baclofen and naloxone

baclofen has been researched along with naloxone in 78 studies

Research

Studies (78)

TimeframeStudies, this research(%)All Research%
pre-199027 (34.62)18.7374
1990's20 (25.64)18.2507
2000's19 (24.36)29.6817
2010's11 (14.10)24.3611
2020's1 (1.28)2.80

Authors

AuthorsStudies
Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Burgis, V; Edwards, JD; Frederickson, RC; Harrell, CE1
Aghajanian, GK; Guyenet, PG1
Jacob, JJ; Ramabadran, K1
Wilson, PR; Yaksh, TL1
Levy, RA; Proudfit, HK1
DeWitte, P; Kalivas, PW; Klitenick, MA1
Rochford, J; Stewart, J1
Bertoni, P; Caffarri, G; Capretti, L; Cavazzini, U; Chiodera, P; Coiro, V; Marcato, A; Rossi, G; Volpi, R1
Holdcroft, A; Nicol, ME1
Miñano, FJ; Sancibrian, M; Serrano, JS1
Bansinath, M; Ramabadran, K; Shukla, VK; Turndorf, H1
Aley, KO; Kulkarni, SK1
Persson, B; Rubenson, A; Sillén, U1
Masotto, C; Negro-Vilar, A; Wisniewski, G1
Masotto, C; Negro-Vilar, A1
Bueno, L; Fargeas, MJ; Fioramonti, J1
Alho, H; Fujimoto, M; Geffard, M; Guidotti, A; Hanbauer, I; Kataoka, Y; Kelly, GD1
Agmo, A; Tarasco, C1
Ho, IK; Sivam, SP2
Baraldi, M; Benelli, A; Caselgrandi, E; Giberti, A; Preti, C; Sandrini, M; Tosi, G; Zanoli, P1
Djavdan, M; Zarrindast, MR1
Graf, PD; Nadel, JA; Tamaoki, J1
Tsai, HY2
Reddy, SV; Yaksh, TL1
Labella, FS; Sawynok, J2
Foong, FW; Satoh, M1
Murakoshi, T; Otsuka, M; Tamai, S; Yanagisawa, M1
Barilli, L; Chiodera, P; Coiro, V; Rossi, G; Roti, E; Volpi, R1
Dackis, CA; Gold, MS; Washton, AM1
Davies, J; Johnston, SE1
Henry, JL1
Childers, SR; Selley, DE; Sim, LJ1
Kelly, MJ; Lagrange, AH; Rønnekleiv, OK1
Bolser, DC; Chapman, RW; Hey, JA; Kreutner, W; Krobatsch, D; Mingo, G1
Lambert, NA; Wilson, WA1
Choi, YS; Do, JC; Kim, YH; Lee, KH; Son, KH; Song, DK; Suh, HW; Woo, MH1
Chieng, B; Christie, MD1
Feuerstein, TJ; Gleichauf, O; Jackisch, R; Landwehrmeyer, GB; Peckys, D; Scheremet, R1
Moises, HC; Rusin, KI1
Chavkin, C; Jin, W1
Bartolini, A; Ipponi, A; Lamberti, C; Malmberg-Aiello, P; Medica, A1
Capasso, A1
Mousa-Ahmadi, E; Zarrindast, MR1
Bocchi, C; Delsignore, R; Fontanesi, B; Gerra, G; Rustichelli, P; Timpano, M; Zaimovic, A; Zambelli, U1
de Castro-Costa, CM; Giffoni, SD; Gifoni, MA; Ramos, RS; Santos, FJ; Santos, Tde J1
Dixon, AK; Freeman, TC; Lee, K; Preston, Z; Richardson, PJ; Widdowson, L1
Mahmoudi, M; Zarrindast, MR1
Bexis, S; Ong, J; White, J1
Balerio, GN; Kemmling, AK; Rubio, MC1
González-Maeso, J; Meana, JJ; Rodríguez-Puertas, R1
Choi, SS; Han, EJ; Han, KJ; Lee, HK; Lee, JK; Lee, TH; Suh, HW1
Balerio, GN; Diaz, SL; Kemmling, AK1
Ang-Lee, MK; Aung, HH; Dey, L; Mehendale, S; Wang, A; Xie, JT; Yuan, CS1
Hemstapat, K; Monteith, GR; Smith, D; Smith, MT1
Martin, TW; Mayhew, JF1
Balerio, GN; Bonavita, CD; Diaz, SL; Kemmling, AK; Rubio, MC1
Bechtholt, AJ; Cunningham, CL1
Addolorato, G; Agabio, R; Carai, MA; Colombo, G; Gessa, GL; Maccioni, P; Orrù, A; Pes, D; Serra, S; Vacca, G1
Fossum, EN; Ingram, SL; Morgan, MM1
Bongianni, F; Cinelli, E; Fontana, GA; Mutolo, D; Pantaleo, T1
Dehpour, AR; Karimian, SM; Mirzaii-Dizgah, I; Riahi, E; Roodsari, HR; Sadeghipour, HR1
Arias, C; Mlewski, EC; Molina, JC; Spear, NE1
Prado, WA; Silva, JR; Silva, ML1
Balerio, GN; Induni, AS; Pedrón, VT; Taravini, IR1
Aso, E; Balerio, GN; Maldonado, R; Moutinho, LM; Varani, AP1
Andrade, CA; Andrade-Franzé, GM; Colombari, DS; De Luca, LA; De Oliveira, LB; Menani, JV1
Duffy, AM; Harte-Hargrove, LC; Milner, TA; Scharfman, HE; Varga-Wesson, A1
Guerdjikova, AI; Keck, PE; McElroy, SL; Mori, N1
Balerio, GN; Pedrón, VT; Varani, AP1
Demirkapu, MJ; Sakallı, E; Topkara, B; Yananli, HR1
Candiotti, KA; Gitlin, M; Rodriguez-Blanco, YF; Sevilla, A; Su, C; Weller, R; Wu, J; Yang, J; Zhang, Y; Zheng, C1

Reviews

4 review(s) available for baclofen and naloxone

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
GABA in morphine analgesia and tolerance.
    Life sciences, 1985, Jul-22, Volume: 37, Issue:3

    Topics: Analgesia; Animals; Baclofen; Benzodiazepines; Bicuculline; Brain Chemistry; Cyclohexanecarboxylic Acids; Drug Tolerance; GABA Antagonists; gamma-Aminobutyric Acid; Mice; Morphine; Muscimol; Naloxone; Picrotoxin; Rats; Receptors, GABA-A; Synaptic Transmission

1985
The sequential use of clonidine and naltrexone in the treatment of opiate addicts.
    Advances in alcohol & substance abuse, 1984,Spring, Volume: 3, Issue:3

    Topics: Adult; Baclofen; Clonidine; Drug Therapy, Combination; Electric Stimulation Therapy; Endorphins; Ethanol; Female; Humans; Locus Coeruleus; Male; Methyldopa; Naloxone; Naltrexone; Opioid-Related Disorders; Substance Withdrawal Syndrome

1984
Psychopharmacologic treatment of eating disorders: emerging findings.
    Current psychiatry reports, 2015, Volume: 17, Issue:5

    Topics: Administration, Intranasal; Anorexia Nervosa; Anti-Obesity Agents; Antidepressive Agents, Second-Generation; Antipsychotic Agents; Baclofen; Binge-Eating Disorder; Bulimia Nervosa; Bupropion; Central Nervous System Stimulants; Chromium Compounds; Humans; Lisdexamfetamine Dimesylate; Morphinans; Naloxone; Narcotic Antagonists; Obesity; Randomized Controlled Trials as Topic

2015

Trials

2 trial(s) available for baclofen and naloxone

ArticleYear
Different effects of baclofen on LH and cortisol responses to naloxone in normal men.
    Psychoneuroendocrinology, 1992, Volume: 17, Issue:6

    Topics: Adrenocorticotropic Hormone; Adult; Baclofen; Dose-Response Relationship, Drug; Double-Blind Method; Humans; Hydrocortisone; Luteinizing Hormone; Male; Naloxone; Premedication; Receptors, GABA-A; Reference Values

1992
Rapid opiate detoxication in outpatient treatment: relationship with naltrexone compliance.
    Journal of substance abuse treatment, 2000, Volume: 18, Issue:2

    Topics: Adolescent; Adrenergic alpha-Agonists; Adult; Anti-Inflammatory Agents, Non-Steroidal; Baclofen; Clonidine; Dose-Response Relationship, Drug; Drug Therapy, Combination; Female; GABA Agents; Heroin Dependence; Humans; Inactivation, Metabolic; Ketoprofen; Male; Methadone; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Oxazepam; Patient Compliance; Substance Withdrawal Syndrome; Treatment Outcome

2000

Other Studies

72 other study(ies) available for baclofen and naloxone

ArticleYear
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
    Journal of medicinal chemistry, 2005, Nov-03, Volume: 48, Issue:22

    Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles

2005
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Dual actions of substance P on nociception: possible role of endogenous opioids.
    Science (New York, N.Y.), 1978, Mar-24, Volume: 199, Issue:4335

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Endorphins; Enkephalins; Mice; Naloxone; Nociceptors; Receptors, Opioid; Structure-Activity Relationship; Substance P

1978
ACh, substance P and met-enkephalin in the locus coeruleus: pharmacological evidence for independent sites of action.
    European journal of pharmacology, 1979, Feb-01, Volume: 53, Issue:4

    Topics: Acetylcholine; Animals; Baclofen; Endorphins; Enkephalins; Locus Coeruleus; Male; Naloxone; Parasympatholytics; Parasympathomimetics; Rats; Receptors, Cholinergic; Substance P; Synaptic Transmission

1979
Facilitatory effect of naloxone and involvement of specific ligand-opiate receptor system in the antinociceptive effects of non-opioid drugs.
    Archives internationales de pharmacodynamie et de therapie, 1978, Volume: 236, Issue:1

    Topics: Analgesics; Animals; Baclofen; Benperidol; Haloperidol; Levodopa; Male; Mice; Naloxone; Phosphodiesterase Inhibitors; Pimozide; Receptors, Opioid; Sympathomimetics

1978
Baclofen is antinociceptive in the spinal intrathecal space of animals.
    European journal of pharmacology, 1978, Oct-15, Volume: 51, Issue:4

    Topics: Aminobutyrates; Analgesics; Animals; Baclofen; Cats; Injections, Spinal; Naloxone; Rats; Stereoisomerism; Time Factors

1978
The analgesic action of baclofen [beta-(4-chlorophenyl)-gamma-aminobutyric acid].
    The Journal of pharmacology and experimental therapeutics, 1977, Volume: 202, Issue:2

    Topics: Aminobutyrates; Analgesics; Animals; Baclofen; Dose-Response Relationship, Drug; Drug Tolerance; Male; Mice; Morphine; Motor Skills; Naloxone; Postural Balance; Reaction Time

1977
Regulation of somatodendritic dopamine release in the ventral tegmental area by opioids and GABA: an in vivo microdialysis study.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:7

    Topics: Afferent Pathways; Animals; Baclofen; Biological Transport; Dendrites; Dialysis; Dopamine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Interneurons; Kinetics; Male; Models, Neurological; Morphine; Muscimol; Naloxone; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tegmentum Mesencephali; Time Factors

1992
Naloxone-induced hypoalgesia: lack of involvement of the GABA-benzodiazepine receptor complex.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:2

    Topics: Analgesia; Animals; Baclofen; Bicuculline; Diazepam; Male; Muscimol; Naloxone; Pain Measurement; Rats; Rats, Wistar; Receptors, GABA-A

1992
Density of intrathecal agents.
    British journal of anaesthesia, 1992, Volume: 68, Issue:1

    Topics: Analgesics, Opioid; Anesthesia, Spinal; Anesthetics, Local; Baclofen; Body Temperature; Cerebrospinal Fluid; Clonidine; Droperidol; Humans; Methadone; Midazolam; Naloxone; Specific Gravity; Temperature

1992
Opioid and prostaglandin mechanisms involved in the effects of GABAergic drugs on body temperature.
    General pharmacology, 1991, Volume: 22, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Body Temperature; Dose-Response Relationship, Drug; Endorphins; gamma-Aminobutyric Acid; Indomethacin; Injections, Intraperitoneal; Muscimol; Naloxone; Prostaglandins; Rats; Rats, Inbred Strains; Receptors, GABA-A

1991
Intracerebroventricular administration of kappa-agonists induces convulsions in mice.
    Brain research bulletin, 1991, Volume: 27, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Baclofen; Benzeneacetamides; Benzomorphans; Cerebral Ventricles; Convulsants; Dizocilpine Maleate; Injections, Intraventricular; Ketamine; Mice; Mice, Inbred Strains; Muscimol; Naloxone; Narcotic Antagonists; Narcotics; Pyrroles; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Seizures; Stereoisomerism; Thiophenes

1991
Baclofen analgesia in mice: a GABAB-mediated response.
    Methods and findings in experimental and clinical pharmacology, 1991, Volume: 13, Issue:10

    Topics: Analgesia; Animals; Baclofen; Female; GABA-A Receptor Antagonists; Male; Mice; Naloxone; Organophosphorus Compounds; Pain; Pain Measurement; Receptors, GABA-A

1991
Central effects of baclofen on the L-dopa induced hyperactive urinary bladder of the rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 330, Issue:3

    Topics: Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Injections, Intraventricular; Levodopa; Male; Naloxone; Rats; Rats, Inbred Strains; Substance P; Urinary Bladder

1985
Different gamma-aminobutyric acid receptor subtypes are involved in the regulation of opiate-dependent and independent luteinizing hormone-releasing hormone secretion.
    Endocrinology, 1989, Volume: 125, Issue:1

    Topics: Animals; Arcuate Nucleus of Hypothalamus; Arginine Vasopressin; Baclofen; Bicuculline; Dinoprostone; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Male; Median Eminence; Muscimol; Naloxone; Narcotics; Oxytocin; Phentolamine; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
Activation of gamma-aminobutyric acid B-receptors abolishes naloxone-stimulated luteinizing hormone release.
    Endocrinology, 1987, Volume: 121, Issue:6

    Topics: Aminooxyacetic Acid; Animals; Baclofen; Gonadotropin-Releasing Hormone; Kinetics; Luteinizing Hormone; Male; Muscimol; Naloxone; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
Central and peripheral action of GABAA and GABAB agonists on small intestine motility in rats.
    European journal of pharmacology, 1988, May-20, Volume: 150, Issue:1-2

    Topics: Animals; Atropine; Baclofen; Bicuculline; Electromyography; Gastrointestinal Motility; Intestine, Small; Male; Muscimol; Naloxone; Phentolamine; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Intrinsic gamma aminobutyric acid receptors modulate the release of catecholamine from canine adrenal gland in situ.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2

    Topics: Adrenal Medulla; Animals; Baclofen; Bicuculline; Chromaffin Granules; Dogs; Electric Stimulation; Epinephrine; Female; Hexamethonium; Hexamethonium Compounds; Histocytochemistry; Isoxazoles; Muscimol; Naloxone; Norepinephrine; Receptors, GABA-A; Splanchnic Nerves

1986
Interactions between naloxone and GABA in the control of locomotor activity in the rat.
    Journal of neural transmission, 1985, Volume: 61, Issue:3-4

    Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Brain; gamma-Aminobutyric Acid; Male; Motor Activity; Naloxone; Neural Inhibition; Rats; Rats, Inbred Strains; Synaptic Transmission

1985
Neurobehavioral, neuroendocrine and neurochemical effects of zinc supplementation in rats.
    Advances in experimental medicine and biology, 1986, Volume: 203

    Topics: Adrenocorticotropic Hormone; Animals; Baclofen; Behavior, Animal; beta-Endorphin; Brain; Diazepam; Endorphins; gamma-Aminobutyric Acid; In Vitro Techniques; Injections, Intraventricular; Naloxone; Pain; Pituitary Gland; Rats; Receptors, GABA-A; Receptors, Opioid; Seizures; Zinc

1986
GABAA-antagonists and baclofen analgesia.
    General pharmacology, 1988, Volume: 19, Issue:5

    Topics: Analgesia; Animals; Baclofen; Bicuculline; GABA Antagonists; Injections, Intraperitoneal; Male; Mice; Morphine; Naloxone; Picrotoxin; Time Factors

1988
Effect of gamma-aminobutyric acid on neurally mediated contraction of guinea pig trachealis smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:1

    Topics: Acetylcholine; Animals; Baclofen; Furosemide; gamma-Aminobutyric Acid; Guinea Pigs; Hemicholinium 3; In Vitro Techniques; Muscimol; Muscle Contraction; Muscle, Smooth; Naloxone; Phentolamine; Propranolol; Trachea

1987
Effect of neuroactive peptides on labeled 5-hydroxytryptamine release from rat spinal cord.
    Proceedings of the National Science Council, Republic of China. Part B, Life sciences, 1984, Volume: 8, Issue:2

    Topics: Animals; Baclofen; beta-Endorphin; Endorphins; Enkephalin, Methionine; Male; Naloxone; Neuropeptides; Neurotensin; Pain; Rats; Rats, Inbred Strains; Secretory Rate; Serotonin; Somatostatin; Spinal Cord; Substance P

1984
Studies in the primate on the analgetic effects associated with intrathecal actions of opiates, alpha-adrenergic agonists and baclofen.
    Anesthesiology, 1981, Volume: 54, Issue:6

    Topics: Adrenergic alpha-Agonists; Analgesia; Animals; Avoidance Learning; Baclofen; Behavior, Animal; Cats; Clonidine; Drug Interactions; Electroshock; Female; Injections, Spinal; Macaca; Macaca mulatta; Male; Meperidine; Morphine; Naloxone; Narcotics; Pain; Phentolamine; Sensory Thresholds; Spinal Cord

1981
Naloxone antagonizes inhibitory and unmasks excitatory effects of baclofen.
    The Journal of pharmacy and pharmacology, 1981, Volume: 33, Issue:9

    Topics: Anesthesia; Animals; Baclofen; Male; Mice; Mice, Inbred Strains; Motor Activity; Naloxone; Reflex; Stereoisomerism

1981
Neurotransmitter-blocking agents influence antinociceptive effects of carbamazepine, baclofen, pentazocine and morphine on bradykinin-induced trigeminal pain.
    Neuropharmacology, 1984, Volume: 23, Issue:6

    Topics: Analgesics; Animals; Atropine; Baclofen; Bicuculline; Bradykinin; Carbamazepine; Haloperidol; Male; Methysergide; Morphine; Naloxone; Neurotransmitter Agents; Pentazocine; Rats; Rats, Inbred Strains; Sympatholytics; Trigeminal Neuralgia; Trigeminal Nucleus, Spinal

1984
Tail-pinch method in vitro and the effects of some antinociceptive compounds.
    European journal of pharmacology, 1984, Nov-13, Volume: 106, Issue:2

    Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Drug Evaluation, Preclinical; Enkephalin, Leucine; Enkephalin, Methionine; Humans; In Vitro Techniques; Morphine; Naloxone; Narcotics; Rats; Rats, Inbred Strains; Somatostatin; Spinal Cord; Stereotyped Behavior; Tail

1984
Further evidence for the possible relationship between neuropeptides and serotonergic neurones in rat spinal cord.
    Japanese journal of pharmacology, 1984, Volume: 35, Issue:2

    Topics: Animals; Baclofen; Enkephalin, Methionine; Male; Naloxone; Nerve Tissue Proteins; Neurons; Potassium; Rats; Rats, Inbred Strains; Serotonin; Spinal Cord; Substance P

1984
Naloxone does not alter the effect of gamma aminobutyric acid derivative, baclofen, on GH release in man.
    Journal of endocrinological investigation, 1983, Volume: 6, Issue:5

    Topics: Adult; Baclofen; Growth Hormone; Humans; Male; Naloxone; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Opioid

1983
Selective antinociceptive effects of tizanidine (DS 103-282), a centrally acting muscle relaxant, on dorsal horn neurones in the feline spinal cord.
    British journal of pharmacology, 1984, Volume: 82, Issue:2

    Topics: Amino Acids; Analgesics; Animals; Baclofen; Cats; Clonidine; Electric Stimulation; Female; Injections, Intravenous; Iontophoresis; Male; Muscle Relaxants, Central; Naloxone; Neurons; Norepinephrine; Spinal Cord

1984
GABAergic drugs, morphine and morphine tolerance: a study in relation to nociception and gastrointestinal transit in mice.
    Neuropharmacology, 1983, Volume: 22, Issue:6

    Topics: Aminooxyacetic Acid; Analgesia; Animals; Baclofen; Bicuculline; Cyclohexanecarboxylic Acids; Digestion; Digestive System; Digestive System Physiological Phenomena; Drug Tolerance; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Morphine; Muscimol; Naloxone; Nociceptors; Oxazoles; Picrotoxin

1983
On the involvement of GABA in the analgesia produced by baclofen, muscimol and morphine.
    Neuropharmacology, 1982, Volume: 21, Issue:5

    Topics: 4-Aminobutyrate Transaminase; Analgesia; Analgesics; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Naloxone; Picrotoxin; Transaminases

1982
Pharmacological studies on the prolonged depressant effects of baclofen on lumbar dorsal horn units in the cat.
    Neuropharmacology, 1982, Volume: 21, Issue:11

    Topics: Animals; Baclofen; Bicuculline; Cats; Depression, Chemical; Drug Interactions; Electric Stimulation; Glycine; Muscimol; Naloxone; Nociceptors; Spinal Cord; Strychnine

1982
In vitro autoradiography of receptor-activated G proteins in rat brain by agonist-stimulated guanylyl 5'-[gamma-[35S]thio]-triphosphate binding.
    Proceedings of the National Academy of Sciences of the United States of America, 1995, Aug-01, Volume: 92, Issue:16

    Topics: Animals; Autoradiography; Baclofen; Benzoxazines; Brain; Cannabinoids; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA-B Receptor Agonists; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Male; Morpholines; Naloxone; Naphthalenes; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid, mu

1995
Estradiol-17 beta and mu-opioid peptides rapidly hyperpolarize GnRH neurons: a cellular mechanism of negative feedback?
    Endocrinology, 1995, Volume: 136, Issue:5

    Topics: Animals; Arcuate Nucleus of Hypothalamus; Baclofen; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Estradiol; Feedback; Female; Gonadotropin-Releasing Hormone; Guinea Pigs; Membrane Potentials; Naloxone; Neurons; Ovariectomy; Potassium Channels; Receptors, Opioid, mu; Tetrodotoxin

1995
Respiratory effects of baclofen and 3-aminopropylphosphinic acid in guinea-pigs.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Administration, Inhalation; Analysis of Variance; Animals; Baclofen; Bicuculline; Carbon Dioxide; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Guinea Pigs; Injections, Intraventricular; Injections, Subcutaneous; Male; Naloxone; Organophosphorus Compounds; Pulmonary Ventilation; Respiration; Tidal Volume

1995
Heterogeneity in presynaptic regulation of GABA release from hippocampal inhibitory neurons.
    Neuron, 1993, Volume: 11, Issue:6

    Topics: Analgesics; Animals; Baclofen; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Evoked Potentials; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Homeostasis; In Vitro Techniques; Male; Naloxone; Nerve Fibers; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Synapses

1993
Antinociceptive effect of smilaxin B administered intracerebroventricularly in the mouse.
    Planta medica, 1996, Volume: 62, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Cerebral Ventricles; Dizocilpine Maleate; Glycosides; Injections, Intraventricular; Injections, Spinal; Male; Methysergide; Mice; Mice, Inbred ICR; Muscimol; Naloxone; Pain; Sincalide; Spinal Cord; Spirostans; Yohimbine

1996
Local opioid withdrawal in rat single periaqueductal gray neurons in vitro.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1996, Nov-15, Volume: 16, Issue:22

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Adrenergic alpha-Agonists; Analgesics, Opioid; Animals; Baclofen; Bicuculline; Clonidine; Drug Tolerance; Electrophysiology; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Male; Membrane Potentials; Morphine; Naloxone; Narcotic Antagonists; Neurons; Organ Culture Techniques; Periaqueductal Gray; Potassium Channels; Rats; Rats, Sprague-Dawley; Sensitivity and Specificity; Substance Withdrawal Syndrome; Tetrodotoxin; Time Factors; Valine

1996
Opioid receptor-mediated control of acetylcholine release in human neocortex tissue.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetylcholine; Adolescent; Adult; Aged; Analgesics; Analysis of Variance; Baclofen; Cerebral Cortex; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; GABA Agonists; Humans; Male; Middle Aged; Muscimol; Naloxone; Naltrexone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid, delta; Tetrodotoxin

1996
Mu-opioid and GABA(B) receptors modulate different types of Ca2+ currents in rat nodose ganglion neurons.
    Neuroscience, 1998, Volume: 85, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analgesics, Opioid; Animals; Baclofen; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Calcium Channels, N-Type; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA Agonists; GABA Antagonists; Naloxone; Narcotic Antagonists; Nerve Tissue Proteins; Neurons; Nifedipine; Nodose Ganglion; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Patch-Clamp Techniques; Peptides; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Spider Venoms

1998
Mu opioids enhance mossy fiber synaptic transmission indirectly by reducing GABAB receptor activation.
    Brain research, 1999, Mar-13, Volume: 821, Issue:2

    Topics: Analgesics, Opioid; Animals; Baclofen; Bicuculline; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA Antagonists; Long-Term Potentiation; Male; Membrane Potentials; Mossy Fibers, Hippocampal; Naloxone; Narcotic Antagonists; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Somatostatin; Synaptic Transmission

1999
Tiagabine antinociception in rodents depends on GABA(B) receptor activation: parallel antinociception testing and medial thalamus GABA microdialysis.
    European journal of pharmacology, 1999, Mar-05, Volume: 368, Issue:2-3

    Topics: Abdomen; Animals; Baclofen; Constriction, Pathologic; Dose-Response Relationship, Drug; Escape Reaction; Extracellular Space; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Microdialysis; Naloxone; Narcotic Antagonists; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Nociceptors; Organophosphorus Compounds; Pain; Pain Measurement; Pain Threshold; Psychomotor Performance; Receptors, GABA-B; Thalamus; Tiagabine

1999
GABAB receptors are involved in the control of acute opiate withdrawal in isolated tissue.
    Progress in neuro-psychopharmacology & biological psychiatry, 1999, Volume: 23, Issue:2

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; GABA Agonists; GABA-B Receptor Antagonists; Guinea Pigs; In Vitro Techniques; Male; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Opioid-Related Disorders; Receptors, GABA-B; Substance Withdrawal Syndrome

1999
Effects of GABAergic system on naloxone-induced jumping in morphine-dependent mice.
    European journal of pharmacology, 1999, Sep-24, Volume: 381, Issue:2-3

    Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Mice; Morphine Dependence; Muscimol; Naloxone; Narcotic Antagonists; Organophosphorus Compounds; Picrotoxin; Substance Withdrawal Syndrome

1999
The effect of baclofen on spontaneous and evoked behavioural expression of experimental neuropathic chronic pain.
    Arquivos de neuro-psiquiatria, 1999, Volume: 57, Issue:3B

    Topics: Animals; Baclofen; Behavior, Animal; Chronic Disease; GABA Agonists; Male; Naloxone; Narcotic Antagonists; Pain; Peripheral Nervous System Diseases; Rats; Rats, Wistar; Sciatic Nerve

1999
Adenosine receptor expression and function in rat striatal cholinergic interneurons.
    British journal of pharmacology, 2000, Volume: 130, Issue:4

    Topics: Acetylcholine; Adenosine; Adenosine Deaminase; Animals; Baclofen; Bicuculline; Caffeine; Cholinergic Fibers; Corpus Striatum; Dose-Response Relationship, Drug; GABA Antagonists; Gene Expression; Male; Membrane Potentials; Naloxone; Narcotic Antagonists; Neurons; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; RNA, Messenger; Tritium; Xanthines

2000
GABA mechanisms and antinociception in mice with ligated sciatic nerve.
    Pharmacology & toxicology, 2001, Volume: 89, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA Antagonists; Ligation; Male; Mice; Mice, Inbred Strains; Morphine; Muscimol; Naloxone; Organophosphorus Compounds; Pain; Pain Measurement; Sciatic Nerve

2001
Attenuation of morphine withdrawal signs by the GABA(B) receptor agonist baclofen.
    Life sciences, 2001, Dec-14, Volume: 70, Issue:4

    Topics: Animals; Baclofen; Behavior, Animal; Drug Antagonism; Drug Combinations; GABA Agonists; GABA Antagonists; Male; Morphine Dependence; Naloxone; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome

2001
Baclofen prevents morphine withdrawal irrespective of seasonal variation.
    Behavioural pharmacology, 2002, Volume: 13, Issue:1

    Topics: Animals; Arousal; Baclofen; Female; Male; Mice; Morphine; Motor Activity; Naloxone; Narcotic Antagonists; Seasons; Substance Withdrawal Syndrome

2002
Quantitative stoichiometry of G-proteins activated by mu-opioid receptors in postmortem human brain.
    European journal of pharmacology, 2002, Sep-27, Volume: 452, Issue:1

    Topics: Alkylation; Analgesics, Opioid; Baclofen; Binding, Competitive; Brain Chemistry; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Inhibitors; Ethylmaleimide; GABA Agonists; GTP-Binding Protein Regulators; GTP-Binding Proteins; Humans; In Vitro Techniques; Kinetics; Membranes; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid, mu; Signal Transduction

2002
Antinociceptive mechanisms of platycodin D administered intracerebroventricularly in the mouse.
    Planta medica, 2002, Volume: 68, Issue:9

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Analgesics; Animals; Baclofen; Carbohydrate Sequence; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Injections, Intraventricular; Injections, Spinal; Male; Methysergide; Mice; Mice, Inbred ICR; Molecular Sequence Data; Muscimol; Naloxone; Narcotic Antagonists; Pain Measurement; Plant Extracts; Platycodon; Receptors, Cholecystokinin; Receptors, N-Methyl-D-Aspartate; Saponins; Serotonin Antagonists; Sincalide; Tail; Triterpenes; Yohimbine

2002
Baclofen reestablishes striatal and cortical dopamine concentrations during naloxone-precipitated withdrawal.
    Neurochemistry international, 2003, Volume: 42, Issue:4

    Topics: Animals; Baclofen; Cerebral Cortex; Chromatography, High Pressure Liquid; Dopamine; Electrochemistry; GABA Agonists; GABA-B Receptor Agonists; Hippocampus; Homovanillic Acid; Hydroxyindoleacetic Acid; Male; Mice; Morphine Dependence; Naloxone; Narcotic Antagonists; Neostriatum; Serotonin; Substance Withdrawal Syndrome

2003
Kavalactones and dihydrokavain modulate GABAergic activity in a rat gastric-brainstem preparation.
    Planta medica, 2002, Volume: 68, Issue:12

    Topics: Animals; Baclofen; Drug Interactions; GABA Agents; GABA Agonists; GABA Antagonists; Kava; Lactones; Muscimol; Naloxone; Narcotic Antagonists; Plant Extracts; Pyrones; Rats; Rats, Sprague-Dawley; Solitary Nucleus; Stomach

2002
Morphine-3-glucuronide's neuro-excitatory effects are mediated via indirect activation of N-methyl-D-aspartic acid receptors: mechanistic studies in embryonic cultured hippocampal neurones.
    Anesthesia and analgesia, 2003, Volume: 97, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aniline Compounds; Animals; Baclofen; Calcium; Calcium Channel Blockers; Cells, Cultured; Central Nervous System Stimulants; Cytosol; Excitatory Amino Acid Antagonists; Fluorescent Dyes; GABA Agonists; Hippocampus; Image Processing, Computer-Assisted; Immunohistochemistry; Microscopy, Fluorescence; Morphine Derivatives; Naloxone; Narcotic Antagonists; Neurons; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Tetrodotoxin; Xanthenes

2003
Baclofen pumps: comment on Anderson et al.
    Paediatric anaesthesia, 2003, Volume: 13, Issue:7

    Topics: Anti-Arrhythmia Agents; Atropine; Baclofen; Child; Coma; GABA Agonists; Humans; Infusion Pumps, Implantable; Morphine; Naloxone; Narcotic Antagonists; Oxygen; Postoperative Complications

2003
Baclofen reestablishes micro-opioid receptor levels modified by morphine withdrawal syndrome in either sex.
    Synapse (New York, N.Y.), 2004, Volume: 54, Issue:1

    Topics: Animals; Baclofen; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Female; GABA Agonists; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Receptors, Opioid, mu; Sex Factors; Substance Withdrawal Syndrome

2004
Ethanol-induced conditioned place preference is expressed through a ventral tegmental area dependent mechanism.
    Behavioral neuroscience, 2005, Volume: 119, Issue:1

    Topics: Animals; Baclofen; Central Nervous System Depressants; Conditioning, Classical; Ethanol; GABA Agonists; Male; Mice; Naloxone; Quaternary Ammonium Compounds; Receptors, GABA-B; Receptors, Opioid; Reinforcement, Psychology; Space Perception; Ventral Tegmental Area

2005
Baclofen-induced reduction of alcohol reinforcement in alcohol-preferring rats.
    Alcohol (Fayetteville, N.Y.), 2005, Volume: 36, Issue:3

    Topics: Alcohol Drinking; Animals; Baclofen; Central Nervous System Depressants; Conditioning, Operant; Dose-Response Relationship, Drug; Ethanol; GABA Agonists; Male; Naloxone; Narcotic Antagonists; Rats; Reinforcement, Psychology; Self Administration; Sucrose

2005
Behavioral and electrophysiological evidence for opioid tolerance in adolescent rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2007, Volume: 32, Issue:3

    Topics: Action Potentials; Age Factors; Animals; Baclofen; Behavior, Animal; Dose-Response Relationship, Drug; Drug Interactions; Drug Tolerance; Electrophysiology; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Agonists; Male; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Neurons; Pain Measurement; Pain Threshold; Periaqueductal Gray; Rats; Rats, Sprague-Dawley; Reaction Time

2007
Modulation of the cough reflex by antitussive agents within the caudal aspect of the nucleus tractus solitarii in the rabbit.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2008, Volume: 295, Issue:1

    Topics: Animals; Antitussive Agents; Baclofen; Cough; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Male; Naloxone; Neurokinin A; Organophosphorus Compounds; Peptide Fragments; Piperidines; Rabbits; Reflex; Solitary Nucleus

2008
Attenuation of morphine withdrawal signs by a GABAB receptor agonist in the locus coeruleus of rats.
    Behavioural brain research, 2009, Jan-03, Volume: 196, Issue:1

    Topics: Analysis of Variance; Animals; Baclofen; Dose-Response Relationship, Drug; Drug Therapy, Combination; GABA Agonists; GABA Antagonists; Injections, Subcutaneous; Locus Coeruleus; Male; Morphine; Morphine Dependence; Motor Activity; Naloxone; Narcotic Antagonists; Narcotics; Organophosphorus Compounds; Rats; Rats, Wistar; Substance Withdrawal Syndrome

2009
Naloxone and baclofen attenuate ethanol's locomotor-activating effects in preweanling Sprague-Dawley rats.
    Behavioral neuroscience, 2009, Volume: 123, Issue:1

    Topics: Analysis of Variance; Animals; Animals, Newborn; Baclofen; Central Nervous System Depressants; Dose-Response Relationship, Drug; Ethanol; GABA Agonists; Male; Motor Activity; Naloxone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley

2009
Analgesia induced by 2- or 100-Hz electroacupuncture in the rat tail-flick test depends on the activation of different descending pain inhibitory mechanisms.
    The journal of pain, 2011, Volume: 12, Issue:1

    Topics: Adjuvants, Anesthesia; Adrenergic alpha-Antagonists; Analgesia; Anesthetics, Intravenous; Animals; Atropine; Baclofen; Bicuculline; Biophysics; Dioxanes; Disease Models, Animal; Electroacupuncture; GABA Agents; Male; Methysergide; Models, Biological; Multivariate Analysis; Naloxone; Narcotic Antagonists; Pain; Pain Management; Pain Measurement; Rats; Rats, Wistar; Reaction Time; Serotonin Antagonists; Tail; Thiopental; Time Factors

2011
Baclofen did not modify sexually dimorphic c-Fos expression during morphine withdrawal syndrome.
    Synapse (New York, N.Y.), 2013, Volume: 67, Issue:3

    Topics: Animals; Baclofen; Female; GABA-B Receptor Agonists; Hippocampus; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Proto-Oncogene Proteins c-fos; Sex Factors; Substance Withdrawal Syndrome

2013
Attenuation by baclofen of nicotine rewarding properties and nicotine withdrawal manifestations.
    Psychopharmacology, 2014, Volume: 231, Issue:15

    Topics: Animals; Anxiety; Avoidance Learning; Baclofen; Conditioning, Psychological; GABA-B Receptor Agonists; Male; Mice; Movement; Naloxone; Narcotic Antagonists; Nicotine; Nicotinic Agonists; Receptors, GABA-B; Reward; Space Perception; Substance Withdrawal Syndrome; Tobacco Use Disorder

2014
Gabaergic and opioid receptors mediate the facilitation of NaCl intake induced by α₂-adrenergic activation in the lateral parabrachial nucleus.
    Behavioural brain research, 2015, Feb-01, Volume: 278

    Topics: Animals; Antihypertensive Agents; Baclofen; Bicuculline; Captopril; Enzyme Inhibitors; Furosemide; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; Imidazoles; Male; Naloxone; Narcotic Antagonists; Parabrachial Nucleus; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, GABA; Receptors, Opioid; Sodium Chloride; Sodium Potassium Chloride Symporter Inhibitors

2015
Opioid receptor-dependent sex differences in synaptic plasticity in the hippocampal mossy fiber pathway of the adult rat.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2015, Jan-28, Volume: 35, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Dendritic Spines; Estrous Cycle; Female; GABA-A Receptor Antagonists; Hippocampus; Long-Term Potentiation; Male; Mossy Fibers, Hippocampal; Naloxone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Opioid; Sex Characteristics; Somatostatin; Synapses

2015
Baclofen prevents the elevated plus maze behavior and BDNF expression during naloxone precipitated morphine withdrawal in male and female mice.
    Synapse (New York, N.Y.), 2016, Volume: 70, Issue:5

    Topics: Animals; Baclofen; Brain; Brain-Derived Neurotrophic Factor; Female; GABA-B Receptor Agonists; Male; Maze Learning; Mice; Morphine; Naloxone; Narcotic Antagonists; Sex Factors; Substance Withdrawal Syndrome

2016
Effects of Injection of Gamma-Aminobutyric Acid Agonists into the Nucleus Accumbens on Naloxone-Induced Morphine Withdrawal.
    Pharmacology, 2017, Volume: 100, Issue:3-4

    Topics: Animals; Baclofen; GABA Agonists; Injections; Locomotion; Male; Morphine Dependence; Muscimol; Naloxone; Narcotic Antagonists; Nucleus Accumbens; Rats, Sprague-Dawley; Substance Withdrawal Syndrome

2017
The mechanism of chronic nicotine exposure and nicotine withdrawal on pain perception in an animal model.
    Neuroscience letters, 2020, 01-10, Volume: 715

    Topics: Animals; Baclofen; Bicuculline; Disease Models, Animal; Down-Regulation; Endorphins; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hyperalgesia; Male; Naloxone; Nicotine; Pain Perception; Pain Threshold; Rats; Receptors, Opioid, mu; Spinal Cord; Substance Withdrawal Syndrome; Time Factors; Up-Regulation

2020