bay h 4502 has been researched along with ketoconazole in 40 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 5 (12.50) | 18.7374 |
1990's | 8 (20.00) | 18.2507 |
2000's | 7 (17.50) | 29.6817 |
2010's | 17 (42.50) | 24.3611 |
2020's | 3 (7.50) | 2.80 |
Authors | Studies |
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Apuzzo, G; Artico, M; Costi, R; Di Santo, R; Massa, S; Retico, A; Simonetti, G; Strippoli, V | 1 |
Artico, M; Botta, M; Ciacci, A; Corelli, F; Costi, R; Di Santo, R; Manetti, F; Massa, S; Tafi, A | 1 |
Ekins, S; Harwood, HJ; Hoover, DJ; Lawton, MP; Mankowski, DC; Treadway, JL | 1 |
Deising, HB; Serfling, A; Wohlrab, J | 1 |
Bartels, M; Hartmann, RW; Hu, Q; Jahn-Hoffmann, K; Lauterbach, T; Müller-Vieira, U; Negri, M; Olgen, S; Zhuang, Y | 1 |
Camoutsis, C; Cirić, A; Geronikaki, A; Glamoclija, J; Omar, K; Soković, M; Zoumpoulakis, P | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Camoutsis, C; Ciric, A; Geronikaki, A; Soković, M; Zervou, M; Zoumpoulakis, P | 1 |
Cirić, A; Geronikaki, A; Glamočlija, J; Liaras, K; Soković, M | 2 |
Camoutsis, Ch; Glamočlija, J; Pairas, G; Pitsas, A; Potamitis, C; Soković, M; Zoumpoulakis, P | 1 |
Bakmiwewa, SM; Ball, HJ; Fatokun, AA; Hunt, NH; Payne, RJ; Tran, A | 1 |
Apostolidis, I; Ćirić, A; Gavalas, A; Geronikaki, A; Glamočlija, J; Hadjipavlou-Litina, D; Liaras, K; Soković, M | 1 |
Avery, VM; Sykes, ML | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Bron, S; Chambon, M; Colau, D; Majjigapu, SR; Michielin, O; Pilotte, L; Röhrig, UF; Turcatti, G; Van den Eynde, BJ; Vogel, P; Zoete, V | 1 |
Apuzzo, G; Artico, M; Ortar, G; Silvestri, R; Simonetti, G; Stefancich, G | 1 |
Aoki, K; Hosaka, J; Uchida, K; Yamaguchi, H | 1 |
Panico, S; Porretta, GC; Scalzo, M; Simonetti, N; Villa, A | 1 |
Cauwenbergh, G | 1 |
Abruzzo, GK; Fromtling, RA; Giltinan, DM; Turnbull, TA | 1 |
Abbott, AB; Odds, FC; Webster, CE | 1 |
Qadripur, SA | 1 |
Espinel-Ingroff, A; Kerkering, TM; Shadomy, S | 1 |
Apuzzo, G; Artico, M; Pagnozzi, E; Retico, A; Silvestri, R; Simonetti, N; Stefancich, G | 1 |
Hegemann, L; Lahijani, KI; Toso, SM; Uitto, J; Webster, GF | 1 |
Inoue, I; Kitajima, Y; Osada, K; Seishima, M | 1 |
Ahmed, S; Keane, J | 1 |
Gee, BC | 1 |
Höltje, HD; Marian, C; Raub, S; Rupp, B | 1 |
Katoh, T | 1 |
Eichenfield, LF; Friedlander, SF | 1 |
Harada, K; Inagaki, K; Kampirapap, K; Koga, H; Maeda, J; Makimura, K; Nanjoh, Y; Neki, D; Reangchainam, S; Tsuboi, R; Yuasa, K | 1 |
Geronikaki, A; Horishny, V; Ivanov, M; Kartsev, V; Kostic, M; Matiychuk, V; Papadopoulou, TA; Petrou, A; Pogodin, P; Poroikov, V; Sokovic, M; Vizirianakis, IS | 1 |
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
Emami, S; Keighobadi, M; Tavangar, P | 1 |
Camoutsis, C; Ciric, A; Eleftheriou, P; Fesatidou, M; Geronikaki, A; Haroun, M; Petrou, A; Sokovic, M; Tratrat, C; Zagaliotis, P | 1 |
Anthi, P; Athina, G; Boris, L; Marija, S; Marina, K; Marina, S; Oliver, R; Victor, K | 1 |
Ciric, A; Geronikaki, A; Glamoclija, J; Kartsev, V; Krysin, MY; Ledenyova, IV; Medvedeva, SM; Petrou, A; Shikhaliev, KS; Sokovic, M | 1 |
Ciric, A; Drumea, M; Geronikaki, A; Glamoclija, J; Kravtsov, V; Lupascu, L; Macaev, F; Petrou, A; Pogrebnoi, S; Smetanscaia, A; Sokovic, M; Stingaci, E; Uncu, L; Valica, V; Zveaghinteva, M | 1 |
5 review(s) available for bay h 4502 and ketoconazole
Article | Year |
---|---|
Approaches to protozoan drug discovery: phenotypic screening.
Topics: Drug Discovery; Humans; Molecular Structure; Neglected Diseases; Phenotype; Plasmodium falciparum; Protozoan Infections; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma cruzi | 2013 |
Seborrhoeic dermatitis.
Topics: Dermatitis, Seborrheic; Humans; Imidazoles; Ketoconazole; Scalp Dermatoses; Selenium Compounds | 2004 |
[Guidelines for diagnosis and treatment of mucocutaneous candidiasis].
Topics: Administration, Oral; Administration, Topical; Antifungal Agents; Candida albicans; Candidiasis, Chronic Mucocutaneous; Drug Administration Schedule; Humans; Imidazoles; Ketoconazole; Microscopy; Morpholines; Naphthalenes; Practice Guidelines as Topic; Terbinafine | 2009 |
Pediatric Onychomycosis: The Emerging Role of Topical Therapy.
Topics: Administration, Topical; Adult; Age Factors; Antifungal Agents; Child; Ciclopirox; Family; Humans; Imidazoles; Incidence; Ketoconazole; Lacquer; Morpholines; Naphthalenes; Onychomycosis; Prevalence; Pyridones; Recurrence; Terbinafine; Tinea Pedis; Treatment Outcome | 2017 |
An overview of azoles targeting sterol 14α-demethylase for antileishmanial therapy.
Topics: 14-alpha Demethylase Inhibitors; Antiprotozoal Agents; Azoles; Humans; Leishmania; Molecular Structure; Sterol 14-Demethylase | 2017 |
35 other study(ies) available for bay h 4502 and ketoconazole
Article | Year |
---|---|
Antifungal agents. 9. 3-Aryl-4-[alpha-(1H-imidazol-1-yl)arylmethyl]pyrroles: a new class of potent anti-Candida agents.
Topics: Adult; Animals; Antifungal Agents; Candida; Candida albicans; Candidiasis; Drug Resistance, Microbial; Female; Humans; Hydrogen-Ion Concentration; Imidazoles; Male; Molecular Structure; Pyrroles; Rabbits; Structure-Activity Relationship | 1995 |
Antifungal agents. 10. New derivatives of 1-[(aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, synthesis, anti-candida activity, and quantitative structure-analysis relationship studies.
Topics: Antifungal Agents; Candida; Imidazoles; Microbial Sensitivity Tests; Models, Molecular; Molecular Conformation; Pyrroles; Quantitative Structure-Activity Relationship; Stereoisomerism | 2002 |
Three-dimensional quantitative structure-activity relationship analysis of human CYP51 inhibitors.
Topics: Amides; Cytochrome P-450 Enzyme Inhibitors; Enzyme Inhibitors; Humans; Indoles; Models, Molecular; Oxidoreductases; Quantitative Structure-Activity Relationship; Sterol 14-Demethylase | 2007 |
Treatment of a clinically relevant plant-pathogenic fungus with an agricultural azole causes cross-resistance to medical azoles and potentiates caspofungin efficacy.
Topics: Amphotericin B; Antifungal Agents; Azoles; Caspofungin; Colletotrichum; Drug Resistance, Fungal; Drug Synergism; Echinocandins; Fungi; Fungicides, Industrial; Humans; In Vitro Techniques; Lipopeptides; Microbial Sensitivity Tests; Microscopy, Fluorescence; Nystatin; Plant Diseases; Skin; Triazoles | 2007 |
Synthesis, biological evaluation, and molecular modeling studies of methylene imidazole substituted biaryls as inhibitors of human 17alpha-hydroxylase-17,20-lyase (CYP17)--part II: Core rigidification and influence of substituents at the methylene bridge.
Topics: Animals; Binding Sites; Biphenyl Compounds; Enzyme Inhibitors; Humans; Imidazoles; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Male; Models, Molecular; Protein Structure, Secondary; Rats; Spectrometry, Mass, Electrospray Ionization; Spectrophotometry, Infrared; Steroid 17-alpha-Hydroxylase; Testosterone | 2008 |
Novel 4-thiazolidinone derivatives as potential antifungal and antibacterial drugs.
Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Fungi; Isomerism; Microbial Sensitivity Tests; Structure-Activity Relationship; Thiazoles | 2010 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Sulfonamide-1,2,4-thiadiazole derivatives as antifungal and antibacterial agents: synthesis, biological evaluation, lipophilicity, and conformational studies.
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Antifungal Agents; Bacteria; Fungi; Microbial Sensitivity Tests; Models, Molecular; Molecular Conformation; Structure-Activity Relationship; Sulfonamides; Thiadiazoles | 2010 |
Thiazole-based chalcones as potent antimicrobial agents. Synthesis and biological evaluation.
Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Chalcones; Fungi; Humans; Mycoses; Structure-Activity Relationship; Thiazoles | 2011 |
Novel (E)-1-(4-methyl-2-(alkylamino)thiazol-5-yl)-3-arylprop-2-en-1-ones as potent antimicrobial agents.
Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Fungi; Humans; Microbial Sensitivity Tests; Mycoses; Structure-Activity Relationship; Thiazoles | 2011 |
Synthesis of novel sulfonamide-1,2,4-triazoles, 1,3,4-thiadiazoles and 1,3,4-oxadiazoles, as potential antibacterial and antifungal agents. Biological evaluation and conformational analysis studies.
Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Fungi; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Oxadiazoles; Thiadiazoles; Triazoles | 2012 |
Identification of selective inhibitors of indoleamine 2,3-dioxygenase 2.
Topics: Animals; Dose-Response Relationship, Drug; Enzyme Inhibitors; HEK293 Cells; Humans; Indoleamine-Pyrrole 2,3,-Dioxygenase; Mice; Models, Molecular; Molecular Structure; Structure-Activity Relationship; Substrate Specificity | 2012 |
Synthesis and biological evaluation of some 5-arylidene-2-(1,3-thiazol-2-ylimino)-1,3-thiazolidin-4-ones as dual anti-inflammatory/antimicrobial agents.
Topics: Animals; Anti-Infective Agents; Anti-Inflammatory Agents; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase Inhibitors; Drug Evaluation, Preclinical; Edema; Gram-Negative Bacteria; Gram-Positive Bacteria; Mice; Microbial Sensitivity Tests; Thiazoles | 2013 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
Detailed analysis and follow-up studies of a high-throughput screening for indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors.
Topics: Animals; Antifungal Agents; Dose-Response Relationship, Drug; Enzyme Inhibitors; High-Throughput Screening Assays; Humans; Indoleamine-Pyrrole 2,3,-Dioxygenase; Mice; Molecular Dynamics Simulation; Molecular Structure; Structure-Activity Relationship | 2014 |
Antibacterial and antifungal agents. XV. Synthesis and antifungal activity of structural analogues of bifonazole and ketoconazole.
Topics: Antifungal Agents; Candida; Imidazoles; Ketoconazole; Microbial Sensitivity Tests | 1992 |
[In vitro antifungal activity of itraconazole, a new triazole antifungal agent, against clinical isolates from patients with dermatomycoses].
Topics: Amphotericin B; Antifungal Agents; Clotrimazole; Dermatomycoses; Humans; Imidazoles; Itraconazole; Ketoconazole; Miconazole; Microbial Sensitivity Tests | 1991 |
Antimicrobial activity of a new derivative: N-(4-chlorobenzyl)-2-(1H-imidazol-1-ylmethyl)benzenamine.
Topics: Aniline Compounds; Animals; Antifungal Agents; Candida; Candida albicans; Gram-Negative Bacteria; Imidazoles; Ketoconazole; Male; Miconazole; Microbial Sensitivity Tests; Rabbits | 1990 |
New and prospective developments in antifungal drugs.
Topics: Administration, Oral; Administration, Topical; Allylamine; Antifungal Agents; Clotrimazole; Dermatomycoses; Drug Compounding; Humans; Imidazoles; Itraconazole; Ketoconazole; Miconazole; Naphthalenes; Terbinafine; Triazoles | 1986 |
Effects of bifonazole, fluconazole, itraconazole, and terbinafine on the chemiluminescence response of immune cells.
Topics: Animals; Antifungal Agents; Cell Survival; Centrifugation; Fluconazole; Imidazoles; In Vitro Techniques; Itraconazole; Ketoconazole; Luminescent Measurements; Luminol; Mice; Mice, Inbred BALB C; Naphthalenes; Phagocytes; Rabbits; Rifampin; Spleen; Terbinafine; Triazoles | 1987 |
Antifungal relative inhibition factors: BAY l-9139, bifonazole, butoconazole, isoconazole, itraconazole (R 51211), oxiconazole, Ro 14-4767/002, sulconazole, terconazole and vibunazole (BAY n-7133) compared in vitro with nine established antifungal agents.
Topics: Antifungal Agents; Aspergillus; Candida; Clotrimazole; Econazole; Imidazoles; In Vitro Techniques; Itraconazole; Ketoconazole; Miconazole; Morpholines; Triazoles | 1984 |
[Antimycotic therapy. 2. Antimycotic chemotherapeutic agents: imidazole derivatives, tolciclate, haloprogin, ciclopiroxolamin].
Topics: Antifungal Agents; Chemical Phenomena; Chemistry; Ciclopirox; Clotrimazole; Dermatomycoses; Econazole; Humans; Imidazoles; Ketoconazole; Miconazole; Phenyl Ethers; Piperazines; Pyridones; Thiocarbamates | 1983 |
In-vitro studies with four new antifungal agents: BAY n 7133, bifonazole (BAY h 4502), ICI 153,066 and Ro 14-4767/002.
Topics: Antifungal Agents; Arthrodermataceae; Blastomyces; Candida; Coccidioides; Cryptococcus neoformans; Drug Evaluation, Preclinical; Histoplasma; Imidazoles; Ketoconazole; Miconazole; Morpholines; Sporothrix; Triazoles | 1984 |
Antifungal agents. VI. In vitro antifungal activities of halobenzoyl esters of cis- and trans-[2-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-ylmethyl)-1,3- dioxolan-4-yl]carbinols.
Topics: Antifungal Agents; Biphenyl Compounds; Candida; Candida albicans; Dioxolanes; Imidazoles; Ketoconazole; Microbial Sensitivity Tests; Stereoisomerism | 1993 |
Direct interaction of antifungal azole-derivatives with calmodulin: a possible mechanism for their therapeutic activity.
Topics: Antifungal Agents; Calmodulin; Clotrimazole; Drug Interactions; Econazole; Imidazoles; Ketoconazole; Kinetics; Miconazole; Phosphodiesterase Inhibitors; Polymyxin B | 1993 |
Different effects of azole-antifungal agents on the regulation of intracellular calcium concentration of Trichophyton rubrum.
Topics: Antifungal Agents; Azoles; Calcium; Chelating Agents; Edetic Acid; Humans; Imidazoles; Intracellular Membranes; Itraconazole; Ketoconazole; Osmolar Concentration; Trichophyton | 1996 |
Modeling study of some inhibitors of 17,20-lyase, a component of the enzyme 17 alpha-hydroxylase/17,20-lyase: a novel approach.
Topics: Binding Sites; Enzyme Inhibitors; Imidazoles; Ketoconazole; Models, Molecular; Protein Conformation; Steroid 17-alpha-Hydroxylase; Substrate Specificity | 1998 |
Molecular design of two sterol 14alpha-demethylase homology models and their interactions with the azole antifungals ketoconazole and bifonazole.
Topics: Amino Acid Sequence; Antifungal Agents; Binding Sites; Candida albicans; Computer-Aided Design; Conserved Sequence; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Enzyme Inhibitors; Fungal Proteins; Humans; Imidazoles; Ketoconazole; Models, Molecular; Molecular Sequence Data; Mycobacterium tuberculosis; Oxidoreductases; Protein Conformation; Sequence Alignment; Sequence Homology, Amino Acid; Sterol 14-Demethylase | 2005 |
In vitro antifungal activity of luliconazole against nondermatophytic moulds.
Topics: Amphotericin B; Antifungal Agents; Clotrimazole; Fluconazole; Fungi; Humans; Imidazoles; Itraconazole; Ketoconazole; Miconazole; Microbial Sensitivity Tests; Morpholines; Sequence Analysis, DNA; Terbinafine; Triazoles; Voriconazole | 2020 |
Synthesis, Biological Evaluation and Molecular Docking Studies of 5-Indolylmethylen-4-oxo-2-thioxothiazolidine Derivatives.
Topics: Ampicillin; Anti-Bacterial Agents; Antifungal Agents; Escherichia coli; Fungi; Imidazoles; Ketoconazole; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Microbial Viability; Molecular Docking Simulation; Molecular Structure; Pseudomonas aeruginosa; Structure-Activity Relationship; Thiazolidines | 2022 |
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
5-Adamantan thiadiazole-based thiazolidinones as antimicrobial agents. Design, synthesis, molecular docking and evaluation.
Topics: Adamantane; Anti-Infective Agents; Binding Sites; Drug Design; Drug Resistance, Bacterial; Escherichia coli; Escherichia coli Proteins; Fungal Proteins; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Molecular Docking Simulation; Protein Structure, Tertiary; Structure-Activity Relationship; Thiadiazoles; Thiazolidines | 2018 |
Design, synthesis and antimicrobial activity of usnic acid derivatives.
Topics: | 2018 |
Appendix A. dithioloquinolinethiones as new potential multitargeted antibacterial and antifungal agents: Synthesis, biological evaluation and molecular docking studies.
Topics: Anti-Bacterial Agents; Antifungal Agents; Carbon-13 Magnetic Resonance Spectroscopy; Chromatography, High Pressure Liquid; Drug Design; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Mass Spectrometry; Microbial Sensitivity Tests; Molecular Docking Simulation; Proton Magnetic Resonance Spectroscopy; Quinolines; Structure-Activity Relationship | 2019 |
New vinyl-1,2,4-triazole derivatives as antimicrobial agents: Synthesis, biological evaluation and molecular docking studies.
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Antifungal Agents; Binding Sites; DNA Gyrase; Drug Design; Erwinia amylovora; Escherichia coli; Escherichia coli Proteins; Fungi; Microbial Sensitivity Tests; Molecular Docking Simulation; Nucleoside-Phosphate Kinase; Structure-Activity Relationship; Triazoles; Xanthomonas campestris | 2020 |