bay-k-8644 has been researched along with bucladesine in 39 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 6 (15.38) | 18.7374 |
1990's | 23 (58.97) | 18.2507 |
2000's | 9 (23.08) | 29.6817 |
2010's | 1 (2.56) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Cuddon, P; Fleming, A; Floto, RA; Goldsmith, P; Jahreiss, L; O'Kane, CJ; Pask, D; Rubinsztein, DC; Saiki, S; Sarkar, S; Siddiqi, FH; Ttofi, EK; Williams, A | 1 |
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
Collison, KA; Matsuda, JJ; Segaloff, DL; Shibata, EF; Volk, KA | 1 |
Mienville, JM | 1 |
Bishopric, NH; Sato, B; Webster, KA | 1 |
Hall, PF; Kawamura, M; Yanagibashi, K | 1 |
Berger, HJ; Pfeifer, A; Rupp, H; Werdan, K | 1 |
Chambers, TJ; Gilgenkrantz, JL; Hall, TJ | 1 |
Andersson, KE; Lindgren, S | 1 |
Delay, MJ; Hochman, D; MacVicar, BA; Weiss, S | 1 |
Kongsamut, S; Miller, RJ | 1 |
Asem, EK; Tsang, BK | 1 |
Warbanow, W; Will-Shahab, L | 2 |
Noronha-Blob, L; Richard, C; U'Prichard, DC | 1 |
Afar, R; Geertsen, S; Quik, M; Trifaró, JM | 1 |
Miras-Portugal, MT; Rodriguez-Pascual, F; Torres, M | 1 |
Akimoto, T; Ichida, S; Kishino, H; Matsuda, N; Nakazaki, S; Wada, T | 1 |
Bellido, T; Boland, R; Fernández, LM; Morelli, S | 1 |
Inada, M; Matsubara, H; Suzuki, J | 1 |
Birkenhäger, JC; Pols, HA; van den Bemd, GC; van Leeuwen, JP | 1 |
Bargas, J; Galarraga, E; Hernández-López, S; Reyes, A | 1 |
Clark, BJ; Pezzi, V; Rainey, WE; Stocco, DM | 1 |
Bernhardt, R; Bird, IM; Denner, K; Mathis, JM; Pezzi, V; Rainey, WE | 1 |
Ando, S; Clark, BJ; Pezzi, V; Rainey, WE; Stocco, DM | 1 |
Fares, N; Gomez, JP; Potreau, D | 1 |
Kubo, T; Taguchi, K; Ueda, M | 1 |
Birder, LA; Finkel, MS; Kanai, AJ; Malinski, T; Mesaros, S; Oddis, CV | 1 |
Bird, IM; Mason, JI; Rainey, WE | 1 |
Murata, T; Yamaguchi, M | 1 |
Dedos, SG; Fugo, H | 1 |
Misawa, H; Yamaguchi, M | 1 |
Hanna, ST; Tang, G; Wang, R; Wu, L; Wu, Y | 1 |
He, JQ; Kamp, TJ | 1 |
Chen, X; Furukawa, S; Goldman, B; Houser, SR; Margulies, KB; Piacentino, V | 1 |
Barclay, JK; Murrant, CL; Reading, SA | 1 |
Sawada, N; Yamaguchi, M | 1 |
Berretta, RM; Chen, X; Harris, DM; Houser, SR; Margulies, KB; Piacentino, V; Zhang, X | 1 |
Teramoto, N; Zhu, HL | 1 |
39 other study(ies) available for bay-k-8644 and bucladesine
Article | Year |
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Novel targets for Huntington's disease in an mTOR-independent autophagy pathway.
Topics: Animals; Autophagy; Calcium Channels, L-Type; Clonidine; Cyclic AMP; Humans; Huntington Disease; Imidazoline Receptors; Minoxidil; Protein Kinases; Signal Transduction; TOR Serine-Threonine Kinases; Type C Phospholipases; Verapamil | 2008 |
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
Evidence that the FSH receptor itself is not a calcium channel.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Bucladesine; Calcium Channels; Cell Line, Transformed; Colforsin; Cyclic AMP; DNA; Electrophysiology; Embryo, Mammalian; Follicle Stimulating Hormone; Humans; Membrane Potentials; Receptors, FSH; Tetraethylammonium; Tetraethylammonium Compounds; Transfection | 1992 |
Voltage-clamp study of calcium currents during differentiation in the NCB-20 neuronal cell line.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcium; Calcium Channels; Cell Differentiation; Cricetinae; Cricetulus; Hybrid Cells; Ion Channel Gating; Membrane Potentials; Mice; Neuroblastoma; Neurons; Tumor Cells, Cultured | 1992 |
Beta-adrenergic regulation of a myocardial actin gene via a cyclic AMP-independent pathway.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Actins; Animals; Animals, Newborn; Blotting, Northern; Bucladesine; Caffeine; Calcimycin; Cells, Cultured; Colforsin; Cyclic AMP; Enkephalins; Gene Expression Regulation; Heart; Heart Ventricles; Isoproterenol; Kinetics; Myocardium; Nifedipine; Potassium Chloride; Propranolol; Protein Precursors; Rats; Receptors, Adrenergic, beta; RNA; RNA, Messenger; Ryanodine | 1992 |
Voltage-dependent Ca2+ channels are involved in regulation of steroid synthesis by bovine but not rat fasciculata cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Cortex Hormones; Adrenocorticotropic Hormone; Animals; Bucladesine; Calcium; Calcium Channel Blockers; Calcium Channels; Cattle; Female; Nifedipine; Potassium; Rats; Rats, Inbred Strains; Zona Fasciculata; Zona Reticularis | 1990 |
Effect of positive inotropic agents on myosin isozyme population and mechanical activity of cultured rat heart myocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Animals, Newborn; Bucladesine; Cardiotonic Agents; Cells, Cultured; Colforsin; Heart; Isoenzymes; Isoproterenol; Myocardial Contraction; Myocardium; Myosins; Ouabain; Phenylephrine; Prazosin; Propranolol; Rats | 1991 |
Regulation of calcitonin release from the 6.23 rat C-cell line by cyclic nucleotide analogues and pharmacological mediators.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcitonin; Carcinoma; Dibutyryl Cyclic GMP; Dinoprostone; Histamine; Isoproterenol; Rats; Thyroid Neoplasms; Tumor Cells, Cultured | 1991 |
Comparison of the effects of milrinone and OPC 3911 with those of isoprenaline, forskolin and dibutyryl-cAMP in rat aorta.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Bucladesine; Calcium; Colforsin; In Vitro Techniques; Isoproterenol; Male; Milrinone; Phenylephrine; Phosphodiesterase Inhibitors; Potassium; Pyridones; Quinolones; Rats; Rats, Inbred Strains; Vasodilation | 1991 |
Modulation of intracellular Ca++ in cultured astrocytes by influx through voltage-activated Ca++ channels.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Astrocytes; Bucladesine; Calcium; Calcium Channels; Cells, Cultured; Electrophysiology; Fluorescent Dyes; Fura-2; Intracellular Membranes; Nifedipine; Potassium | 1991 |
Nerve growth factor modulates the drug sensitivity of neurotransmitter release from PC-12 cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcium; Cell Differentiation; Dihydropyridines; Nerve Growth Factors; Nifedipine; Nitrendipine; Norepinephrine; Pheochromocytoma; Potassium; Pyridines; Rats; Secretory Rate | 1986 |
Effects of calcium channel activators BAY-K8644 and CGP-28392 on steroidogenesis in granulosa cells of the domestic hen.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcium; Chickens; Colforsin; Female; Granulosa Cells; Luteinizing Hormone; Progesterone; Pyridines; Steroids | 1987 |
Decreased contractile response after exposure of the rat aorta to Db cAMP or IBMX.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Bucladesine; Calcimycin; Calcium Chloride; Cyclic AMP; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Theophylline | 1987 |
Voltage-sensitive calcium channels in differentiated neuroblastoma X glioma hybrid (NG108-15) cells: characterization by quin 2 fluorescence.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aminoquinolines; Animals; Bucladesine; Calcium; Cricetinae; Dihydropyridines; Fluorescent Dyes; Glioma; Humans; Hybrid Cells; Ion Channels; Membrane Potentials; Neuroblastoma; Potassium Chloride; Sodium; Tetrodotoxin; Veratridine | 1988 |
Altered effect of BAY K 8644 after exposure of the rat aorta to IBMX or Db cAMP.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta; Bucladesine; Cyclic AMP; Dihydropyridines; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Rats; Rats, Inbred Strains; Theophylline | 1988 |
Regulation of alpha-bungarotoxin sites in chromaffin cells in culture by nicotinic receptor ligands, K+, and cAMP.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenal Medulla; alpha7 Nicotinic Acetylcholine Receptor; Biological Transport; Bucladesine; Bungarotoxins; Carbachol; Cells, Cultured; Colforsin; Enzyme Activation; Gallopamil; Nicotine; Norepinephrine; Potassium; Receptors, Cholinergic; Receptors, Nicotinic; Tubocurarine | 1988 |
Modulation of the dihydropyridine-insensitive Ca2+ influx by 8-bromo-guanosine-3':5'-monophosphate, cyclic (8-Br-cGMP) in bovine adrenal chromaffin cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Bucladesine; Calcium; Calcium Channels; Cattle; Cells, Cultured; Cyclic GMP; Dihydropyridines; Neomycin; Nerve Tissue Proteins; omega-Agatoxin IVA; omega-Conotoxin GVIA; Peptides; Potassium Chloride; Second Messenger Systems; Spider Venoms | 1994 |
Specific bindings of [3H](+)PN200-110 and [125I]omega-conotoxin to crude membranes from differentiated NG108-15 cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain; Bucladesine; Cell Differentiation; Cell Membrane; Diltiazem; Glioma; Hybrid Cells; Isradipine; Mollusk Venoms; Neuroblastoma; Nitrendipine; omega-Conotoxin GVIA; Potassium Chloride; Rats; Tumor Cells, Cultured; Verapamil | 1993 |
Evidence for the participation of protein kinase C and 3',5'-cyclic AMP-dependent protein kinase in the stimulation of muscle cell proliferation by 1,25-dihydroxy-vitamin D3.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Alkaloids; Animals; Bucladesine; Calcitriol; Calcium; Calcium Channels; Cell Division; Cells, Cultured; Chick Embryo; Colforsin; Diglycerides; DNA; Dose-Response Relationship, Drug; Muscles; Nifedipine; Protein Kinase C; Protein Kinases; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors | 1993 |
Shaker-related potassium channel, Kv1.4, mRNA regulation in cultured rat heart myocytes and differential expression of Kv1.4 and Kv1.5 genes in myocardial development and hypertrophy.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aging; Animals; Animals, Newborn; Atrial Natriuretic Factor; Base Sequence; Bucladesine; Cardiomegaly; Cells, Cultured; DNA Primers; Gene Expression Regulation; Heart; Heart Ventricles; Molecular Sequence Data; Myocardium; Nifedipine; Oligonucleotides, Antisense; Polymerase Chain Reaction; Potassium Channels; Rats; Rats, Sprague-Dawley; Rats, Wistar; RNA, Messenger | 1993 |
Evidence for coordinated regulation of osteoblast function by 1,25-dihydroxyvitamin D3 and parathyroid hormone.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcitriol; Calcium; Calcium Channel Agonists; Cell Line; Colforsin; Cyclic AMP; Cytochrome P-450 Enzyme System; Drug Synergism; Enzyme Activation; Humans; Osteoblasts; Osteocalcin; Parathyroid Hormone; Protein Kinase C; Rats; Receptors, Calcitriol; RNA, Messenger; Signal Transduction; Steroid Hydroxylases; Tetradecanoylphorbol Acetate; Up-Regulation; Vitamin D3 24-Hydroxylase | 1996 |
Dopamine modulates the afterhyperpolarization in neostriatal neurones.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Bucladesine; Calcium Channel Agonists; Dopamine; Dopamine D2 Receptor Antagonists; In Vitro Techniques; Neostriatum; Neurons; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1996 |
The steroidogenic acute regulatory protein is induced by angiotensin II and K+ in H295R adrenocortical cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aldosterone; Angiotensin II; Bucladesine; Calcium Channel Agonists; Cell Line; Cyclic AMP-Dependent Protein Kinases; Humans; Phosphoproteins; Potassium; Protein Kinase C; Tetradecanoylphorbol Acetate; Time Factors | 1995 |
Differential regulation of 11 beta-hydroxylase and aldosterone synthase in human adrenocortical H295R cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Cortex; Angiotensin II; Base Sequence; Bucladesine; Calcium Channel Agonists; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cytochrome P-450 CYP11B2; Gene Expression Regulation; Humans; Molecular Sequence Data; Nifedipine; Potassium; Protein Kinase C; Steroid 11-beta-Hydroxylase; Tetradecanoylphorbol Acetate | 1996 |
Role of calmodulin-dependent protein kinase II in the acute stimulation of aldosterone production.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Cortex; Aldosterone; Angiotensin II; Benzylamines; Bucladesine; Calcium Channel Agonists; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cell Line; Enzyme Inhibitors; Humans; Hydroxycholesterols; Imidazoles; Phosphoproteins; Potassium; Sulfonamides | 1996 |
Effects of Bay K 8644 on L-type calcium current from newborn rat cardiomyocytes in primary culture.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic beta-Agonists; Animals; Animals, Newborn; Bucladesine; Calcium; Calcium Channel Agonists; Calcium Channels; Cells, Cultured; Heart; Isoproterenol; Membrane Potentials; Myocardium; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Phosphorylation; Rats; Rats, Wistar | 1996 |
Effects of cAMP and cGMP on L-type calcium channel currents in rat mesenteric artery cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Colforsin; Cyclic AMP; Cyclic GMP; In Vitro Techniques; Isoquinolines; Male; Membrane Potentials; Mesenteric Arteries; Muscle, Smooth, Vascular; Nifedipine; Nitroglycerin; Patch-Clamp Techniques; Rats; Rats, Wistar | 1997 |
Beta-adrenergic regulation of constitutive nitric oxide synthase in cardiac myocytes.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aging; Animals; Animals, Newborn; Bucladesine; Calcimycin; Cells, Cultured; Dobutamine; Enzyme Induction; Guanosine Diphosphate; Heart; Interleukin-1; Isoproterenol; Myocardial Contraction; Myocardium; Nitric Oxide; Nitric Oxide Synthase; Norepinephrine; omega-N-Methylarginine; Rats; Receptors, Adrenergic, beta; Terbutaline; Thionucleotides; Trifluoperazine | 1997 |
Protein kinase A, protein kinase C, and Ca(2+)-regulated expression of 21-hydroxylase cytochrome P450 in H295R human adrenocortical cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Cortex; Angiotensin II; Bucladesine; Calcium; Calcium Channel Agonists; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Gene Expression Regulation, Enzymologic; Humans; Potassium; Protein Kinase C; RNA, Messenger; Signal Transduction; Steroid 21-Hydroxylase; Tetradecanoylphorbol Acetate | 1998 |
Promoter characterization of the rat gene for Ca2+-binding protein regucalcin. Transcriptional regulation by signaling factors.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Base Sequence; Bucladesine; Calcium-Binding Proteins; Carboxylic Ester Hydrolases; Chromosome Mapping; Dexamethasone; Estradiol; Insulin; Intracellular Signaling Peptides and Proteins; Molecular Sequence Data; Polymerase Chain Reaction; Promoter Regions, Genetic; Rats; Sulfotransferases; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1999 |
Interactions between Ca2+ and cAMP in ecdysteroid secretion from the prothoracic glands of Bombyx mori.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bombyx; Bucladesine; Calcimycin; Calcium; Colforsin; Cyclic AMP; Drug Interactions; Ecdysterone; Enzyme Inhibitors; Phosphodiesterase Inhibitors; Second Messenger Systems; Signal Transduction; Thionucleotides; Verapamil | 1999 |
Involvement of hepatic nuclear factor I binding motif in transcriptional regulation of Ca(2+)-binding protein regucalcin gene.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Amino Acid Motifs; Animals; Base Sequence; Binding Sites; Bucladesine; Calcium-Binding Proteins; Carboxylic Ester Hydrolases; CCAAT-Enhancer-Binding Proteins; DNA; DNA Primers; DNA-Binding Proteins; Gene Expression Regulation; In Vitro Techniques; Insulin; Intracellular Signaling Peptides and Proteins; Liver; Liver Neoplasms, Experimental; Male; Molecular Sequence Data; Mutation; NFI Transcription Factors; Promoter Regions, Genetic; Protein Binding; Rats; Rats, Wistar; Sulfotransferases; Tetradecanoylphorbol Acetate; Transcription Factors; Tumor Cells, Cultured; Y-Box-Binding Protein 1 | 2000 |
Altered L-type Ca(2+) channel currents in vascular smooth muscle cells from experimental diabetic rats.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arteries; Bucladesine; Calcium Channels, L-Type; Cells, Cultured; Cyclic AMP; Diabetes Mellitus, Experimental; Dihydropyridines; Electric Conductivity; Glucose; Male; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Tail | 2000 |
L-type Ca2+ channels gaining respect in heart failure.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic beta-Agonists; Bucladesine; Calcium Channel Agonists; Calcium Channels, L-Type; Heart Failure; Heart Ventricles; Humans; Isoproterenol; Membrane Potentials | 2002 |
L-type Ca2+ channel density and regulation are altered in failing human ventricular myocytes and recover after support with mechanical assist devices.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic beta-Agonists; Bucladesine; Calcium Channel Agonists; Calcium Channels, L-Type; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Heart Failure; Heart Ventricles; Heart-Assist Devices; Humans; Isoproterenol; Membrane Potentials; Middle Aged; Okadaic Acid; Phosphoprotein Phosphatases; Phosphorylation; Protein Phosphatase 2 | 2002 |
Increased cAMP as a positive inotropic factor for mammalian skeletal muscle in vitro.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic beta-Agonists; Animals; Bucladesine; Caffeine; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Cyclic AMP; Dantrolene; Diltiazem; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Mice; Muscle Relaxants, Central; Muscle, Skeletal; Sarcolemma; Sarcoplasmic Reticulum; Time Factors | 2003 |
Overexpression of RGPR-p117 enhances regucalcin gene promoter activity in cloned normal rat kidney proximal tubular epithelial cells: involvement of TTGGC motif.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Base Sequence; Bucladesine; Calcium-Binding Proteins; Carboxylic Ester Hydrolases; Clone Cells; Consensus Sequence; DNA; DNA-Binding Proteins; Epithelial Cells; Gene Expression; Genes, Reporter; Hormones; Intracellular Signaling Peptides and Proteins; Kidney Tubules, Proximal; Luciferases; Promoter Regions, Genetic; Rats; RNA, Messenger; Sequence Deletion; Signal Transduction; Sulfotransferases; Tetradecanoylphorbol Acetate; Transfection; Two-Hybrid System Techniques | 2006 |
Reduced effects of BAY K 8644 on L-type Ca2+ current in failing human cardiac myocytes are related to abnormal adrenergic regulation.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenergic beta-Agonists; Bucladesine; Calcium Channel Agonists; Calcium Channels, L-Type; Cardiotonic Agents; Catecholamines; Drug Resistance; Heart Failure; Heart Ventricles; Heart-Assist Devices; Humans; Isoproterenol; Membrane Potentials; Myocardial Contraction; Myocytes, Cardiac; Phosphorylation | 2008 |
Antagonistic actions of S(-)-Bay K 8644 on cyclic nucleotide-induced inhibition of voltage-dependent Ba(2+) currents in guinea pig gastric antrum.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Bucladesine; Calcium Channel Agonists; Calcium Channels, L-Type; Colforsin; Cyclic GMP; Female; Guinea Pigs; In Vitro Techniques; Male; Myocytes, Smooth Muscle; Nitroprusside; Patch-Clamp Techniques; Pyloric Antrum; Stereoisomerism; Vasodilator Agents | 2008 |