bay-k-8644 and 4-aminopyridine

bay-k-8644 has been researched along with 4-aminopyridine in 28 studies

Research

Studies (28)

TimeframeStudies, this research(%)All Research%
pre-19902 (7.14)18.7374
1990's15 (53.57)18.2507
2000's6 (21.43)29.6817
2010's5 (17.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Kaneda, M; Kaneko, A; Ueda, Y1
Sanders, KM; Thornbury, KD; Ward, SM1
Deitmer, P; Lammel, E; Noack, T1
Furukawa, T; Katsuragi, T; Ogawa, S; Shirakabe, K; Soejima, O1
Barrett, EF; Morita, K1
Mantovani, P; Palmi, M; Petkov, VV; Sgaragli, GP1
Jonkman, FA; Korstanje, C; Van Kemenade, JE; Van Zwieten, PA1
Massieu, L; Tapia, R1
Bonev, AD; Mawe, GM; Nelson, MT; Zhang, L1
Bilodeau, L; Durroux, T; Gallo-Payet, N; Guillon, G; Payet, MD1
Bertaccini, G; Coruzzi, G; Poli, E; Pozzoli, C1
Hume, RI; Lin, X; Nuttall, AL1
Brady, G; Docherty, JR1
Hu, Q; Huang, F; Shi, Y1
Maggi, CA; Santicioli, P1
Cotton, KD; Hollywood, MA; McHale, NG; Thornbury, KD1
Apaydin, S; Ates, M; Gelal, A; Guven, H; Tuncok, Y1
Ghisdal, P; Gomez, JP; Morel, N1
Malvin, GM; Walker, BR1
Flameng, W; Macianskiene, R; Moccia, F; Mubagwa, K; Sipido, KR1
Nedergaard, OA; Uhrenholt, TR1
Keum, EM; Kim, SC; Lee, MY; Myung, SC; Park, SY1
Arcanjo, DD; Cavalcanti, SC; Oliveira, AP; Oliveira, NN; Oliveira, Rde C; Quintans-Júnior, LJ; Santos, MR; Silva-Filho, JC1
Fan, X; Hess, EJ; Hughes, KE; Jinnah, HA1
Boehm, S; Geier, P; Gupta, KD; Kubista, H; Lagler, M; Rubi, L; Schandl, U; Spies, D1
Cavalcante, Fde A; Correia, AC; da Silva, BA; de Souza, IL; Paredes-Gamero, EJ; Santos, BV; Silva, Mda C; Vasconcelos, LH1

Other Studies

28 other study(ies) available for bay-k-8644 and 4-aminopyridine

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Voltage-dependent ionic currents in solitary horizontal cells isolated from cat retina.
    Journal of neurophysiology, 1992, Volume: 68, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Action Potentials; Animals; Calcium Channels; Cats; Cells, Cultured; Cesium; Electric Conductivity; Membrane Potentials; Nifedipine; Potassium Channels; Retinal Ganglion Cells; Sodium; Sodium Channels; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin

1992
Outward currents in longitudinal colonic muscle cells contribute to spiking electrical behavior.
    The American journal of physiology, 1992, Volume: 263, Issue:1 Pt 1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Action Potentials; Animals; Calcium; Colon; Dogs; Electrophysiology; Female; Male; Muscle, Smooth; Nifedipine; Tetraethylammonium; Tetraethylammonium Compounds

1992
Characterization of membrane currents in single smooth muscle cells from the guinea-pig gastric antrum.
    The Journal of physiology, 1992, Volume: 451

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Caffeine; Calcium; Guinea Pigs; In Vitro Techniques; Kinetics; Membrane Potentials; Muscle, Smooth; Nifedipine; Potassium; Pyloric Antrum; Tetraethylammonium; Tetraethylammonium Compounds

1992
Involvement of dihydropyridine-sensitive Ca2+ channels in adenosine-evoked inhibition of acetylcholine release from guinea pig ileal preparation.
    Journal of neurochemistry, 1990, Volume: 55, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Acetylcholine; Adenosine; Animals; Atropine; Bethanechol; Bethanechol Compounds; Calcium Channels; Chromatography, High Pressure Liquid; Dihydropyridines; Electric Stimulation; Guinea Pigs; Ileum; Male; Muscle, Smooth; Nifedipine; Physostigmine; Tetrodotoxin; Theophylline

1990
Evidence for two calcium-dependent potassium conductances in lizard motor nerve terminals.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1990, Volume: 10, Issue:8

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Action Potentials; Animals; Apamin; Caffeine; Calcium; Charybdotoxin; Egtazic Acid; Electric Conductivity; Lizards; Motor Neurons; Muscle Contraction; Nerve Endings; Potassium; Procaine; Scorpion Venoms; Tetraethylammonium; Tetraethylammonium Compounds

1990
4-Aminopyridine activates an inhibitory alpha 1-adrenergic mechanism unmasked by nifedipin on the electrically stimulated rat vas deferens.
    Acta physiologica et pharmacologica Bulgarica, 1990, Volume: 16, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Calcium; Electric Stimulation; Epididymis; In Vitro Techniques; Male; Muscle, Smooth; Nifedipine; Potassium Channels; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vas Deferens

1990
Bay k 8644, a calcium entry promoter, as an antidote in verapamil intoxication in rabbits.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 287, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Aminopyridines; Animals; Antidotes; Atrioventricular Node; Blood Pressure; Cardiovascular Agents; Electrocardiography; Female; Heart Rate; Hydrogen-Ion Concentration; In Vitro Techniques; Ion Channels; Male; Pyridines; Rabbits; Verapamil

1987
Relationship of dihydropyridine binding sites with calcium-dependent neurotransmitter release in synaptosomes.
    Journal of neurochemistry, 1988, Volume: 51, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Aminopyridines; Animals; Brain; Calcium; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; gamma-Aminobutyric Acid; Ion Channels; Isradipine; Lanthanum; Male; Mice; Neurotransmitter Agents; Nifedipine; Nitrendipine; Oxadiazoles; Potassium; Receptors, Nicotinic; Ruthenium Red; Synaptosomes

1988
Ionic basis of the action potential of guinea pig gallbladder smooth muscle cells.
    The American journal of physiology, 1993, Volume: 265, Issue:6 Pt 1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Action Potentials; Animals; Calcium Channels; Cell Membrane; Charybdotoxin; Electrophysiology; Female; Gallbladder; Guinea Pigs; In Vitro Techniques; Male; Membrane Potentials; Muscle, Smooth; Nifedipine; Potassium Channel Blockers; Potassium Channels; Scorpion Venoms; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Time Factors

1993
Characterization of K+ and Ca2+ ionic currents in glomerulosa cells from human adrenal glands.
    Endocrinology, 1994, Volume: 134, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Action Potentials; Adolescent; Adult; Aldosterone; Barium; Cadmium; Calcium Channels; Cells, Cultured; Electric Conductivity; Humans; Kinetics; Membrane Potentials; Nickel; Nifedipine; Potassium Channels; Tetraethylammonium; Tetraethylammonium Compounds; Zona Glomerulosa

1994
Signal transducing mechanisms coupled to histamine H3 receptors and alpha-2 adrenoceptors in the guinea pig duodenum: possible involvement of N-type Ca++ channels.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Calcium Channel Blockers; Calcium Channels; Clonidine; Duodenum; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; omega-Conotoxin GVIA; Peptides; Receptors, Adrenergic, alpha-2; Receptors, Histamine H3; Signal Transduction

1994
Dihydropyridines and verapamil inhibit voltage-dependent K+ current in isolated outer hair cells of the guinea pig.
    Hearing research, 1995, Volume: 88, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Cochlea; Guinea Pigs; Hair Cells, Auditory, Outer; Membrane Potentials; Nifedipine; Nimodipine; Patch-Clamp Techniques; Potassium Channel Blockers; Quinine; Verapamil

1995
Prejunctional actions of K+ channel blockers in rat vas deferens.
    European journal of pharmacology, 1995, Dec-20, Volume: 287, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Adenosine Triphosphate; Anesthetics; Animals; Apamin; Calcium; Charybdotoxin; Electric Stimulation; Enzyme Activation; Isometric Contraction; Male; Neuromuscular Junction; Norepinephrine; Phorbol 12,13-Dibutyrate; Potassium Channel Blockers; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Structure-Activity Relationship; Tetraethylammonium; Tetraethylammonium Compounds; Vas Deferens; Xylazine

1995
Inhibition of Toosendanin on the delayed rectifier potassium current in neuroblastoma x glioma NG108-15 cells.
    Brain research, 1997, Mar-14, Volume: 751, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Delayed Rectifier Potassium Channels; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Glioma; Hybrid Cells; Mice; Neuroblastoma; Neuromuscular Blocking Agents; Nifedipine; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Rats; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1997
Pharmacological modulation of electromechanical coupling in the proximal and distal regions of the guinea-pig renal pelvis.
    Journal of autonomic pharmacology, 1997, Volume: 17, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Action Potentials; Animals; Calcium Channel Blockers; Calcium-Transporting ATPases; Charybdotoxin; Electrophysiology; Enzyme Inhibitors; Guinea Pigs; Indoles; Kidney Pelvis; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Potassium Channels; Sarcoplasmic Reticulum; Tetraethylammonium; Tetraethylammonium Compounds

1997
Outward currents in smooth muscle cells isolated from sheep mesenteric lymphatics.
    The Journal of physiology, 1997, Aug-15, Volume: 503 ( Pt 1)

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Calcium Channel Blockers; Calcium Channels; Female; In Vitro Techniques; Lymphatic System; Male; Membrane Potentials; Muscle, Smooth; Mycotoxins; Nifedipine; Patch-Clamp Techniques; Peptides; Potassium Channels; Sheep; Tetraethylammonium; Tetraethylammonium Compounds

1997
The effects of 4-aminopyridine and Bay K 8644 on verapamil-induced cardiovascular toxicity in anesthetized rats.
    Journal of toxicology. Clinical toxicology, 1998, Volume: 36, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Blood Pressure; Bradycardia; Calcium Channel Agonists; Calcium Channel Blockers; Cardiovascular System; Dose-Response Relationship, Drug; Heart Rate; Hypotension; Male; Random Allocation; Rats; Rats, Wistar; Verapamil

1998
Changes of the potassium currents in rat aortic smooth muscle cells during postnatal development.
    Pflugers Archiv : European journal of physiology, 2000, Volume: 441, Issue:2-3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Aging; Animals; Aorta, Thoracic; Calcium; Calcium Channel Agonists; Charybdotoxin; Electric Conductivity; Male; Membrane Potentials; Muscle Contraction; Muscle Development; Muscle, Smooth, Vascular; Norepinephrine; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Rats; Rats, Wistar; Tetraethylammonium; Vasoconstriction

2000
Sites and ionic mechanisms of hypoxic vasoconstriction in frog skin.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2001, Volume: 280, Issue:5

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Arterioles; Calcium Channels, L-Type; Homeostasis; Hypoxia; Mammals; Muscle, Smooth, Vascular; Nifedipine; Nitrogen; Oxygen; Potassium Channel Blockers; Skin; Time Factors; Vasoconstriction; Vasoconstrictor Agents; Venules; Xenopus laevis

2001
Channels involved in transient currents unmasked by removal of extracellular calcium in cardiac cells.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 282, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cesium; Chelating Agents; Diltiazem; Drug Resistance; Egtazic Acid; Electric Conductivity; Heart Ventricles; Isoproterenol; Kinetics; Magnesium; Membrane Potentials; Myocardium; Nifedipine; Patch-Clamp Techniques; Potassium; Receptors, Adrenergic, beta; Swine; Verapamil

2002
Calcium channels involved in noradrenaline release from sympathetic neurones in rabbit carotid artery.
    Pharmacology & toxicology, 2003, Volume: 92, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, N-Type; Carotid Artery, Common; Electric Stimulation; Female; Male; Neurons; Nifedipine; Nimodipine; Norepinephrine; omega-Conotoxin GVIA; Potassium Channel Blockers; Rabbits; Sympathetic Nervous System; Time Factors

2003
Vasomotor action of insulin on the rabbit normal cavernous smooth muscle.
    European journal of pharmacology, 2006, Apr-24, Volume: 536, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Calcium Channels; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Indomethacin; Insulin; Male; Membrane Potentials; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Penis; Potassium Channel Blockers; Potassium Channels; Prostaglandins; Prostaglandins H; Rabbits; Tetraethylammonium; Vasoconstrictor Agents

2006
Investigation of mechanisms involved in (-)-borneol-induced vasorelaxant response on rat thoracic aorta.
    Basic & clinical pharmacology & toxicology, 2012, Volume: 110, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Aorta, Thoracic; Calcium Chloride; Camphanes; Endothelium, Vascular; Glyburide; Phenylephrine; Potassium Channels; Potassium Chloride; Rats; Tetraethylammonium; Vasodilator Agents

2012
Selective and sustained α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor activation in cerebellum induces dystonia in mice.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Benzothiadiazines; Cerebellum; Dose-Response Relationship, Drug; Dystonia; Female; Male; Mice; Mice, Inbred C57BL; Quisqualic Acid; Receptors, AMPA; Receptors, Kainic Acid

2012
Raised activity of L-type calcium channels renders neurons prone to form paroxysmal depolarization shifts.
    Neuromolecular medicine, 2013, Volume: 15, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Anthracenes; Caffeine; Calcium Channels, L-Type; Calcium Signaling; Cells, Cultured; Dimethyl Sulfoxide; Epilepsy; Excitatory Postsynaptic Potentials; Hippocampus; Hydrogen Peroxide; Isradipine; Magnesium; Neurons; Oxidative Stress; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley

2013
Flavonoid galetin 3,6-dimethyl ether attenuates guinea pig ileum contraction through K(+) channel activation and decrease in cytosolic calcium concentration.
    European journal of pharmacology, 2015, Nov-15, Volume: 767

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Apamin; Calcium; Calcium Chloride; Carbachol; Cell Survival; Cesium; Chlorides; Flavonoids; Glyburide; Guinea Pigs; Histamine; Histamine Antagonists; Ileum; Muscle Cells; Muscle Contraction; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Tetraethylammonium

2015