bay-k-8644 and colforsin

bay-k-8644 has been researched along with colforsin in 108 studies

Research

Studies (108)

TimeframeStudies, this research(%)All Research%
pre-199021 (19.44)18.7374
1990's69 (63.89)18.2507
2000's14 (12.96)29.6817
2010's4 (3.70)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Cuddon, P; Fleming, A; Floto, RA; Goldsmith, P; Jahreiss, L; O'Kane, CJ; Pask, D; Rubinsztein, DC; Saiki, S; Sarkar, S; Siddiqi, FH; Ttofi, EK; Williams, A1
Desnos, C; Laran, MP; Scherman, D1
Greer, MA; Sato, N; Wang, X1
Castrén, E; Hartikka, J; Lindholm, D; Thoenen, H; Zafra, F1
Harbon, S; Khac, LD; Mokhtari, A; Renner, M1
Chiba, S; Furukawa, Y; Karasawa, Y1
Collison, KA; Matsuda, JJ; Segaloff, DL; Shibata, EF; Volk, KA1
Inagami, T; Ishido, M; Miyazaki, H; Murakami, K; Ohnishi, J; Shibata, T1
Zatz, M1
Broadley, KJ; Urquhart, RA2
Bishopric, NH; Sato, B; Webster, KA1
Birkenhäger, JC; Buurman, CJ; Pols, HA; Schilte, JP; van Leeuwen, JP1
Kasper, G; Marquez, CR; Zatz, M1
Collins, BJ; Cuttler, L; Staib, NE; Szabo, M1
Leppäluoto, J; Ruskoaho, H; Vuolteenaho, O1
Amino, N; Miyai, K; Tada, H; Takada, K1
Boutjdir, M; Fischmeister, R; Hanf, R; Méry, PF; Shrier, A1
Bowling, N; Gengo, PJ; Hayes, JS; Kauffman, RF; Utterback, B; Wyss, VL1
Lory, P; Nargeot, J; Nerbonne, JM; Richard, S; Tiaho, F1
Lynch, C1
Watkins, WD; Whorton, AR; Xuan, YT1
Dubyak, GR; Jones, SW; Marks, TN1
Berger, HJ; Pfeifer, A; Rupp, H; Werdan, K1
Heisler, S1
Andersson, KE; Lindgren, S1
Sperelakis, N; Tripathi, O1
Forder, J; Rasmussen, H; Scriabine, A1
Park, S; Rasmussen, H1
Blinks, JR; Endoh, M; Taira, N; Yanagisawa, T1
Assayag, E; Heisler, S; Labrie, F; Mehri, Y; Simard, J1
Hess, P; Lansman, JB; Nilius, B; Tsien, RW1
Chiu, AT; McCall, DE; Timmermans, PB1
Ganten, D; Lang, RE; Ruskoaho, H; Toth, M; Unger, T1
Bjøro, T; Gautvik, KM; Gordeladze, J; Haug, E; Iversen, JG; Ostberg, BC; Sand, O; Torjesen, PA1
Höllt, V; Kley, N; Loeffler, JP; Pittius, CW1
Asem, EK; Tsang, BK1
Birnbaumer, L; Brown, AM; Codina, J; Imoto, Y; Reeves, JP; Yatani, A1
Ahn, HY; Karaki, H; Urakawa, N1
Afar, R; Geertsen, S; Quik, M; Trifaró, JM1
Bose, D; Bouchard, RA; Hryshko, LV; Kobayashi, T1
Akahane, K; Chiba, S; Furukawa, Y; Ogiwara, Y; Saegusa, K1
Auguet, M; Braquet, P; Clostre, F; Delaflotte, S; Pirotzky, E1
Haleen, SJ; Major, TC; Pugsley, TA; Sircar, I; Steffen, RP; Taylor, MD; Weishaar, RE1
Adler-Graschinsky, E; Elgoyhen, B1
Calixto, JB1
Brown, AM; Imoto, Y; Schwartz, A; Yatani, A1
Kojima, I; Kojima, K; Rasmussen, H1
Eiter, C; Kroesen, S; Laslop, A; Tschernitz, C; Winkler, H1
Buckingham, JC; Cowell, AM; Flower, J; Taylor, AD1
Chu, A; Mészáros, LG; Reinach, P; Socci, R1
Ernsberger, P; Evinger, MJ; Joh, TH; Regunathan, S; Reis, DJ1
Huizinga, JD; Liu, LW1
Cherington, V; Riseberg, JC; Tischler, AS1
Buckingham, JC; Flower, RJ; Loxley, HD; Taylor, AD1
Bargas, J; Greengard, P; Hemmings, HC; Nairn, AC; Surmeier, DJ1
Calissano, P; Galli, C; Meucci, O; Schettini, G; Scorziello, A; Werge, TM1
Chang, JP; Jobin, RM; Neumann, CM; Van Goor, F; Wong, AO1
Abernethy, WB; Butterworth, JF; Leith, JP; Prielipp, RC; Zaloga, GP1
Chiba, S; Furukawa, Y; Inoue, Y; Oguchi, T; Sawaki, S1
Prostran, M; Todorović, Z; Varagić, VM1
Mulderry, PK1
Bellido, T; Boland, R; Fernández, LM; Morelli, S1
Ammälä, C; Ashcroft, FM; Rorsman, P1
Biden, TJ; Browne, CL1
Klein, DC; Vanecek, J1
Buckingham, JC; Flower, RJ; Taylor, AD1
Birkenhäger, JC; Pols, HA; van den Bemd, GC; van Leeuwen, JP1
Aggarwal, R; Boyden, PA1
Brabant, G; Mader, T; Rossig, L; Schöfl, C; von zur Mühlen, A1
Chang, JP; Jobin, RM; Neumann, CM; Van Goor, F1
Bernhardt, R; Bird, IM; Denner, K; Mathis, JM; Pezzi, V; Rainey, WE1
O'Neil, RG; Zhang, MI1
Delpech, N; Potreau, D; Soustre, H1
Dou, CL; Levine, JM1
Kubo, T; Taguchi, K; Ueda, M1
Bond, M; McConnell, BK; Morano, I; Moravec, CS1
Crawford, FA; Doscher, MA; Hebbar, L; Houck, WV; Joshi, JD; Mukherjee, R; Spinale, FG; Thomas, CV; Wang, YH1
Graybiel, AM; Liu, FC1
Bird, IM; Mason, JI; Rainey, WE1
Baker, H; Cigola, E; Franzen, L; Lee, JW; Volpe, BT1
Gohshi, A; Honda, K; Kamiya, H; Motoya, T; Takano, Y; Tominaga, K; Yamada, K1
Gong, GX; Scholz, PM; Tse, J; Weiss, HR; Yan, L1
Beales, IL; Calam, J; Jordinson, M1
Addicks, K; Bloch, W; Bohlen, H; Fleischmann, BK; Hescheler, J; Ji, GJ; Kolossov, E; Liu, Q; Manzke, O; Viatchenko-Karpinski, S1
Abi-Gerges, N; Faivre, V; Fischmeister, R; Mebazaa, A; Méry, PF; Paqueron, X; Payen, D; Tavernier, B1
Betancourt-Calle, S; Bollag, WB; Calle, RA; Jung, EM; Rasmussen, H1
Dedos, SG; Fugo, H1
Pei, JM; Wang, HX; Wong, TM; Yu, XC1
Chen, HL; Jea, JC; Liu, TC; Pu, HF; Tan, SK1
Chik, CL; Ho, AK; Negishi, T1
Coyne, MD; Gwathmey, JK; Kim, CS1
Bauer, R; Doblinger, A; Hoflehner, J; Kapeller, I; Laslop, A1
Buckingham, JC; Christian, HC; Flower, RJ; Morris, JF; Taylor, AD1
Betancourt-Calle, S; Bollag, WB; Calle, RA; Isales, CM; Rasmussen, H; White, S1
Birkenbeil, H; Dedos, SG1
Hino, N; Masumiya, H; Ochi, R; Tsujikawa, H1
Barbuti, A; Palmiter, RD; Protas, L; Qu, J; Robinson, RB; Rybin, VO; Steinberg, SF1
Lo, MJ; Wang, PS1
Gupte, SA; Masumiya, H; Ochi, R; Okada, T; Song, Y; Tsujikawa, H; Watanabe, M1
Bian, JS; Hu, LF; Pan, TT; Yong, QC1
Teramoto, N; Zhu, HL1
Cui, H; Fu, W; Gao, J; Lu, B; Wang, H; Wang, Y; Yu, X; Yu, Y; Zhang, L1
Biraud, M; Cario-Toumaniantz, C; Chevalier, J; Derkinderen, P; Lebouvier, T; Mahé, MM; Neunlist, M; Paillusson, S; Tasselli, M1
Gurgul-Convey, E; Kaminski, MT; Lenzen, S1
Cao, L; Cao, YX; Li, S; Mi, YN; Ping, NN1
Lenzen, S; Teraoku, H1

Reviews

1 review(s) available for bay-k-8644 and colforsin

ArticleYear
Scattered light intensity fluctuation in the canine ventricular myocardium: correlation with inotropic drug effect.
    Canadian journal of physiology and pharmacology, 1988, Volume: 66, Issue:9

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Colforsin; Dobutamine; Dogs; Heart; Light; Myocardial Contraction; Ouabain; Scattering, Radiation; Temperature

1988

Other Studies

107 other study(ies) available for bay-k-8644 and colforsin

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Novel targets for Huntington's disease in an mTOR-independent autophagy pathway.
    Nature chemical biology, 2008, Volume: 4, Issue:5

    Topics: Animals; Autophagy; Calcium Channels, L-Type; Clonidine; Cyclic AMP; Humans; Huntington Disease; Imidazoline Receptors; Minoxidil; Protein Kinases; Signal Transduction; TOR Serine-Threonine Kinases; Type C Phospholipases; Verapamil

2008
Regulation of the chromaffin granule catecholamine transporter in cultured bovine adrenal medullary cells: stimulus-biosynthesis coupling.
    Journal of neurochemistry, 1992, Volume: 59, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholinesterase; Adrenal Medulla; Animals; Biological Transport; Carbachol; Carrier Proteins; Catecholamine Plasma Membrane Transport Proteins; Catecholamines; Cattle; Cells, Cultured; Chromaffin Granules; Chromogranin A; Chromogranins; Colforsin; Cyclic AMP; Cycloheximide; Dactinomycin; Dopamine beta-Hydroxylase; Membrane Proteins; Membrane Transport Proteins; Nifedipine; Potassium; Protein Kinase C; Tetrabenazine; Time Factors; Tritium; Tyrosine 3-Monooxygenase

1992
Lidocaine inhibits prolactin secretion in GH4C1 cells by blocking calcium influx.
    Molecular and cellular endocrinology, 1992, Volume: 87, Issue:1-3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenoma; Animals; Calcium; Colforsin; Lidocaine; Pituitary Neoplasms; Potassium; Procaine; Prolactin; Rats; Tetradecanoylphorbol Acetate; Tetrodotoxin; Tumor Cells, Cultured

1992
Regulation of brain-derived neurotrophic factor and nerve growth factor mRNA in primary cultures of hippocampal neurons and astrocytes.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:12

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Astrocytes; Brain-Derived Neurotrophic Factor; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Cytokines; Glutamates; Glutamic Acid; Growth Substances; Hippocampus; Ionomycin; Isoquinolines; Kainic Acid; Kinetics; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Nifedipine; Norepinephrine; Piperazines; Potassium; Protein Kinase Inhibitors; Quisqualic Acid; Rats; RNA, Messenger; Tetradecanoylphorbol Acetate

1992
Activation of beta-adrenergic receptors inhibits Ca2+ entry-mediated generation of inositol phosphates in the guinea pig myometrium, a cyclic AMP-independent event.
    Molecular pharmacology, 1992, Volume: 41, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aluminum; Animals; Calcium; Calcium Channels; Carbachol; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Drug Antagonism; Female; Fluorine; Guinea Pigs; Inositol Phosphates; Ionomycin; Isoproterenol; Myometrium; Nifedipine; Oxytocin; Pertussis Toxin; Receptors, Adrenergic, beta; Type C Phospholipases; Verapamil; Virulence Factors, Bordetella

1992
Cyclic-AMP-dependent positive chrono- and inotropic responses in the blood-perfused dog atrium.
    Advances in second messenger and phosphoprotein research, 1992, Volume: 25

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Colforsin; Depression, Chemical; Dogs; Heart Atria; Heart Rate; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Perfusion; Stimulation, Chemical

1992
Evidence that the FSH receptor itself is not a calcium channel.
    Endocrinology, 1992, Volume: 131, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Bucladesine; Calcium Channels; Cell Line, Transformed; Colforsin; Cyclic AMP; DNA; Electrophysiology; Embryo, Mammalian; Follicle Stimulating Hormone; Humans; Membrane Potentials; Receptors, FSH; Tetraethylammonium; Tetraethylammonium Compounds; Transfection

1992
The rat angiotensin II AT1A receptor couples with three different signal transduction pathways.
    Biochemical and biophysical research communications, 1992, Jul-31, Volume: 186, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Angiotensin II; Animals; Binding, Competitive; Calcium; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Egtazic Acid; Kinetics; Neomycin; Nicardipine; Rats; Receptors, Angiotensin; Recombinant Proteins; Signal Transduction; Transfection; Type C Phospholipases

1992
Agents that affect calcium influx can change cyclic nucleotide levels in cultured chick pineal cells.
    Brain research, 1992, Jun-26, Volume: 583, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Cells, Cultured; Chickens; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Egtazic Acid; Kinetics; Nitrendipine; Pineal Gland

1992
The effects of P1- and muscarinic-receptor agonists upon cAMP-dependent and independent inotropic responses of guinea-pig cardiac preparations.
    General pharmacology, 1992, Volume: 23, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Carbachol; Colforsin; Cyclic AMP; Guinea Pigs; Heart; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Papillary Muscles; Phenylisopropyladenosine; Receptors, Muscarinic; Receptors, Purinergic

1992
Beta-adrenergic regulation of a myocardial actin gene via a cyclic AMP-independent pathway.
    The Journal of biological chemistry, 1992, Oct-15, Volume: 267, Issue:29

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Actins; Animals; Animals, Newborn; Blotting, Northern; Bucladesine; Caffeine; Calcimycin; Cells, Cultured; Colforsin; Cyclic AMP; Enkephalins; Gene Expression Regulation; Heart; Heart Ventricles; Isoproterenol; Kinetics; Myocardium; Nifedipine; Potassium Chloride; Propranolol; Protein Precursors; Rats; Receptors, Adrenergic, beta; RNA; RNA, Messenger; Ryanodine

1992
The indirect negative inotropic effects of the P1-receptor agonist, L-phenylisopropyladenosine, in guinea-pig isolated cardiac preparations: comparison with cromakalim.
    Canadian journal of physiology and pharmacology, 1992, Volume: 70, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atrial Function; Atrial Function, Left; Benzopyrans; Cardiotonic Agents; Colforsin; Cromakalim; Depression, Chemical; Guinea Pigs; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Papillary Muscles; Phenylisopropyladenosine; Pyrroles; Stimulation, Chemical; Time Factors

1992
Role of calcium and cAMP in heterologous up-regulation of the 1,25-dihydroxyvitamin D3 receptor in an osteoblast cell line.
    Cell calcium, 1990, Volume: 11, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenine; Adenylyl Cyclase Inhibitors; Calcitriol; Calcium; Cell Line; Colforsin; Cyclic AMP; Dinoprostone; Nitrendipine; Osteoblasts; Parathyroid Hormone; Receptors, Calcitriol; Receptors, Steroid; Up-Regulation; Verapamil

1990
Vasoactive intestinal peptide stimulates chick pineal melatonin production and interacts with other stimulatory and inhibitory agents but does not show alpha 1-adrenergic potentiation.
    Journal of neurochemistry, 1990, Volume: 55, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Chickens; Colforsin; Drug Interactions; Isoproterenol; Kinetics; Light; Melatonin; Nitrendipine; Norepinephrine; Phenylephrine; Pineal Gland; Receptors, Adrenergic, alpha; Vasoactive Intestinal Peptide; Yohimbine

1990
Biphasic action of forskolin on growth hormone and prolactin secretion by rat anterior pituitary cells in vitro.
    Endocrinology, 1990, Volume: 127, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Calcimycin; Cells, Cultured; Cholera Toxin; Colforsin; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Activation; Female; Growth Hormone; Growth Hormone-Releasing Hormone; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Somatostatin; Virulence Factors, Bordetella

1990
Phorbol esters enhance stretch-induced atrial natriuretic peptide secretion.
    Endocrinology, 1990, Volume: 127, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atrial Natriuretic Factor; Colforsin; Heart; Heart Atria; Male; Physical Stimulation; Radioimmunoassay; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate

1990
Relationship between proliferation and cell cycle-dependent Ca2+ influx induced by a combination of thyrotropin and insulin-like growth factor-I in rat thyroid cells.
    The Journal of clinical investigation, 1990, Volume: 86, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Cell Cycle; Cell Division; Cell Line; Cobalt; Colforsin; DNA; Drug Combinations; Insulin-Like Growth Factor I; Kinetics; Lanthanum; Pertussis Toxin; Rats; Thyroid Gland; Thyrotropin; Virulence Factors, Bordetella

1990
High affinity forskolin inhibition of L-type Ca2+ current in cardiac cells.
    Molecular pharmacology, 1990, Volume: 38, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Colforsin; Cyclic AMP; In Vitro Techniques; Kinetics; Myocardium; Phosphorylation; Rana esculenta

1990
Cardiac inotropic responses to calcium and forskolin are not altered by prolonged isoproterenol infusion.
    European journal of pharmacology, 1990, Oct-09, Volume: 187, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Colforsin; Cyclic AMP; Drug Interactions; Heart; In Vitro Techniques; Infusions, Intravenous; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Nifedipine; Radioligand Assay; Rats; Receptors, Adrenergic, beta

1990
Cyclic-AMP-dependent phosphorylation modulates the stereospecific activation of cardiac Ca channels by Bay K 8644.
    Pflugers Archiv : European journal of physiology, 1990, Volume: 417, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Colforsin; Cyclic AMP; Drug Combinations; Electric Conductivity; Heart; Isoproterenol; Membrane Potentials; Myocardium; Phosphorylation; Rats

1990
Pharmacological evidence for two types of myocardial sarcoplasmic reticulum Ca2+ release.
    The American journal of physiology, 1991, Volume: 260, Issue:3 Pt 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Anesthetics, Local; Animals; Caffeine; Calcium; Colforsin; Guinea Pigs; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Myocardium; Ryanodine; Sarcolemma; Sodium

1991
Regulation of endothelin-mediated calcium mobilization in vascular smooth muscle cells by isoproterenol.
    The American journal of physiology, 1991, Volume: 260, Issue:3 Pt 1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Cell Line; Colforsin; Cyclic AMP; Endothelins; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Isoproterenol; Kinetics; Muscle, Smooth, Vascular; Potassium; Propranolol

1991
Calcium currents in the A7r5 smooth muscle-derived cell line.
    Pflugers Archiv : European journal of physiology, 1990, Volume: 417, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta; Biological Transport; Calcium; Calcium Channels; Cell Line; Colforsin; Cytosol; Dihydropyridines; Electric Conductivity; Fluorescence; Isoproterenol; Ligands; Muscle, Smooth, Vascular; Nifedipine; Potassium

1990
Effect of positive inotropic agents on myosin isozyme population and mechanical activity of cultured rat heart myocytes.
    Circulation research, 1991, Volume: 68, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Animals, Newborn; Bucladesine; Cardiotonic Agents; Cells, Cultured; Colforsin; Heart; Isoenzymes; Isoproterenol; Myocardial Contraction; Myocardium; Myosins; Ouabain; Phenylephrine; Prazosin; Propranolol; Rats

1991
Chloride channel blockers inhibit ACTH secretion from mouse pituitary tumor cells.
    The American journal of physiology, 1991, Volume: 260, Issue:4 Pt 1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adenylate Cyclase Toxin; Adrenocorticotropic Hormone; Animals; Cell Line; Chloride Channels; Colforsin; Corticotropin-Releasing Hormone; Ion Channels; Kinetics; Membrane Proteins; Mice; ortho-Aminobenzoates; Osmolar Concentration; Pertussis Toxin; Pituitary Neoplasms; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella

1991
Comparison of the effects of milrinone and OPC 3911 with those of isoprenaline, forskolin and dibutyryl-cAMP in rat aorta.
    General pharmacology, 1991, Volume: 22, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Bucladesine; Calcium; Colforsin; In Vitro Techniques; Isoproterenol; Male; Milrinone; Phenylephrine; Phosphodiesterase Inhibitors; Potassium; Pyridones; Quinolones; Rats; Rats, Inbred Strains; Vasodilation

1991
Effects of 8-bromo-cyclic GMP on slow channel mediated action potentials of 3-days-old embryonic chick ventricle.
    Journal of developmental physiology, 1991, Volume: 16, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Chick Embryo; Colforsin; Cyclic GMP; Heart Ventricles; Ion Channels; Isoproterenol; Ventricular Function

1991
Plasma membrane calcium flux, protein kinase C activation and smooth muscle contraction.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Cell Membrane; Colforsin; Drug Synergism; Enzyme Activation; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nitrendipine; Ouabain; Perfusion; Phospholipids; Potassium; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate; Vasoconstriction

1985
Activation of tracheal smooth muscle contraction: synergism between Ca2+ and activators of protein kinase C.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:24

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcimycin; Calcium; Cattle; Colforsin; Diterpenes; Drug Synergism; Enzyme Activation; Ethers; In Vitro Techniques; Ionomycin; Muscle Contraction; Muscle, Smooth; Nifedipine; Protein Kinase C; Terpenes; Tetradecanoylphorbol Acetate; Trachea

1985
Effects of new inotropic agents on cyclic nucleotide metabolism and calcium transients in canine ventricular muscle.
    Circulation, 1986, Volume: 73, Issue:3 Pt 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aequorin; Aminopyridines; Amrinone; Animals; Calcium; Carbachol; Cardiotonic Agents; Colforsin; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Enoximone; Female; Imidazoles; Male; Milrinone; Myocardial Contraction; Myocardium; Nifedipine; Nucleotides, Cyclic; Pyrazines; Pyridones; Quinolines; Time Factors

1986
Atrial natriuretic factor does not affect basal, forskolin- and CRF-stimulated adenylate cyclase activity, cAMP formation or ACTH secretion, but does stimulate cGMP synthesis in anterior pituitary.
    Molecular and cellular endocrinology, 1986, Volume: 44, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenocorticotropic Hormone; Animals; Atrial Natriuretic Factor; Cell Line; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; Cyclic GMP; Growth Hormone; Kinetics; Mice; Nifedipine; Pituitary Gland, Anterior; Potassium Chloride; Tetradecanoylphorbol Acetate

1986
A novel type of cardiac calcium channel in ventricular cells.
    Biomedica biochimica acta, 1986, Volume: 45, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Colforsin; Electric Conductivity; Guinea Pigs; In Vitro Techniques; Ion Channels; Isoproterenol; Membrane Potentials; Nifedipine; Ventricular Function

1986
Pharmacological characteristics of receptor-operated and potential-operated Ca2+ channels in rat aorta.
    European journal of pharmacology, 1986, Aug-07, Volume: 127, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Calcium; Colforsin; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Nifedipine; Norepinephrine; Potassium; Rats; Rats, Inbred Strains; Receptors, Cell Surface

1986
The phorbol ester induced atrial natriuretic peptide secretion is stimulated by forskolin and Bay K8644 and inhibited by 8-bromo-cyclic GMP.
    Biochemical and biophysical research communications, 1986, Aug-29, Volume: 139, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atrial Natriuretic Factor; Calcium; Colforsin; Cyclic AMP; Cyclic GMP; Depression, Chemical; Perfusion; Rats; Stimulation, Chemical; Tetradecanoylphorbol Acetate

1986
Vasoactive intestinal peptide and peptide with N-terminal histidine and C-terminal isoleucine increase prolactin secretion in cultured rat pituitary cells (GH4C1) via a cAMP-dependent mechanism which involves transient elevation of intracellular Ca2+.
    Molecular and cellular endocrinology, 1987, Volume: 49, Issue:2-3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Animals; Calcium; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP; Membrane Potentials; Peptide PHI; Pituitary Gland; Prolactin; Rats; Secretory Rate; Thyrotropin-Releasing Hormone; Vasoactive Intestinal Peptide; Verapamil

1987
Involvement of ion channels in the induction of proenkephalin A gene expression by nicotine and cAMP in bovine chromaffin cells.
    The Journal of biological chemistry, 1987, Mar-25, Volume: 262, Issue:9

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adrenal Glands; Animals; Calcium; Cattle; Cells, Cultured; Chromaffin System; Colforsin; Cyclic AMP; Enkephalins; Gallopamil; Gene Expression Regulation; Ion Channels; Nicotine; Nifedipine; Protein Precursors; RNA, Messenger; Sodium; Tubocurarine; Verapamil

1987
Effects of calcium channel activators BAY-K8644 and CGP-28392 on steroidogenesis in granulosa cells of the domestic hen.
    Biochemical and biophysical research communications, 1987, Jul-15, Volume: 146, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcium; Chickens; Colforsin; Female; Granulosa Cells; Luteinizing Hormone; Progesterone; Pyridines; Steroids

1987
A G protein directly regulates mammalian cardiac calcium channels.
    Science (New York, N.Y.), 1987, Nov-27, Volume: 238, Issue:4831

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Colforsin; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guinea Pigs; Heart; Ion Channels; Isoproterenol; Leupeptins; Membrane Potentials; Phosphorylation; Thionucleotides; Ventricular Function

1987
Inhibitory effects of caffeine on contractions and calcium movement in vascular and intestinal smooth muscle.
    British journal of pharmacology, 1988, Volume: 93, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Caffeine; Calcium; Calcium Radioisotopes; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Norepinephrine; Rabbits

1988
Regulation of alpha-bungarotoxin sites in chromaffin cells in culture by nicotinic receptor ligands, K+, and cAMP.
    Molecular pharmacology, 1988, Volume: 34, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenal Medulla; alpha7 Nicotinic Acetylcholine Receptor; Biological Transport; Bucladesine; Bungarotoxins; Carbachol; Cells, Cultured; Colforsin; Enzyme Activation; Gallopamil; Nicotine; Norepinephrine; Potassium; Receptors, Cholinergic; Receptors, Nicotinic; Tubocurarine

1988
Differential vagal inhibition of the positive chronotropic and inotropic responses to cardiotonics in the isolated dog atrium.
    European journal of pharmacology, 1989, Feb-14, Volume: 161, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cardiotonic Agents; Colforsin; Dobutamine; Dogs; Electric Stimulation; Heart; Heart Rate; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Vagus Nerve

1989
Effects of atrial natriuretic factor (ANF) on phenylephrine-triggered intra- and extracellular calcium dependent contraction in rat aorta.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Atrial Natriuretic Factor; Calcium; Colforsin; Cyclic AMP; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phenylephrine; Rats; Rats, Inbred Strains

1989
PD 122860: a novel dihydropyridine with sodium channel stimulating and calcium channel blocking properties.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Colforsin; Coronary Circulation; Dihydropyridines; Electrocardiography; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Ouabain; Rats; Rats, Inbred Strains; Reference Values; Sodium Channels; Veratridine

1989
Diminution by benzodiazepines of the chronotropic responses to noradrenaline in rat isolated atria.
    European journal of pharmacology, 1989, May-30, Volume: 164, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Colforsin; Cyclic AMP; Diazepam; Female; Flumazenil; Heart; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains

1989
Interactions between forskolin, calcium and Bay K 8644 in K+-depolarized rat uterine muscle.
    General pharmacology, 1989, Volume: 20, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Chloride; Colforsin; Female; In Vitro Techniques; Potassium; Rats; Uterine Contraction; Uterus

1989
New positive inotropic agent OPC-8212 modulates single Ca2+ channels in ventricular myocytes of guinea pig.
    Journal of cardiovascular pharmacology, 1989, Volume: 13, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Caffeine; Calcium Channels; Cardiotonic Agents; Colforsin; Cyclic AMP; Depression, Chemical; Dose-Response Relationship, Drug; Guinea Pigs; Heart Ventricles; Isoproterenol; Myocardium; Phosphorylation; Pyrazines; Quinolines

1989
Role of calcium and cAMP in the action of adrenocorticotropin on aldosterone secretion.
    The Journal of biological chemistry, 1985, Apr-10, Volume: 260, Issue:7

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Glands; Adrenocorticotropic Hormone; Aldosterone; Animals; Calcimycin; Calcium; Cattle; Colforsin; Cyclic AMP; Diterpenes; Dose-Response Relationship, Drug; Nifedipine; Phospholipids

1985
Biosynthesis of large dense-core vesicles in PC12 cells: effects of depolarization and second messengers on the mRNA levels of their constituents.
    Brain research. Molecular brain research, 1995, Volume: 31, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Chromaffin Granules; Colforsin; Membrane Potentials; PC12 Cells; Rats; RNA, Messenger; Second Messenger Systems; Solubility; Stimulation, Chemical; Tetradecanoylphorbol Acetate

1995
Lipocortin 1 mediates an early inhibitory action of glucocorticoids on the secretion of ACTH by the rat anterior pituitary gland in vitro.
    Neuroendocrinology, 1993, Volume: 58, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Animals; Annexin A1; Colforsin; Corticotropin-Releasing Hormone; Culture Techniques; Cycloheximide; Dactinomycin; Dexamethasone; Male; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Recombinant Proteins

1993
In situ Ca(2+)-induced Ca2+ release from a ryanodine-sensitive intracellular Ca2+ store in corneal epithelial cells.
    Comparative biochemistry and physiology. B, Comparative biochemistry, 1993, Volume: 106, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding Sites; Caffeine; Calcium; Calcium Channels; Cattle; Colforsin; Cornea; Cyclic AMP; Epithelial Cells; Epithelium; Muscle Proteins; Radioimmunoassay; Ryanodine; Ryanodine Receptor Calcium Release Channel; Signal Transduction

1993
A single transmitter regulates gene expression through two separate mechanisms: cholinergic regulation of phenylethanolamine N-methyltransferase mRNA via nicotinic and muscarinic pathways.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenal Medulla; Animals; Atropine; Binding, Competitive; Calcimycin; Calcium; Carbachol; Cattle; Cells, Cultured; Colforsin; Epinephrine; Gene Expression Regulation, Enzymologic; Hexamethonium; Hexamethonium Compounds; Kinetics; Muscarine; Nicotine; Phenylethanolamine N-Methyltransferase; Piperidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Receptors, Nicotinic; RNA, Messenger

1994
Canine colonic circular muscle generates action potentials without the pacemaker component.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Barium; Calcium Channels; Colforsin; Colon; Dogs; Electric Stimulation; Electrophysiology; Female; Gallopamil; In Vitro Techniques; Male; Microelectrodes; Muscle, Smooth; Neuromuscular Depolarizing Agents; Potassium; Potassium Channels

1994
Multiple mitogenic signalling pathways in chromaffin cells: a model for cell cycle regulation in the nervous system.
    Neuroscience letters, 1994, Feb-28, Volume: 168, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Cell Cycle; Cell Division; Cells, Cultured; Colforsin; Dexamethasone; Ethers, Cyclic; Female; Models, Neurological; Nerve Endings; Nerve Growth Factors; Okadaic Acid; Phosphoprotein Phosphatases; Potassium Chloride; Rats; Rats, Inbred F344; Signal Transduction; Tetradecanoylphorbol Acetate; Tetrodotoxin; Veratridine

1994
Lipocortin 1 and hypothalamo-pituitary function in the rat.
    Annals of the New York Academy of Sciences, 1994, Nov-30, Volume: 746

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Animals; Annexin A1; Antibodies, Monoclonal; Arginine Vasopressin; Colforsin; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Hypothalamo-Hypophyseal System; Hypothalamus; In Vitro Techniques; Interleukin-1; Pituitary Gland, Anterior; Rats

1994
Modulation of calcium currents by a D1 dopaminergic protein kinase/phosphatase cascade in rat neostriatal neurons.
    Neuron, 1995, Volume: 14, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Kinetics; Membrane Potentials; Neostriatum; Neurons; Nifedipine; Phosphoprotein Phosphatases; Protein Phosphatase 1; Rats; Rats, Wistar; Receptors, Dopamine D1; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors

1995
Apoptosis in cerebellar granule cells is blocked by high KCl, forskolin, and IGF-1 through distinct mechanisms of action: the involvement of intracellular calcium and RNA synthesis.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Apoptosis; Calcium; Cerebellum; Colforsin; Electrophysiology; Insulin-Like Growth Factor I; Intracellular Membranes; Neurons; Nifedipine; Potassium; Potassium Chloride; Rats; Rats, Wistar; RNA; Transcription, Genetic

1995
Signal transduction pathways in GnRH- and dopamine D1-stimulated growth hormone secretion in the goldfish.
    The Chinese journal of physiology, 1994, Volume: 37, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Colforsin; Cyclic AMP; Dopamine; Goldfish; Gonadotropin-Releasing Hormone; Growth Hormone; Phospholipases A; Phospholipases A2; Pituitary Gland; Protein Kinase C; Signal Transduction; Verapamil

1994
Calcium entry attenuates adenylyl cyclase activity. A possible mechanism for calcium-induced catecholamine resistance.
    Chest, 1995, Volume: 107, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Epinephrine; Extracellular Space; Humans; Lymphocytes

1995
Zatebradine attenuates cyclic AMP-related positive chronotropic but not inotropic responses in isolated, perfused right atria of the dog.
    Clinical and experimental pharmacology & physiology, 1995, Volume: 22, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic Agonists; Animals; Benzazepines; Cardiovascular Agents; Colforsin; Dogs; Heart Atria; Heart Rate; Myocardial Contraction; Stimulation, Chemical

1995
The effect of nickel chloride on the isolated hemidiaphragm of the rat.
    General pharmacology, 1995, Volume: 26, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Colforsin; Diaphragm; Electric Stimulation; Female; In Vitro Techniques; Isometric Contraction; Lidocaine; Male; Nickel; Rats; Time Factors; Verapamil

1995
Synergistic regulation of vasoactive intestinal polypeptide expression by cyclic AMP and calcium in newborn but not adult rat sensory neurons in culture.
    Neuroscience, 1993, Volume: 53, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Aging; Animals; Animals, Newborn; Axons; Calcitonin Gene-Related Peptide; Calcium; Colforsin; Cyclic AMP; Female; Ganglia, Spinal; Immunohistochemistry; Male; Nerve Growth Factors; Neurons, Afferent; Rats; Rats, Wistar; Signal Transduction; Substance P; Vasoactive Intestinal Peptide

1993
Evidence for the participation of protein kinase C and 3',5'-cyclic AMP-dependent protein kinase in the stimulation of muscle cell proliferation by 1,25-dihydroxy-vitamin D3.
    Molecular and cellular endocrinology, 1993, Volume: 90, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Bucladesine; Calcitriol; Calcium; Calcium Channels; Cell Division; Cells, Cultured; Chick Embryo; Colforsin; Diglycerides; DNA; Dose-Response Relationship, Drug; Muscles; Nifedipine; Protein Kinase C; Protein Kinases; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors

1993
Calcium-independent potentiation of insulin release by cyclic AMP in single beta-cells.
    Nature, 1993, May-27, Volume: 363, Issue:6427

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Activation; Exocytosis; Fluorometry; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Protein Kinase Inhibitors; Protein Kinases

1993
Cross-talk between muscarinic- and adenosine-receptor signalling in the regulation of cytosolic free Ca2+ and insulin secretion.
    The Biochemical journal, 1993, Aug-01, Volume: 293 ( Pt 3)

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine; Atropine; Calcium; Calcium Channels; Carbachol; Cells, Cultured; Colforsin; Cytosol; Enzyme Activation; Glyceraldehyde; Insulin; Insulin Secretion; Ion Channel Gating; Muscarinic Antagonists; Receptors, Muscarinic; Receptors, Purinergic; Signal Transduction; Type C Phospholipases

1993
Mechanism of melatonin signal transduction in the neonatal rat pituitary.
    Neurochemistry international, 1995, Volume: 27, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Calcimycin; Calcium; Colforsin; Cyclic AMP; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Melatonin; Nifedipine; Organ Culture Techniques; Pituitary Gland, Anterior; Rats; Receptors, Cell Surface; Receptors, Melatonin; Signal Transduction

1995
Dexamethasone inhibits the release of TSH from the rat anterior pituitary gland in vitro by mechanisms dependent on de novo protein synthesis and lipocortin 1.
    The Journal of endocrinology, 1995, Volume: 147, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Annexin A1; Calcium Channel Blockers; Colforsin; Depression, Chemical; Dexamethasone; In Vitro Techniques; Male; Pituitary Gland, Anterior; Protein Biosynthesis; Rats; Rats, Sprague-Dawley; Thyrotropin; Thyrotropin-Releasing Hormone; Vasoactive Intestinal Peptide

1995
Evidence for coordinated regulation of osteoblast function by 1,25-dihydroxyvitamin D3 and parathyroid hormone.
    Biochimica et biophysica acta, 1996, Jun-05, Volume: 1312, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcitriol; Calcium; Calcium Channel Agonists; Cell Line; Colforsin; Cyclic AMP; Cytochrome P-450 Enzyme System; Drug Synergism; Enzyme Activation; Humans; Osteoblasts; Osteocalcin; Parathyroid Hormone; Protein Kinase C; Rats; Receptors, Calcitriol; RNA, Messenger; Signal Transduction; Steroid Hydroxylases; Tetradecanoylphorbol Acetate; Up-Regulation; Vitamin D3 24-Hydroxylase

1996
Altered pharmacologic responsiveness of reduced L-type calcium currents in myocytes surviving in the infarcted heart.
    Journal of cardiovascular electrophysiology, 1996, Volume: 7, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Colforsin; Cyclic AMP; Dogs; Heart; Isoproterenol; Myocardial Infarction

1996
CYCLIC adenosine 3',5'-monophosphate potentiates Ca2+ signaling and insulin secretion by phospholipase C-linked hormones in HIT cells.
    Endocrinology, 1996, Volume: 137, Issue:7

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Arginine Vasopressin; Bombesin; Calcium; Calcium-Transporting ATPases; Cell Line; Colforsin; Cricetinae; Cyclic AMP; Egtazic Acid; Enzyme Inhibitors; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Mesocricetus; Nifedipine; Signal Transduction; Terpenes; Thapsigargin; Time Factors

1996
Interactions between signaling pathways in mediating GnRH-stimulated GTH release from goldfish pituitary cells: protein kinase C, but not cyclic AMP is an important mediator of GnRH-stimulated gonadotropin secretion in goldfish.
    General and comparative endocrinology, 1996, Volume: 102, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Arachidonic Acid; Calcium Channel Agonists; Cells, Cultured; Chickens; Colforsin; Cyclic AMP; Diglycerides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Goldfish; Gonadotropin-Releasing Hormone; Gonadotropins, Pituitary; Male; Microspheres; Naphthalenes; Pituitary Gland; Potassium; Protein Kinase C; Salmon; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate

1996
Differential regulation of 11 beta-hydroxylase and aldosterone synthase in human adrenocortical H295R cells.
    Molecular and cellular endocrinology, 1996, Jul-23, Volume: 121, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Cortex; Angiotensin II; Base Sequence; Bucladesine; Calcium Channel Agonists; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cytochrome P-450 CYP11B2; Gene Expression Regulation; Humans; Molecular Sequence Data; Nifedipine; Potassium; Protein Kinase C; Steroid 11-beta-Hydroxylase; Tetradecanoylphorbol Acetate

1996
Regulated calcium channel in apical membranes renal proximal tubule cells.
    The American journal of physiology, 1996, Volume: 271, Issue:5 Pt 1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Calcium; Calcium Channels; Cations, Monovalent; Cell Membrane; Cells, Cultured; Colforsin; Epithelium; Ion Channel Gating; Kidney Tubules, Proximal; Membrane Potentials; Nifedipine; Patch-Clamp Techniques; Rabbits; Substrate Specificity; Tetradecanoylphorbol Acetate

1996
Endothelin-1 inhibits L-type Ca2+ current enhanced by isoprenaline in rat atrial myocytes.
    Journal of cardiovascular pharmacology, 1997, Volume: 29, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic beta-Agonists; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Cyclic AMP; Endothelin-1; Heart Atria; Isoproterenol; Myocardium; Patch-Clamp Techniques; Protein Kinase Inhibitors; Rats

1997
Identification of a neuronal cell surface receptor for a growth inhibitory chondroitin sulfate proteoglycan (NG2).
    Journal of neurochemistry, 1997, Volume: 68, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding Sites; Calcium Channel Agonists; Cellular Senescence; Cerebellum; Chondroitin Sulfate Proteoglycans; Colforsin; Cyclic AMP; Growth Inhibitors; Ionomycin; Neurites; Neurons; Pertussis Toxin; Rats; Receptors, Cell Surface; Virulence Factors, Bordetella

1997
Effects of cAMP and cGMP on L-type calcium channel currents in rat mesenteric artery cells.
    Japanese journal of pharmacology, 1997, Volume: 74, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Colforsin; Cyclic AMP; Cyclic GMP; In Vitro Techniques; Isoquinolines; Male; Membrane Potentials; Mesenteric Arteries; Muscle, Smooth, Vascular; Nifedipine; Nitroglycerin; Patch-Clamp Techniques; Rats; Rats, Wistar

1997
Troponin I phosphorylation in spontaneously hypertensive rat heart: effect of beta-adrenergic stimulation.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 2

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Calcium; Calcium-Binding Proteins; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Electric Stimulation; Enzyme Inhibitors; Heart; Heart Ventricles; Hypertension; Isoproterenol; Marine Toxins; Myocardial Contraction; Myocardium; Myosin Light Chains; Norepinephrine; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Troponin I

1997
Downstream defects in beta-adrenergic signaling and relation to myocyte contractility after cardioplegic arrest.
    The Journal of thoracic and cardiovascular surgery, 1998, Volume: 115, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Colforsin; Heart Arrest, Induced; Isoproterenol; Myocardial Contraction; Receptors, Adrenergic, beta; Signal Transduction; Swine; Time Factors; Ventricular Dysfunction, Left

1998
Region-dependent dynamics of cAMP response element-binding protein phosphorylation in the basal ganglia.
    Proceedings of the National Academy of Sciences of the United States of America, 1998, Apr-14, Volume: 95, Issue:8

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Animals, Newborn; Basal Ganglia; Benzazepines; Calcium; Calcium Channels; Calcium Channels, L-Type; Colforsin; Corpus Striatum; Cyclic AMP Response Element-Binding Protein; Dopamine Agonists; Kinetics; N-Methylaspartate; Organ Culture Techniques; Organ Specificity; Phosphorylation; Rats; Rats, Sprague-Dawley; Time Factors

1998
Protein kinase A, protein kinase C, and Ca(2+)-regulated expression of 21-hydroxylase cytochrome P450 in H295R human adrenocortical cells.
    The Journal of clinical endocrinology and metabolism, 1998, Volume: 83, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Cortex; Angiotensin II; Bucladesine; Calcium; Calcium Channel Agonists; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Gene Expression Regulation, Enzymologic; Humans; Potassium; Protein Kinase C; RNA, Messenger; Signal Transduction; Steroid 21-Hydroxylase; Tetradecanoylphorbol Acetate

1998
Tyrosine hydroxylase expression in primary cultures of olfactory bulb: role of L-type calcium channels.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Oct-01, Volume: 18, Issue:19

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Cells, Cultured; Colforsin; Mice; Mice, Inbred C57BL; Mice, Inbred CBA; Nerve Tissue Proteins; Neurites; Nifedipine; Olfactory Bulb; Potassium Chloride; Stimulation, Chemical; Time Factors; Tyrosine 3-Monooxygenase

1998
Changes in adrenocorticotropic hormone (ACTH) release from the cultured anterior pituitary cells of streptozotocin-induced diabetic rats.
    Biological & pharmaceutical bulletin, 1998, Volume: 21, Issue:8

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Animals; Cells, Cultured; Colforsin; Corticotropin-Releasing Hormone; Diabetes Mellitus, Experimental; Male; Pituitary Gland, Anterior; Rats; Rats, Wistar; Streptozocin

1998
Relationship between decreased function and O2 consumption caused by cyclic GMP in cardiac myocytes and L-type calcium channels.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1998, Volume: 198, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analysis of Variance; Animals; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Cyclic GMP; Heart; Muscle Contraction; Myocardium; Nifedipine; Nitroprusside; Oxygen Consumption; Rabbits; Radioimmunoassay

1998
Soybean agglutinin stimulated cholecystokinin release from cultured rabbit jejunal cells requires calcium influx via L-type calcium channels.
    Peptides, 1998, Volume: 19, Issue:9

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Animals; Calcium; Calcium Channels; Calcium Channels, L-Type; Cell Separation; Cells, Cultured; Cholecystokinin; Colforsin; Enzyme Activation; Jejunum; Lectins; Male; Phenylalanine; Plant Lectins; Protein Kinase C; Rabbits; Radioimmunoassay; Somatostatin; Soybean Proteins; Staurosporine; Verapamil

1998
Functional characteristics of ES cell-derived cardiac precursor cells identified by tissue-specific expression of the green fluorescent protein.
    The Journal of cell biology, 1998, Dec-28, Volume: 143, Issue:7

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Actins; Animals; Caffeine; Calcium; Calcium Channels; Calcium Channels, L-Type; Calcium Signaling; Calcium-Transporting ATPases; Cell Differentiation; Colforsin; Fetal Heart; Fetal Proteins; Gene Expression Regulation, Developmental; Genes, Reporter; Green Fluorescent Proteins; Inositol 1,4,5-Trisphosphate Receptors; Luminescent Proteins; Mice; Muscle Proteins; Myocardial Contraction; Organ Specificity; Patch-Clamp Techniques; Promoter Regions, Genetic; Receptors, Cytoplasmic and Nuclear; Recombinant Fusion Proteins; Ryanodine Receptor Calcium Release Channel; Stem Cells

1998
Sequential changes in autonomic regulation of cardiac myocytes after in vivo endotoxin injection in rat.
    American journal of respiratory and critical care medicine, 1999, Volume: 160, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adenylyl Cyclases; Adrenergic Antagonists; Adrenergic beta-Agonists; Animals; Autonomic Nervous System; Calcium Channel Agonists; Calcium Channels, L-Type; Colforsin; Diterpenes; Electrophysiology; Endotoxemia; Endotoxins; Enzyme Activators; Escherichia coli; Heart; Hemodynamics; In Vitro Techniques; Injections, Intravenous; Isoproterenol; Male; Myocardium; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Rats; Sepsis

1999
Effects of angiotensin II and adrenocorticotropic hormone on myristoylated alanine-rich C-kinase substrate phosphorylation in glomerulosa cells.
    Molecular and cellular endocrinology, 1999, Aug-20, Volume: 154, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Aldosterone; Angiotensin II; Animals; Calcium Channel Agonists; Cattle; Cells, Cultured; Colforsin; Humans; Intracellular Signaling Peptides and Proteins; Membrane Proteins; Myristoylated Alanine-Rich C Kinase Substrate; Phosphorylation; Protein Kinase C; Proteins; Zona Glomerulosa

1999
Interactions between Ca2+ and cAMP in ecdysteroid secretion from the prothoracic glands of Bombyx mori.
    Molecular and cellular endocrinology, 1999, Aug-20, Volume: 154, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bombyx; Bucladesine; Calcimycin; Calcium; Colforsin; Cyclic AMP; Drug Interactions; Ecdysterone; Enzyme Inhibitors; Phosphodiesterase Inhibitors; Second Messenger Systems; Signal Transduction; Thionucleotides; Verapamil

1999
Anti-arrhythmic effect of kappa-opioid receptor stimulation in the perfused rat heart: involvement of a cAMP-dependent pathway.
    Journal of molecular and cellular cardiology, 1999, Volume: 31, Issue:10

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Calcium; Colforsin; Cyclic AMP; Cytosol; Electric Stimulation; Electrocardiography; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Naltrexone; Norepinephrine; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa

1999
Muscarinic regulation of basal versus thyrotropin-releasing hormone-induced prolactin secretion in rat anterior pituitary cells. differential roles of nitric oxide and intracellular calcium mobilization.
    Neuroendocrinology, 1999, Volume: 70, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Calcium Signaling; Colforsin; Cyclic AMP; Female; Neurons; Nitric Oxide; Pertussis Toxin; Pituitary Gland; Prolactin; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Thyrotropin-Releasing Hormone; Virulence Factors, Bordetella

1999
Ceramide enhances growth hormone (GH)-releasing hormone-stimulated cyclic adenosine 3',5'-monophosphate accumulation but inhibits GH release in rat anterior pituitary cells.
    Endocrinology, 1999, Volume: 140, Issue:12

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Ceramides; Colforsin; Cyclic AMP; Glucosyltransferases; Growth Hormone; Growth Hormone-Releasing Hormone; Ionomycin; Ionophores; Male; Meperidine; Pituitary Gland, Anterior; Potassium Chloride; Rats; Rats, Sprague-Dawley

1999
Voltage-dependent calcium channels in ventricular cells of rainbow trout: effect of temperature changes in vitro.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2000, Volume: 278, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adaptation, Physiological; Animals; Barium; Body Temperature; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cardiotonic Agents; Cold Temperature; Colforsin; Heart Ventricles; In Vitro Techniques; Ion Channel Gating; Isoproterenol; Membrane Potentials; Muscle Fibers, Skeletal; Myocardial Contraction; Myocardium; Nifedipine; Oncorhynchus mykiss; Patch-Clamp Techniques; Pyrroles; Tetrodotoxin

2000
Regulation of the biosynthesis and processing of chromogranins in organotypic slices: influence of depolarization, forskolin and differentiating factors.
    The European journal of neuroscience, 2000, Volume: 12, Issue:8

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aspartic Acid Endopeptidases; Calcium Channel Agonists; Cell Differentiation; Chromogranin A; Chromogranins; Colforsin; Gene Expression; Hippocampus; In Situ Hybridization; Membrane Potentials; Nerve Growth Factors; Neurons; Organ Culture Techniques; Potassium; Proprotein Convertase 2; Proprotein Convertases; Proteins; Rats; Rats, Sprague-Dawley; RNA, Messenger; Stimulation, Chemical; Subtilisins

2000
Evidence from immunoneutralization and antisense studies that the inhibitory actions of glucocorticoids on growth hormone release in vitro require annexin 1 (lipocortin 1).
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Annexin A1; Antibodies, Monoclonal; Colforsin; Corticosterone; Dexamethasone; DNA, Antisense; Glucocorticoids; Growth Hormone; Growth Hormone-Releasing Hormone; In Vitro Techniques; Male; Microscopy, Electron; Pituitary Gland; Rats; Rats, Sprague-Dawley

2000
Differential effects of agonists of aldosterone secretion on steroidogenic acute regulatory phosphorylation.
    Molecular and cellular endocrinology, 2001, Feb-28, Volume: 173, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Aldosterone; Angiotensin II; Animals; Blotting, Western; Calcium Channel Agonists; Cattle; Cells, Cultured; Colforsin; Electrophoresis, Gel, Two-Dimensional; Phosphoproteins; Phosphorylation; Potassium Chloride; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate; Vasoconstrictor Agents; Zona Glomerulosa

2001
Inhibition of cAMP signalling cascade-mediated Ca2+ influx by a prothoracicostatic peptide (Mas-MIP I) via dihydropyridine-sensitive Ca2+ channels in the prothoracic glands of the silkworm, Bombyx mori.
    Insect biochemistry and molecular biology, 2003, Volume: 33, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bombyx; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Cells, Cultured; Colforsin; Cyclic AMP; Dihydropyridines; Exocrine Glands; Kinetics; Larva; Signal Transduction

2003
Modulation of manganese currents by 1, 4-dihydropyridines, isoproterenol and forskolin in rabbit ventricular cells.
    Pflugers Archiv : European journal of physiology, 2003, Volume: 446, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic beta-Agonists; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Colforsin; Cyclic AMP; Dihydropyridines; Electrophysiology; Heart Ventricles; In Vitro Techniques; Ion Channel Gating; Ion Channels; Isoproterenol; Manganese; Membrane Potentials; Myocardium; Myocytes, Cardiac; Nitrendipine; Patch-Clamp Techniques; Rabbits; Signal Transduction

2003
Neuropeptide Y is an essential in vivo developmental regulator of cardiac ICa,L.
    Circulation research, 2003, Nov-14, Volume: 93, Issue:10

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Animals, Newborn; Calcium Channel Agonists; Calcium Channels, L-Type; Cell Separation; Colforsin; Female; Gene Expression Regulation, Developmental; Heart Ventricles; Male; Mice; Mice, Transgenic; Myocardium; Myocytes, Cardiac; Neuropeptide Y; Patch-Clamp Techniques

2003
Relative and combined effects of estradiol and prolactin on corticosterone secretion in ovariectomized rats.
    The Chinese journal of physiology, 2003, Sep-30, Volume: 46, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adrenocorticotropic Hormone; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Colforsin; Corticosterone; Cyclic AMP; Drug Synergism; Estradiol; Female; Injections, Intravenous; Nifedipine; Ovariectomy; Phosphodiesterase Inhibitors; Prolactin; Rats; Rats, Sprague-Dawley; Signal Transduction

2003
Cholesterol depletion modulates basal L-type Ca2+ current and abolishes its -adrenergic enhancement in ventricular myocytes.
    American journal of physiology. Heart and circulatory physiology, 2008, Volume: 294, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; beta-Cyclodextrins; Calcium Channel Agonists; Calcium Channels, L-Type; Calcium Signaling; Cholesterol; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic CMP; Dose-Response Relationship, Drug; Enzyme Activators; Heart Ventricles; In Vitro Techniques; Isoproterenol; Membrane Microdomains; Membrane Potentials; Myocytes, Cardiac; Rabbits; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Time Factors

2008
Negative regulation of beta-adrenergic function by hydrogen sulphide in the rat hearts.
    Journal of molecular and cellular cardiology, 2008, Volume: 44, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Calcium Signaling; Colforsin; Cyclic AMP; Electric Stimulation; Hydrogen Sulfide; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Myocytes, Cardiac; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta

2008
Antagonistic actions of S(-)-Bay K 8644 on cyclic nucleotide-induced inhibition of voltage-dependent Ba(2+) currents in guinea pig gastric antrum.
    Naunyn-Schmiedeberg's archives of pharmacology, 2008, Volume: 378, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Bucladesine; Calcium Channel Agonists; Calcium Channels, L-Type; Colforsin; Cyclic GMP; Female; Guinea Pigs; In Vitro Techniques; Male; Myocytes, Smooth Muscle; Nitroprusside; Patch-Clamp Techniques; Pyloric Antrum; Stereoisomerism; Vasodilator Agents

2008
Antiarrhythmic effect of acupuncture pretreatment in rats subjected to simulative global ischemia and reperfusion--involvement of adenylate cyclase, protein kinase A, and L-type Ca2+ channel.
    The journal of physiological sciences : JPS, 2008, Volume: 58, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Arrhythmias, Cardiac; Calcium Channel Agonists; Calcium Channels, L-Type; Calcium Signaling; Colforsin; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Electroacupuncture; Electrocardiography; Enzyme Activation; Enzyme Activators; Heart Rate; Male; Myocardial Reperfusion Injury; Myocytes, Cardiac; Perfusion; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1

2008
α-Synuclein expression is induced by depolarization and cyclic AMP in enteric neurons.
    Journal of neurochemistry, 2010, Volume: 115, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; alpha-Synuclein; Animals; Blotting, Western; Calcium Channel Agonists; Calcium Channels, L-Type; Colforsin; Cyclic AMP; Electrophysiology; Enteric Nervous System; Female; Immunohistochemistry; Indicators and Reagents; Mice; Mice, Inbred C57BL; Neurons; Phosphopyruvate Hydratase; Pregnancy; ras Proteins; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Reverse Transcriptase Polymerase Chain Reaction

2010
Physiological characterization of the human EndoC-βH1 β-cell line.
    Biochemical and biophysical research communications, 2015, Aug-14, Volume: 464, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Diphosphate; Adenosine Triphosphate; Biological Transport; Calcium Channels; Cell Line; Colforsin; Founder Effect; Gene Expression; Glucokinase; Glucose; Glucose Transporter Type 1; Glucose Transporter Type 2; Glutamine; Glyburide; Humans; Insulin; Insulin-Secreting Cells; Keto Acids; Leucine; Mannoheptulose; Phosphorylation; Potassium Channels, Inwardly Rectifying

2015
H2S induces vasoconstriction of rat cerebral arteries via cAMP/adenylyl cyclase pathway.
    Toxicology and applied pharmacology, 2015, Dec-15, Volume: 289, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Calcium Channel Agonists; Calcium Channels, L-Type; Cerebral Arteries; Colforsin; Cyclic AMP; Endothelium; Hydrogen Sulfide; Isoproterenol; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Rats; Rats, Sprague-Dawley; Sulfides; Vasoconstriction

2015
Dynamics of Insulin Secretion from EndoC-
    Journal of diabetes research, 2017, Volume: 2017

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Cell Line; Colforsin; Exocytosis; Glucose; Glyburide; Humans; Insulin; Insulin Secretion; Insulin-Secreting Cells; Mannoheptulose; Signal Transduction

2017