of atrial natriuretic peptide on agonist-induced Ca2+ signal generation.
    The Journal of clinical investigation, 1987, Volume: 80, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aequorin; Angiotensin II; Animals; Aorta, Thoracic; Atrial Natriuretic Factor; Caffeine; Calcium; Histamine; Kinetics; Luminescent Proteins; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Rabbits

1987
Is airway hyperresponsiveness a smooth muscle abnormality?
    Progress in clinical and biological research, 1988, Volume: 263

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Bronchi; Bronchial Spasm; Calcium; Carbachol; Histamine; Humans; Immunization; In Vitro Techniques; Ion Channels; Muscle Contraction; Muscle, Smooth

1988
Dependence of stress on cross-bridge phosphorylation in vascular smooth muscle.
    The American journal of physiology, 1989, Volume: 256, Issue:1 Pt 1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Ethers; Histamine; Ionomycin; Kinetics; Muscle Contraction; Muscle, Smooth, Vascular; Myosins; Phorbol 12,13-Dibutyrate; Phosphoproteins; Potassium; Swine

1989
Sensitization alters contractile responses and calcium influx in human airway smooth muscle.
    The Journal of allergy and clinical immunology, 1989, Volume: 84, Issue:4 Pt 1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aged; Bronchi; Calcium; Carbachol; Female; Histamine; Humans; Immunization; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Potassium Chloride

1989
The selective potentiation of noradrenaline-induced tone by Bay K 8644 in the rabbit basilar artery.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1989, Volume: 9, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Basilar Artery; Drug Synergism; Histamine; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Rabbits

1989
Mechanism of contraction to endothelin in isolated porcine coronary artery.
    The American journal of physiology, 1989, Volume: 257, Issue:6 Pt 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium; Calcium Channels; Coronary Vessels; Dinoprost; Endothelins; Endothelium, Vascular; Histamine; In Vitro Techniques; Kinetics; Membrane Potentials; Muscle, Smooth, Vascular; Nicardipine; Peptides; Potassium Chloride; Receptors, Nicotinic; Swine; Vasoconstriction

1989
Pharmacological evidence that flow- and potassium-induced contraction of rabbit facial vein may involve the same calcium entry pathway.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Face; Histamine; In Vitro Techniques; Male; Potassium; Rabbits; Regional Blood Flow; Vasoconstriction; Veins

1994
Effects of the potassium channel openers cromakalim and pinacidil on catecholamine secretion and calcium mobilization in cultured bovine adrenal chromaffin cells.
    Biochemical pharmacology, 1994, May-18, Volume: 47, Issue:10

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Barium; Benzopyrans; Bradykinin; Calcimycin; Calcium; Carbachol; Catecholamines; Cattle; Cells, Cultured; Cromakalim; Guanidines; Histamine; Pinacidil; Potassium; Potassium Channels; Pyrroles; Rubidium Radioisotopes

1994
Role of protein kinase C-mediated pathway in the pathogenesis of coronary artery spasm in a swine model.
    Circulation, 1994, Volume: 90, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Calcium; Coronary Vasospasm; Disease Models, Animal; Histamine; Male; Phorbol 12,13-Dibutyrate; Protein Kinase C; Serotonin; Staurosporine; Swine; Swine, Miniature

1994
Ionic mechanisms involved in the secretory effects of histamine in the rat adrenal medulla.
    European journal of pharmacology, 1993, Sep-14, Volume: 241, Issue:2-3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Calcium; Catecholamines; Female; Histamine; In Vitro Techniques; Nitrendipine; Rats; Rats, Sprague-Dawley; Sodium

1993
Coronary artery spasm does not depend on the intracellular calcium store but is substantially mediated by the protein kinase C-mediated pathway in a swine model with interleukin-1 beta in vivo.
    Circulation, 1996, Jul-15, Volume: 94, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium-Transporting ATPases; Coronary Vasospasm; Cytosol; Enzyme Activation; Histamine; Interleukin-1; Male; Muscle, Smooth, Vascular; Nifedipine; Phorbol 12,13-Dibutyrate; Protein Kinase C; Ryanodine; Sarcoplasmic Reticulum; Serotonin; Sphingosine; Staurosporine; Swine; Terpenes; Thapsigargin

1996
The effect of L-type calcium channel modulators on the mobilization of intracellular calcium stores in guinea-pig intestinal smooth muscle.
    British journal of pharmacology, 1996, Volume: 119, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Diazoxide; Fura-2; Guinea Pigs; Histamine; Ileum; Isometric Contraction; Muscle, Smooth; Nimodipine; Ryanodine; Thapsigargin

1996
Voltage-gated Ca2+ currents in rat gastric enterochromaffin-like cells.
    The American journal of physiology, 1998, Volume: 274, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Enterochromaffin-like Cells; Female; Gastric Fundus; Gastric Mucosa; Histamine; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Verapamil

1998
Different contributions of voltage-sensitive Ca2+ channels to histamine-induced catecholamine release and tyrosine hydroxylase activation in bovine adrenal chromaffin cells.
    Cell calcium, 1999, Volume: 25, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Glands; Animals; Calcium Channel Blockers; Calcium Channels; Catecholamines; Cattle; Chromaffin Cells; Dose-Response Relationship, Drug; GTP-Binding Proteins; Histamine; Nitrendipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; Peptides; Spider Venoms; Tetrodotoxin; Tyrosine 3-Monooxygenase

1999
Role of neuropeptide-sensitive L-type Ca(2+) channels in histamine release in gastric enterochromaffin-like cells.
    The American journal of physiology, 1999, Volume: 277, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylate Cyclase Toxin; Animals; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Dihydropyridines; DNA Primers; Enterochromaffin-like Cells; Galanin; Gastric Acid; Gastric Mucosa; Gastrins; Gene Expression; GTP-Binding Proteins; Histamine; Histamine Release; Membrane Potentials; Neuropeptides; Neurotransmitter Agents; omega-Conotoxin GVIA; Peptide YY; Pertussis Toxin; Pituitary Adenylate Cyclase-Activating Polypeptide; Potassium; Rabbits; Rats; Receptors, Histamine H2; Somatostatin; Stomach; Tetraethylammonium; Virulence Factors, Bordetella

1999
Enhancement of acetylcholine-induced desensitization of guinea-pig ileal longitudinal muscle in Ca2+-free conditions.
    Journal of autonomic pharmacology, 1999, Volume: 19, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium; Calcium Channel Agonists; Desensitization, Immunologic; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Histamine; Ileum; Ion Channel Gating; Male; Muscle, Smooth; Protein Kinase C; Vasodilator Agents

1999
Diminished inibitory action of ethanol on the contraction of gallbladder isolated from chronically ethanol-fed Guinea pigs.
    Pharmacology, 2002, Volume: 65, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Body Weight; Calcium Channel Agonists; Dose-Response Relationship, Drug; Ethanol; Gallbladder; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Phorbol 12,13-Dibutyrate; Potassium Chloride; Verapamil

2002
The initial inositol 1,4,5-trisphosphate response induced by histamine is strongly amplified by Ca(2+) release from internal stores in smooth muscle.
    Cell calcium, 2002, Volume: 31, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Androstadienes; Animals; Calcium; Carbachol; Cimetidine; Extracellular Space; Guinea Pigs; Histamine; Histamine Agonists; Inositol 1,4,5-Trisphosphate; Kinetics; Lithium; Muscle, Smooth; Pyrilamine; Ryanodine; Thapsigargin; Type C Phospholipases; Urinary Bladder; Wortmannin

2002
Somatostatin, misoprostol and galanin inhibit gastrin- and PACAP-stimulated secretion of histamine and pancreastatin from ECL cells by blocking specific Ca2+ channels.
    Regulatory peptides, 2005, Aug-15, Volume: 130, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Ulcer Agents; Calcium; Calcium Channels; Cells, Cultured; Chromogranin A; Dose-Response Relationship, Drug; Enterochromaffin-like Cells; Exocytosis; Galanin; Gastrins; Histamine; Hormones; Male; Microscopy, Video; Misoprostol; Models, Biological; Nifedipine; Pancreatic Hormones; Peptides, Cyclic; Rats; Rats, Sprague-Dawley; Somatostatin; Time Factors

2005
Acute exposure to a moderate strength static magnetic field reduces edema formation in rats.
    American journal of physiology. Heart and circulatory physiology, 2008, Volume: 294, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arginine; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Carrageenan; Disease Models, Animal; Dose-Response Relationship, Radiation; Edema; Electromagnetic Fields; Histamine; Inflammation; Male; Muscle, Smooth, Vascular; Nitric Oxide; Nitric Oxide Synthase; Rats; Rats, Sprague-Dawley; Severity of Illness Index; Signal Transduction; Time Factors

2008
Ent-7α-acetoxytrachyloban-18-oic acid and ent-7α-hydroxytrachyloban-18-oic acid from Xylopia langsdorfiana A. St-Hil. & Tul. modulate K(+) and Ca(2+) channels to reduce cytosolic calcium concentration on guinea pig ileum.
    European journal of pharmacology, 2012, Mar-05, Volume: 678, Issue:1-3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Calcium Chloride; Cells, Cultured; Cytosol; Diterpenes; Dose-Response Relationship, Drug; Drug Interactions; Female; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Parasympatholytics; Potassium Channels; Xylopia

2012
Effects of dehydroeffusol on spasmogen-induced contractile responses of rat intestinal smooth muscles.
    Planta medica, 2014, Volume: 80, Issue:12

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Histamine; Jejunum; Magnoliopsida; Male; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Phenanthrenes; Pilocarpine; Plant Extracts; Potassium Chloride; Rats, Sprague-Dawley

2014
Flavonoid galetin 3,6-dimethyl ether attenuates guinea pig ileum contraction through K(+) channel activation and decrease in cytosolic calcium concentration.
    European journal of pharmacology, 2015, Nov-15, Volume: 767

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Apamin; Calcium; Calcium Chloride; Carbachol; Cell Survival; Cesium; Chlorides; Flavonoids; Glyburide; Guinea Pigs; Histamine; Histamine Antagonists; Ileum; Muscle Cells; Muscle Contraction; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Tetraethylammonium

2015