Page last updated: 2024-08-23

balsalazide and mesalamine

balsalazide has been researched along with mesalamine in 83 studies

Research

Studies (83)

TimeframeStudies, this research(%)All Research%
pre-19903 (3.61)18.7374
1990's17 (20.48)18.2507
2000's49 (59.04)29.6817
2010's12 (14.46)24.3611
2020's2 (2.41)2.80

Authors

AuthorsStudies
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Giaffer, MH; Holdsworth, CD; O'Brien, CJ1
Baron, JH; Barrison, IG; Giaffer, MH; Hoare, AM; Holdsworth, CD; Lennard-Jones, JE; Manjunatha, S; McIntyre, PB; Polson, RJ; Rodrigues, CA1
Brown, P; Gibson, JA; Green, JR; Kerr, GD; Rowlinson, A; Swan, CH; Swarbrick, ET; Thornton, P1
Baron, JH; Barrison, IG; Lennard-Jones, JE; McIntyre, PB; Rodrigues, CA; Thornton, PC; Walker, JG1
Lennard-Jones, JE; McIntyre, PB1
Baron, JH; Chan, RP; Gilbert, AP; Lennard-Jones, JE; Pope, DJ; Sacra, PJ1
Kataoka, M; Kawasaki, M; Kimura, I; Nagahama, S; Sato, M1
Kataoka, M; Kokuba, Y; Kumamoto, T; Matsuda, A1
Gibson, JA; Green, JR; Hodgson, HJ; Holdsworth, CD; Kerr, GD; Leicester, RJ; Lobo, AJ; Parkins, KJ; Taylor, MD1
Prakash, A; Spencer, CM1
Gross, V1
Kataoka, M; Kimura, I; Kokuba, Y; Kumamoto, T; Matsuda, A1
Kataoka, M; Kawasaki, M; Kimura, I; Kokuba, Y; Matsuda, A; Nagahama, S1
Crowe, JP; Gibson, JA; Green, JR; Holdsworth, CD; Kerr, GD; Lobo, AJ; Schofield, KJ; Swarbrick, ET; Taylor, MD1
Kataoka, M; Kawasaki, M; Kimura, I; Kokurba, Y; Matsuda, A1
Hanauer, SB3
Blake, DR; Millar, AD; Rampton, DS; Simmonds, NJ1
Regueiro, MD1
Lowry, PW; Sandborn, WJ; Szumlanski, CL; Weinshilboum, RM1
Green, JR1
Adhiyaman, V; Froese, S; Vaishnavi, A2
Johnson, LK; Kim, YS; MacGregor, DJ; Sleisenger, MH1
Ragunath, K; Williams, JG1
Franklin, CL; Lipsky, JJ; Loftus, EV; Lowry, PW; Mays, DC; Sandborn, WJ; Szumlanski, CL; Tremaine, WJ; Weaver, AL; Weinshilboum, RM1
Brandes, JW; Ewald, U; Hämling, J; Howaldt, S; Koop, I; Krakamp, B; Kruis, W; Mönnikes, H; Pallant, D; Schreiber, S; Schütz, E; Stolte, M; Theuer, D1
Gibson, JA; Green, JR; Kerr, GD; Mansfield, JC; Thornton, PC1
Cann, PA; Giaffer, MH; Holdsworth, CD; Mansfield, JC; McKenna, D; Thornton, PC1
Farrell, RJ; Peppercorn, MA1
Bell, JK; Johnson, LK; Koval, G; Levine, DS; Pruitt, R; Riff, DS; Sales, D; Wruble, L1
Goa, KL; Muijsers, RB1
Hussar, DA1
Schroeder, KW1
Cross, A; Doty, P; Hanson, J; Hardi, R; Johanson, J; Johnson, LK; Koval, G; Pruitt, R; Riff, D; Safdi, M; Winston, B; Wruble, L1
Green, JR; Johnson, LK; Pruitt, RE1
Cohen, RD1
Cummings, JH; Edmond, LM; Hopkins, MJ; Magee, EA1
Biancone, L; De Nigris, F; Fantini, M; Fina, D; Geremia, A; Pallone, F; Tosti, C1
Bjorkman, DJ; Kane, SV1
Bjorkman, D; Kane, SV; Loftus, EV1
Gibson, JA; Green, JR; Kerr, GD; Swan, CH; Swarbrick, ET; Thornton, PC1
Buch, A; Hanauer, SB; Sandborn, WJ1
Baker, DE; Kane, S1
Brandimarte, G; Forti, G; Gigliobianco, A; Giorgetti, GM; Modeo, ME; Tursi, A1
Chang, EB; Hanauer, SB; Kles, KA; Musch, MW; Turner, JR; Vavricka, SR1
Bettenhausen, D; Jahraus, CD; Rubin, DT; Scherl, EJ1
Bettenhausen, D; Jahraus, CD; Malik, U; Sellitti, M; St Clair, WH1
Baker, DE1
Sandborn, WJ1
Choudhary, C; Cohn, JR; Kung, SJ; McGeady, SJ1
Mackowiak, JI1
Aguirre, A; Brass, C; Margarone, J; Markiewicz, M; Suresh, L1
Aiello, F; Brandimarte, G; Elisei, W; Giorgetti, GM; Tursi, A1
Assem, ES; Pearce, FL; Peh, KH; Wan, BC1
Austin, D; Hogg, KJ; Jamieson, N; Robertson, E1
Abdollahi, M; Nikfar, S; Rahimi, R; Rezaie, A1
Tursi, A2
Moss, AC; Patil, SA1
Hu, J; Liu, XC; Mei, Q; Xu, JM2
Forbes, WP; Gordon, GL; Huang, S; Lamet, M; Mareya, S; Pruitt, R; Scherl, EJ; Shaw, A1
Attard, TM; Bortey, E; Forbes, WP; Heyman, MB; Pieniaszek, HJ; Pohl, JF; Quiros, JA; Walker, K1
Rajapakse, R; Wiggins, JB1
Gum, JR; Hayes, A; Johnson, LK; Kim, YS; McQuaid, KR; Sleisenger, MH; Terdiman, JP; Weinberg, VK1
Abuhammad, A; Laurieri, N; Lowe, E; Ryan, A; Sim, E; Wang, CJ; Westwood, I1
Candlish, W; Gravil, J; McGrane, J; Paravasthu, M1
Laurieri, N; Ryan, A; Sim, E; Wang, CJ; Westwood, I1
Rothenberg, ME; Sonu, I; Wong, R1
Lee, CS; Lee, JJ; Mulberg, AE; Nelson, RM; Papadopoulos, EJ; Rodriguez, WJ; Sachs, HC; Sun, H1
Coman, RM; Gjymishka, A; Glover, SC1
Dhaneshwar, SS1
Byeon, JS; Cho, EA; Chung, EJ; Do, EJ; Hwang, SW; Kim, JH; Kim, SY; Lee, HJ; Myung, SJ; Park, S; Park, SH; Ryu, YM; Yang, DH; Yang, SK; Ye, BD1
Jeong, HJ; Kim, EM; Kim, IH; Kim, SH; Kim, SL; Kim, SW; Kim, YN; Lee, SO; Lee, ST; Liu, YC; Park, YR; Seo, SY1
Kuriyama, A; Matsumura, M; Urushidani, S1
Choi, YS; Kim, DS; Kim, JK; Kim, WJ; Lee, DH1
Bracher, F; Dietschreit, JCB; Ghazy, E; Glas, C; Jung, M; Ochsenfeld, C; Sippl, W; Urban, L; Wössner, N1
Damkier, P; Eisenberg, ML; Kjeldsen, J; Lindahl-Jacobsen, R; Streett, SE; Wensink, MJ1

Reviews

20 review(s) available for balsalazide and mesalamine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Balsalazide.
    Drugs, 1998, Volume: 56, Issue:1

    Topics: Aminosalicylic Acids; Anti-Ulcer Agents; Colitis, Ulcerative; Drug Tolerance; Humans; Mesalamine; Phenylhydrazines

1998
Review article: balsalazide therapy in ulcerative colitis.
    Alimentary pharmacology & therapeutics, 2001, Volume: 15, Issue:10

    Topics: Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Clinical Trials as Topic; Colitis, Ulcerative; Humans; Mesalamine; Phenylhydrazines; Prodrugs

2001
Equimolar doses of balsalazide and mesalamine: are we comparing apples and oranges?
    The American journal of gastroenterology, 2002, Volume: 97, Issue:6

    Topics: Aminosalicylic Acids; Anti-Ulcer Agents; Colitis, Ulcerative; Dose-Response Relationship, Drug; Humans; Mesalamine; Phenylhydrazines

2002
Balsalazide: a review of its therapeutic use in mild-to-moderate ulcerative colitis.
    Drugs, 2002, Volume: 62, Issue:11

    Topics: Aminosalicylic Acids; Anti-Ulcer Agents; Colitis, Ulcerative; Databases, Bibliographic; Female; Humans; Male; Mesalamine; Phenylhydrazines; Randomized Controlled Trials as Topic; Sex Factors; Treatment Outcome

2002
Role of mesalazine in acute and long-term treatment of ulcerative colitis and its complications.
    Scandinavian journal of gastroenterology. Supplement, 2002, Issue:236

    Topics: Acute Disease; Administration, Oral; Administration, Rectal; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Colitis, Ulcerative; Enema; Humans; Mesalamine; Phenylhydrazines; Prodrugs; Sulfasalazine; Time Factors

2002
Review article: maintenance treatment of Crohn's disease.
    Alimentary pharmacology & therapeutics, 2003, Volume: 17 Suppl 2

    Topics: Adrenal Cortex Hormones; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Antibodies, Monoclonal; Crohn Disease; Gastrointestinal Agents; Humans; Immunosuppressive Agents; Mesalamine; Phenylhydrazines; Remission Induction; Secondary Prevention; Sulfasalazine; Tumor Necrosis Factor-alpha

2003
The efficacy of oral 5-ASAs in the treatment of active ulcerative colitis: a systematic review.
    Reviews in gastroenterological disorders, 2003,Fall, Volume: 3, Issue:4

    Topics: Administration, Oral; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Clinical Trials as Topic; Colitis, Ulcerative; Humans; Mesalamine; Phenylhydrazines; Treatment Outcome

2003
Systematic review: short-term adverse effects of 5-aminosalicylic acid agents in the treatment of ulcerative colitis.
    Alimentary pharmacology & therapeutics, 2004, Jan-15, Volume: 19, Issue:2

    Topics: Administration, Oral; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Colitis, Ulcerative; Double-Blind Method; Humans; Mesalamine; Phenylhydrazines; Randomized Controlled Trials as Topic

2004
The short- and long-term safety of 5-aminosalicylate products in the treatment of ulcerative colitis.
    Reviews in gastroenterological disorders, 2004,Spring, Volume: 4, Issue:2

    Topics: Adolescent; Adult; Aminosalicylic Acids; Child; Clinical Trials as Topic; Colitis, Ulcerative; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Labeling; Female; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Product Surveillance, Postmarketing; Sensitivity and Specificity; Sulfasalazine

2004
Safety of balsalazide therapy in the treatment of inflammatory bowel disease.
    Reviews in gastroenterological disorders, 2005,Summer, Volume: 5, Issue:3

    Topics: Aminosalicylic Acids; Anti-Ulcer Agents; Clinical Trials as Topic; Humans; Inflammatory Bowel Diseases; Mesalamine; Phenylhydrazines; Safety

2005
Treatment of ulcerative colitis with oral mesalamine: advances in drug formulation, efficacy expectations and dose response, compliance, and chemoprevention.
    Reviews in gastroenterological disorders, 2006,Spring, Volume: 6, Issue:2

    Topics: Administration, Oral; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Chemistry, Pharmaceutical; Chemoprevention; Clinical Trials as Topic; Colitis, Ulcerative; Delayed-Action Preparations; Dose-Response Relationship, Drug; Humans; Mesalamine; Patient Compliance; Phenylhydrazines; Remission Induction; Sulfasalazine

2006
Comparison of mesalazine and balsalazide in induction and maintenance of remission in patients with ulcerative colitis: a meta-analysis.
    Digestive diseases and sciences, 2009, Volume: 54, Issue:4

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Colitis, Ulcerative; Female; Humans; Male; Mesalamine; Phenylhydrazines; Remission Induction

2009
Balsalazide plus high-potency probiotic preparation (VSL[sharp]3) in the treatment of acute mild-to-moderate ulcerative colitis and uncomplicated diverticulitis of the colon.
    Journal of clinical gastroenterology, 2008, Volume: 42 Suppl 3 Pt 1

    Topics: Clinical Trials as Topic; Colitis, Ulcerative; Diverticulitis, Colonic; Drug Therapy, Combination; Gastrointestinal Agents; Humans; Mesalamine; Phenylhydrazines; Probiotics; Prodrugs; Treatment Outcome

2008
Balsalazide disodium for the treatment of ulcerative colitis.
    Expert review of gastroenterology & hepatology, 2008, Volume: 2, Issue:2

    Topics: Colitis, Ulcerative; Gastrointestinal Agents; Humans; Mesalamine; Phenylhydrazines

2008
Balsalazide in treating colonic diseases.
    Expert opinion on drug metabolism & toxicology, 2009, Volume: 5, Issue:12

    Topics: Colitis, Ulcerative; Colonic Diseases; Gastrointestinal Agents; Humans; Mesalamine; Phenylhydrazines; Prodrugs; Treatment Outcome

2009
Balsalazide: a novel 5-aminosalicylate prodrug for the treatment of active ulcerative colitis.
    Expert opinion on drug metabolism & toxicology, 2009, Volume: 5, Issue:10

    Topics: Clinical Trials as Topic; Colitis, Ulcerative; Delayed-Action Preparations; Gastrointestinal Agents; Humans; Mesalamine; Phenylhydrazines; Prodrugs; Remission Induction

2009
Febrile pleuropericarditis, a potentially life-threatening adverse event of balsalazide--case report and literature review of the side effects of 5-aminosalicylates.
    Expert review of clinical immunology, 2014, Volume: 10, Issue:5

    Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Colitis, Ulcerative; Fever; Humans; Male; Mesalamine; Pericarditis; Phenylhydrazines

2014
Colon-specific prodrugs of 4-aminosalicylic acid for inflammatory bowel disease.
    World journal of gastroenterology, 2014, Apr-07, Volume: 20, Issue:13

    Topics: Aminosalicylic Acid; Aminosalicylic Acids; Clinical Trials as Topic; Colon; Fatty Acids, Omega-3; Heparin, Low-Molecular-Weight; Humans; Inflammatory Bowel Diseases; Mesalamine; Phenylhydrazines; Prodrugs; Sulfasalazine

2014
5-aminosalicylic acid agents for prevention of recurrent diverticulitis: A systematic review and meta-analysis.
    Journal of gastroenterology and hepatology, 2018, Volume: 33, Issue:1

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Aminosalicylic Acids; Anti-Inflammatory Agents; Databases, Bibliographic; Diverticulitis; Female; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Randomized Controlled Trials as Topic; Recurrence; Secondary Prevention; Sulfasalazine; Treatment Outcome; Young Adult

2018

Trials

20 trial(s) available for balsalazide and mesalamine

ArticleYear
Improved maintenance of remission in ulcerative colitis by balsalazide 4 g/day compared with 2 g/day.
    Alimentary pharmacology & therapeutics, 1992, Volume: 6, Issue:4

    Topics: Adult; Aged; Aged, 80 and over; Aminosalicylic Acids; Colitis, Ulcerative; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Sulfasalazine

1992
Short report: comparison of two doses of balsalazide in maintaining ulcerative colitis in remission over 12 months.
    Alimentary pharmacology & therapeutics, 1992, Volume: 6, Issue:5

    Topics: Adult; Aged; Aminosalicylic Acids; Colitis, Ulcerative; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Prospective Studies; Time Factors

1992
Balsalazide in the maintenance treatment of patients with ulcerative colitis, a double-blind comparison with sulphasalazine.
    Alimentary pharmacology & therapeutics, 1988, Volume: 2, Issue:3

    Topics: Adult; Aged; Aminosalicylic Acids; Colitis, Ulcerative; Double-Blind Method; Female; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Sulfasalazine

1988
Studies of two novel sulfasalazine analogs, ipsalazide and balsalazide.
    Digestive diseases and sciences, 1983, Volume: 28, Issue:7

    Topics: Aminosalicylic Acids; Animals; Chemical Phenomena; Chemistry; Clinical Trials as Topic; Colitis, Ulcerative; Feces; Female; Humans; Male; Mesalamine; Mice; Mice, Inbred Strains; Phenylhydrazines; Rats; Rats, Inbred Strains; Time Factors

1983
Balsalazide is more effective and better tolerated than mesalamine in the treatment of acute ulcerative colitis. The Abacus Investigator Group.
    Gastroenterology, 1998, Volume: 114, Issue:1

    Topics: Adult; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Colitis, Ulcerative; Double-Blind Method; Female; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Treatment Outcome

1998
Maintenance of remission of ulcerative colitis: a comparison between balsalazide 3 g daily and mesalazine 1.2 g daily over 12 months. ABACUS Investigator group.
    Alimentary pharmacology & therapeutics, 1998, Volume: 12, Issue:12

    Topics: Adolescent; Adult; Aged; Aminosalicylic Acids; Anti-Ulcer Agents; Colitis, Ulcerative; Delayed-Action Preparations; Double-Blind Method; Female; Headache; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Secondary Prevention; Time Factors; Treatment Failure

1998
Balsalazide led to greater remission rates and tolerance than mesalamine in acute ulcerative colitis.
    Gut, 1999, Volume: 44, Issue:4

    Topics: Acute Disease; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Colitis, Ulcerative; Female; Humans; Male; Mesalamine; Phenylhydrazines; Randomized Controlled Trials as Topic

1999
Low dose balsalazide (1.5 g twice daily) and mesalazine (0.5 g three times daily) maintained remission of ulcerative colitis but high dose balsalazide (3.0 g twice daily) was superior in preventing relapses.
    Gut, 2001, Volume: 49, Issue:6

    Topics: Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Colitis, Ulcerative; Colon; Double-Blind Method; Drug Administration Schedule; Female; Humans; Male; Mesalamine; Phenylhydrazines; Prodrugs

2001
A double-blind comparison of balsalazide, 6.75 g daily, and sulfasalazine, 3 g daily, in patients with newly diagnosed or relapsed active ulcerative colitis.
    Alimentary pharmacology & therapeutics, 2002, Volume: 16, Issue:1

    Topics: Administration, Oral; Adrenal Cortex Hormones; Adult; Aged; Aminosalicylic Acids; Anti-Ulcer Agents; Colitis, Ulcerative; Double-Blind Method; Female; Gastrointestinal Agents; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Severity of Illness Index; Sigmoidoscopy; Sulfasalazine; Treatment Outcome

2002
A double-blind comparison of balsalazide, 6.75 g, and sulfasalazine, 3 g, as sole therapy in the management of ulcerative colitis.
    Alimentary pharmacology & therapeutics, 2002, Volume: 16, Issue:1

    Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Aminosalicylic Acids; Anti-Ulcer Agents; Colitis, Ulcerative; Double-Blind Method; Female; Gastrointestinal Agents; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Severity of Illness Index; Sigmoidoscopy; Sulfasalazine; Treatment Outcome

2002
A randomized, double blind, dose-response comparison of balsalazide (6.75 g), balsalazide (2.25 g), and mesalamine (2.4 g) in the treatment of active, mild-to-moderate ulcerative colitis.
    The American journal of gastroenterology, 2002, Volume: 97, Issue:6

    Topics: Adult; Aged; Aged, 80 and over; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Colitis, Ulcerative; Dose-Response Relationship, Drug; Double-Blind Method; Female; Homeostasis; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Safety; Severity of Illness Index

2002
Balsalazide is superior to mesalamine in the time to improvement of signs and symptoms of acute mild-to-moderate ulcerative colitis.
    The American journal of gastroenterology, 2002, Volume: 97, Issue:12

    Topics: Acute Disease; Adolescent; Adult; Aged; Aged, 80 and over; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Child; Colitis, Ulcerative; Double-Blind Method; Humans; Mesalamine; Middle Aged; Phenylhydrazines; Safety; Treatment Outcome

2002
Patient-led variable dosing with balsalazide as long-term therapy for maintenance in ulcerative colitis: a 3-year prospective observational study.
    Alimentary pharmacology & therapeutics, 2004, Feb-15, Volume: 19, Issue:4

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Aminosalicylic Acids; Cohort Studies; Colitis, Ulcerative; Female; Humans; Male; Mesalamine; Middle Aged; Patient Participation; Phenylhydrazines; Prognosis; Prospective Studies; Recurrence; Treatment Outcome

2004
Comparative pharmacokinetics of equimolar doses of 5-aminosalicylate administered as oral mesalamine (Asacol) and balsalazide: a randomized, single-dose, crossover study in healthy volunteers.
    Alimentary pharmacology & therapeutics, 2004, May-15, Volume: 19, Issue:10

    Topics: Administration, Oral; Adult; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Cross-Over Studies; Female; Humans; Male; Mesalamine; Phenylhydrazines

2004
Low-dose balsalazide plus a high-potency probiotic preparation is more effective than balsalazide alone or mesalazine in the treatment of acute mild-to-moderate ulcerative colitis.
    Medical science monitor : international medical journal of experimental and clinical research, 2004, Volume: 10, Issue:11

    Topics: Adult; Aged; Aminosalicylic Acids; Colitis, Ulcerative; Drug Therapy, Combination; Female; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Probiotics

2004
Prevention of acute radiation-induced proctosigmoiditis by balsalazide: a randomized, double-blind, placebo controlled trial in prostate cancer patients.
    International journal of radiation oncology, biology, physics, 2005, Dec-01, Volume: 63, Issue:5

    Topics: Acute Disease; Aged; Aminosalicylic Acids; Anti-Ulcer Agents; Colon, Sigmoid; Double-Blind Method; Humans; Male; Mesalamine; Phenylhydrazines; Pilot Projects; Proctocolitis; Prostatic Neoplasms; Radiation Injuries; Rectum

2005
Balsalazide and/or high-potency probiotic mixture (VSL#3) in maintaining remission after attack of acute, uncomplicated diverticulitis of the colon.
    International journal of colorectal disease, 2007, Volume: 22, Issue:9

    Topics: Acute Disease; Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Bifidobacterium; Diverticulitis, Colonic; Drug Therapy, Combination; Female; Follow-Up Studies; Gastrointestinal Agents; Humans; Lacticaseibacillus casei; Male; Mesalamine; Middle Aged; Phenylhydrazines; Pilot Projects; Probiotics; Recurrence; Treatment Outcome

2007
Safety and efficacy of a new 3.3 g b.i.d. tablet formulation in patients with mild-to-moderately-active ulcerative colitis: a multicenter, randomized, double-blind, placebo-controlled study.
    The American journal of gastroenterology, 2009, Volume: 104, Issue:6

    Topics: Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Colitis, Ulcerative; Disease Progression; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Follow-Up Studies; Gastrointestinal Hemorrhage; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Prospective Studies; Rectum; Severity of Illness Index; Sigmoidoscopy; Tablets; Treatment Outcome

2009
Safety, efficacy, and pharmacokinetics of balsalazide in pediatric patients with mild-to-moderate active ulcerative colitis: results of a randomized, double-blind study.
    Journal of pediatric gastroenterology and nutrition, 2009, Volume: 49, Issue:5

    Topics: Adolescent; Aminosalicylic Acids; Anti-Inflammatory Agents; Child; Colitis, Ulcerative; Colon; Double-Blind Method; Female; Humans; Male; Mesalamine; Phenylhydrazines

2009
Chemoprevention of colonic polyps with balsalazide: an exploratory, double-blind, placebo-controlled study.
    Digestive diseases and sciences, 2009, Volume: 54, Issue:11

    Topics: Adenoma; Aged; Apoptosis; Colon, Sigmoid; Colonic Neoplasms; Colonic Polyps; Double-Blind Method; Gastrointestinal Agents; Humans; Male; Mesalamine; Middle Aged; Phenylhydrazines; Prospective Studies

2009

Other Studies

43 other study(ies) available for balsalazide and mesalamine

ArticleYear
Clinical tolerance to three 5-aminosalicylic acid releasing preparations in patients with inflammatory bowel disease intolerant or allergic to sulphasalazine.
    Alimentary pharmacology & therapeutics, 1992, Volume: 6, Issue:1

    Topics: Aminosalicylic Acids; Drug Hypersensitivity; Female; Humans; Inflammatory Bowel Diseases; Male; Mesalamine; Phenylhydrazines; Sulfapyridine; Sulfasalazine

1992
Reversal with balsalazide of infertility caused by sulphsalazine.
    British medical journal (Clinical research ed.), 1984, Jun-02, Volume: 288, Issue:6431

    Topics: Adult; Aminosalicylic Acids; Colitis, Ulcerative; Humans; Infertility, Male; Male; Mesalamine; Phenylhydrazines; Sperm Count; Sulfasalazine

1984
[Pharmacological studies of BX661A. 5-[4-(2-carboxyethylcarbamoyl)-phenylazo]-salicylic acid disodium salt dihydrate (1). Therapeutic effects on dextran sulfate sodium (DSS)-induced ulcerative colitis (UC) model in rats].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1997, Volume: 109, Issue:2

    Topics: Administration, Oral; Aminosalicylic Acids; Animals; Anthracenes; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Colitis, Ulcerative; Dextran Sulfate; Male; Mesalamine; Phenylhydrazines; Rats; Rats, Sprague-Dawley; Sulfapyridine; Sulfasalazine

1997
Inhibition by aminosalicylates of lipid peroxidation in large intestinal mucosa after mesenteric ischemia/reperfusion in the rat.
    Japanese journal of pharmacology, 1997, Volume: 75, Issue:2

    Topics: Aminosalicylic Acids; Animals; Anti-Inflammatory Agents, Non-Steroidal; Intestinal Mucosa; Intestine, Large; Lipid Peroxidation; Male; Mesalamine; Phenylhydrazines; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Splanchnic Circulation

1997
Efficacy of different mesalamine-releasing drugs.
    Gastroenterology, 1998, Volume: 115, Issue:5

    Topics: Acute Disease; Aminosalicylic Acids; Anti-Ulcer Agents; Clinical Trials as Topic; Colitis, Ulcerative; Humans; Mesalamine; Phenylhydrazines; Research Design

1998
Effects of BX661A, a new therapeutic agent for ulcerative colitis, on reactive oxygen species in comparison with salazosulfapyridine and its metabolite sulfapyridine.
    Arzneimittel-Forschung, 1998, Volume: 48, Issue:10

    Topics: Aminosalicylic Acids; Anti-Ulcer Agents; Colitis, Ulcerative; Cytochrome c Group; Hydrogen Peroxide; Hypochlorous Acid; Kinetics; Mesalamine; Phenylhydrazines; Reactive Oxygen Species; Sulfapyridine; Sulfasalazine; Superoxides

1998
Determination of the active moiety of BX661A, a new therapeutic agent for ulcerative colitis, by studying its therapeutic effects on ulcerative colitis induced by dextran sulfate sodium in rats.
    Arzneimittel-Forschung, 1998, Volume: 48, Issue:11

    Topics: Alanine; Aminosalicylic Acids; Animals; Anti-Ulcer Agents; Colitis, Ulcerative; Colon; Dextran Sulfate; Drug Interactions; Male; Mesalamine; Phenylhydrazines; Rats; Rats, Sprague-Dawley; Sulfapyridine; Sulfasalazine

1998
Effects of BX661A, a new therapeutic agent for ulcerative colitis, on chemotaxis and reactive oxygen species production in polymorphonuclear leukocytes in comparison with salazosulfapyridine and its metabolite sulfapyridine.
    Arzneimittel-Forschung, 1998, Volume: 48, Issue:12

    Topics: Aminosalicylic Acids; Animals; Anti-Ulcer Agents; Chemotaxis, Leukocyte; Colitis, Ulcerative; Guinea Pigs; Humans; In Vitro Techniques; Male; Mesalamine; Neutrophils; Phenylhydrazines; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Sulfapyridine; Sulfasalazine

1998
Antioxidant effects of aminosalicylates and potential new drugs for inflammatory bowel disease: assessment in cell-free systems and inflamed human colorectal biopsies.
    Alimentary pharmacology & therapeutics, 1999, Volume: 13, Issue:3

    Topics: Adrenal Cortex Hormones; Adult; Aged; Aminosalicylic Acid; Aminosalicylic Acids; Anti-Infective Agents; Anti-Inflammatory Agents; Anti-Ulcer Agents; Antioxidants; Cell-Free System; Colitis; Female; Humans; In Vitro Techniques; Inflammatory Bowel Diseases; Luminescent Measurements; Male; Mesalamine; Metronidazole; Middle Aged; Phenylhydrazines; Proctitis; Steroids

1999
Will the real 5-aminosalicylic acid please stand up?
    Inflammatory bowel diseases, 1999, Volume: 5, Issue:2

    Topics: Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Colitis, Ulcerative; Humans; Mesalamine; Phenylhydrazines

1999
Balsalazide and azathiprine or 6-mercaptopurine: evidence for a potentially serious drug interaction.
    Gastroenterology, 1999, Volume: 116, Issue:6

    Topics: Aminosalicylic Acids; Anti-Ulcer Agents; Antirheumatic Agents; Azathioprine; Drug Interactions; Drug Therapy, Combination; Humans; Inflammatory Bowel Diseases; Mercaptopurine; Mesalamine; Phenylhydrazines

1999
Balsalazide and azathioprine or 6-mercaptopurine.
    Gastroenterology, 1999, Volume: 117, Issue:6

    Topics: Administration, Oral; Aminosalicylic Acids; Antimetabolites; Azathioprine; Drug Interactions; Humans; Inhibitory Concentration 50; Mercaptopurine; Mesalamine; Methyltransferases; Phenylhydrazines; Prodrugs

1999
Hypersensitivity reaction to balsalazide.
    BMJ (Clinical research ed.), 2000, Mar-04, Volume: 320, Issue:7235

    Topics: Aminosalicylic Acids; Anti-Ulcer Agents; Drug Hypersensitivity; Female; Humans; Mesalamine; Middle Aged; Phenylhydrazines

2000
Chemoprevention of colon cancer carcinogenesis by balsalazide: inhibition of azoxymethane-induced aberrant crypt formation in the rat colon and intestinal tumor formation in the B6-Min/+ mouse.
    International journal of oncology, 2000, Volume: 17, Issue:1

    Topics: Aminosalicylic Acids; Animals; Anti-Ulcer Agents; Anticarcinogenic Agents; Azoxymethane; Cell Division; Colonic Neoplasms; Genes, APC; Humans; Indomethacin; Intestinal Mucosa; Intestinal Neoplasms; Mesalamine; Mice; Mice, Mutant Strains; Phenylhydrazines; Prodrugs; Rats; Rats, Inbred F344; Tumor Cells, Cultured

2000
Oral balsalazide (Colazal) for ulcerative colitis.
    The Medical letter on drugs and therapeutics, 2001, Jul-23, Volume: 43, Issue:1109

    Topics: Abdominal Pain; Administration, Oral; Aminosalicylic Acids; Anti-Ulcer Agents; Colitis, Ulcerative; Diarrhea; Dose-Response Relationship, Drug; Double-Blind Method; Drug Hypersensitivity; Drug Interactions; Mesalamine; Nausea; Phenylhydrazines; Randomized Controlled Trials as Topic

2001
Drug points: Hypersensitivity reaction to balsalazide.
    BMJ (Clinical research ed.), 2001, Sep-01, Volume: 323, Issue:7311

    Topics: Aminosalicylic Acids; Anti-Ulcer Agents; Drug Hypersensitivity; Female; Humans; Mesalamine; Middle Aged; Pericarditis; Phenylhydrazines

2001
Leucopenia resulting from a drug interaction between azathioprine or 6-mercaptopurine and mesalamine, sulphasalazine, or balsalazide.
    Gut, 2001, Volume: 49, Issue:5

    Topics: Adult; Aminosalicylic Acids; Analysis of Variance; Anti-Inflammatory Agents, Non-Steroidal; Azathioprine; Binomial Distribution; Chromatography, High Pressure Liquid; Confidence Intervals; Drug Interactions; Female; Humans; Immunosuppressive Agents; Leukopenia; Male; Mercaptopurine; Mesalamine; Methyltransferases; Phenylhydrazines; Sulfasalazine; Thioguanine

2001
Balsalazide disodium.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2002, Jan-01, Volume: 59, Issue:1

    Topics: Aminosalicylic Acids; Anti-Ulcer Agents; Colitis, Ulcerative; Drug Interactions; Female; Humans; Male; Mesalamine; Phenylhydrazines; Pregnancy

2002
New drugs 2002, part 1.
    Nursing, 2002, Volume: 32, Issue:1

    Topics: Amides; Aminosalicylic Acids; Anti-Ulcer Agents; Antipsychotic Agents; Bimatoprost; Cloprostenol; Cyclohexanes; Drug Approval; Drug Therapy; Drug-Related Side Effects and Adverse Reactions; Galantamine; Glaucoma; Gonadotropin-Releasing Hormone; Humans; Hypoglycemic Agents; Insulin; Insulin Glargine; Insulin, Long-Acting; Lipids; Mesalamine; Nateglinide; Nootropic Agents; Phenylalanine; Phenylhydrazines; Piperazines; Thiazoles; Travoprost

2002
Caution in the interpretation of safety and efficacy differences in clinical trials comparing aminosalicylates for ulcerative colitis.
    The American journal of gastroenterology, 2003, Volume: 98, Issue:1

    Topics: Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Clinical Trials as Topic; Colitis, Ulcerative; Data Interpretation, Statistical; Humans; Mesalamine; Phenylhydrazines

2003
Treatment of ulcerative colitis with balsalazide: response to editorial by Drs. Farrell and Peppercorn and letter to the editor by Dr. Hanauer.
    The American journal of gastroenterology, 2003, Volume: 98, Issue:1

    Topics: Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Colitis, Ulcerative; Humans; Mesalamine; Phenylhydrazines

2003
The mesalamine wars heat up-enter balsalazide.
    Gastroenterology, 2003, Volume: 124, Issue:2

    Topics: Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Colitis, Ulcerative; Dose-Response Relationship, Drug; Humans; Mesalamine; Phenylhydrazines; Randomized Controlled Trials as Topic

2003
Treatment of ulcerative colitis with balsalazide: response to Drs Johnson, Green, and Pruitt.
    The American journal of gastroenterology, 2003, Volume: 98, Issue:3

    Topics: Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Colitis, Ulcerative; Humans; Mesalamine; Phenylhydrazines; United Kingdom; United States

2003
The effect of 5-aminosalicylic acid-containing drugs on sulfide production by sulfate-reducing and amino acid-fermenting bacteria.
    Inflammatory bowel diseases, 2003, Volume: 9, Issue:1

    Topics: Amino Acids; Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Desulfovibrio; Feces; Fermentation; Fusobacterium; Humans; In Vitro Techniques; Inflammatory Bowel Diseases; Mesalamine; Phenylhydrazines; Sulfasalazine; Sulfides

2003
Comparative analysis of the in vitro prosecretory effects of balsalazide, sulfasalazine, olsalazine, and mesalamine in rabbit distal ileum.
    Inflammatory bowel diseases, 2005, Volume: 11, Issue:3

    Topics: Aminosalicylic Acids; Animals; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Colitis, Ulcerative; Diarrhea; Disease Models, Animal; Gastrointestinal Agents; Ileum; Mesalamine; Phenylhydrazines; Prodrugs; Rabbits; Random Allocation; Sulfasalazine; Tissue Culture Techniques

2005
Inflammation's role in rectal cancer following prostate radiotherapy, and emerging evidence for a protective role for balsalazide.
    Gastroenterology, 2005, Volume: 129, Issue:2

    Topics: Aminosalicylic Acids; Dose-Response Relationship, Drug; Drug Administration Schedule; Humans; Male; Mesalamine; Neoplasms, Radiation-Induced; Phenylhydrazines; Primary Prevention; Prognosis; Prostatic Neoplasms; Radiation Injuries; Rectal Neoplasms; Risk Assessment; Treatment Outcome

2005
Lack of cross-reactivity between 5-aminosalicylic acid-based drugs: a case report and review of the literature.
    Annals of allergy, asthma & immunology : official publication of the American College of Allergy, Asthma, & Immunology, 2006, Volume: 97, Issue:3

    Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Crohn Disease; Cross Reactions; Drug Hypersensitivity; Exanthema; Herpes Simplex; Humans; Immunosuppressive Agents; Male; Mercaptopurine; Mesalamine; Phenylhydrazines; Prednisone

2006
A two-stage decision analysis to assess the cost of 5-aminosalicylic acid failure and the economics of balsalazide versus mesalamine in the treatment of ulcerative colitis.
    Managed care interface, 2006, Volume: 19, Issue:10

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Colitis, Ulcerative; Decision Support Techniques; Humans; Mesalamine; Phenylhydrazines; Treatment Failure; United States

2006
Pyostomatitis vegetans: A clinical marker of silent ulcerative colitis.
    Journal of oral and maxillofacial surgery : official journal of the American Association of Oral and Maxillofacial Surgeons, 2007, Volume: 65, Issue:2

    Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Colitis, Ulcerative; Diagnosis, Differential; Gastrointestinal Agents; Humans; Male; Mesalamine; Phenylhydrazines; Stomatitis

2007
Effect of sulphasalazine and balsalazide on histamine release from mast cells.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2007, Volume: 56 Suppl 1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cell Line; Gastrointestinal Agents; Histamine Release; Humans; Hydrogen Peroxide; Inflammatory Bowel Diseases; Mast Cells; Mesalamine; Oxidants; Phenylhydrazines; Rats; Sulfasalazine

2007
Balsalazide-induced myocarditis.
    International journal of cardiology, 2008, Nov-28, Volume: 130, Issue:3

    Topics: Adult; Colitis, Ulcerative; Gastrointestinal Agents; Humans; Male; Mesalamine; Myocarditis; Phenylhydrazines

2008
[Effect of balsalazide on intestinal mucosal permeability of dextran sulfate sodium-induced colitis in mice].
    Zhonghua wei chang wai ke za zhi = Chinese journal of gastrointestinal surgery, 2009, Volume: 12, Issue:2

    Topics: Animals; Colitis; Dextran Sulfate; Female; Intestinal Mucosa; Male; Mesalamine; Mice; Mice, Inbred C57BL; Permeability; Phenylhydrazines

2009
Balsalazine decreases intestinal mucosal permeability of dextran sulfate sodium-induced colitis in mice.
    Acta pharmacologica Sinica, 2009, Volume: 30, Issue:7

    Topics: Animals; Colitis; Dextran Sulfate; Gastrointestinal Agents; Glutathione Peroxidase; Interferon-gamma; Intestinal Absorption; Intestinal Mucosa; Malondialdehyde; Mesalamine; Mice; Mice, Inbred C57BL; Peroxidase; Phenylhydrazines; Superoxide Dismutase; Tumor Necrosis Factor-alpha

2009
Role of tyrosine 131 in the active site of paAzoR1, an azoreductase with specificity for the inflammatory bowel disease prodrug balsalazide.
    Acta crystallographica. Section F, Structural biology and crystallization communications, 2010, Jan-01, Volume: 66, Issue:Pt 1

    Topics: Azo Compounds; Catalysis; Catalytic Domain; Crystallography, X-Ray; Enzyme Stability; Hot Temperature; Kinetics; Mesalamine; Mutagenesis, Site-Directed; NAD; NADH, NADPH Oxidoreductases; Nitroreductases; Phenylhydrazines; Protein Folding; Pseudomonas aeruginosa; Tyrosine

2010
Unilateral balsalazide-induced eosinophilic pneumonia in an ulcerative colitis patient.
    The journal of the Royal College of Physicians of Edinburgh, 2010, Volume: 40, Issue:3

    Topics: Adult; Biopsy; Colitis, Ulcerative; Female; Gastrointestinal Agents; Humans; Mesalamine; Phenylhydrazines; Pulmonary Eosinophilia; Radiography, Thoracic; Tomography, X-Ray Computed

2010
Reaction mechanism of azoreductases suggests convergent evolution with quinone oxidoreductases.
    Protein & cell, 2010, Volume: 1, Issue:8

    Topics: Benzoquinones; Catalytic Domain; Enzyme Stability; Evolution, Molecular; Flavins; Hot Temperature; Kinetics; Mesalamine; NAD; NADH, NADPH Oxidoreductases; NADP; Nitroreductases; Osmolar Concentration; Oxidation-Reduction; Phenylhydrazines; Phylogeny; Protein Binding; Pseudomonas aeruginosa; Spectrophotometry, Ultraviolet

2010
5-ASA induced recurrent myopericarditis and cardiac tamponade in a patient with ulcerative colitis.
    Digestive diseases and sciences, 2013, Volume: 58, Issue:8

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Cardiac Tamponade; Colitis, Ulcerative; Female; Humans; Mesalamine; Pericarditis; Phenylhydrazines; Sulfasalazine; Young Adult

2013
Alternate endpoints and clinical outcome assessments in pediatric ulcerative colitis registration trials.
    Journal of pediatric gastroenterology and nutrition, 2014, Volume: 58, Issue:1

    Topics: Antibodies, Monoclonal; Colitis, Ulcerative; Humans; Infliximab; Mesalamine; Outcome Assessment, Health Care; Phenylhydrazines

2014
Suppression of colitis-associated carcinogenesis through modulation of IL-6/STAT3 pathway by balsalazide and VSL#3.
    Journal of gastroenterology and hepatology, 2016, Volume: 31, Issue:8

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Anticarcinogenic Agents; Azoxymethane; bcl-2-Associated X Protein; Cell Transformation, Neoplastic; Colitis; Colon; Colorectal Neoplasms; Dextran Sulfate; Disease Models, Animal; Gastrointestinal Agents; Inflammation Mediators; Interleukin-6; Macrophages; Male; Mesalamine; Mice, Inbred C57BL; Phenylhydrazines; Phosphorylation; Probiotics; Proto-Oncogene Proteins c-bcl-2; Signal Transduction; STAT3 Transcription Factor; Time Factors

2016
Combined Parthenolide and Balsalazide Have Enhanced Antitumor Efficacy Through Blockade of NF-κB Activation.
    Molecular cancer research : MCR, 2017, Volume: 15, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Carcinogenesis; Cell Proliferation; Colitis; Colorectal Neoplasms; Drug Synergism; Female; Humans; Mesalamine; Mice; Mice, Inbred BALB C; NF-kappa B; Phenylhydrazines; Sesquiterpenes; Signal Transduction

2017
Efficacy of topical 5-aminosalicylate monotherapy in patients with ulcerative proctitis with skip inflammation.
    Journal of gastroenterology and hepatology, 2018, Volume: 33, Issue:6

    Topics: Administration, Ophthalmic; Administration, Topical; Adolescent; Adult; Aged; Aged, 80 and over; Anti-Inflammatory Agents, Non-Steroidal; Dermatitis; Disease Progression; Drug Therapy, Combination; Female; Follow-Up Studies; Humans; Maintenance Chemotherapy; Male; Mesalamine; Middle Aged; Phenylhydrazines; Proctocolitis; Remission Induction; Treatment Outcome; Young Adult

2018
Identification of the subtype-selective Sirt5 inhibitor balsalazide through systematic SAR analysis and rationalization via theoretical investigations.
    European journal of medicinal chemistry, 2020, Nov-15, Volume: 206

    Topics: Drug Design; Histone Deacetylase Inhibitors; Mesalamine; Molecular Docking Simulation; Phenylhydrazines; Protein Conformation; Salicylic Acid; Sirtuins; Structure-Activity Relationship

2020
Balsalazide Exposure During the Development of Fertilizing Sperm May Be Associated With Offspring Birth Defects.
    Inflammatory bowel diseases, 2022, 10-03, Volume: 28, Issue:10

    Topics: Congenital Abnormalities; Humans; Male; Mesalamine; Phenylhydrazines; Semen; Spermatozoa

2022