bay-k-8644 has been researched along with glyburide in 29 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (3.45) | 18.7374 |
1990's | 13 (44.83) | 18.2507 |
2000's | 8 (27.59) | 29.6817 |
2010's | 7 (24.14) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J | 1 |
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
Huang, TF; Ko, FN; Su, MJ; Teng, CM; Wang, ML; Wu, TS; Yu, SM | 1 |
Eltze, M | 1 |
Asano, M; Masuzawa-Ito, K; Matsuda, T; Oyama, H; Shibuya, M; Sugita, K; Suzuki, Y | 1 |
Chiba, S; Furukawa, Y; Inoue, Y; Oguchi, T; Sawaki, S | 1 |
Cailmail, S; Gaudin, C; Hartleb, M; Lebrec, D; Moreau, R | 1 |
Allescher, HD; Franck, H; Puschmann, A; Schusdziarra, V | 1 |
Maggi, CA; Meini, S; Santicioli, P | 1 |
Berkovich, A; De Stefanis, P; Guidotti, A; Impagnatiello, F | 1 |
Giuliani, S; Maggi, CA; Santicioli, P | 1 |
Champion, HC; Kadowitz, PJ | 1 |
Fuhlendorff, J; Gromada, J; Madsen, P; Springborg, J; Varming, AR | 1 |
Allescher, HD; Franck, H; Puschmann, A; Schusdziarra, V; Storr, M | 1 |
Bataille, D; Blache, P; Dalle, S; Le Brigand, L; Le-Nguyen, D | 1 |
Böhm-Pinger, MM; Dittrich, M; Fischer, IR; Fleischmann, BK; Gryshchenko, O; Hescheler, J; Igelmund, P; Soest, J; Viatchenko-Karpinski, S | 1 |
Berg Nyborg, NC; Sheykhzade, M | 1 |
Babaya, N; Hamada, Y; Ikegami, H; Kawaguchi, Y; Nojima, K; Ogihara, T; Shibata, M; Ueda, H; Yamada, K; Yamato, E | 1 |
Dennedy, MC; Houlihan, DD; Morrison, JJ | 1 |
Ito, Y; Naito, S; Teramoto, N; Tomoda, T; Yunoki, T | 1 |
He, RR; Liu, YX; Wu, YM; Xiao, L; Zhang, H | 1 |
He, RR; Liu, YX; Wang, FW; Wang, R; Wu, YM; Xiao, L | 1 |
Arcanjo, DD; Cavalcanti, SC; Oliveira, AP; Oliveira, NN; Oliveira, Rde C; Quintans-Júnior, LJ; Santos, MR; Silva-Filho, JC | 1 |
He, RR; Li, Q; Liu, S; Wu, YM; Xu, M | 1 |
Gurgul-Convey, E; Kaminski, MT; Lenzen, S | 1 |
Cavalcante, Fde A; Correia, AC; da Silva, BA; de Souza, IL; Paredes-Gamero, EJ; Santos, BV; Silva, Mda C; Vasconcelos, LH | 1 |
Guo, Q; Jin, S; Wang, R; Wu, Y; Xiao, L; Xue, H | 1 |
Lenzen, S; Teraoku, H | 1 |
29 other study(ies) available for bay-k-8644 and glyburide
Article | Year |
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Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection | 2009 |
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
Vasorelaxing effect in rat thoracic aorta caused by fraxinellone and dictamine isolated from the Chinese herb Dictamnus dasycarpus Turcz: comparison with cromakalim and Ca2+ channel blockers.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Aorta, Thoracic; Benzofurans; Benzopyrans; Calcium; Calcium Channel Blockers; Cromakalim; Cyclic AMP; Cyclic GMP; Drugs, Chinese Herbal; Female; Glyburide; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Potassium Channels; Potassium Chloride; Pyrroles; Quinolines; Rats; Rats, Inbred Strains; Verapamil | 1992 |
Competitive antagonism by glibenclamide of cromakalim inhibition of twitch contractions in rabbit vas deferens.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Benzopyrans; Calcium Channel Blockers; Cromakalim; Electric Stimulation; Glyburide; In Vitro Techniques; Male; Muscle, Smooth; Potassium Channels; Pyrroles; Rabbits; Vas Deferens | 1989 |
Functional role of charybdotoxin-sensitive K+ channels in the resting state of cerebral, coronary and mesenteric arteries of the dog.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Apamin; Arteries; Calcium; Calcium Radioisotopes; Capillary Permeability; Cerebral Arteries; Charybdotoxin; Coronary Vessels; Dogs; Female; Glyburide; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Potassium; Potassium Channels; Rubidium; Rubidium Radioisotopes; Scorpion Venoms; Sensitivity and Specificity; Tetraethylammonium; Tetraethylammonium Compounds | 1993 |
Selective inhibition by E4080, a novel bradycardic agent, of positive chronotropic responses to norepinephrine in isolated dog hearts.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atropine; Biological Clocks; Catechols; Cyclic AMP; Dogs; Glyburide; Heart; Heart Rate; Imidazoles; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Potassium Channels; Sinoatrial Node; Vasodilator Agents | 1993 |
Vascular hyporesponsiveness to endothelin 1 in rats with cirrhosis.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arginine; Blood Pressure; Dose-Response Relationship, Drug; Endothelins; Glyburide; Hemodynamics; Liver Cirrhosis, Experimental; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Rats; Rats, Sprague-Dawley | 1994 |
Functional evidence for a glibenclamide-sensitive K+ channel in rat ileal smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Benzopyrans; Calcitonin Gene-Related Peptide; Carbachol; Cromakalim; Glyburide; Ileum; Male; Muscle Contraction; Muscle, Smooth; Potassium Channels; Pyrroles; Rats; Rats, Wistar | 1994 |
Propagation of impulses in the guinea-pig ureter and its blockade by calcitonin gene-related peptide (CGRP).
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Benzopyrans; Calcitonin Gene-Related Peptide; Cromakalim; Electric Stimulation; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Pyrroles; Tetrodotoxin; Ureter | 1995 |
Inhibitory effect of ODN, a naturally occurring processing product of diazepam binding inhibitor, on secretagogues-induced insulin secretion.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Amino Acid Sequence; Animals; Calcium; Cricetinae; Cyclic AMP; Diazepam Binding Inhibitor; Dose-Response Relationship, Drug; Glucose; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Insulinoma; Ion Channels; Islets of Langerhans; Male; Molecular Sequence Data; Neuropeptides; Nitroprusside; Peptide Fragments; Rats; Time Factors; Tumor Cells, Cultured | 1995 |
CGRP inhibition of electromechanical coupling in the guinea-pig isolated renal pelvis.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Arginine; Calcitonin Gene-Related Peptide; Calcium; Carbazoles; Enzyme Inhibitors; Glyburide; Guinea Pigs; In Vitro Techniques; Indoles; Isoquinolines; Kidney Pelvis; Male; Membrane Potentials; Nitroarginine; Potassium Channels; Ryanodine; Sucrose; Sulfonamides; Terpenes; Tetrodotoxin; Thapsigargin | 1995 |
Vasodilator responses to acetylcholine, bradykinin, and substance P are mediated by a TEA-sensitive mechanism.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Albuterol; Alprostadil; Analysis of Variance; Angiotensin II; Animals; Benzopyrans; Blood Pressure; Bradykinin; Cats; Cromakalim; Endothelium, Vascular; Female; Glyburide; Heart Rate; Hindlimb; Hydrazines; Isradipine; Male; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitrogen Oxides; Nitroprusside; Norepinephrine; Penicillamine; Prostaglandin Endoperoxides, Synthetic; Pyrroles; S-Nitroso-N-Acetylpenicillamine; Substance P; Tetraethylammonium; Tetraethylammonium Compounds; Thromboxane A2; Vasoactive Intestinal Peptide; Vasodilation; Vasodilator Agents | 1997 |
Increase in [Ca2+]i and subsequent insulin release from beta TC3-cells with the L-type Ca(2+)-channel activator, FPL 64176.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Antigens, Polyomavirus Transforming; Calcium; Calcium Channel Agonists; Calcium Channels; Calcium Channels, L-Type; Dose-Response Relationship, Drug; Glyburide; Insulin; Insulin Secretion; Insulinoma; Kinetics; Mice; Mice, Transgenic; Pancreatic Neoplasms; Promoter Regions, Genetic; Pyrroles; Simian virus 40; Tumor Cells, Cultured | 1997 |
Involvement of intracellular Ca2+ stores in inhibitory effects of NO donor SIN-1 and cGMP.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Triphosphate; Animals; Apamin; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Carbachol; Charybdotoxin; Cyclic GMP; Egtazic Acid; Glyburide; Ileum; In Vitro Techniques; Indoles; Kinetics; Male; Molsidomine; Muscle Contraction; Muscle, Smooth; Peptides; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium; Tetrodotoxin; Thionucleotides | 1998 |
Miniglucagon: a local regulator of islet physiology.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Calcium Channels, L-Type; Cell Line; Cell Membrane; Glucagon; Glucagon-Like Peptide 1; Glucagon-Like Peptides; Glucose; Glyburide; Homeostasis; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Membrane Potentials; Peptide Fragments; Peptides | 1998 |
Role of ATP-dependent K(+) channels in the electrical excitability of early embryonic stem cell-derived cardiomyocytes.
Topics: 2,4-Dinitrophenol; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Calcium Channel Agonists; Cardiotonic Agents; Cell Differentiation; Charybdotoxin; Cromakalim; Enzyme Inhibitors; Glyburide; Isoproterenol; KATP Channels; Membrane Potentials; Mice; Myocardial Contraction; Myocardium; Organoids; Patch-Clamp Techniques; Potassium Channels; Potassium Channels, Inwardly Rectifying; Stem Cells; Thapsigargin | 1999 |
Mechanism of CGRP-induced relaxation in rat intramural coronary arteries.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analysis of Variance; Animals; Calcitonin Gene-Related Peptide; Calcium; Calcium Channel Agonists; Charybdotoxin; Coronary Vessels; Drug Interactions; Enzyme Inhibitors; Felodipine; Fluorescent Dyes; Fura-2; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Male; Osmolar Concentration; Peptides; Potassium; Potassium Channels; Rats; Rats, Sprague-Dawley; Rest; Thapsigargin; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents | 2001 |
Insulin secretion to glucose as well as nonglucose stimuli is impaired in spontaneously diabetic Nagoya-Shibata-Yasuda mice.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arginine; Blood Glucose; Calcium Channel Agonists; Cell Separation; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Disease Models, Animal; Dose-Response Relationship, Drug; Glucose; Glucose Tolerance Test; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Mice, Inbred C3H; Mice, Inbred Strains; Stimulation, Chemical | 2001 |
Polyamine effects on human myometrial contractility.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Agonists; Calcium Channel Agonists; Cesarean Section; Female; Gestational Age; Glyburide; Humans; Hysterectomy; Methylene Blue; Myometrium; Oxytocin; Phenylephrine; Polyamines; Pregnancy; Spermine; Uterine Contraction | 2002 |
Multiple actions of U-37883A, an ATP-sensitive K+ channel blocker, on membrane currents in pig urethra.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adamantane; Adenosine Triphosphate; Analysis of Variance; Animals; Barium; Calcium Channel Agonists; Cromakalim; Dose-Response Relationship, Drug; Female; Glyburide; In Vitro Techniques; Membrane Potentials; Morpholines; Muscle Cells; Nitroprusside; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Swine; Time Factors; Urethra; Vasodilator Agents | 2005 |
Hydrogen sulfide facilitates carotid sinus baroreflex in anesthetized rats.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkynes; Animals; Baroreflex; Blood Pressure; Calcium Channel Agonists; Carotid Sinus; Cystathionine gamma-Lyase; Glyburide; Glycine; Hydrogen Sulfide; Male; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Sulfides | 2006 |
Hydrogen sulfide facilitates carotid sinus baroreceptor activity in anesthetized male rats.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkynes; Anesthesia; Animals; Carotid Sinus; Glyburide; Glycine; Hydrogen Sulfide; Male; Pressoreceptors; Rats; Rats, Sprague-Dawley | 2007 |
Investigation of mechanisms involved in (-)-borneol-induced vasorelaxant response on rat thoracic aorta.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Aorta, Thoracic; Calcium Chloride; Camphanes; Endothelium, Vascular; Glyburide; Phenylephrine; Potassium Channels; Potassium Chloride; Rats; Tetraethylammonium; Vasodilator Agents | 2012 |
Electrophysiological effects of hydrogen sulfide on human atrial fibers.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Calcium Channel Agonists; Calcium Channels, L-Type; Cystathionine gamma-Lyase; Electrophysiology; Glyburide; Heart Atria; Humans; Hydrogen Sulfide; In Vitro Techniques; KATP Channels; Sulfides | 2011 |
Physiological characterization of the human EndoC-βH1 β-cell line.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Diphosphate; Adenosine Triphosphate; Biological Transport; Calcium Channels; Cell Line; Colforsin; Founder Effect; Gene Expression; Glucokinase; Glucose; Glucose Transporter Type 1; Glucose Transporter Type 2; Glutamine; Glyburide; Humans; Insulin; Insulin-Secreting Cells; Keto Acids; Leucine; Mannoheptulose; Phosphorylation; Potassium Channels, Inwardly Rectifying | 2015 |
Flavonoid galetin 3,6-dimethyl ether attenuates guinea pig ileum contraction through K(+) channel activation and decrease in cytosolic calcium concentration.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Apamin; Calcium; Calcium Chloride; Carbachol; Cell Survival; Cesium; Chlorides; Flavonoids; Glyburide; Guinea Pigs; Histamine; Histamine Antagonists; Ileum; Muscle Cells; Muscle Contraction; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Tetraethylammonium | 2015 |
Perfusion of isolated carotid sinus with hydrogen sulfide attenuated the renal sympathetic nerve activity in anesthetized male rats.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkynes; Animals; Baroreflex; Carotid Sinus; Glyburide; Glycine; Hydrogen Sulfide; In Vitro Techniques; Male; Perfusion; Rats, Sprague-Dawley; Sympathetic Nervous System | 2016 |
Dynamics of Insulin Secretion from EndoC-
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Cell Line; Colforsin; Exocytosis; Glucose; Glyburide; Humans; Insulin; Insulin Secretion; Insulin-Secreting Cells; Mannoheptulose; Signal Transduction | 2017 |