baclofen and piperidines

baclofen has been researched along with piperidines in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19903 (11.54)18.7374
1990's8 (30.77)18.2507
2000's7 (26.92)29.6817
2010's7 (26.92)24.3611
2020's1 (3.85)2.80

Authors

AuthorsStudies
Waldmeier, PC1
Gerlach, J1
Desideri, N; Galli, A; Sestili, I; Stein, ML1
Bardgett, ME; Gray, BC; Miller, JW1
Ferrendelli, JA; Miller, JW1
Curtis, DR; Gynther, BD; Malik, R1
Ottervanger, JP; Schutter, N; Verhaar, HJ1
Bizec, JL; Cabane, J; Derenne, JP; Guelaud, C; Similowski, T; Whitelaw, WA1
Chen, Y; Matsuki, N; Saito, H1
Itoh, Y; Kimura, K; Oka, M; Shimidzu, T; Ukai, Y; Yoshikuni, Y1
Bousquet, P; Feldman, J; Lienhard, JP; Monassier, L; Riehl, V; Tibiriça, E1
Bousquet, P; Brandt, CM; Monassier, L1
Adriaensen, H; Colpaert, FC; Deseure, K; Koek, W1
Gallate, JE; McGregor, IS1
Khodayar, MJ; Naderi, N; Shafaghi, B; Zarindast, MR1
Argiolas, A; Mascia, MS; Melis, MR; Melis, T; Sanna, F; Succu, S1
Bongianni, F; Cinelli, E; Fontana, GA; Mutolo, D; Pantaleo, T1
Hasanein, P; Keshavarz, S; Moghaddam, AH; Rezvani, ME; Roohbakhsh, A1
Bernardi, G; Castelli, M; Cavasinni, F; Centonze, D; De Chiara, V; Errico, F; Mataluni, G; Musella, A; Rossi, S; Sacchetti, L; Siracusano, A; Usiello, A1
Bongianni, F; Cinelli, E; Mutolo, D; Pantaleo, T1
Au, J; Berry-Kravis, E; Hagerman, R; Lauterborn, J1
Bidlack, JM; Dean, RL; Deaver, DR; Eyerman, D; Todtenkopf, MS; Turncliff, RZ1
Niere, F; Raab-Graham, KF; Workman, ER1
Cui, CL; Ge, FF; Li, YJ; Ping, XJ; Qi, C; Shen, F; Sun, LL; Sun, XW; Xing, GG1
Ganji, A; Komaki, A; Komaki, H; Nazari, M; Salehi, I; Sarihi, A; Shahidi, S1
Axelsson, SFA; Horiguchi, N; Horst, NK; Robbins, TW; Roberts, AC1

Reviews

1 review(s) available for baclofen and piperidines

ArticleYear
Fragile X syndrome and targeted treatment trials.
    Results and problems in cell differentiation, 2012, Volume: 54

    Topics: Animals; Anti-Bacterial Agents; Antioxidants; Baclofen; Brain-Derived Neurotrophic Factor; Central Nervous System Stimulants; Clinical Trials as Topic; Dendritic Spines; Donepezil; Dopamine; Enzyme Inhibitors; Fragile X Mental Retardation Protein; Fragile X Syndrome; Humans; Indans; Lithium Compounds; Melatonin; Mice; Mice, Knockout; Minocycline; Nootropic Agents; Piperidines; Receptor, Metabotropic Glutamate 5; Receptors, GABA; Receptors, Metabotropic Glutamate; Signal Transduction; Vitamin E

2012

Trials

1 trial(s) available for baclofen and piperidines

ArticleYear
Effects of centrally-acting glutamatergic modulators on cardiovascular responses to stress in humans.
    Journal of cardiology, 2001, Volume: 37 Suppl 1

    Topics: Administration, Oral; Adult; Baclofen; Cold Temperature; Double-Blind Method; Excitatory Amino Acid Antagonists; Exercise Test; GABA Agonists; Heart Rate; Hemodynamics; Humans; Intelligence Tests; Piperidines; Stress, Physiological

2001

Other Studies

24 other study(ies) available for baclofen and piperidines

ArticleYear
Analysis of the activation of dopamine metabolism by a serotonin uptake inhibitor.
    European journal of pharmacology, 1979, Dec-20, Volume: 60, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Benzofurans; Corpus Striatum; Dopamine; Female; Haloperidol; Homovanillic Acid; Piperidines; Rats; Scopolamine; Serotonin Antagonists; Time Factors

1979
The relationship between parkinsonism and tardive dyskinesia.
    The American journal of psychiatry, 1977, Volume: 134, Issue:7

    Topics: Age Factors; Aminobutyrates; Baclofen; Basal Ganglia; Biperiden; Choline; Dopamine; Dyskinesia, Drug-Induced; Humans; Levodopa; Methyltyrosines; Mouth; Parkinson Disease; Piperidines; Tranquilizing Agents

1977
Synthesis and binding properties to GABA receptors of 3-hydroxypyridinyl- and 3-hydroxypiperidinyl-analogues of baclofen.
    Archiv der Pharmazie, 1992, Volume: 325, Issue:1

    Topics: Aminobutyrates; Animals; Baclofen; Binding, Competitive; Brain; Piperidines; Propionates; Pyridines; Rats; Receptors, GABA-A

1992
The role of the laterodorsal tegmental nucleus of the rat in experimental seizures.
    Neuroscience, 1991, Volume: 43, Issue:1

    Topics: Alcian Blue; Animals; Baclofen; Bicuculline; Female; Histocytochemistry; In Vitro Techniques; Microinjections; Pentylenetetrazole; Piperidines; Rats; Rats, Inbred Strains; Seizures; Strychnine; Tegmentum Mesencephali; Thalamic Nuclei

1991
Characterization of GABAergic seizure regulation in the midline thalamus.
    Neuropharmacology, 1990, Volume: 29, Issue:7

    Topics: Animals; Baclofen; Bicuculline; Electroencephalography; Epilepsy; Female; Flurazepam; gamma-Aminobutyric Acid; Pentobarbital; Pentylenetetrazole; Piperidines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Thalamic Nuclei

1990
A pharmacological study of group I muscle afferent terminals and synaptic excitation in the intermediate nucleus and Clarke's column of the cat spinal cord.
    Experimental brain research, 1986, Volume: 64, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Cats; gamma-Aminobutyric Acid; Interneurons; Muscles; Neurons, Afferent; Piperidines; Spinal Cord; Synaptic Transmission

1986
[Intestinal pseudo-obstruction during use of baclofen].
    Nederlands tijdschrift voor geneeskunde, 1995, Sep-16, Volume: 139, Issue:37

    Topics: Aged; Anti-Ulcer Agents; Baclofen; Bisacodyl; Cathartics; Cisapride; Humans; Intestinal Pseudo-Obstruction; Male; Muscle Relaxants, Central; Piperidines; Radiography

1995
Baclofen therapy for chronic hiccup.
    The European respiratory journal, 1995, Volume: 8, Issue:2

    Topics: Anti-Ulcer Agents; Baclofen; Chronic Disease; Cisapride; Dose-Response Relationship, Drug; Female; Gastroesophageal Reflux; Hiccup; Humans; Male; Middle Aged; Omeprazole; Piperidines; Treatment Outcome

1995
Ethanol-induced emesis in the house musk shrew, Suncus murinus.
    Life sciences, 1997, Volume: 60, Issue:4-5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetaldehyde; Alcohol Deterrents; Animals; Antiemetics; Baclofen; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Depressants; Disulfiram; Dose-Response Relationship, Drug; Ethanol; Female; GABA Antagonists; Indoles; Injections, Intraperitoneal; Injections, Intraventricular; Injections, Subcutaneous; Male; Piperidines; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Tiopronin; Tropisetron; Vagotomy; Vomiting

1997
Involvement of metabotropic glutamate receptors in Gi- and Gs-dependent modulation of adenylate cyclase activity induced by a novel cognition enhancer NS-105 in rat brain.
    Brain research, 1997, Apr-18, Volume: 754, Issue:1-2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic alpha-Agonists; Alanine; Animals; Baclofen; Brimonidine Tartrate; Cell Membrane; Cerebral Cortex; Cholera Toxin; Cognition; Colforsin; Cyclic AMP; Cycloleucine; Excitatory Amino Acid Antagonists; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Isoproterenol; Kinetics; Male; Manganese; Pertussis Toxin; Piperidines; Proline; Quinoxalines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, Neurotransmitter; Virulence Factors, Bordetella; Yohimbine

1997
Effects of ifenprodil and baclofen on exercise-induced increase of myocardial oxygen demand in normotensive rats.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: Animals; Baclofen; Baroreflex; Blood Pressure; Excitatory Amino Acid Antagonists; Exercise Test; GABA Agonists; Male; Myocardium; Oxygen Consumption; Physical Exertion; Piperidines; Rats; Rats, Inbred WKY; Receptors, Glutamate; Synapses

1999
The 5-HT(1A) receptor agonist F 13640 attenuates mechanical allodynia in a rat model of trigeminal neuropathic pain.
    European journal of pharmacology, 2002, Dec-05, Volume: 456, Issue:1-3

    Topics: Aminopyridines; Animals; Baclofen; Behavior, Animal; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Morphine; Muscle Relaxants, Central; Narcotics; Pain; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Stress, Mechanical; Trigeminal Neuralgia

2002
Rats on the grog: novel pharmacotherapies for alcohol craving.
    Addictive behaviors, 2004, Volume: 29, Issue:7

    Topics: Alcoholism; Animals; Baclofen; Beer; Behavior, Addictive; Cannabinoid Receptor Antagonists; Corticotropin-Releasing Hormone; Humans; Models, Animal; Naltrexone; Narcotic Antagonists; Neuropeptide Y; Piperidines; Pyrazoles; Rats; Receptors, Corticotropin-Releasing Hormone; Receptors, GABA-B; Research Design; Rimonabant

2004
Interaction between gamma-aminobutyric acid GABAB and cannabinoid CB1 receptors in spinal pain pathways in rat.
    European journal of pharmacology, 2005, May-09, Volume: 514, Issue:2-3

    Topics: Analysis of Variance; Animals; Baclofen; Cyclohexanols; Dose-Response Relationship, Drug; Drug Interactions; Formaldehyde; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Injections, Spinal; Male; Pain; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, GABA-B; Rimonabant; Signal Transduction; Spinal Cord

2005
The cannabinoid CB1 receptor antagonist SR 141716A induces penile erection by increasing extra-cellular glutamic acid in the paraventricular nucleus of male rats.
    Behavioural brain research, 2006, May-15, Volume: 169, Issue:2

    Topics: Anesthetics, Local; Animals; Baclofen; Behavior, Animal; Cannabinoid Receptor Antagonists; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Extracellular Space; GABA Agonists; Glutamic Acid; Male; Microdialysis; Microinjections; Models, Biological; Muscimol; Paraventricular Hypothalamic Nucleus; Penile Erection; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Tetrodotoxin

2006
Modulation of the cough reflex by antitussive agents within the caudal aspect of the nucleus tractus solitarii in the rabbit.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2008, Volume: 295, Issue:1

    Topics: Animals; Antitussive Agents; Baclofen; Cough; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Male; Naloxone; Neurokinin A; Organophosphorus Compounds; Peptide Fragments; Piperidines; Rabbits; Reflex; Solitary Nucleus

2008
Role of endocannabinoid system in the ventral hippocampus of rats in the modulation of anxiety-like behaviours.
    Basic & clinical pharmacology & toxicology, 2009, Volume: 105, Issue:5

    Topics: Amidohydrolases; Animals; Anxiety; Baclofen; Behavior, Animal; Benzamides; Bicuculline; Cannabinoid Receptor Modulators; Carbamates; Dose-Response Relationship, Drug; Endocannabinoids; GABA Antagonists; Hippocampus; Male; Maze Learning; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2009
Voluntary exercise and sucrose consumption enhance cannabinoid CB1 receptor sensitivity in the striatum.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2010, Volume: 35, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Corpus Striatum; Dose-Response Relationship, Drug; Dronabinol; Drug Administration Schedule; Drug Interactions; Excitatory Amino Acid Antagonists; Exploratory Behavior; Food Preferences; GABA Agonists; GABA Antagonists; Inhibitory Postsynaptic Potentials; Male; Methoxyhydroxyphenylglycol; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Physical Conditioning, Animal; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Reward; Statistics, Nonparametric; Stress, Psychological; Sucrose; Time Factors

2010
Depression of cough reflex by microinjections of antitussive agents into caudal ventral respiratory group of the rabbit.
    Journal of applied physiology (Bethesda, Md. : 1985), 2010, Volume: 109, Issue:4

    Topics: Abdominal Muscles; Animals; Antitussive Agents; Baclofen; Cough; Diaphragm; Electromyography; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Hemodynamics; Male; Microinjections; Neurokinin A; Peptide Fragments; Phrenic Nerve; Physical Stimulation; Piperidines; Rabbits; Reflex; Respiratory Center; Respiratory Mechanics; Solitary Nucleus

2010
Effects of oral loperamide on efficacy of naltrexone, baclofen and AM-251 in blocking ethanol self-administration in rats.
    Pharmacology, biochemistry, and behavior, 2012, Volume: 100, Issue:3

    Topics: Administration, Oral; Alcohol Deterrents; Alcohol Drinking; Animals; Animals, Outbred Strains; Baclofen; Behavior, Animal; Drug Synergism; Drug Therapy, Combination; GABA-B Receptor Agonists; Loperamide; Male; Naltrexone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, Opioid, kappa; Receptors, Opioid, mu

2012
mTORC1-dependent protein synthesis underlying rapid antidepressant effect requires GABABR signaling.
    Neuropharmacology, 2013, Volume: 73

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Brain-Derived Neurotrophic Factor; Calcium; Calcium Channels, L-Type; Cells, Cultured; Cytoskeletal Proteins; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-B Receptor Agonists; Hippocampus; Humans; Immobility Response, Tonic; Male; Mechanistic Target of Rapamycin Complex 1; Mice; Multiprotein Complexes; Nerve Tissue Proteins; Organophosphorus Compounds; Piperidines; Prefrontal Cortex; Primary Cell Culture; Receptors, AMPA; Receptors, GABA-B; Signal Transduction; TOR Serine-Threonine Kinases

2013
Re-exposure to morphine-associated context facilitated long-term potentiation in the vSUB-NAc glutamatergic pathway via GluN2B-containing receptor activation.
    Addiction biology, 2017, Volume: 22, Issue:2

    Topics: Analgesics, Opioid; Animals; Baclofen; Behavior, Animal; Conditioning, Operant; GABA-A Receptor Agonists; GABA-B Receptor Agonists; Hippocampus; Long-Term Potentiation; Male; Memory; Morphine; Muscimol; Nucleus Accumbens; Phenols; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

2017
Interactive effects of AM251 and baclofen on synaptic plasticity in the rat dentate gyrus.
    Brain research, 2016, 11-15, Volume: 1651

    Topics: Anesthetics, Intravenous; Animals; Baclofen; Cannabinoid Receptor Antagonists; Dentate Gyrus; Drug Interactions; Electric Stimulation; Evoked Potentials; GABA-B Receptor Agonists; Long-Term Potentiation; Male; Microelectrodes; Piperidines; Pyrazoles; Random Allocation; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, GABA-B; Synaptic Potentials; Urethane

2016
Flexible versus Fixed Spatial Self-Ordered Response Sequencing: Effects of Inactivation and Neurochemical Modulation of Ventrolateral Prefrontal Cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2021, 08-25, Volume: 41, Issue:34

    Topics: Animals; Antipsychotic Agents; Baclofen; Callithrix; Cognition Disorders; Dopamine; Dopamine D2 Receptor Antagonists; Fluorobenzenes; GABA Agonists; gamma-Aminobutyric Acid; Goals; Memory, Short-Term; Muscimol; Piperidines; Prefrontal Cortex; Psychomotor Performance; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Spatial Behavior; Sulpiride

2021