baclofen and verapamil

baclofen has been researched along with verapamil in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19902 (13.33)18.7374
1990's4 (26.67)18.2507
2000's5 (33.33)29.6817
2010's4 (26.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Antonsson, M; Bengtsson, O; Bredberg, U; Fridén, M; Hammarlund-Udenaes, M; Jerndal, G; Wan, H; Winiwarter, S1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Ahlin, G; Bergström, F; Bredberg, U; Fridén, M; Hammarlund-Udenaes, M; Rehngren, M; Wan, H1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Bourdelais, AJ; Kalivas, PW1
Carignani, C; Marchetti, C; Robello, M1
Entrikin, RK; Patterson, GT; Wilson, BW1
Benitez, JG; Brunswick, JE; Hodgman, M; Martin, TG; Roberge, RJ1
Acs, Z; Horváth, G; Makara, GB; Mergl, Z; Nagy, I1
Gadoth, N; Hering-Hanit, R1
Ban, JY; Lee, BY; Seong, YH1

Reviews

1 review(s) available for baclofen and verapamil

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

1 trial(s) available for baclofen and verapamil

ArticleYear
The use of baclofen in cluster headache.
    Current pain and headache reports, 2001, Volume: 5, Issue:1

    Topics: Adrenal Cortex Hormones; Adult; Aged; Autonomic Nervous System; Baclofen; Cluster Headache; Drug Administration Schedule; Humans; Male; Middle Aged; Pilot Projects; Treatment Outcome; Verapamil

2001

Other Studies

13 other study(ies) available for baclofen and verapamil

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Structure-brain exposure relationships in rat and human using a novel data set of unbound drug concentrations in brain interstitial and cerebrospinal fluids.
    Journal of medicinal chemistry, 2009, Oct-22, Volume: 52, Issue:20

    Topics: Animals; Blood-Brain Barrier; Brain; Extracellular Fluid; Humans; Linear Models; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Rats; Rats, Sprague-Dawley

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Measurement of unbound drug exposure in brain: modeling of pH partitioning explains diverging results between the brain slice and brain homogenate methods.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:3

    Topics: Animals; Biological Transport; Brain; Chemical Phenomena; Dialysis; Hydrogen-Ion Concentration; In Vitro Techniques; Lysosomes; Male; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Tissue Distribution

2011
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Modulation of extracellular gamma-aminobutyric acid in the ventral pallidum using in vivo microdialysis.
    Journal of neurochemistry, 1992, Volume: 58, Issue:6

    Topics: Animals; Baclofen; Calcium Channels; Dialysis; Dose-Response Relationship, Drug; Extracellular Space; gamma-Aminobutyric Acid; Globus Pallidus; Magnesium Chloride; Male; Muscimol; Neurons; Potassium; Rats; Rats, Inbred Strains; Sodium Channels; Tetrodotoxin; Verapamil; Veratridine

1992
Voltage-dependent calcium currents in dissociated granule cells from rat cerebellum.
    Neuroscience, 1991, Volume: 43, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Baclofen; Bicuculline; Calcium Channels; Cerebellum; Electrophysiology; gamma-Aminobutyric Acid; Membrane Potentials; Rats; Rats, Inbred Strains; Verapamil

1991
Baclofen, procainamide, verapamil, and prenylamine in hereditary muscular dystrophy of the chicken.
    Experimental neurology, 1981, Volume: 74, Issue:1

    Topics: Acetylcholinesterase; Animals; Baclofen; Chickens; Creatine Kinase; Male; Muscles; Muscular Dystrophy, Animal; Prenylamine; Procainamide; Thorax; Verapamil

1981
Supraventricular tachyarrhythmia associated with baclofen overdose.
    Journal of toxicology. Clinical toxicology, 1994, Volume: 32, Issue:3

    Topics: Adenosine; Adult; Baclofen; Drug Overdose; Electrocardiography; Humans; Intubation, Intratracheal; Male; Suicide, Attempted; Tachycardia, Supraventricular; Verapamil

1994
gamma-Aminobutyric acid-induced elevation of intracellular calcium concentration in pituitary cells of neonatal rats.
    Neuroendocrinology, 1993, Volume: 57, Issue:6

    Topics: Animals; Animals, Newborn; Baclofen; Calcium; Female; Fura-2; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Nifedipine; Picrotoxin; Pituitary Gland; Potassium Chloride; Rats; Rats, Wistar; Receptors, GABA-A; Verapamil

1993
Chronic stimulation of GABAA receptor with muscimol reduces amyloid beta protein (25-35)-induced neurotoxicity in cultured rat cortical cells.
    Neuroscience research, 2005, Volume: 52, Issue:4

    Topics: Amyloid beta-Peptides; Analysis of Variance; Animals; Baclofen; Blotting, Western; Calcium; Calcium Channel Blockers; Caspase 3; Caspases; Cell Death; Cell Survival; Cells, Cultured; Cerebral Cortex; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Enzyme Inhibitors; Female; GABA Agonists; Glutamic Acid; Muscimol; Neurons; Neuroprotective Agents; NG-Nitroarginine Methyl Ester; Peptide Fragments; Pregnancy; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, GABA-A; Tetrazolium Salts; Thiazoles; Time Factors; Verapamil

2005