bay-k-8644 has been researched along with colforsin in 108 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 21 (19.44) | 18.7374 |
1990's | 69 (63.89) | 18.2507 |
2000's | 14 (12.96) | 29.6817 |
2010's | 4 (3.70) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Cuddon, P; Fleming, A; Floto, RA; Goldsmith, P; Jahreiss, L; O'Kane, CJ; Pask, D; Rubinsztein, DC; Saiki, S; Sarkar, S; Siddiqi, FH; Ttofi, EK; Williams, A | 1 |
Desnos, C; Laran, MP; Scherman, D | 1 |
Greer, MA; Sato, N; Wang, X | 1 |
Castrén, E; Hartikka, J; Lindholm, D; Thoenen, H; Zafra, F | 1 |
Harbon, S; Khac, LD; Mokhtari, A; Renner, M | 1 |
Chiba, S; Furukawa, Y; Karasawa, Y | 1 |
Collison, KA; Matsuda, JJ; Segaloff, DL; Shibata, EF; Volk, KA | 1 |
Inagami, T; Ishido, M; Miyazaki, H; Murakami, K; Ohnishi, J; Shibata, T | 1 |
Zatz, M | 1 |
Broadley, KJ; Urquhart, RA | 2 |
Bishopric, NH; Sato, B; Webster, KA | 1 |
Birkenhäger, JC; Buurman, CJ; Pols, HA; Schilte, JP; van Leeuwen, JP | 1 |
Kasper, G; Marquez, CR; Zatz, M | 1 |
Collins, BJ; Cuttler, L; Staib, NE; Szabo, M | 1 |
Leppäluoto, J; Ruskoaho, H; Vuolteenaho, O | 1 |
Amino, N; Miyai, K; Tada, H; Takada, K | 1 |
Boutjdir, M; Fischmeister, R; Hanf, R; Méry, PF; Shrier, A | 1 |
Bowling, N; Gengo, PJ; Hayes, JS; Kauffman, RF; Utterback, B; Wyss, VL | 1 |
Lory, P; Nargeot, J; Nerbonne, JM; Richard, S; Tiaho, F | 1 |
Lynch, C | 1 |
Watkins, WD; Whorton, AR; Xuan, YT | 1 |
Dubyak, GR; Jones, SW; Marks, TN | 1 |
Berger, HJ; Pfeifer, A; Rupp, H; Werdan, K | 1 |
Heisler, S | 1 |
Andersson, KE; Lindgren, S | 1 |
Sperelakis, N; Tripathi, O | 1 |
Forder, J; Rasmussen, H; Scriabine, A | 1 |
Park, S; Rasmussen, H | 1 |
Blinks, JR; Endoh, M; Taira, N; Yanagisawa, T | 1 |
Assayag, E; Heisler, S; Labrie, F; Mehri, Y; Simard, J | 1 |
Hess, P; Lansman, JB; Nilius, B; Tsien, RW | 1 |
Chiu, AT; McCall, DE; Timmermans, PB | 1 |
Ganten, D; Lang, RE; Ruskoaho, H; Toth, M; Unger, T | 1 |
Bjøro, T; Gautvik, KM; Gordeladze, J; Haug, E; Iversen, JG; Ostberg, BC; Sand, O; Torjesen, PA | 1 |
Höllt, V; Kley, N; Loeffler, JP; Pittius, CW | 1 |
Asem, EK; Tsang, BK | 1 |
Birnbaumer, L; Brown, AM; Codina, J; Imoto, Y; Reeves, JP; Yatani, A | 1 |
Ahn, HY; Karaki, H; Urakawa, N | 1 |
Afar, R; Geertsen, S; Quik, M; Trifaró, JM | 1 |
Bose, D; Bouchard, RA; Hryshko, LV; Kobayashi, T | 1 |
Akahane, K; Chiba, S; Furukawa, Y; Ogiwara, Y; Saegusa, K | 1 |
Auguet, M; Braquet, P; Clostre, F; Delaflotte, S; Pirotzky, E | 1 |
Haleen, SJ; Major, TC; Pugsley, TA; Sircar, I; Steffen, RP; Taylor, MD; Weishaar, RE | 1 |
Adler-Graschinsky, E; Elgoyhen, B | 1 |
Calixto, JB | 1 |
Brown, AM; Imoto, Y; Schwartz, A; Yatani, A | 1 |
Kojima, I; Kojima, K; Rasmussen, H | 1 |
Eiter, C; Kroesen, S; Laslop, A; Tschernitz, C; Winkler, H | 1 |
Buckingham, JC; Cowell, AM; Flower, J; Taylor, AD | 1 |
Chu, A; Mészáros, LG; Reinach, P; Socci, R | 1 |
Ernsberger, P; Evinger, MJ; Joh, TH; Regunathan, S; Reis, DJ | 1 |
Huizinga, JD; Liu, LW | 1 |
Cherington, V; Riseberg, JC; Tischler, AS | 1 |
Buckingham, JC; Flower, RJ; Loxley, HD; Taylor, AD | 1 |
Bargas, J; Greengard, P; Hemmings, HC; Nairn, AC; Surmeier, DJ | 1 |
Calissano, P; Galli, C; Meucci, O; Schettini, G; Scorziello, A; Werge, TM | 1 |
Chang, JP; Jobin, RM; Neumann, CM; Van Goor, F; Wong, AO | 1 |
Abernethy, WB; Butterworth, JF; Leith, JP; Prielipp, RC; Zaloga, GP | 1 |
Chiba, S; Furukawa, Y; Inoue, Y; Oguchi, T; Sawaki, S | 1 |
Prostran, M; Todorović, Z; Varagić, VM | 1 |
Mulderry, PK | 1 |
Bellido, T; Boland, R; Fernández, LM; Morelli, S | 1 |
Ammälä, C; Ashcroft, FM; Rorsman, P | 1 |
Biden, TJ; Browne, CL | 1 |
Klein, DC; Vanecek, J | 1 |
Buckingham, JC; Flower, RJ; Taylor, AD | 1 |
Birkenhäger, JC; Pols, HA; van den Bemd, GC; van Leeuwen, JP | 1 |
Aggarwal, R; Boyden, PA | 1 |
Brabant, G; Mader, T; Rossig, L; Schöfl, C; von zur Mühlen, A | 1 |
Chang, JP; Jobin, RM; Neumann, CM; Van Goor, F | 1 |
Bernhardt, R; Bird, IM; Denner, K; Mathis, JM; Pezzi, V; Rainey, WE | 1 |
O'Neil, RG; Zhang, MI | 1 |
Delpech, N; Potreau, D; Soustre, H | 1 |
Dou, CL; Levine, JM | 1 |
Kubo, T; Taguchi, K; Ueda, M | 1 |
Bond, M; McConnell, BK; Morano, I; Moravec, CS | 1 |
Crawford, FA; Doscher, MA; Hebbar, L; Houck, WV; Joshi, JD; Mukherjee, R; Spinale, FG; Thomas, CV; Wang, YH | 1 |
Graybiel, AM; Liu, FC | 1 |
Bird, IM; Mason, JI; Rainey, WE | 1 |
Baker, H; Cigola, E; Franzen, L; Lee, JW; Volpe, BT | 1 |
Gohshi, A; Honda, K; Kamiya, H; Motoya, T; Takano, Y; Tominaga, K; Yamada, K | 1 |
Gong, GX; Scholz, PM; Tse, J; Weiss, HR; Yan, L | 1 |
Beales, IL; Calam, J; Jordinson, M | 1 |
Addicks, K; Bloch, W; Bohlen, H; Fleischmann, BK; Hescheler, J; Ji, GJ; Kolossov, E; Liu, Q; Manzke, O; Viatchenko-Karpinski, S | 1 |
Abi-Gerges, N; Faivre, V; Fischmeister, R; Mebazaa, A; Méry, PF; Paqueron, X; Payen, D; Tavernier, B | 1 |
Betancourt-Calle, S; Bollag, WB; Calle, RA; Jung, EM; Rasmussen, H | 1 |
Dedos, SG; Fugo, H | 1 |
Pei, JM; Wang, HX; Wong, TM; Yu, XC | 1 |
Chen, HL; Jea, JC; Liu, TC; Pu, HF; Tan, SK | 1 |
Chik, CL; Ho, AK; Negishi, T | 1 |
Coyne, MD; Gwathmey, JK; Kim, CS | 1 |
Bauer, R; Doblinger, A; Hoflehner, J; Kapeller, I; Laslop, A | 1 |
Buckingham, JC; Christian, HC; Flower, RJ; Morris, JF; Taylor, AD | 1 |
Betancourt-Calle, S; Bollag, WB; Calle, RA; Isales, CM; Rasmussen, H; White, S | 1 |
Birkenbeil, H; Dedos, SG | 1 |
Hino, N; Masumiya, H; Ochi, R; Tsujikawa, H | 1 |
Barbuti, A; Palmiter, RD; Protas, L; Qu, J; Robinson, RB; Rybin, VO; Steinberg, SF | 1 |
Lo, MJ; Wang, PS | 1 |
Gupte, SA; Masumiya, H; Ochi, R; Okada, T; Song, Y; Tsujikawa, H; Watanabe, M | 1 |
Bian, JS; Hu, LF; Pan, TT; Yong, QC | 1 |
Teramoto, N; Zhu, HL | 1 |
Cui, H; Fu, W; Gao, J; Lu, B; Wang, H; Wang, Y; Yu, X; Yu, Y; Zhang, L | 1 |
Biraud, M; Cario-Toumaniantz, C; Chevalier, J; Derkinderen, P; Lebouvier, T; Mahé, MM; Neunlist, M; Paillusson, S; Tasselli, M | 1 |
Gurgul-Convey, E; Kaminski, MT; Lenzen, S | 1 |
Cao, L; Cao, YX; Li, S; Mi, YN; Ping, NN | 1 |
Lenzen, S; Teraoku, H | 1 |
1 review(s) available for bay-k-8644 and colforsin
Article | Year |
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Scattered light intensity fluctuation in the canine ventricular myocardium: correlation with inotropic drug effect.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Colforsin; Dobutamine; Dogs; Heart; Light; Myocardial Contraction; Ouabain; Scattering, Radiation; Temperature | 1988 |
107 other study(ies) available for bay-k-8644 and colforsin
Article | Year |
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Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Novel targets for Huntington's disease in an mTOR-independent autophagy pathway.
Topics: Animals; Autophagy; Calcium Channels, L-Type; Clonidine; Cyclic AMP; Humans; Huntington Disease; Imidazoline Receptors; Minoxidil; Protein Kinases; Signal Transduction; TOR Serine-Threonine Kinases; Type C Phospholipases; Verapamil | 2008 |
Regulation of the chromaffin granule catecholamine transporter in cultured bovine adrenal medullary cells: stimulus-biosynthesis coupling.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholinesterase; Adrenal Medulla; Animals; Biological Transport; Carbachol; Carrier Proteins; Catecholamine Plasma Membrane Transport Proteins; Catecholamines; Cattle; Cells, Cultured; Chromaffin Granules; Chromogranin A; Chromogranins; Colforsin; Cyclic AMP; Cycloheximide; Dactinomycin; Dopamine beta-Hydroxylase; Membrane Proteins; Membrane Transport Proteins; Nifedipine; Potassium; Protein Kinase C; Tetrabenazine; Time Factors; Tritium; Tyrosine 3-Monooxygenase | 1992 |
Lidocaine inhibits prolactin secretion in GH4C1 cells by blocking calcium influx.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenoma; Animals; Calcium; Colforsin; Lidocaine; Pituitary Neoplasms; Potassium; Procaine; Prolactin; Rats; Tetradecanoylphorbol Acetate; Tetrodotoxin; Tumor Cells, Cultured | 1992 |
Regulation of brain-derived neurotrophic factor and nerve growth factor mRNA in primary cultures of hippocampal neurons and astrocytes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Astrocytes; Brain-Derived Neurotrophic Factor; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Cytokines; Glutamates; Glutamic Acid; Growth Substances; Hippocampus; Ionomycin; Isoquinolines; Kainic Acid; Kinetics; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Nifedipine; Norepinephrine; Piperazines; Potassium; Protein Kinase Inhibitors; Quisqualic Acid; Rats; RNA, Messenger; Tetradecanoylphorbol Acetate | 1992 |
Activation of beta-adrenergic receptors inhibits Ca2+ entry-mediated generation of inositol phosphates in the guinea pig myometrium, a cyclic AMP-independent event.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aluminum; Animals; Calcium; Calcium Channels; Carbachol; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Drug Antagonism; Female; Fluorine; Guinea Pigs; Inositol Phosphates; Ionomycin; Isoproterenol; Myometrium; Nifedipine; Oxytocin; Pertussis Toxin; Receptors, Adrenergic, beta; Type C Phospholipases; Verapamil; Virulence Factors, Bordetella | 1992 |
Cyclic-AMP-dependent positive chrono- and inotropic responses in the blood-perfused dog atrium.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Colforsin; Depression, Chemical; Dogs; Heart Atria; Heart Rate; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Perfusion; Stimulation, Chemical | 1992 |
Evidence that the FSH receptor itself is not a calcium channel.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Bucladesine; Calcium Channels; Cell Line, Transformed; Colforsin; Cyclic AMP; DNA; Electrophysiology; Embryo, Mammalian; Follicle Stimulating Hormone; Humans; Membrane Potentials; Receptors, FSH; Tetraethylammonium; Tetraethylammonium Compounds; Transfection | 1992 |
The rat angiotensin II AT1A receptor couples with three different signal transduction pathways.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Angiotensin II; Animals; Binding, Competitive; Calcium; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Egtazic Acid; Kinetics; Neomycin; Nicardipine; Rats; Receptors, Angiotensin; Recombinant Proteins; Signal Transduction; Transfection; Type C Phospholipases | 1992 |
Agents that affect calcium influx can change cyclic nucleotide levels in cultured chick pineal cells.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Cells, Cultured; Chickens; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Egtazic Acid; Kinetics; Nitrendipine; Pineal Gland | 1992 |
The effects of P1- and muscarinic-receptor agonists upon cAMP-dependent and independent inotropic responses of guinea-pig cardiac preparations.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Carbachol; Colforsin; Cyclic AMP; Guinea Pigs; Heart; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Papillary Muscles; Phenylisopropyladenosine; Receptors, Muscarinic; Receptors, Purinergic | 1992 |
Beta-adrenergic regulation of a myocardial actin gene via a cyclic AMP-independent pathway.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Actins; Animals; Animals, Newborn; Blotting, Northern; Bucladesine; Caffeine; Calcimycin; Cells, Cultured; Colforsin; Cyclic AMP; Enkephalins; Gene Expression Regulation; Heart; Heart Ventricles; Isoproterenol; Kinetics; Myocardium; Nifedipine; Potassium Chloride; Propranolol; Protein Precursors; Rats; Receptors, Adrenergic, beta; RNA; RNA, Messenger; Ryanodine | 1992 |
The indirect negative inotropic effects of the P1-receptor agonist, L-phenylisopropyladenosine, in guinea-pig isolated cardiac preparations: comparison with cromakalim.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atrial Function; Atrial Function, Left; Benzopyrans; Cardiotonic Agents; Colforsin; Cromakalim; Depression, Chemical; Guinea Pigs; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Papillary Muscles; Phenylisopropyladenosine; Pyrroles; Stimulation, Chemical; Time Factors | 1992 |
Role of calcium and cAMP in heterologous up-regulation of the 1,25-dihydroxyvitamin D3 receptor in an osteoblast cell line.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenine; Adenylyl Cyclase Inhibitors; Calcitriol; Calcium; Cell Line; Colforsin; Cyclic AMP; Dinoprostone; Nitrendipine; Osteoblasts; Parathyroid Hormone; Receptors, Calcitriol; Receptors, Steroid; Up-Regulation; Verapamil | 1990 |
Vasoactive intestinal peptide stimulates chick pineal melatonin production and interacts with other stimulatory and inhibitory agents but does not show alpha 1-adrenergic potentiation.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Chickens; Colforsin; Drug Interactions; Isoproterenol; Kinetics; Light; Melatonin; Nitrendipine; Norepinephrine; Phenylephrine; Pineal Gland; Receptors, Adrenergic, alpha; Vasoactive Intestinal Peptide; Yohimbine | 1990 |
Biphasic action of forskolin on growth hormone and prolactin secretion by rat anterior pituitary cells in vitro.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Calcimycin; Cells, Cultured; Cholera Toxin; Colforsin; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Activation; Female; Growth Hormone; Growth Hormone-Releasing Hormone; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Somatostatin; Virulence Factors, Bordetella | 1990 |
Phorbol esters enhance stretch-induced atrial natriuretic peptide secretion.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atrial Natriuretic Factor; Colforsin; Heart; Heart Atria; Male; Physical Stimulation; Radioimmunoassay; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate | 1990 |
Relationship between proliferation and cell cycle-dependent Ca2+ influx induced by a combination of thyrotropin and insulin-like growth factor-I in rat thyroid cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Cell Cycle; Cell Division; Cell Line; Cobalt; Colforsin; DNA; Drug Combinations; Insulin-Like Growth Factor I; Kinetics; Lanthanum; Pertussis Toxin; Rats; Thyroid Gland; Thyrotropin; Virulence Factors, Bordetella | 1990 |
High affinity forskolin inhibition of L-type Ca2+ current in cardiac cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Colforsin; Cyclic AMP; In Vitro Techniques; Kinetics; Myocardium; Phosphorylation; Rana esculenta | 1990 |
Cardiac inotropic responses to calcium and forskolin are not altered by prolonged isoproterenol infusion.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Colforsin; Cyclic AMP; Drug Interactions; Heart; In Vitro Techniques; Infusions, Intravenous; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Nifedipine; Radioligand Assay; Rats; Receptors, Adrenergic, beta | 1990 |
Cyclic-AMP-dependent phosphorylation modulates the stereospecific activation of cardiac Ca channels by Bay K 8644.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Colforsin; Cyclic AMP; Drug Combinations; Electric Conductivity; Heart; Isoproterenol; Membrane Potentials; Myocardium; Phosphorylation; Rats | 1990 |
Pharmacological evidence for two types of myocardial sarcoplasmic reticulum Ca2+ release.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Anesthetics, Local; Animals; Caffeine; Calcium; Colforsin; Guinea Pigs; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Myocardium; Ryanodine; Sarcolemma; Sodium | 1991 |
Regulation of endothelin-mediated calcium mobilization in vascular smooth muscle cells by isoproterenol.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Cell Line; Colforsin; Cyclic AMP; Endothelins; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Isoproterenol; Kinetics; Muscle, Smooth, Vascular; Potassium; Propranolol | 1991 |
Calcium currents in the A7r5 smooth muscle-derived cell line.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta; Biological Transport; Calcium; Calcium Channels; Cell Line; Colforsin; Cytosol; Dihydropyridines; Electric Conductivity; Fluorescence; Isoproterenol; Ligands; Muscle, Smooth, Vascular; Nifedipine; Potassium | 1990 |
Effect of positive inotropic agents on myosin isozyme population and mechanical activity of cultured rat heart myocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Animals, Newborn; Bucladesine; Cardiotonic Agents; Cells, Cultured; Colforsin; Heart; Isoenzymes; Isoproterenol; Myocardial Contraction; Myocardium; Myosins; Ouabain; Phenylephrine; Prazosin; Propranolol; Rats | 1991 |
Chloride channel blockers inhibit ACTH secretion from mouse pituitary tumor cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adenylate Cyclase Toxin; Adrenocorticotropic Hormone; Animals; Cell Line; Chloride Channels; Colforsin; Corticotropin-Releasing Hormone; Ion Channels; Kinetics; Membrane Proteins; Mice; ortho-Aminobenzoates; Osmolar Concentration; Pertussis Toxin; Pituitary Neoplasms; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1991 |
Comparison of the effects of milrinone and OPC 3911 with those of isoprenaline, forskolin and dibutyryl-cAMP in rat aorta.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Bucladesine; Calcium; Colforsin; In Vitro Techniques; Isoproterenol; Male; Milrinone; Phenylephrine; Phosphodiesterase Inhibitors; Potassium; Pyridones; Quinolones; Rats; Rats, Inbred Strains; Vasodilation | 1991 |
Effects of 8-bromo-cyclic GMP on slow channel mediated action potentials of 3-days-old embryonic chick ventricle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Chick Embryo; Colforsin; Cyclic GMP; Heart Ventricles; Ion Channels; Isoproterenol; Ventricular Function | 1991 |
Plasma membrane calcium flux, protein kinase C activation and smooth muscle contraction.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Cell Membrane; Colforsin; Drug Synergism; Enzyme Activation; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nitrendipine; Ouabain; Perfusion; Phospholipids; Potassium; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate; Vasoconstriction | 1985 |
Activation of tracheal smooth muscle contraction: synergism between Ca2+ and activators of protein kinase C.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcimycin; Calcium; Cattle; Colforsin; Diterpenes; Drug Synergism; Enzyme Activation; Ethers; In Vitro Techniques; Ionomycin; Muscle Contraction; Muscle, Smooth; Nifedipine; Protein Kinase C; Terpenes; Tetradecanoylphorbol Acetate; Trachea | 1985 |
Effects of new inotropic agents on cyclic nucleotide metabolism and calcium transients in canine ventricular muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aequorin; Aminopyridines; Amrinone; Animals; Calcium; Carbachol; Cardiotonic Agents; Colforsin; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Enoximone; Female; Imidazoles; Male; Milrinone; Myocardial Contraction; Myocardium; Nifedipine; Nucleotides, Cyclic; Pyrazines; Pyridones; Quinolines; Time Factors | 1986 |
Atrial natriuretic factor does not affect basal, forskolin- and CRF-stimulated adenylate cyclase activity, cAMP formation or ACTH secretion, but does stimulate cGMP synthesis in anterior pituitary.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenocorticotropic Hormone; Animals; Atrial Natriuretic Factor; Cell Line; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; Cyclic GMP; Growth Hormone; Kinetics; Mice; Nifedipine; Pituitary Gland, Anterior; Potassium Chloride; Tetradecanoylphorbol Acetate | 1986 |
A novel type of cardiac calcium channel in ventricular cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Colforsin; Electric Conductivity; Guinea Pigs; In Vitro Techniques; Ion Channels; Isoproterenol; Membrane Potentials; Nifedipine; Ventricular Function | 1986 |
Pharmacological characteristics of receptor-operated and potential-operated Ca2+ channels in rat aorta.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Calcium; Colforsin; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Nifedipine; Norepinephrine; Potassium; Rats; Rats, Inbred Strains; Receptors, Cell Surface | 1986 |
The phorbol ester induced atrial natriuretic peptide secretion is stimulated by forskolin and Bay K8644 and inhibited by 8-bromo-cyclic GMP.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atrial Natriuretic Factor; Calcium; Colforsin; Cyclic AMP; Cyclic GMP; Depression, Chemical; Perfusion; Rats; Stimulation, Chemical; Tetradecanoylphorbol Acetate | 1986 |
Vasoactive intestinal peptide and peptide with N-terminal histidine and C-terminal isoleucine increase prolactin secretion in cultured rat pituitary cells (GH4C1) via a cAMP-dependent mechanism which involves transient elevation of intracellular Ca2+.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Animals; Calcium; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP; Membrane Potentials; Peptide PHI; Pituitary Gland; Prolactin; Rats; Secretory Rate; Thyrotropin-Releasing Hormone; Vasoactive Intestinal Peptide; Verapamil | 1987 |
Involvement of ion channels in the induction of proenkephalin A gene expression by nicotine and cAMP in bovine chromaffin cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adrenal Glands; Animals; Calcium; Cattle; Cells, Cultured; Chromaffin System; Colforsin; Cyclic AMP; Enkephalins; Gallopamil; Gene Expression Regulation; Ion Channels; Nicotine; Nifedipine; Protein Precursors; RNA, Messenger; Sodium; Tubocurarine; Verapamil | 1987 |
Effects of calcium channel activators BAY-K8644 and CGP-28392 on steroidogenesis in granulosa cells of the domestic hen.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcium; Chickens; Colforsin; Female; Granulosa Cells; Luteinizing Hormone; Progesterone; Pyridines; Steroids | 1987 |
A G protein directly regulates mammalian cardiac calcium channels.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Colforsin; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guinea Pigs; Heart; Ion Channels; Isoproterenol; Leupeptins; Membrane Potentials; Phosphorylation; Thionucleotides; Ventricular Function | 1987 |
Inhibitory effects of caffeine on contractions and calcium movement in vascular and intestinal smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Caffeine; Calcium; Calcium Radioisotopes; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Norepinephrine; Rabbits | 1988 |
Regulation of alpha-bungarotoxin sites in chromaffin cells in culture by nicotinic receptor ligands, K+, and cAMP.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenal Medulla; alpha7 Nicotinic Acetylcholine Receptor; Biological Transport; Bucladesine; Bungarotoxins; Carbachol; Cells, Cultured; Colforsin; Enzyme Activation; Gallopamil; Nicotine; Norepinephrine; Potassium; Receptors, Cholinergic; Receptors, Nicotinic; Tubocurarine | 1988 |
Differential vagal inhibition of the positive chronotropic and inotropic responses to cardiotonics in the isolated dog atrium.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cardiotonic Agents; Colforsin; Dobutamine; Dogs; Electric Stimulation; Heart; Heart Rate; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Vagus Nerve | 1989 |
Effects of atrial natriuretic factor (ANF) on phenylephrine-triggered intra- and extracellular calcium dependent contraction in rat aorta.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Atrial Natriuretic Factor; Calcium; Colforsin; Cyclic AMP; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phenylephrine; Rats; Rats, Inbred Strains | 1989 |
PD 122860: a novel dihydropyridine with sodium channel stimulating and calcium channel blocking properties.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Colforsin; Coronary Circulation; Dihydropyridines; Electrocardiography; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Ouabain; Rats; Rats, Inbred Strains; Reference Values; Sodium Channels; Veratridine | 1989 |
Diminution by benzodiazepines of the chronotropic responses to noradrenaline in rat isolated atria.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Colforsin; Cyclic AMP; Diazepam; Female; Flumazenil; Heart; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains | 1989 |
Interactions between forskolin, calcium and Bay K 8644 in K+-depolarized rat uterine muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Chloride; Colforsin; Female; In Vitro Techniques; Potassium; Rats; Uterine Contraction; Uterus | 1989 |
New positive inotropic agent OPC-8212 modulates single Ca2+ channels in ventricular myocytes of guinea pig.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Caffeine; Calcium Channels; Cardiotonic Agents; Colforsin; Cyclic AMP; Depression, Chemical; Dose-Response Relationship, Drug; Guinea Pigs; Heart Ventricles; Isoproterenol; Myocardium; Phosphorylation; Pyrazines; Quinolines | 1989 |
Role of calcium and cAMP in the action of adrenocorticotropin on aldosterone secretion.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Glands; Adrenocorticotropic Hormone; Aldosterone; Animals; Calcimycin; Calcium; Cattle; Colforsin; Cyclic AMP; Diterpenes; Dose-Response Relationship, Drug; Nifedipine; Phospholipids | 1985 |
Biosynthesis of large dense-core vesicles in PC12 cells: effects of depolarization and second messengers on the mRNA levels of their constituents.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Chromaffin Granules; Colforsin; Membrane Potentials; PC12 Cells; Rats; RNA, Messenger; Second Messenger Systems; Solubility; Stimulation, Chemical; Tetradecanoylphorbol Acetate | 1995 |
Lipocortin 1 mediates an early inhibitory action of glucocorticoids on the secretion of ACTH by the rat anterior pituitary gland in vitro.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Animals; Annexin A1; Colforsin; Corticotropin-Releasing Hormone; Culture Techniques; Cycloheximide; Dactinomycin; Dexamethasone; Male; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Recombinant Proteins | 1993 |
In situ Ca(2+)-induced Ca2+ release from a ryanodine-sensitive intracellular Ca2+ store in corneal epithelial cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding Sites; Caffeine; Calcium; Calcium Channels; Cattle; Colforsin; Cornea; Cyclic AMP; Epithelial Cells; Epithelium; Muscle Proteins; Radioimmunoassay; Ryanodine; Ryanodine Receptor Calcium Release Channel; Signal Transduction | 1993 |
A single transmitter regulates gene expression through two separate mechanisms: cholinergic regulation of phenylethanolamine N-methyltransferase mRNA via nicotinic and muscarinic pathways.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenal Medulla; Animals; Atropine; Binding, Competitive; Calcimycin; Calcium; Carbachol; Cattle; Cells, Cultured; Colforsin; Epinephrine; Gene Expression Regulation, Enzymologic; Hexamethonium; Hexamethonium Compounds; Kinetics; Muscarine; Nicotine; Phenylethanolamine N-Methyltransferase; Piperidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Receptors, Nicotinic; RNA, Messenger | 1994 |
Canine colonic circular muscle generates action potentials without the pacemaker component.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Barium; Calcium Channels; Colforsin; Colon; Dogs; Electric Stimulation; Electrophysiology; Female; Gallopamil; In Vitro Techniques; Male; Microelectrodes; Muscle, Smooth; Neuromuscular Depolarizing Agents; Potassium; Potassium Channels | 1994 |
Multiple mitogenic signalling pathways in chromaffin cells: a model for cell cycle regulation in the nervous system.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Cell Cycle; Cell Division; Cells, Cultured; Colforsin; Dexamethasone; Ethers, Cyclic; Female; Models, Neurological; Nerve Endings; Nerve Growth Factors; Okadaic Acid; Phosphoprotein Phosphatases; Potassium Chloride; Rats; Rats, Inbred F344; Signal Transduction; Tetradecanoylphorbol Acetate; Tetrodotoxin; Veratridine | 1994 |
Lipocortin 1 and hypothalamo-pituitary function in the rat.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Animals; Annexin A1; Antibodies, Monoclonal; Arginine Vasopressin; Colforsin; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Hypothalamo-Hypophyseal System; Hypothalamus; In Vitro Techniques; Interleukin-1; Pituitary Gland, Anterior; Rats | 1994 |
Modulation of calcium currents by a D1 dopaminergic protein kinase/phosphatase cascade in rat neostriatal neurons.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Kinetics; Membrane Potentials; Neostriatum; Neurons; Nifedipine; Phosphoprotein Phosphatases; Protein Phosphatase 1; Rats; Rats, Wistar; Receptors, Dopamine D1; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors | 1995 |
Apoptosis in cerebellar granule cells is blocked by high KCl, forskolin, and IGF-1 through distinct mechanisms of action: the involvement of intracellular calcium and RNA synthesis.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Apoptosis; Calcium; Cerebellum; Colforsin; Electrophysiology; Insulin-Like Growth Factor I; Intracellular Membranes; Neurons; Nifedipine; Potassium; Potassium Chloride; Rats; Rats, Wistar; RNA; Transcription, Genetic | 1995 |
Signal transduction pathways in GnRH- and dopamine D1-stimulated growth hormone secretion in the goldfish.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Colforsin; Cyclic AMP; Dopamine; Goldfish; Gonadotropin-Releasing Hormone; Growth Hormone; Phospholipases A; Phospholipases A2; Pituitary Gland; Protein Kinase C; Signal Transduction; Verapamil | 1994 |
Calcium entry attenuates adenylyl cyclase activity. A possible mechanism for calcium-induced catecholamine resistance.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Epinephrine; Extracellular Space; Humans; Lymphocytes | 1995 |
Zatebradine attenuates cyclic AMP-related positive chronotropic but not inotropic responses in isolated, perfused right atria of the dog.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic Agonists; Animals; Benzazepines; Cardiovascular Agents; Colforsin; Dogs; Heart Atria; Heart Rate; Myocardial Contraction; Stimulation, Chemical | 1995 |
The effect of nickel chloride on the isolated hemidiaphragm of the rat.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Colforsin; Diaphragm; Electric Stimulation; Female; In Vitro Techniques; Isometric Contraction; Lidocaine; Male; Nickel; Rats; Time Factors; Verapamil | 1995 |
Synergistic regulation of vasoactive intestinal polypeptide expression by cyclic AMP and calcium in newborn but not adult rat sensory neurons in culture.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Aging; Animals; Animals, Newborn; Axons; Calcitonin Gene-Related Peptide; Calcium; Colforsin; Cyclic AMP; Female; Ganglia, Spinal; Immunohistochemistry; Male; Nerve Growth Factors; Neurons, Afferent; Rats; Rats, Wistar; Signal Transduction; Substance P; Vasoactive Intestinal Peptide | 1993 |
Evidence for the participation of protein kinase C and 3',5'-cyclic AMP-dependent protein kinase in the stimulation of muscle cell proliferation by 1,25-dihydroxy-vitamin D3.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Bucladesine; Calcitriol; Calcium; Calcium Channels; Cell Division; Cells, Cultured; Chick Embryo; Colforsin; Diglycerides; DNA; Dose-Response Relationship, Drug; Muscles; Nifedipine; Protein Kinase C; Protein Kinases; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors | 1993 |
Calcium-independent potentiation of insulin release by cyclic AMP in single beta-cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Activation; Exocytosis; Fluorometry; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Protein Kinase Inhibitors; Protein Kinases | 1993 |
Cross-talk between muscarinic- and adenosine-receptor signalling in the regulation of cytosolic free Ca2+ and insulin secretion.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine; Atropine; Calcium; Calcium Channels; Carbachol; Cells, Cultured; Colforsin; Cytosol; Enzyme Activation; Glyceraldehyde; Insulin; Insulin Secretion; Ion Channel Gating; Muscarinic Antagonists; Receptors, Muscarinic; Receptors, Purinergic; Signal Transduction; Type C Phospholipases | 1993 |
Mechanism of melatonin signal transduction in the neonatal rat pituitary.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Calcimycin; Calcium; Colforsin; Cyclic AMP; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Melatonin; Nifedipine; Organ Culture Techniques; Pituitary Gland, Anterior; Rats; Receptors, Cell Surface; Receptors, Melatonin; Signal Transduction | 1995 |
Dexamethasone inhibits the release of TSH from the rat anterior pituitary gland in vitro by mechanisms dependent on de novo protein synthesis and lipocortin 1.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Annexin A1; Calcium Channel Blockers; Colforsin; Depression, Chemical; Dexamethasone; In Vitro Techniques; Male; Pituitary Gland, Anterior; Protein Biosynthesis; Rats; Rats, Sprague-Dawley; Thyrotropin; Thyrotropin-Releasing Hormone; Vasoactive Intestinal Peptide | 1995 |
Evidence for coordinated regulation of osteoblast function by 1,25-dihydroxyvitamin D3 and parathyroid hormone.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcitriol; Calcium; Calcium Channel Agonists; Cell Line; Colforsin; Cyclic AMP; Cytochrome P-450 Enzyme System; Drug Synergism; Enzyme Activation; Humans; Osteoblasts; Osteocalcin; Parathyroid Hormone; Protein Kinase C; Rats; Receptors, Calcitriol; RNA, Messenger; Signal Transduction; Steroid Hydroxylases; Tetradecanoylphorbol Acetate; Up-Regulation; Vitamin D3 24-Hydroxylase | 1996 |
Altered pharmacologic responsiveness of reduced L-type calcium currents in myocytes surviving in the infarcted heart.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Colforsin; Cyclic AMP; Dogs; Heart; Isoproterenol; Myocardial Infarction | 1996 |
CYCLIC adenosine 3',5'-monophosphate potentiates Ca2+ signaling and insulin secretion by phospholipase C-linked hormones in HIT cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Arginine Vasopressin; Bombesin; Calcium; Calcium-Transporting ATPases; Cell Line; Colforsin; Cricetinae; Cyclic AMP; Egtazic Acid; Enzyme Inhibitors; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Mesocricetus; Nifedipine; Signal Transduction; Terpenes; Thapsigargin; Time Factors | 1996 |
Interactions between signaling pathways in mediating GnRH-stimulated GTH release from goldfish pituitary cells: protein kinase C, but not cyclic AMP is an important mediator of GnRH-stimulated gonadotropin secretion in goldfish.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Arachidonic Acid; Calcium Channel Agonists; Cells, Cultured; Chickens; Colforsin; Cyclic AMP; Diglycerides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Goldfish; Gonadotropin-Releasing Hormone; Gonadotropins, Pituitary; Male; Microspheres; Naphthalenes; Pituitary Gland; Potassium; Protein Kinase C; Salmon; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate | 1996 |
Differential regulation of 11 beta-hydroxylase and aldosterone synthase in human adrenocortical H295R cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Cortex; Angiotensin II; Base Sequence; Bucladesine; Calcium Channel Agonists; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cytochrome P-450 CYP11B2; Gene Expression Regulation; Humans; Molecular Sequence Data; Nifedipine; Potassium; Protein Kinase C; Steroid 11-beta-Hydroxylase; Tetradecanoylphorbol Acetate | 1996 |
Regulated calcium channel in apical membranes renal proximal tubule cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Calcium; Calcium Channels; Cations, Monovalent; Cell Membrane; Cells, Cultured; Colforsin; Epithelium; Ion Channel Gating; Kidney Tubules, Proximal; Membrane Potentials; Nifedipine; Patch-Clamp Techniques; Rabbits; Substrate Specificity; Tetradecanoylphorbol Acetate | 1996 |
Endothelin-1 inhibits L-type Ca2+ current enhanced by isoprenaline in rat atrial myocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic beta-Agonists; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Cyclic AMP; Endothelin-1; Heart Atria; Isoproterenol; Myocardium; Patch-Clamp Techniques; Protein Kinase Inhibitors; Rats | 1997 |
Identification of a neuronal cell surface receptor for a growth inhibitory chondroitin sulfate proteoglycan (NG2).
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding Sites; Calcium Channel Agonists; Cellular Senescence; Cerebellum; Chondroitin Sulfate Proteoglycans; Colforsin; Cyclic AMP; Growth Inhibitors; Ionomycin; Neurites; Neurons; Pertussis Toxin; Rats; Receptors, Cell Surface; Virulence Factors, Bordetella | 1997 |
Effects of cAMP and cGMP on L-type calcium channel currents in rat mesenteric artery cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Colforsin; Cyclic AMP; Cyclic GMP; In Vitro Techniques; Isoquinolines; Male; Membrane Potentials; Mesenteric Arteries; Muscle, Smooth, Vascular; Nifedipine; Nitroglycerin; Patch-Clamp Techniques; Rats; Rats, Wistar | 1997 |
Troponin I phosphorylation in spontaneously hypertensive rat heart: effect of beta-adrenergic stimulation.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Calcium; Calcium-Binding Proteins; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Electric Stimulation; Enzyme Inhibitors; Heart; Heart Ventricles; Hypertension; Isoproterenol; Marine Toxins; Myocardial Contraction; Myocardium; Myosin Light Chains; Norepinephrine; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Troponin I | 1997 |
Downstream defects in beta-adrenergic signaling and relation to myocyte contractility after cardioplegic arrest.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Colforsin; Heart Arrest, Induced; Isoproterenol; Myocardial Contraction; Receptors, Adrenergic, beta; Signal Transduction; Swine; Time Factors; Ventricular Dysfunction, Left | 1998 |
Region-dependent dynamics of cAMP response element-binding protein phosphorylation in the basal ganglia.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Animals, Newborn; Basal Ganglia; Benzazepines; Calcium; Calcium Channels; Calcium Channels, L-Type; Colforsin; Corpus Striatum; Cyclic AMP Response Element-Binding Protein; Dopamine Agonists; Kinetics; N-Methylaspartate; Organ Culture Techniques; Organ Specificity; Phosphorylation; Rats; Rats, Sprague-Dawley; Time Factors | 1998 |
Protein kinase A, protein kinase C, and Ca(2+)-regulated expression of 21-hydroxylase cytochrome P450 in H295R human adrenocortical cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Cortex; Angiotensin II; Bucladesine; Calcium; Calcium Channel Agonists; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Gene Expression Regulation, Enzymologic; Humans; Potassium; Protein Kinase C; RNA, Messenger; Signal Transduction; Steroid 21-Hydroxylase; Tetradecanoylphorbol Acetate | 1998 |
Tyrosine hydroxylase expression in primary cultures of olfactory bulb: role of L-type calcium channels.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Cells, Cultured; Colforsin; Mice; Mice, Inbred C57BL; Mice, Inbred CBA; Nerve Tissue Proteins; Neurites; Nifedipine; Olfactory Bulb; Potassium Chloride; Stimulation, Chemical; Time Factors; Tyrosine 3-Monooxygenase | 1998 |
Changes in adrenocorticotropic hormone (ACTH) release from the cultured anterior pituitary cells of streptozotocin-induced diabetic rats.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Animals; Cells, Cultured; Colforsin; Corticotropin-Releasing Hormone; Diabetes Mellitus, Experimental; Male; Pituitary Gland, Anterior; Rats; Rats, Wistar; Streptozocin | 1998 |
Relationship between decreased function and O2 consumption caused by cyclic GMP in cardiac myocytes and L-type calcium channels.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analysis of Variance; Animals; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Cyclic GMP; Heart; Muscle Contraction; Myocardium; Nifedipine; Nitroprusside; Oxygen Consumption; Rabbits; Radioimmunoassay | 1998 |
Soybean agglutinin stimulated cholecystokinin release from cultured rabbit jejunal cells requires calcium influx via L-type calcium channels.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Animals; Calcium; Calcium Channels; Calcium Channels, L-Type; Cell Separation; Cells, Cultured; Cholecystokinin; Colforsin; Enzyme Activation; Jejunum; Lectins; Male; Phenylalanine; Plant Lectins; Protein Kinase C; Rabbits; Radioimmunoassay; Somatostatin; Soybean Proteins; Staurosporine; Verapamil | 1998 |
Functional characteristics of ES cell-derived cardiac precursor cells identified by tissue-specific expression of the green fluorescent protein.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Actins; Animals; Caffeine; Calcium; Calcium Channels; Calcium Channels, L-Type; Calcium Signaling; Calcium-Transporting ATPases; Cell Differentiation; Colforsin; Fetal Heart; Fetal Proteins; Gene Expression Regulation, Developmental; Genes, Reporter; Green Fluorescent Proteins; Inositol 1,4,5-Trisphosphate Receptors; Luminescent Proteins; Mice; Muscle Proteins; Myocardial Contraction; Organ Specificity; Patch-Clamp Techniques; Promoter Regions, Genetic; Receptors, Cytoplasmic and Nuclear; Recombinant Fusion Proteins; Ryanodine Receptor Calcium Release Channel; Stem Cells | 1998 |
Sequential changes in autonomic regulation of cardiac myocytes after in vivo endotoxin injection in rat.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adenylyl Cyclases; Adrenergic Antagonists; Adrenergic beta-Agonists; Animals; Autonomic Nervous System; Calcium Channel Agonists; Calcium Channels, L-Type; Colforsin; Diterpenes; Electrophysiology; Endotoxemia; Endotoxins; Enzyme Activators; Escherichia coli; Heart; Hemodynamics; In Vitro Techniques; Injections, Intravenous; Isoproterenol; Male; Myocardium; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Rats; Sepsis | 1999 |
Effects of angiotensin II and adrenocorticotropic hormone on myristoylated alanine-rich C-kinase substrate phosphorylation in glomerulosa cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Aldosterone; Angiotensin II; Animals; Calcium Channel Agonists; Cattle; Cells, Cultured; Colforsin; Humans; Intracellular Signaling Peptides and Proteins; Membrane Proteins; Myristoylated Alanine-Rich C Kinase Substrate; Phosphorylation; Protein Kinase C; Proteins; Zona Glomerulosa | 1999 |
Interactions between Ca2+ and cAMP in ecdysteroid secretion from the prothoracic glands of Bombyx mori.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bombyx; Bucladesine; Calcimycin; Calcium; Colforsin; Cyclic AMP; Drug Interactions; Ecdysterone; Enzyme Inhibitors; Phosphodiesterase Inhibitors; Second Messenger Systems; Signal Transduction; Thionucleotides; Verapamil | 1999 |
Anti-arrhythmic effect of kappa-opioid receptor stimulation in the perfused rat heart: involvement of a cAMP-dependent pathway.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Calcium; Colforsin; Cyclic AMP; Cytosol; Electric Stimulation; Electrocardiography; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Naltrexone; Norepinephrine; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa | 1999 |
Muscarinic regulation of basal versus thyrotropin-releasing hormone-induced prolactin secretion in rat anterior pituitary cells. differential roles of nitric oxide and intracellular calcium mobilization.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Calcium Signaling; Colforsin; Cyclic AMP; Female; Neurons; Nitric Oxide; Pertussis Toxin; Pituitary Gland; Prolactin; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Thyrotropin-Releasing Hormone; Virulence Factors, Bordetella | 1999 |
Ceramide enhances growth hormone (GH)-releasing hormone-stimulated cyclic adenosine 3',5'-monophosphate accumulation but inhibits GH release in rat anterior pituitary cells.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Ceramides; Colforsin; Cyclic AMP; Glucosyltransferases; Growth Hormone; Growth Hormone-Releasing Hormone; Ionomycin; Ionophores; Male; Meperidine; Pituitary Gland, Anterior; Potassium Chloride; Rats; Rats, Sprague-Dawley | 1999 |
Voltage-dependent calcium channels in ventricular cells of rainbow trout: effect of temperature changes in vitro.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adaptation, Physiological; Animals; Barium; Body Temperature; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cardiotonic Agents; Cold Temperature; Colforsin; Heart Ventricles; In Vitro Techniques; Ion Channel Gating; Isoproterenol; Membrane Potentials; Muscle Fibers, Skeletal; Myocardial Contraction; Myocardium; Nifedipine; Oncorhynchus mykiss; Patch-Clamp Techniques; Pyrroles; Tetrodotoxin | 2000 |
Regulation of the biosynthesis and processing of chromogranins in organotypic slices: influence of depolarization, forskolin and differentiating factors.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aspartic Acid Endopeptidases; Calcium Channel Agonists; Cell Differentiation; Chromogranin A; Chromogranins; Colforsin; Gene Expression; Hippocampus; In Situ Hybridization; Membrane Potentials; Nerve Growth Factors; Neurons; Organ Culture Techniques; Potassium; Proprotein Convertase 2; Proprotein Convertases; Proteins; Rats; Rats, Sprague-Dawley; RNA, Messenger; Stimulation, Chemical; Subtilisins | 2000 |
Evidence from immunoneutralization and antisense studies that the inhibitory actions of glucocorticoids on growth hormone release in vitro require annexin 1 (lipocortin 1).
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Annexin A1; Antibodies, Monoclonal; Colforsin; Corticosterone; Dexamethasone; DNA, Antisense; Glucocorticoids; Growth Hormone; Growth Hormone-Releasing Hormone; In Vitro Techniques; Male; Microscopy, Electron; Pituitary Gland; Rats; Rats, Sprague-Dawley | 2000 |
Differential effects of agonists of aldosterone secretion on steroidogenic acute regulatory phosphorylation.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Aldosterone; Angiotensin II; Animals; Blotting, Western; Calcium Channel Agonists; Cattle; Cells, Cultured; Colforsin; Electrophoresis, Gel, Two-Dimensional; Phosphoproteins; Phosphorylation; Potassium Chloride; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate; Vasoconstrictor Agents; Zona Glomerulosa | 2001 |
Inhibition of cAMP signalling cascade-mediated Ca2+ influx by a prothoracicostatic peptide (Mas-MIP I) via dihydropyridine-sensitive Ca2+ channels in the prothoracic glands of the silkworm, Bombyx mori.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bombyx; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Cells, Cultured; Colforsin; Cyclic AMP; Dihydropyridines; Exocrine Glands; Kinetics; Larva; Signal Transduction | 2003 |
Modulation of manganese currents by 1, 4-dihydropyridines, isoproterenol and forskolin in rabbit ventricular cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic beta-Agonists; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Colforsin; Cyclic AMP; Dihydropyridines; Electrophysiology; Heart Ventricles; In Vitro Techniques; Ion Channel Gating; Ion Channels; Isoproterenol; Manganese; Membrane Potentials; Myocardium; Myocytes, Cardiac; Nitrendipine; Patch-Clamp Techniques; Rabbits; Signal Transduction | 2003 |
Neuropeptide Y is an essential in vivo developmental regulator of cardiac ICa,L.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Animals, Newborn; Calcium Channel Agonists; Calcium Channels, L-Type; Cell Separation; Colforsin; Female; Gene Expression Regulation, Developmental; Heart Ventricles; Male; Mice; Mice, Transgenic; Myocardium; Myocytes, Cardiac; Neuropeptide Y; Patch-Clamp Techniques | 2003 |
Relative and combined effects of estradiol and prolactin on corticosterone secretion in ovariectomized rats.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adrenocorticotropic Hormone; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Colforsin; Corticosterone; Cyclic AMP; Drug Synergism; Estradiol; Female; Injections, Intravenous; Nifedipine; Ovariectomy; Phosphodiesterase Inhibitors; Prolactin; Rats; Rats, Sprague-Dawley; Signal Transduction | 2003 |
Cholesterol depletion modulates basal L-type Ca2+ current and abolishes its -adrenergic enhancement in ventricular myocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; beta-Cyclodextrins; Calcium Channel Agonists; Calcium Channels, L-Type; Calcium Signaling; Cholesterol; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic CMP; Dose-Response Relationship, Drug; Enzyme Activators; Heart Ventricles; In Vitro Techniques; Isoproterenol; Membrane Microdomains; Membrane Potentials; Myocytes, Cardiac; Rabbits; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Time Factors | 2008 |
Negative regulation of beta-adrenergic function by hydrogen sulphide in the rat hearts.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Calcium Signaling; Colforsin; Cyclic AMP; Electric Stimulation; Hydrogen Sulfide; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Myocytes, Cardiac; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 2008 |
Antagonistic actions of S(-)-Bay K 8644 on cyclic nucleotide-induced inhibition of voltage-dependent Ba(2+) currents in guinea pig gastric antrum.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Bucladesine; Calcium Channel Agonists; Calcium Channels, L-Type; Colforsin; Cyclic GMP; Female; Guinea Pigs; In Vitro Techniques; Male; Myocytes, Smooth Muscle; Nitroprusside; Patch-Clamp Techniques; Pyloric Antrum; Stereoisomerism; Vasodilator Agents | 2008 |
Antiarrhythmic effect of acupuncture pretreatment in rats subjected to simulative global ischemia and reperfusion--involvement of adenylate cyclase, protein kinase A, and L-type Ca2+ channel.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Arrhythmias, Cardiac; Calcium Channel Agonists; Calcium Channels, L-Type; Calcium Signaling; Colforsin; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Electroacupuncture; Electrocardiography; Enzyme Activation; Enzyme Activators; Heart Rate; Male; Myocardial Reperfusion Injury; Myocytes, Cardiac; Perfusion; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1 | 2008 |
α-Synuclein expression is induced by depolarization and cyclic AMP in enteric neurons.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; alpha-Synuclein; Animals; Blotting, Western; Calcium Channel Agonists; Calcium Channels, L-Type; Colforsin; Cyclic AMP; Electrophysiology; Enteric Nervous System; Female; Immunohistochemistry; Indicators and Reagents; Mice; Mice, Inbred C57BL; Neurons; Phosphopyruvate Hydratase; Pregnancy; ras Proteins; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Reverse Transcriptase Polymerase Chain Reaction | 2010 |
Physiological characterization of the human EndoC-βH1 β-cell line.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Diphosphate; Adenosine Triphosphate; Biological Transport; Calcium Channels; Cell Line; Colforsin; Founder Effect; Gene Expression; Glucokinase; Glucose; Glucose Transporter Type 1; Glucose Transporter Type 2; Glutamine; Glyburide; Humans; Insulin; Insulin-Secreting Cells; Keto Acids; Leucine; Mannoheptulose; Phosphorylation; Potassium Channels, Inwardly Rectifying | 2015 |
H2S induces vasoconstriction of rat cerebral arteries via cAMP/adenylyl cyclase pathway.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Calcium Channel Agonists; Calcium Channels, L-Type; Cerebral Arteries; Colforsin; Cyclic AMP; Endothelium; Hydrogen Sulfide; Isoproterenol; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Rats; Rats, Sprague-Dawley; Sulfides; Vasoconstriction | 2015 |
Dynamics of Insulin Secretion from EndoC-
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Cell Line; Colforsin; Exocytosis; Glucose; Glyburide; Humans; Insulin; Insulin Secretion; Insulin-Secreting Cells; Mannoheptulose; Signal Transduction | 2017 |