baclofen has been researched along with naloxone in 78 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 27 (34.62) | 18.7374 |
1990's | 20 (25.64) | 18.2507 |
2000's | 19 (24.36) | 29.6817 |
2010's | 11 (14.10) | 24.3611 |
2020's | 1 (1.28) | 2.80 |
Authors | Studies |
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Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Burgis, V; Edwards, JD; Frederickson, RC; Harrell, CE | 1 |
Aghajanian, GK; Guyenet, PG | 1 |
Jacob, JJ; Ramabadran, K | 1 |
Wilson, PR; Yaksh, TL | 1 |
Levy, RA; Proudfit, HK | 1 |
DeWitte, P; Kalivas, PW; Klitenick, MA | 1 |
Rochford, J; Stewart, J | 1 |
Bertoni, P; Caffarri, G; Capretti, L; Cavazzini, U; Chiodera, P; Coiro, V; Marcato, A; Rossi, G; Volpi, R | 1 |
Holdcroft, A; Nicol, ME | 1 |
Miñano, FJ; Sancibrian, M; Serrano, JS | 1 |
Bansinath, M; Ramabadran, K; Shukla, VK; Turndorf, H | 1 |
Aley, KO; Kulkarni, SK | 1 |
Persson, B; Rubenson, A; Sillén, U | 1 |
Masotto, C; Negro-Vilar, A; Wisniewski, G | 1 |
Masotto, C; Negro-Vilar, A | 1 |
Bueno, L; Fargeas, MJ; Fioramonti, J | 1 |
Alho, H; Fujimoto, M; Geffard, M; Guidotti, A; Hanbauer, I; Kataoka, Y; Kelly, GD | 1 |
Agmo, A; Tarasco, C | 1 |
Ho, IK; Sivam, SP | 2 |
Baraldi, M; Benelli, A; Caselgrandi, E; Giberti, A; Preti, C; Sandrini, M; Tosi, G; Zanoli, P | 1 |
Djavdan, M; Zarrindast, MR | 1 |
Graf, PD; Nadel, JA; Tamaoki, J | 1 |
Tsai, HY | 2 |
Reddy, SV; Yaksh, TL | 1 |
Labella, FS; Sawynok, J | 2 |
Foong, FW; Satoh, M | 1 |
Murakoshi, T; Otsuka, M; Tamai, S; Yanagisawa, M | 1 |
Barilli, L; Chiodera, P; Coiro, V; Rossi, G; Roti, E; Volpi, R | 1 |
Dackis, CA; Gold, MS; Washton, AM | 1 |
Davies, J; Johnston, SE | 1 |
Henry, JL | 1 |
Childers, SR; Selley, DE; Sim, LJ | 1 |
Kelly, MJ; Lagrange, AH; Rønnekleiv, OK | 1 |
Bolser, DC; Chapman, RW; Hey, JA; Kreutner, W; Krobatsch, D; Mingo, G | 1 |
Lambert, NA; Wilson, WA | 1 |
Choi, YS; Do, JC; Kim, YH; Lee, KH; Son, KH; Song, DK; Suh, HW; Woo, MH | 1 |
Chieng, B; Christie, MD | 1 |
Feuerstein, TJ; Gleichauf, O; Jackisch, R; Landwehrmeyer, GB; Peckys, D; Scheremet, R | 1 |
Moises, HC; Rusin, KI | 1 |
Chavkin, C; Jin, W | 1 |
Bartolini, A; Ipponi, A; Lamberti, C; Malmberg-Aiello, P; Medica, A | 1 |
Capasso, A | 1 |
Mousa-Ahmadi, E; Zarrindast, MR | 1 |
Bocchi, C; Delsignore, R; Fontanesi, B; Gerra, G; Rustichelli, P; Timpano, M; Zaimovic, A; Zambelli, U | 1 |
de Castro-Costa, CM; Giffoni, SD; Gifoni, MA; Ramos, RS; Santos, FJ; Santos, Tde J | 1 |
Dixon, AK; Freeman, TC; Lee, K; Preston, Z; Richardson, PJ; Widdowson, L | 1 |
Mahmoudi, M; Zarrindast, MR | 1 |
Bexis, S; Ong, J; White, J | 1 |
Balerio, GN; Kemmling, AK; Rubio, MC | 1 |
González-Maeso, J; Meana, JJ; Rodríguez-Puertas, R | 1 |
Choi, SS; Han, EJ; Han, KJ; Lee, HK; Lee, JK; Lee, TH; Suh, HW | 1 |
Balerio, GN; Diaz, SL; Kemmling, AK | 1 |
Ang-Lee, MK; Aung, HH; Dey, L; Mehendale, S; Wang, A; Xie, JT; Yuan, CS | 1 |
Hemstapat, K; Monteith, GR; Smith, D; Smith, MT | 1 |
Martin, TW; Mayhew, JF | 1 |
Balerio, GN; Bonavita, CD; Diaz, SL; Kemmling, AK; Rubio, MC | 1 |
Bechtholt, AJ; Cunningham, CL | 1 |
Addolorato, G; Agabio, R; Carai, MA; Colombo, G; Gessa, GL; Maccioni, P; Orrù, A; Pes, D; Serra, S; Vacca, G | 1 |
Fossum, EN; Ingram, SL; Morgan, MM | 1 |
Bongianni, F; Cinelli, E; Fontana, GA; Mutolo, D; Pantaleo, T | 1 |
Dehpour, AR; Karimian, SM; Mirzaii-Dizgah, I; Riahi, E; Roodsari, HR; Sadeghipour, HR | 1 |
Arias, C; Mlewski, EC; Molina, JC; Spear, NE | 1 |
Prado, WA; Silva, JR; Silva, ML | 1 |
Balerio, GN; Induni, AS; Pedrón, VT; Taravini, IR | 1 |
Aso, E; Balerio, GN; Maldonado, R; Moutinho, LM; Varani, AP | 1 |
Andrade, CA; Andrade-Franzé, GM; Colombari, DS; De Luca, LA; De Oliveira, LB; Menani, JV | 1 |
Duffy, AM; Harte-Hargrove, LC; Milner, TA; Scharfman, HE; Varga-Wesson, A | 1 |
Guerdjikova, AI; Keck, PE; McElroy, SL; Mori, N | 1 |
Balerio, GN; Pedrón, VT; Varani, AP | 1 |
Demirkapu, MJ; Sakallı, E; Topkara, B; Yananli, HR | 1 |
Candiotti, KA; Gitlin, M; Rodriguez-Blanco, YF; Sevilla, A; Su, C; Weller, R; Wu, J; Yang, J; Zhang, Y; Zheng, C | 1 |
4 review(s) available for baclofen and naloxone
Article | Year |
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DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
GABA in morphine analgesia and tolerance.
Topics: Analgesia; Animals; Baclofen; Benzodiazepines; Bicuculline; Brain Chemistry; Cyclohexanecarboxylic Acids; Drug Tolerance; GABA Antagonists; gamma-Aminobutyric Acid; Mice; Morphine; Muscimol; Naloxone; Picrotoxin; Rats; Receptors, GABA-A; Synaptic Transmission | 1985 |
The sequential use of clonidine and naltrexone in the treatment of opiate addicts.
Topics: Adult; Baclofen; Clonidine; Drug Therapy, Combination; Electric Stimulation Therapy; Endorphins; Ethanol; Female; Humans; Locus Coeruleus; Male; Methyldopa; Naloxone; Naltrexone; Opioid-Related Disorders; Substance Withdrawal Syndrome | 1984 |
Psychopharmacologic treatment of eating disorders: emerging findings.
Topics: Administration, Intranasal; Anorexia Nervosa; Anti-Obesity Agents; Antidepressive Agents, Second-Generation; Antipsychotic Agents; Baclofen; Binge-Eating Disorder; Bulimia Nervosa; Bupropion; Central Nervous System Stimulants; Chromium Compounds; Humans; Lisdexamfetamine Dimesylate; Morphinans; Naloxone; Narcotic Antagonists; Obesity; Randomized Controlled Trials as Topic | 2015 |
2 trial(s) available for baclofen and naloxone
Article | Year |
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Different effects of baclofen on LH and cortisol responses to naloxone in normal men.
Topics: Adrenocorticotropic Hormone; Adult; Baclofen; Dose-Response Relationship, Drug; Double-Blind Method; Humans; Hydrocortisone; Luteinizing Hormone; Male; Naloxone; Premedication; Receptors, GABA-A; Reference Values | 1992 |
Rapid opiate detoxication in outpatient treatment: relationship with naltrexone compliance.
Topics: Adolescent; Adrenergic alpha-Agonists; Adult; Anti-Inflammatory Agents, Non-Steroidal; Baclofen; Clonidine; Dose-Response Relationship, Drug; Drug Therapy, Combination; Female; GABA Agents; Heroin Dependence; Humans; Inactivation, Metabolic; Ketoprofen; Male; Methadone; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Oxazepam; Patient Compliance; Substance Withdrawal Syndrome; Treatment Outcome | 2000 |
72 other study(ies) available for baclofen and naloxone
Article | Year |
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2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles | 2005 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
Dual actions of substance P on nociception: possible role of endogenous opioids.
Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Endorphins; Enkephalins; Mice; Naloxone; Nociceptors; Receptors, Opioid; Structure-Activity Relationship; Substance P | 1978 |
ACh, substance P and met-enkephalin in the locus coeruleus: pharmacological evidence for independent sites of action.
Topics: Acetylcholine; Animals; Baclofen; Endorphins; Enkephalins; Locus Coeruleus; Male; Naloxone; Parasympatholytics; Parasympathomimetics; Rats; Receptors, Cholinergic; Substance P; Synaptic Transmission | 1979 |
Facilitatory effect of naloxone and involvement of specific ligand-opiate receptor system in the antinociceptive effects of non-opioid drugs.
Topics: Analgesics; Animals; Baclofen; Benperidol; Haloperidol; Levodopa; Male; Mice; Naloxone; Phosphodiesterase Inhibitors; Pimozide; Receptors, Opioid; Sympathomimetics | 1978 |
Baclofen is antinociceptive in the spinal intrathecal space of animals.
Topics: Aminobutyrates; Analgesics; Animals; Baclofen; Cats; Injections, Spinal; Naloxone; Rats; Stereoisomerism; Time Factors | 1978 |
The analgesic action of baclofen [beta-(4-chlorophenyl)-gamma-aminobutyric acid].
Topics: Aminobutyrates; Analgesics; Animals; Baclofen; Dose-Response Relationship, Drug; Drug Tolerance; Male; Mice; Morphine; Motor Skills; Naloxone; Postural Balance; Reaction Time | 1977 |
Regulation of somatodendritic dopamine release in the ventral tegmental area by opioids and GABA: an in vivo microdialysis study.
Topics: Afferent Pathways; Animals; Baclofen; Biological Transport; Dendrites; Dialysis; Dopamine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Interneurons; Kinetics; Male; Models, Neurological; Morphine; Muscimol; Naloxone; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tegmentum Mesencephali; Time Factors | 1992 |
Naloxone-induced hypoalgesia: lack of involvement of the GABA-benzodiazepine receptor complex.
Topics: Analgesia; Animals; Baclofen; Bicuculline; Diazepam; Male; Muscimol; Naloxone; Pain Measurement; Rats; Rats, Wistar; Receptors, GABA-A | 1992 |
Density of intrathecal agents.
Topics: Analgesics, Opioid; Anesthesia, Spinal; Anesthetics, Local; Baclofen; Body Temperature; Cerebrospinal Fluid; Clonidine; Droperidol; Humans; Methadone; Midazolam; Naloxone; Specific Gravity; Temperature | 1992 |
Opioid and prostaglandin mechanisms involved in the effects of GABAergic drugs on body temperature.
Topics: Animals; Baclofen; Bicuculline; Body Temperature; Dose-Response Relationship, Drug; Endorphins; gamma-Aminobutyric Acid; Indomethacin; Injections, Intraperitoneal; Muscimol; Naloxone; Prostaglandins; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1991 |
Intracerebroventricular administration of kappa-agonists induces convulsions in mice.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Baclofen; Benzeneacetamides; Benzomorphans; Cerebral Ventricles; Convulsants; Dizocilpine Maleate; Injections, Intraventricular; Ketamine; Mice; Mice, Inbred Strains; Muscimol; Naloxone; Narcotic Antagonists; Narcotics; Pyrroles; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Seizures; Stereoisomerism; Thiophenes | 1991 |
Baclofen analgesia in mice: a GABAB-mediated response.
Topics: Analgesia; Animals; Baclofen; Female; GABA-A Receptor Antagonists; Male; Mice; Naloxone; Organophosphorus Compounds; Pain; Pain Measurement; Receptors, GABA-A | 1991 |
Central effects of baclofen on the L-dopa induced hyperactive urinary bladder of the rat.
Topics: Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Injections, Intraventricular; Levodopa; Male; Naloxone; Rats; Rats, Inbred Strains; Substance P; Urinary Bladder | 1985 |
Different gamma-aminobutyric acid receptor subtypes are involved in the regulation of opiate-dependent and independent luteinizing hormone-releasing hormone secretion.
Topics: Animals; Arcuate Nucleus of Hypothalamus; Arginine Vasopressin; Baclofen; Bicuculline; Dinoprostone; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Male; Median Eminence; Muscimol; Naloxone; Narcotics; Oxytocin; Phentolamine; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
Activation of gamma-aminobutyric acid B-receptors abolishes naloxone-stimulated luteinizing hormone release.
Topics: Aminooxyacetic Acid; Animals; Baclofen; Gonadotropin-Releasing Hormone; Kinetics; Luteinizing Hormone; Male; Muscimol; Naloxone; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
Central and peripheral action of GABAA and GABAB agonists on small intestine motility in rats.
Topics: Animals; Atropine; Baclofen; Bicuculline; Electromyography; Gastrointestinal Motility; Intestine, Small; Male; Muscimol; Naloxone; Phentolamine; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Intrinsic gamma aminobutyric acid receptors modulate the release of catecholamine from canine adrenal gland in situ.
Topics: Adrenal Medulla; Animals; Baclofen; Bicuculline; Chromaffin Granules; Dogs; Electric Stimulation; Epinephrine; Female; Hexamethonium; Hexamethonium Compounds; Histocytochemistry; Isoxazoles; Muscimol; Naloxone; Norepinephrine; Receptors, GABA-A; Splanchnic Nerves | 1986 |
Interactions between naloxone and GABA in the control of locomotor activity in the rat.
Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Brain; gamma-Aminobutyric Acid; Male; Motor Activity; Naloxone; Neural Inhibition; Rats; Rats, Inbred Strains; Synaptic Transmission | 1985 |
Neurobehavioral, neuroendocrine and neurochemical effects of zinc supplementation in rats.
Topics: Adrenocorticotropic Hormone; Animals; Baclofen; Behavior, Animal; beta-Endorphin; Brain; Diazepam; Endorphins; gamma-Aminobutyric Acid; In Vitro Techniques; Injections, Intraventricular; Naloxone; Pain; Pituitary Gland; Rats; Receptors, GABA-A; Receptors, Opioid; Seizures; Zinc | 1986 |
GABAA-antagonists and baclofen analgesia.
Topics: Analgesia; Animals; Baclofen; Bicuculline; GABA Antagonists; Injections, Intraperitoneal; Male; Mice; Morphine; Naloxone; Picrotoxin; Time Factors | 1988 |
Effect of gamma-aminobutyric acid on neurally mediated contraction of guinea pig trachealis smooth muscle.
Topics: Acetylcholine; Animals; Baclofen; Furosemide; gamma-Aminobutyric Acid; Guinea Pigs; Hemicholinium 3; In Vitro Techniques; Muscimol; Muscle Contraction; Muscle, Smooth; Naloxone; Phentolamine; Propranolol; Trachea | 1987 |
Effect of neuroactive peptides on labeled 5-hydroxytryptamine release from rat spinal cord.
Topics: Animals; Baclofen; beta-Endorphin; Endorphins; Enkephalin, Methionine; Male; Naloxone; Neuropeptides; Neurotensin; Pain; Rats; Rats, Inbred Strains; Secretory Rate; Serotonin; Somatostatin; Spinal Cord; Substance P | 1984 |
Studies in the primate on the analgetic effects associated with intrathecal actions of opiates, alpha-adrenergic agonists and baclofen.
Topics: Adrenergic alpha-Agonists; Analgesia; Animals; Avoidance Learning; Baclofen; Behavior, Animal; Cats; Clonidine; Drug Interactions; Electroshock; Female; Injections, Spinal; Macaca; Macaca mulatta; Male; Meperidine; Morphine; Naloxone; Narcotics; Pain; Phentolamine; Sensory Thresholds; Spinal Cord | 1981 |
Naloxone antagonizes inhibitory and unmasks excitatory effects of baclofen.
Topics: Anesthesia; Animals; Baclofen; Male; Mice; Mice, Inbred Strains; Motor Activity; Naloxone; Reflex; Stereoisomerism | 1981 |
Neurotransmitter-blocking agents influence antinociceptive effects of carbamazepine, baclofen, pentazocine and morphine on bradykinin-induced trigeminal pain.
Topics: Analgesics; Animals; Atropine; Baclofen; Bicuculline; Bradykinin; Carbamazepine; Haloperidol; Male; Methysergide; Morphine; Naloxone; Neurotransmitter Agents; Pentazocine; Rats; Rats, Inbred Strains; Sympatholytics; Trigeminal Neuralgia; Trigeminal Nucleus, Spinal | 1984 |
Tail-pinch method in vitro and the effects of some antinociceptive compounds.
Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Drug Evaluation, Preclinical; Enkephalin, Leucine; Enkephalin, Methionine; Humans; In Vitro Techniques; Morphine; Naloxone; Narcotics; Rats; Rats, Inbred Strains; Somatostatin; Spinal Cord; Stereotyped Behavior; Tail | 1984 |
Further evidence for the possible relationship between neuropeptides and serotonergic neurones in rat spinal cord.
Topics: Animals; Baclofen; Enkephalin, Methionine; Male; Naloxone; Nerve Tissue Proteins; Neurons; Potassium; Rats; Rats, Inbred Strains; Serotonin; Spinal Cord; Substance P | 1984 |
Naloxone does not alter the effect of gamma aminobutyric acid derivative, baclofen, on GH release in man.
Topics: Adult; Baclofen; Growth Hormone; Humans; Male; Naloxone; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Opioid | 1983 |
Selective antinociceptive effects of tizanidine (DS 103-282), a centrally acting muscle relaxant, on dorsal horn neurones in the feline spinal cord.
Topics: Amino Acids; Analgesics; Animals; Baclofen; Cats; Clonidine; Electric Stimulation; Female; Injections, Intravenous; Iontophoresis; Male; Muscle Relaxants, Central; Naloxone; Neurons; Norepinephrine; Spinal Cord | 1984 |
GABAergic drugs, morphine and morphine tolerance: a study in relation to nociception and gastrointestinal transit in mice.
Topics: Aminooxyacetic Acid; Analgesia; Animals; Baclofen; Bicuculline; Cyclohexanecarboxylic Acids; Digestion; Digestive System; Digestive System Physiological Phenomena; Drug Tolerance; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Morphine; Muscimol; Naloxone; Nociceptors; Oxazoles; Picrotoxin | 1983 |
On the involvement of GABA in the analgesia produced by baclofen, muscimol and morphine.
Topics: 4-Aminobutyrate Transaminase; Analgesia; Analgesics; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Naloxone; Picrotoxin; Transaminases | 1982 |
Pharmacological studies on the prolonged depressant effects of baclofen on lumbar dorsal horn units in the cat.
Topics: Animals; Baclofen; Bicuculline; Cats; Depression, Chemical; Drug Interactions; Electric Stimulation; Glycine; Muscimol; Naloxone; Nociceptors; Spinal Cord; Strychnine | 1982 |
In vitro autoradiography of receptor-activated G proteins in rat brain by agonist-stimulated guanylyl 5'-[gamma-[35S]thio]-triphosphate binding.
Topics: Animals; Autoradiography; Baclofen; Benzoxazines; Brain; Cannabinoids; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA-B Receptor Agonists; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Male; Morpholines; Naloxone; Naphthalenes; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid, mu | 1995 |
Estradiol-17 beta and mu-opioid peptides rapidly hyperpolarize GnRH neurons: a cellular mechanism of negative feedback?
Topics: Animals; Arcuate Nucleus of Hypothalamus; Baclofen; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Estradiol; Feedback; Female; Gonadotropin-Releasing Hormone; Guinea Pigs; Membrane Potentials; Naloxone; Neurons; Ovariectomy; Potassium Channels; Receptors, Opioid, mu; Tetrodotoxin | 1995 |
Respiratory effects of baclofen and 3-aminopropylphosphinic acid in guinea-pigs.
Topics: Administration, Inhalation; Analysis of Variance; Animals; Baclofen; Bicuculline; Carbon Dioxide; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Guinea Pigs; Injections, Intraventricular; Injections, Subcutaneous; Male; Naloxone; Organophosphorus Compounds; Pulmonary Ventilation; Respiration; Tidal Volume | 1995 |
Heterogeneity in presynaptic regulation of GABA release from hippocampal inhibitory neurons.
Topics: Analgesics; Animals; Baclofen; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Evoked Potentials; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Homeostasis; In Vitro Techniques; Male; Naloxone; Nerve Fibers; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Synapses | 1993 |
Antinociceptive effect of smilaxin B administered intracerebroventricularly in the mouse.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Cerebral Ventricles; Dizocilpine Maleate; Glycosides; Injections, Intraventricular; Injections, Spinal; Male; Methysergide; Mice; Mice, Inbred ICR; Muscimol; Naloxone; Pain; Sincalide; Spinal Cord; Spirostans; Yohimbine | 1996 |
Local opioid withdrawal in rat single periaqueductal gray neurons in vitro.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Adrenergic alpha-Agonists; Analgesics, Opioid; Animals; Baclofen; Bicuculline; Clonidine; Drug Tolerance; Electrophysiology; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Male; Membrane Potentials; Morphine; Naloxone; Narcotic Antagonists; Neurons; Organ Culture Techniques; Periaqueductal Gray; Potassium Channels; Rats; Rats, Sprague-Dawley; Sensitivity and Specificity; Substance Withdrawal Syndrome; Tetrodotoxin; Time Factors; Valine | 1996 |
Opioid receptor-mediated control of acetylcholine release in human neocortex tissue.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetylcholine; Adolescent; Adult; Aged; Analgesics; Analysis of Variance; Baclofen; Cerebral Cortex; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; GABA Agonists; Humans; Male; Middle Aged; Muscimol; Naloxone; Naltrexone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid, delta; Tetrodotoxin | 1996 |
Mu-opioid and GABA(B) receptors modulate different types of Ca2+ currents in rat nodose ganglion neurons.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analgesics, Opioid; Animals; Baclofen; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Calcium Channels, N-Type; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA Agonists; GABA Antagonists; Naloxone; Narcotic Antagonists; Nerve Tissue Proteins; Neurons; Nifedipine; Nodose Ganglion; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Patch-Clamp Techniques; Peptides; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Spider Venoms | 1998 |
Mu opioids enhance mossy fiber synaptic transmission indirectly by reducing GABAB receptor activation.
Topics: Analgesics, Opioid; Animals; Baclofen; Bicuculline; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA Antagonists; Long-Term Potentiation; Male; Membrane Potentials; Mossy Fibers, Hippocampal; Naloxone; Narcotic Antagonists; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Somatostatin; Synaptic Transmission | 1999 |
Tiagabine antinociception in rodents depends on GABA(B) receptor activation: parallel antinociception testing and medial thalamus GABA microdialysis.
Topics: Abdomen; Animals; Baclofen; Constriction, Pathologic; Dose-Response Relationship, Drug; Escape Reaction; Extracellular Space; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Microdialysis; Naloxone; Narcotic Antagonists; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Nociceptors; Organophosphorus Compounds; Pain; Pain Measurement; Pain Threshold; Psychomotor Performance; Receptors, GABA-B; Thalamus; Tiagabine | 1999 |
GABAB receptors are involved in the control of acute opiate withdrawal in isolated tissue.
Topics: Animals; Baclofen; Dose-Response Relationship, Drug; GABA Agonists; GABA-B Receptor Antagonists; Guinea Pigs; In Vitro Techniques; Male; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Opioid-Related Disorders; Receptors, GABA-B; Substance Withdrawal Syndrome | 1999 |
Effects of GABAergic system on naloxone-induced jumping in morphine-dependent mice.
Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Mice; Morphine Dependence; Muscimol; Naloxone; Narcotic Antagonists; Organophosphorus Compounds; Picrotoxin; Substance Withdrawal Syndrome | 1999 |
The effect of baclofen on spontaneous and evoked behavioural expression of experimental neuropathic chronic pain.
Topics: Animals; Baclofen; Behavior, Animal; Chronic Disease; GABA Agonists; Male; Naloxone; Narcotic Antagonists; Pain; Peripheral Nervous System Diseases; Rats; Rats, Wistar; Sciatic Nerve | 1999 |
Adenosine receptor expression and function in rat striatal cholinergic interneurons.
Topics: Acetylcholine; Adenosine; Adenosine Deaminase; Animals; Baclofen; Bicuculline; Caffeine; Cholinergic Fibers; Corpus Striatum; Dose-Response Relationship, Drug; GABA Antagonists; Gene Expression; Male; Membrane Potentials; Naloxone; Narcotic Antagonists; Neurons; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; RNA, Messenger; Tritium; Xanthines | 2000 |
GABA mechanisms and antinociception in mice with ligated sciatic nerve.
Topics: Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA Antagonists; Ligation; Male; Mice; Mice, Inbred Strains; Morphine; Muscimol; Naloxone; Organophosphorus Compounds; Pain; Pain Measurement; Sciatic Nerve | 2001 |
Attenuation of morphine withdrawal signs by the GABA(B) receptor agonist baclofen.
Topics: Animals; Baclofen; Behavior, Animal; Drug Antagonism; Drug Combinations; GABA Agonists; GABA Antagonists; Male; Morphine Dependence; Naloxone; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome | 2001 |
Baclofen prevents morphine withdrawal irrespective of seasonal variation.
Topics: Animals; Arousal; Baclofen; Female; Male; Mice; Morphine; Motor Activity; Naloxone; Narcotic Antagonists; Seasons; Substance Withdrawal Syndrome | 2002 |
Quantitative stoichiometry of G-proteins activated by mu-opioid receptors in postmortem human brain.
Topics: Alkylation; Analgesics, Opioid; Baclofen; Binding, Competitive; Brain Chemistry; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Inhibitors; Ethylmaleimide; GABA Agonists; GTP-Binding Protein Regulators; GTP-Binding Proteins; Humans; In Vitro Techniques; Kinetics; Membranes; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid, mu; Signal Transduction | 2002 |
Antinociceptive mechanisms of platycodin D administered intracerebroventricularly in the mouse.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Analgesics; Animals; Baclofen; Carbohydrate Sequence; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Injections, Intraventricular; Injections, Spinal; Male; Methysergide; Mice; Mice, Inbred ICR; Molecular Sequence Data; Muscimol; Naloxone; Narcotic Antagonists; Pain Measurement; Plant Extracts; Platycodon; Receptors, Cholecystokinin; Receptors, N-Methyl-D-Aspartate; Saponins; Serotonin Antagonists; Sincalide; Tail; Triterpenes; Yohimbine | 2002 |
Baclofen reestablishes striatal and cortical dopamine concentrations during naloxone-precipitated withdrawal.
Topics: Animals; Baclofen; Cerebral Cortex; Chromatography, High Pressure Liquid; Dopamine; Electrochemistry; GABA Agonists; GABA-B Receptor Agonists; Hippocampus; Homovanillic Acid; Hydroxyindoleacetic Acid; Male; Mice; Morphine Dependence; Naloxone; Narcotic Antagonists; Neostriatum; Serotonin; Substance Withdrawal Syndrome | 2003 |
Kavalactones and dihydrokavain modulate GABAergic activity in a rat gastric-brainstem preparation.
Topics: Animals; Baclofen; Drug Interactions; GABA Agents; GABA Agonists; GABA Antagonists; Kava; Lactones; Muscimol; Naloxone; Narcotic Antagonists; Plant Extracts; Pyrones; Rats; Rats, Sprague-Dawley; Solitary Nucleus; Stomach | 2002 |
Morphine-3-glucuronide's neuro-excitatory effects are mediated via indirect activation of N-methyl-D-aspartic acid receptors: mechanistic studies in embryonic cultured hippocampal neurones.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aniline Compounds; Animals; Baclofen; Calcium; Calcium Channel Blockers; Cells, Cultured; Central Nervous System Stimulants; Cytosol; Excitatory Amino Acid Antagonists; Fluorescent Dyes; GABA Agonists; Hippocampus; Image Processing, Computer-Assisted; Immunohistochemistry; Microscopy, Fluorescence; Morphine Derivatives; Naloxone; Narcotic Antagonists; Neurons; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Tetrodotoxin; Xanthenes | 2003 |
Baclofen pumps: comment on Anderson et al.
Topics: Anti-Arrhythmia Agents; Atropine; Baclofen; Child; Coma; GABA Agonists; Humans; Infusion Pumps, Implantable; Morphine; Naloxone; Narcotic Antagonists; Oxygen; Postoperative Complications | 2003 |
Baclofen reestablishes micro-opioid receptor levels modified by morphine withdrawal syndrome in either sex.
Topics: Animals; Baclofen; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Female; GABA Agonists; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Receptors, Opioid, mu; Sex Factors; Substance Withdrawal Syndrome | 2004 |
Ethanol-induced conditioned place preference is expressed through a ventral tegmental area dependent mechanism.
Topics: Animals; Baclofen; Central Nervous System Depressants; Conditioning, Classical; Ethanol; GABA Agonists; Male; Mice; Naloxone; Quaternary Ammonium Compounds; Receptors, GABA-B; Receptors, Opioid; Reinforcement, Psychology; Space Perception; Ventral Tegmental Area | 2005 |
Baclofen-induced reduction of alcohol reinforcement in alcohol-preferring rats.
Topics: Alcohol Drinking; Animals; Baclofen; Central Nervous System Depressants; Conditioning, Operant; Dose-Response Relationship, Drug; Ethanol; GABA Agonists; Male; Naloxone; Narcotic Antagonists; Rats; Reinforcement, Psychology; Self Administration; Sucrose | 2005 |
Behavioral and electrophysiological evidence for opioid tolerance in adolescent rats.
Topics: Action Potentials; Age Factors; Animals; Baclofen; Behavior, Animal; Dose-Response Relationship, Drug; Drug Interactions; Drug Tolerance; Electrophysiology; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Agonists; Male; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Neurons; Pain Measurement; Pain Threshold; Periaqueductal Gray; Rats; Rats, Sprague-Dawley; Reaction Time | 2007 |
Modulation of the cough reflex by antitussive agents within the caudal aspect of the nucleus tractus solitarii in the rabbit.
Topics: Animals; Antitussive Agents; Baclofen; Cough; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Male; Naloxone; Neurokinin A; Organophosphorus Compounds; Peptide Fragments; Piperidines; Rabbits; Reflex; Solitary Nucleus | 2008 |
Attenuation of morphine withdrawal signs by a GABAB receptor agonist in the locus coeruleus of rats.
Topics: Analysis of Variance; Animals; Baclofen; Dose-Response Relationship, Drug; Drug Therapy, Combination; GABA Agonists; GABA Antagonists; Injections, Subcutaneous; Locus Coeruleus; Male; Morphine; Morphine Dependence; Motor Activity; Naloxone; Narcotic Antagonists; Narcotics; Organophosphorus Compounds; Rats; Rats, Wistar; Substance Withdrawal Syndrome | 2009 |
Naloxone and baclofen attenuate ethanol's locomotor-activating effects in preweanling Sprague-Dawley rats.
Topics: Analysis of Variance; Animals; Animals, Newborn; Baclofen; Central Nervous System Depressants; Dose-Response Relationship, Drug; Ethanol; GABA Agonists; Male; Motor Activity; Naloxone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley | 2009 |
Analgesia induced by 2- or 100-Hz electroacupuncture in the rat tail-flick test depends on the activation of different descending pain inhibitory mechanisms.
Topics: Adjuvants, Anesthesia; Adrenergic alpha-Antagonists; Analgesia; Anesthetics, Intravenous; Animals; Atropine; Baclofen; Bicuculline; Biophysics; Dioxanes; Disease Models, Animal; Electroacupuncture; GABA Agents; Male; Methysergide; Models, Biological; Multivariate Analysis; Naloxone; Narcotic Antagonists; Pain; Pain Management; Pain Measurement; Rats; Rats, Wistar; Reaction Time; Serotonin Antagonists; Tail; Thiopental; Time Factors | 2011 |
Baclofen did not modify sexually dimorphic c-Fos expression during morphine withdrawal syndrome.
Topics: Animals; Baclofen; Female; GABA-B Receptor Agonists; Hippocampus; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Proto-Oncogene Proteins c-fos; Sex Factors; Substance Withdrawal Syndrome | 2013 |
Attenuation by baclofen of nicotine rewarding properties and nicotine withdrawal manifestations.
Topics: Animals; Anxiety; Avoidance Learning; Baclofen; Conditioning, Psychological; GABA-B Receptor Agonists; Male; Mice; Movement; Naloxone; Narcotic Antagonists; Nicotine; Nicotinic Agonists; Receptors, GABA-B; Reward; Space Perception; Substance Withdrawal Syndrome; Tobacco Use Disorder | 2014 |
Gabaergic and opioid receptors mediate the facilitation of NaCl intake induced by α₂-adrenergic activation in the lateral parabrachial nucleus.
Topics: Animals; Antihypertensive Agents; Baclofen; Bicuculline; Captopril; Enzyme Inhibitors; Furosemide; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; Imidazoles; Male; Naloxone; Narcotic Antagonists; Parabrachial Nucleus; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, GABA; Receptors, Opioid; Sodium Chloride; Sodium Potassium Chloride Symporter Inhibitors | 2015 |
Opioid receptor-dependent sex differences in synaptic plasticity in the hippocampal mossy fiber pathway of the adult rat.
Topics: Animals; Baclofen; Bicuculline; Dendritic Spines; Estrous Cycle; Female; GABA-A Receptor Antagonists; Hippocampus; Long-Term Potentiation; Male; Mossy Fibers, Hippocampal; Naloxone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Opioid; Sex Characteristics; Somatostatin; Synapses | 2015 |
Baclofen prevents the elevated plus maze behavior and BDNF expression during naloxone precipitated morphine withdrawal in male and female mice.
Topics: Animals; Baclofen; Brain; Brain-Derived Neurotrophic Factor; Female; GABA-B Receptor Agonists; Male; Maze Learning; Mice; Morphine; Naloxone; Narcotic Antagonists; Sex Factors; Substance Withdrawal Syndrome | 2016 |
Effects of Injection of Gamma-Aminobutyric Acid Agonists into the Nucleus Accumbens on Naloxone-Induced Morphine Withdrawal.
Topics: Animals; Baclofen; GABA Agonists; Injections; Locomotion; Male; Morphine Dependence; Muscimol; Naloxone; Narcotic Antagonists; Nucleus Accumbens; Rats, Sprague-Dawley; Substance Withdrawal Syndrome | 2017 |
The mechanism of chronic nicotine exposure and nicotine withdrawal on pain perception in an animal model.
Topics: Animals; Baclofen; Bicuculline; Disease Models, Animal; Down-Regulation; Endorphins; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hyperalgesia; Male; Naloxone; Nicotine; Pain Perception; Pain Threshold; Rats; Receptors, Opioid, mu; Spinal Cord; Substance Withdrawal Syndrome; Time Factors; Up-Regulation | 2020 |