bay-k-8644 and gamma-aminobutyric acid

bay-k-8644 has been researched along with gamma-aminobutyric acid in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19902 (9.52)18.7374
1990's8 (38.10)18.2507
2000's9 (42.86)29.6817
2010's2 (9.52)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Ascioti, C; De Sarro, A; De Sarro, G; di Paola, ED; Vidal, MJ1
Dohi, T; Kitayama, S; Morita, K; Tsujimoto, A1
Astier, H; Roussel, JP1
Kuramoto, K; Morita, Y; Sorimachi, M; Yamagami, K1
Carignani, C; Marchetti, C; Robello, M1
Bockaert, J; Kemp, DE; Pin, JP; Sebben, M; Weiss, S1
Massieu, L; Tapia, R1
Borges, S; Gleason, E; Wilson, M1
Roldan, ER; Shi, QX1
Akaike, N; Ishibashi, H; Rhee, JS1
Pan, ZH1
Cormier, R; Covey, DF; Fu, T; Isenberg, KE; Mennerick, S; Xu, W; Zorumski, CF1
Baran, H; Hörtnagl, H; Kepplinger, B1
Bernardi, G; Giacomini, P; Lavaroni, F; Spadoni, F; Stefani, A1
Kagaya, A; Kurata, K; Morinobu, S; Takebayashi, M; Yamawaki, S1
Akaike, N; Ishibashi, H; Lawlor, GF; Rhee, JS; Wang, ZM; Watanabe, Y1
Darcy, DP; Isaacson, JS; Murphy, GJ1
Holmgaard, K; Jensen, K; Lambert, JD1
Aceves, J; Caballero-Florán, I; Erlij, D; Florán, B; Ochoa-Sánchez, N; Paz-Bermúdez, F; Recillas-Morales, S; Sánchez-Vega, L; Silva, I1

Other Studies

21 other study(ies) available for bay-k-8644 and gamma-aminobutyric acid

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Effects of antiepileptic drugs, calcium channel blockers and other compounds on seizures induced by activation of voltage-dependent L calcium channel in DBA/2 mice.
    General pharmacology, 1992, Volume: 23, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine; Amino Acids; Animals; Anticonvulsants; Calcium Channel Blockers; Calcium Channels; Electroencephalography; Electrophysiology; Female; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Mice; Mice, Inbred DBA; Receptors, Opioid, kappa; Seizures; Synaptic Transmission

1992
GABAergic modulation of catecholamine release from cultured bovine adrenal chromaffin cells. Evidence for the involvement of Cl(-)-dependent Ca2+ entry.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 341, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenal Glands; Animals; Calcium; Calcium Radioisotopes; Catecholamines; Cattle; Cells, Cultured; Chlorides; Chromaffin System; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Ion Channels; Muscimol; Pentobarbital; Time Factors; Veratridine

1990
Involvement of dihydropyridine-sensitive calcium channels in the GABAA potentiation of TRH-induced TSH release.
    European journal of pharmacology, 1990, Nov-06, Volume: 190, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Drug Synergism; GABA Antagonists; gamma-Aminobutyric Acid; GTP-Binding Proteins; In Vitro Techniques; Isonicotinic Acids; Male; Nifedipine; omega-Conotoxins; Peptides, Cyclic; Pertussis Toxin; Pituitary Gland; Pyridazines; Rats; Rats, Inbred Strains; Thyrotropin; Thyrotropin-Releasing Hormone; Virulence Factors, Bordetella

1990
GABA inhibits the rise in cytosolic free calcium concentration in depolarized immature cerebellar Purkinje cells.
    Neuroscience letters, 1991, Jan-28, Volume: 122, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aging; Animals; Calcium; Cerebellum; Cytosol; Gallopamil; gamma-Aminobutyric Acid; Kinetics; Purkinje Cells; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Veratridine

1991
Voltage-dependent calcium currents in dissociated granule cells from rat cerebellum.
    Neuroscience, 1991, Volume: 43, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Baclofen; Bicuculline; Calcium Channels; Cerebellum; Electrophysiology; gamma-Aminobutyric Acid; Membrane Potentials; Rats; Rats, Inbred Strains; Verapamil

1991
Release of endogenous amino acids from striatal neurons in primary culture.
    Journal of neurochemistry, 1986, Volume: 47, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Amino Acids; Animals; Calcium; Cells, Cultured; Chromatography, High Pressure Liquid; Corpus Striatum; Embryo, Mammalian; gamma-Aminobutyric Acid; Mice; Neurons; Nifedipine; Potassium; Time Factors; Veratrine

1986
Relationship of dihydropyridine binding sites with calcium-dependent neurotransmitter release in synaptosomes.
    Journal of neurochemistry, 1988, Volume: 51, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Aminopyridines; Animals; Brain; Calcium; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; gamma-Aminobutyric Acid; Ion Channels; Isradipine; Lanthanum; Male; Mice; Neurotransmitter Agents; Nifedipine; Nitrendipine; Oxadiazoles; Potassium; Receptors, Nicotinic; Ruthenium Red; Synaptosomes

1988
Control of transmitter release from retinal amacrine cells by Ca2+ influx and efflux.
    Neuron, 1994, Volume: 13, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Chick Embryo; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Retina; Sodium; Synapses; Synaptic Transmission

1994
Evidence that a GABAA-like receptor is involved in progesterone-induced acrosomal exocytosis in mouse spermatozoa.
    Biology of reproduction, 1995, Volume: 52, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acrosome; Animals; Bicuculline; Calcium Channels; Exocytosis; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Nifedipine; Progesterone; Receptors, GABA-A; Sperm Capacitation; Spermatozoa; Verapamil

1995
Calcium channels in the GABAergic presynaptic nerve terminals projecting to meynert neurons of the rat.
    Journal of neurochemistry, 1999, Volume: 72, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cholinergic Fibers; Electrophysiology; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Neural Inhibition; Nicardipine; omega-Conotoxin GVIA; omega-Conotoxins; Organ Culture Techniques; Peptides; Presynaptic Terminals; Rats; Rats, Wistar; Ryanodine; Substantia Innominata; Tetrodotoxin; Thapsigargin

1999
Differential expression of high- and two types of low-voltage-activated calcium currents in rod and cone bipolar cells of the rat retina.
    Journal of neurophysiology, 2000, Volume: 83, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Axons; Bicuculline; Cadmium; Calcium Channel Blockers; Calcium Channels, L-Type; Cells, Cultured; Evoked Potentials; gamma-Aminobutyric Acid; Membrane Potentials; Nickel; Nimodipine; Protein Kinase C; Quinine; Rats; Rats, Long-Evans; Receptors, GABA; Retinal Cone Photoreceptor Cells; Retinal Rod Photoreceptor Cells; Tetrodotoxin

2000
Slow death of postnatal hippocampal neurons by GABA(A) receptor overactivation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, May-01, Volume: 20, Issue:9

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Cell Death; Cells, Cultured; Excitatory Amino Acid Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; N-Methylaspartate; Neurons; Potassium Chloride; Rats; Receptors, GABA-A

2000
Clonidine modulates BAY K 8644-induced rat behavior and neurotransmitter changes in the brain.
    European journal of pharmacology, 2000, Jul-28, Volume: 401, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 3,4-Dihydroxyphenylacetic Acid; Adrenergic alpha-Agonists; Animals; Behavior, Animal; Brain; Calcium Channel Agonists; Clonidine; Dopamine; gamma-Aminobutyric Acid; Homovanillic Acid; Male; Neurotransmitter Agents; Norepinephrine; Rats; Rats, Sprague-Dawley; Serotonin

2000
The effects of gabapentin on different ligand- and voltage-gated currents in isolated cortical neurons.
    Epilepsy research, 2001, Volume: 43, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetates; Amines; Animals; Anticonvulsants; Calcium Channel Agonists; Calcium Channels; Cerebral Cortex; Cyclohexanecarboxylic Acids; Gabapentin; gamma-Aminobutyric Acid; Glutamic Acid; Male; Neurons; Potassium Channels; Pyramidal Cells; Rats; Rats, Wistar; Sodium Channels

2001
Effect of beta-estradiol on voltage-gated Ca(2+) channels in rat hippocampal neurons: a comparison with dehydroepiandrosterone.
    European journal of pharmacology, 2001, Mar-30, Volume: 416, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Androstenedione; Animals; Azlocillin; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Corticosterone; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; Dizocilpine Maleate; Estradiol; Estrogen Antagonists; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hippocampus; Imidazolidines; N-Methylaspartate; Neurons; Nifedipine; Rats; Rats, Wistar; Tamoxifen

2001
Inhibitory effects of 1,4-DHP antagonists on synaptic GABA release modulated by BAY-K 8644 in mechanically dissociated rat substantia innominata.
    Life sciences, 2002, Jul-26, Volume: 71, Issue:10

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channels, L-Type; Dihydropyridines; Electrophysiology; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Male; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Patch-Clamp Techniques; Presynaptic Terminals; Rats; Rats, Wistar; Substantia Innominata; Synapses

2002
Intraglomerular inhibition: signaling mechanisms of an olfactory microcircuit.
    Nature neuroscience, 2005, Volume: 8, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Animals, Newborn; Bicuculline; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Signaling; Chelating Agents; Dendrites; Diagnostic Imaging; Dihydropyridines; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Neural Conduction; Neural Inhibition; Neural Networks, Computer; Neurons; Nickel; Nimodipine; Olfactory Bulb; Patch-Clamp Techniques; Phosphinic Acids; Potassium; Propanolamines; Pyrimidines; Rats; Rats, Sprague-Dawley; Signal Transduction; Synapses; Synaptic Transmission; Tetrodotoxin; Time Factors; Valine

2005
Imaging of Ca2+ responses mediated by presynaptic L-type channels on GABAergic boutons of cultured hippocampal neurons.
    Brain research, 2009, Jan-16, Volume: 1249

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels, L-Type; Calcium Channels, N-Type; Cells, Cultured; gamma-Aminobutyric Acid; Hippocampus; Isradipine; Membrane Potentials; Neurons; Patch-Clamp Techniques; Presynaptic Terminals; Rats; Rats, Wistar; Receptors, Presynaptic

2009
L-type Ca²⁺ channel activity determines modulation of GABA release by dopamine in the substantia nigra reticulata and the globus pallidus of the rat.
    Neuroscience, 2014, Jan-03, Volume: 256

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Agatoxins; Analysis of Variance; Animals; Calcium Channel Agonists; Calcium Channels, L-Type; Dopamine; Dopamine Agents; gamma-Aminobutyric Acid; Globus Pallidus; In Vitro Techniques; Male; Nifedipine; Potassium Chloride; Rats; Rats, Wistar; Substantia Nigra; Tritium

2014