baclofen has been researched along with enkephalin, ala(2)-mephe(4)-gly(5)- in 50 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 24 (48.00) | 18.2507 |
2000's | 19 (38.00) | 29.6817 |
2010's | 6 (12.00) | 24.3611 |
2020's | 1 (2.00) | 2.80 |
Authors | Studies |
---|---|
Kelly, MJ; Loose, MD; Ronnekleiv, OK | 2 |
Dunwiddie, TV; Lupica, CR; Proctor, WR | 1 |
Alberch, J; Arenas, E; Marsal, J | 1 |
Childers, SR; Selley, DE; Sim, LJ | 1 |
Kelly, MJ; Lagrange, AH; Rønnekleiv, OK | 1 |
Narahashi, T; Nomura, K; Reuveny, E | 1 |
Kalivas, PW; Klitenick, MA | 1 |
Lambert, NA; Wilson, WA | 1 |
Churchill, L; Hooks, MS; Johnson, K; Kalivas, PW; Klitenick, MA | 1 |
Feldman, JL; Johnson, SM; Smith, JC | 1 |
Christie, MJ; Osborne, PB; Vaughan, CW; Wilson, HI | 1 |
Kelly, MJ; Lagrange, AH; Rønnekleiv, OK; Wagner, EJ | 1 |
Feuerstein, TJ; Gleichauf, O; Jackisch, R; Landwehrmeyer, GB; Peckys, D; Scheremet, R | 1 |
Avoli, M; Barbarosie, M; Köhling, R | 1 |
Kelly, MJ; Lagrange, AH; Rønnekleiv, OK; Wagner, EJ; Zhang, G | 1 |
Jan, LY; Lüscher, C; Malenka, RC; Nicoll, RA; Stoffel, M | 1 |
Grudt, TJ; Henderson, G | 1 |
Moises, HC; Rusin, KI | 1 |
Lupica, CR; Svoboda, KR | 1 |
Churchill, L; Kalivas, PW; Klitenick, MA | 1 |
Chavkin, C; Jin, W | 1 |
Christie, MJ; Connor, M; Pintar, JE; Schuller, A | 1 |
Dun, NJ; Hwang, BH; Mizoguchi, H; Nagase, H; Narita, M; Oji, DE; Tseng, LF | 1 |
Kelly, MJ; Reyes-Vazquez, C; Ronnekleiv, OK; Wagner, EJ | 1 |
Hayward, MD; Kelly, MJ; Low, MJ; Ronnekleiv, OK; Slugg, RM | 1 |
Duffy, P; Jackson, D; Kalivas, PW; Romanidies, A; Wyndham, L | 1 |
Bodnar, RJ; Christian, G; Echo, JA; Lamonte, N; Ragnauth, A; Znamensky, V | 1 |
Ackerman, TF; Bodnar, RJ; Echo, JA; Lamonte, N | 1 |
González-Maeso, J; Meana, JJ; Rodríguez-Puertas, R | 1 |
Bosch, MA; Ibrahim, N; Kelly, MJ; Low, MJ; Qiu, J; Rubinstein, M; Rønnekleiv, OK; Smart, JL | 1 |
Ackerman, TF; Bodnar, RJ; Lamonte, N | 1 |
Balerio, GN; Bonavita, CD; Diaz, SL; Kemmling, AK; Rubio, MC | 1 |
Melnick, IV; Safronov, BV; Santos, SF | 1 |
Avoli, M; D'Antuono, M; de Guzman, P; Kano, T | 1 |
Bagley, EE; Chieng, BC; Christie, MJ; Connor, M | 1 |
Antonelli, MC; Balerio, GN; Barros, VG; Diaz, SL; Rubio, MC | 1 |
Chiu, K; Evans, CJ; Kieffer, BL; Maidment, NT; Walwyn, WM; Wei, W; Xie, CW | 1 |
Hammond, DL; Jongeling, AC; Zhang, L | 1 |
Colón, J; Luján, R; Marker, CL; Wickman, K | 1 |
Castiglioni, AJ; Lipscombe, D; Raingo, J | 1 |
Bongianni, F; Cinelli, E; Fontana, GA; Mutolo, D; Pantaleo, T | 1 |
Cai, YQ; Pan, HL; Wu, ZZ | 1 |
Bongianni, F; Cinelli, E; Mutolo, D; Pantaleo, T | 1 |
Bourova, L; Dlouha, K; Kagan, D; Novotny, J; Svoboda, P; Vosahlikova, M | 1 |
Chen, W; Marvizón, JC; Zhang, G | 1 |
Ikeda, SR; Ono, F; Won, YJ | 1 |
Bailey, CP; Dewey, WL; Gabra, BH; Henderson, G; Hull, LC | 1 |
Du, X; Gamper, N; Huang, D; Huang, S; Peers, C; Zhang, H | 1 |
Carlson, HN; Christensen, BA; Pratt, WE | 1 |
50 other study(ies) available for baclofen and enkephalin, ala(2)-mephe(4)-gly(5)-
Article | Year |
---|---|
Estrogen suppresses mu-opioid- and GABAB-mediated hyperpolarization of hypothalamic arcuate neurons.
Topics: Animals; Arcuate Nucleus of Hypothalamus; Baclofen; beta-Endorphin; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Estradiol; Evoked Potentials; Female; gamma-Aminobutyric Acid; Guinea Pigs; Hypothalamus; In Vitro Techniques; Membrane Potentials; Neurons; Ovariectomy; Receptors, Opioid; Receptors, Opioid, mu; Tetrodotoxin | 1992 |
Dissociation of mu and delta opioid receptor-mediated reductions in evoked and spontaneous synaptic inhibition in the rat hippocampus in vitro.
Topics: 2-Amino-5-phosphonovalerate; Analgesics; Animals; Axons; Baclofen; Bicuculline; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Evoked Potentials; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Male; Neurons; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu; Synapses | 1992 |
Neurons in the rat arcuate nucleus are hyperpolarized by GABAB and mu-opioid receptor agonists: evidence for convergence at a ligand-gated potassium conductance.
Topics: Animals; Arcuate Nucleus of Hypothalamus; Baclofen; beta-Endorphin; Cell Polarity; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Female; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Opioid; Receptors, Opioid, mu | 1991 |
GABAA and GABAB antagonists prevent the opioid inhibition of endogenous acetylcholine release evoked by glutamate from rat neostriatal slices.
Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Corpus Striatum; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; GABA Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Morphine; Narcotics; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
In vitro autoradiography of receptor-activated G proteins in rat brain by agonist-stimulated guanylyl 5'-[gamma-[35S]thio]-triphosphate binding.
Topics: Animals; Autoradiography; Baclofen; Benzoxazines; Brain; Cannabinoids; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA-B Receptor Agonists; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Male; Morpholines; Naloxone; Naphthalenes; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid, mu | 1995 |
Estradiol-17 beta and mu-opioid peptides rapidly hyperpolarize GnRH neurons: a cellular mechanism of negative feedback?
Topics: Animals; Arcuate Nucleus of Hypothalamus; Baclofen; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Estradiol; Feedback; Female; Gonadotropin-Releasing Hormone; Guinea Pigs; Membrane Potentials; Naloxone; Neurons; Ovariectomy; Potassium Channels; Receptors, Opioid, mu; Tetrodotoxin | 1995 |
Opioid inhibition and desensitization of calcium channel currents in rat dorsal root ganglion neurons.
Topics: Analgesics; Animals; Baclofen; Calcium Channel Blockers; Cyclic AMP-Dependent Protein Kinases; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ganglia, Spinal; Guanosine 5'-O-(3-Thiotriphosphate); Neurons; Protein Kinase C; Rats; Rats, Sprague-Dawley | 1994 |
Behavioral and neurochemical studies of opioid effects in the pedunculopontine nucleus and mediodorsal thalamus.
Topics: Amino Acid Sequence; Animals; Baclofen; Behavior, Animal; Dopamine; Dorsomedial Hypothalamic Nucleus; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Extracellular Space; Haloperidol; Male; Microinjections; Molecular Sequence Data; Motor Activity; Nucleus Accumbens; Pons; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Synaptic Transmission; Ventral Tegmental Area | 1994 |
Heterogeneity in presynaptic regulation of GABA release from hippocampal inhibitory neurons.
Topics: Analgesics; Animals; Baclofen; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Evoked Potentials; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Homeostasis; In Vitro Techniques; Male; Naloxone; Nerve Fibers; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Synapses | 1993 |
Involvement of the ventral tegmental area in locomotion elicited from the nucleus accumbens or ventral pallidum.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Globus Pallidus; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Ventral Tegmental Area | 1996 |
Modulation of respiratory rhythm in vitro: role of Gi/o protein-mediated mechanisms.
Topics: Analgesics; Animals; Baclofen; Clonidine; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; gamma-Aminobutyric Acid; GTP-Binding Proteins; In Vitro Techniques; Rats; Respiration; Serotonin | 1996 |
Opioid inhibition of rat periaqueductal grey neurones with identified projections to rostral ventromedial medulla in vitro.
Topics: Analgesics; Animals; Baclofen; Brain; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Methionine; Enkephalins; Fluorescent Dyes; GABA Agonists; In Vitro Techniques; Microspheres; Narcotics; Neurons; Patch-Clamp Techniques; Periaqueductal Gray; Rats; Rats, Sprague-Dawley; Rhodamines | 1996 |
Estrogen rapidly attenuates a GABAB response in hypothalamic neurons.
Topics: Animals; Baclofen; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Estradiol; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Hypothalamus; Neurons; Potassium Channels; Receptors, GABA; Receptors, Opioid, mu | 1996 |
Opioid receptor-mediated control of acetylcholine release in human neocortex tissue.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetylcholine; Adolescent; Adult; Aged; Analgesics; Analysis of Variance; Baclofen; Cerebral Cortex; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; GABA Agonists; Humans; Male; Middle Aged; Muscimol; Naloxone; Naltrexone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid, delta; Tetrodotoxin | 1996 |
Anoxia blocks the presynaptic control of GABA release at inhibitory terminals in the rat hippocampus.
Topics: 4-Aminopyridine; 6-Cyano-7-nitroquinoxaline-2,3-dione; Analgesics; Animals; Baclofen; Cell Hypoxia; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Evoked Potentials; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hippocampus; Interneurons; Male; Neurons; Rats; Rats, Sprague-Dawley; Synapses; Synaptic Transmission | 1996 |
Tolerance to mu-opioid receptor agonists but not cross-tolerance to gamma-aminobutyric acid(B) receptor agonists in arcuate A12 dopamine neurons with chronic morphine treatment.
Topics: Animals; Arcuate Nucleus of Hypothalamus; Baclofen; Drug Tolerance; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Female; GABA-B Receptor Agonists; Guinea Pigs; Hypothalamus; In Vitro Techniques; Membrane Potentials; Morphine; Morphine Dependence; Neurons; Receptors, Opioid, mu; Tetrodotoxin; Tyrosine 3-Monooxygenase | 1997 |
G protein-coupled inwardly rectifying K+ channels (GIRKs) mediate postsynaptic but not presynaptic transmitter actions in hippocampal neurons.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analgesics; Animals; Baclofen; Down-Regulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Excitatory Amino Acid Antagonists; Female; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Agonists; GTP-Binding Proteins; Hippocampus; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Potassium Channels; Potassium Channels, Inwardly Rectifying; Presynaptic Terminals; Pyramidal Cells; Receptors, Adrenergic, alpha-1; Receptors, GABA-B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Synaptic Membranes; Transcription, Genetic | 1997 |
Glycine and GABAA receptor-mediated synaptic transmission in rat substantia gelatinosa: inhibition by mu-opioid and GABAB agonists.
Topics: Analgesics, Opioid; Animals; Baclofen; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Excitatory Postsynaptic Potentials; Female; GABA Agents; GABA Antagonists; GABA-B Receptor Agonists; Glycine Agents; In Vitro Techniques; Male; Membrane Potentials; Narcotic Antagonists; Patch-Clamp Techniques; Peptide Fragments; Peptides; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Glycine; Receptors, Opioid, mu; Somatostatin; Strychnine; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin | 1998 |
Mu-opioid and GABA(B) receptors modulate different types of Ca2+ currents in rat nodose ganglion neurons.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analgesics, Opioid; Animals; Baclofen; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Calcium Channels, N-Type; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA Agonists; GABA Antagonists; Naloxone; Narcotic Antagonists; Nerve Tissue Proteins; Neurons; Nifedipine; Nodose Ganglion; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Patch-Clamp Techniques; Peptides; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Spider Venoms | 1998 |
Opioid inhibition of hippocampal interneurons via modulation of potassium and hyperpolarization-activated cation (Ih) currents.
Topics: Analgesics; Analgesics, Opioid; Animals; Baclofen; Barium; Cardiovascular Agents; Cations; Cell Size; Cells, Cultured; Cesium; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; GABA Agonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hippocampus; Interneurons; Male; Membrane Potentials; Potassium; Potassium Channels; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu | 1998 |
Dopamine depletion reorganizes projections from the nucleus accumbens and ventral pallidum that mediate opioid-induced motor activity.
Topics: Analgesics, Opioid; Animals; Baclofen; Dopamine; Dopamine Antagonists; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fluphenazine; GABA Agonists; Globus Pallidus; Locomotion; Male; Microinjections; Motor Activity; Motor Neurons; Muscimol; Neural Pathways; Nucleus Accumbens; Oxidopamine; Rats; Rats, Sprague-Dawley; Sympatholytics | 1998 |
Mu opioids enhance mossy fiber synaptic transmission indirectly by reducing GABAB receptor activation.
Topics: Analgesics, Opioid; Animals; Baclofen; Bicuculline; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA Antagonists; Long-Term Potentiation; Male; Membrane Potentials; Mossy Fibers, Hippocampal; Naloxone; Narcotic Antagonists; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Somatostatin; Synaptic Transmission | 1999 |
Mu-opioid receptor modulation of calcium channel current in periaqueductal grey neurons from C57B16/J mice and mutant mice lacking MOR-1.
Topics: Animals; Baclofen; Calcium Channels; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Oligopeptides; Periaqueductal Gray; Receptors, Opioid, mu | 1999 |
Identification of the G-protein-coupled ORL1 receptor in the mouse spinal cord by [35S]-GTPgammaS binding and immunohistochemistry.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Atropine; Autoradiography; Baclofen; Binding, Competitive; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Haloperidol; Immunohistochemistry; In Vitro Techniques; Male; Membranes; Mice; Mice, Inbred ICR; Naltrexone; Narcotic Antagonists; Nociceptin; Nociceptin Receptor; Opioid Peptides; Peptide Fragments; Propranolol; Receptors, Opioid; Somatostatin; Spinal Cord; Sulfur Radioisotopes; Yohimbine | 1999 |
The role of intrinsic and agonist-activated conductances in determining the firing patterns of preoptic area neurons in the guinea pig.
Topics: 4-Aminopyridine; Action Potentials; Animals; Baclofen; Barium Compounds; Cesium; Chlorides; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Excitatory Amino Acid Agonists; Female; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Neurons; Nickel; Ovariectomy; Patch-Clamp Techniques; Potassium Channels; Preoptic Area; Pyrimidines; Reaction Time; Tetrodotoxin | 2000 |
Effect of the mu-opioid agonist DAMGO on medial basal hypothalamic neurons in beta-endorphin knockout mice.
Topics: Animals; Baclofen; beta-Endorphin; Dose-Response Relationship, Drug; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Female; GABA Agonists; Hypothalamus, Middle; Mice; Mice, Knockout; Neurons; Potassium Channels; Pro-Opiomelanocortin; Receptors, Opioid, mu; Reference Values | 2000 |
Involvement of pallidothalamic circuitry in working memory.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analgesics, Opioid; Animals; Baclofen; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Excitatory Amino Acid Agonists; Extracellular Space; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Maze Learning; Mediodorsal Thalamic Nucleus; Memory, Short-Term; Motor Activity; Neural Inhibition; Neural Pathways; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, GABA-B; Receptors, Opioid, mu | 2001 |
gamma-Aminobutyric acid receptor subtype antagonists differentially alter opioid-induced feeding in the shell region of the nucleus accumbens in rats.
Topics: Animals; Baclofen; Bicuculline; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Naltrexone; Narcotic Antagonists; Narcotics; Neurons; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Receptors, Opioid | 2001 |
Alterations in food intake elicited by GABA and opioid agonists and antagonists administered into the ventral tegmental area region of rats.
Topics: Administration, Oral; Analgesics, Opioid; Animals; Baclofen; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Food Preferences; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Microinjections; Muscimol; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Receptors, Opioid, mu; Ventral Tegmental Area | 2002 |
Quantitative stoichiometry of G-proteins activated by mu-opioid receptors in postmortem human brain.
Topics: Alkylation; Analgesics, Opioid; Baclofen; Binding, Competitive; Brain Chemistry; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Inhibitors; Ethylmaleimide; GABA Agonists; GTP-Binding Protein Regulators; GTP-Binding Proteins; Humans; In Vitro Techniques; Kinetics; Membranes; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid, mu; Signal Transduction | 2002 |
Hypothalamic proopiomelanocortin neurons are glucose responsive and express K(ATP) channels.
Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Antihypertensive Agents; ATP-Binding Cassette Transporters; Baclofen; Diazoxide; Electric Conductivity; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Female; GABA Agonists; GABA-B Receptor Agonists; Glucose; Green Fluorescent Proteins; Hypothalamus; Indicators and Reagents; Luminescent Proteins; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Neurons; Patch-Clamp Techniques; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pro-Opiomelanocortin; Receptors, Drug; Receptors, GABA-B; Receptors, Opioid, mu; RNA, Messenger; Sulfonylurea Receptors | 2003 |
Lack of intersite GABA receptor subtype antagonist effects upon mu opioid receptor agonist-induced feeding elicited from either the ventral tegmental area or nucleus accumbens shell in rats.
Topics: Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Male; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Tegmentum Mesencephali | 2003 |
Baclofen reestablishes micro-opioid receptor levels modified by morphine withdrawal syndrome in either sex.
Topics: Animals; Baclofen; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Female; GABA Agonists; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Receptors, Opioid, mu; Sex Factors; Substance Withdrawal Syndrome | 2004 |
Selective postsynaptic inhibition of tonic-firing neurons in substantia gelatinosa by mu-opioid agonist.
Topics: Analgesics, Opioid; Animals; Baclofen; Barium; Cell Shape; Cesium; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Evoked Potentials; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Agonists; In Vitro Techniques; Interneurons; Neurons; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Opioid, mu; Receptors, Presynaptic; Substantia Gelatinosa | 2004 |
Ripple activity in the dentate gyrus of dishinibited hippocampus-entorhinal cortex slices.
Topics: Analgesics, Opioid; Animals; Anti-Ulcer Agents; Baclofen; Carbenoxolone; Cell Communication; Cortical Synchronization; Dentate Gyrus; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Entorhinal Cortex; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Gap Junctions; Hippocampus; Mice; Octanols; Organ Culture Techniques; Picrotoxin; Receptors, Neurotransmitter | 2005 |
Opioid tolerance in periaqueductal gray neurons isolated from mice chronically treated with morphine.
Topics: Analgesics, Opioid; Animals; Baclofen; Calcium Channels; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GABA Agonists; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Morphine; Neurons; Pain Measurement; Periaqueductal Gray; Receptors, Opioid, mu | 2005 |
Morphine withdrawal syndrome and its prevention with baclofen: Autoradiographic study of mu-opioid receptors in prepubertal male and female mice.
Topics: Aging; Animals; Autoradiography; Baclofen; Binding Sites; Brain; Disease Models, Animal; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Female; GABA Agonists; Male; Mice; Morphine; Morphine Dependence; Narcotic Antagonists; Narcotics; Receptors, Opioid, mu; Sex Characteristics; Substance Withdrawal Syndrome | 2006 |
Mu opioid receptor-effector coupling and trafficking in dorsal root ganglia neurons.
Topics: Analgesics, Opioid; Analysis of Variance; Animals; Animals, Newborn; Baclofen; Cells, Cultured; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Flow Cytometry; GABA Agonists; Ganglia, Spinal; Membrane Potentials; Mice; Mice, Knockout; Morphine; Neurons; Patch-Clamp Techniques; Protein Transport; Receptors, Opioid, mu; Time Factors; Transfection | 2006 |
Suitability of the retrograde tracer Dil for electrophysiological studies of brainstem neurons: adverse ramifications for G-protein coupled receptor agonists.
Topics: Amino Acids; Analysis of Variance; Animals; Animals, Newborn; Baclofen; Brain Stem; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Immunohistochemistry; In Vitro Techniques; Male; Membrane Potentials; Neurons; Neurotransmitter Agents; Patch-Clamp Techniques; Rats; Receptors, G-Protein-Coupled; Statistics, Nonparametric; Tryptophan Hydroxylase | 2007 |
Distinct populations of spinal cord lamina II interneurons expressing G-protein-gated potassium channels.
Topics: Analgesics, Opioid; Analysis of Variance; Animals; Baclofen; Blotting, Western; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Agonists; Immunohistochemistry; Immunoprecipitation; In Vitro Techniques; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Microscopy, Immunoelectron; Organophosphorus Compounds; Receptors, GABA; Receptors, Opioid, mu; Spinal Cord; Synapses | 2006 |
Alternative splicing controls G protein-dependent inhibition of N-type calcium channels in nociceptors.
Topics: Alternative Splicing; Analgesics, Opioid; Animals; Baclofen; Calcium; Calcium Channels, N-Type; Cell Line; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Inhibitors; Exons; GABA Agonists; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Membrane Potentials; Molecular Sequence Data; Neural Inhibition; Nociceptors; Patch-Clamp Techniques; Rats; Transfection | 2007 |
Modulation of the cough reflex by antitussive agents within the caudal aspect of the nucleus tractus solitarii in the rabbit.
Topics: Animals; Antitussive Agents; Baclofen; Cough; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Male; Naloxone; Neurokinin A; Organophosphorus Compounds; Peptide Fragments; Piperidines; Rabbits; Reflex; Solitary Nucleus | 2008 |
A functional link between T-type calcium channels and mu-opioid receptor expression in adult primary sensory neurons.
Topics: Analgesics, Opioid; Animals; Baclofen; Biophysics; Calcium Channel Blockers; Calcium Channels, T-Type; Capsaicin; Cells, Cultured; Drug Interactions; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GABA Agonists; Ganglia, Spinal; Gene Expression; Guanosine 5'-O-(3-Thiotriphosphate); Lectins; Male; Membrane Potentials; omega-Conotoxin GVIA; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Sensory Receptor Cells | 2009 |
Depression of cough reflex by microinjections of antitussive agents into caudal ventral respiratory group of the rabbit.
Topics: Abdominal Muscles; Animals; Antitussive Agents; Baclofen; Cough; Diaphragm; Electromyography; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Hemodynamics; Male; Microinjections; Neurokinin A; Peptide Fragments; Phrenic Nerve; Physical Stimulation; Piperidines; Rabbits; Reflex; Respiratory Center; Respiratory Mechanics; Solitary Nucleus | 2010 |
Long-term adaptation to high doses of morphine causes desensitization of mu-OR- and delta-OR-stimulated G-protein response in forebrain cortex but does not decrease the amount of G-protein alpha subunits.
Topics: Adaptation, Physiological; Animals; Baclofen; Behavior, Animal; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GTP-Binding Protein alpha Subunits; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Male; Morphine; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, mu; Substance Withdrawal Syndrome; Time Factors | 2010 |
Src family kinases mediate the inhibition of substance P release in the rat spinal cord by μ-opioid receptors and GABA(B) receptors, but not α2 adrenergic receptors.
Topics: Animals; Baclofen; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Male; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, GABA-B; Receptors, Opioid, mu; Spinal Cord; src-Family Kinases; Substance P | 2010 |
Identification and modulation of voltage-gated Ca2+ currents in zebrafish Rohon-Beard neurons.
Topics: Animals; Animals, Genetically Modified; Baclofen; Calcium Channels; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; gamma-Aminobutyric Acid; Green Fluorescent Proteins; Models, Animal; Neurotransmitter Agents; Patch-Clamp Techniques; Sensory Receptor Cells; Zebrafish | 2011 |
Reversal of morphine analgesic tolerance by ethanol in the mouse.
Topics: Analgesics, Opioid; Animals; Baclofen; Bicuculline; Central Nervous System Depressants; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Ethanol; GABA Antagonists; Hypnotics and Sedatives; Immersion; Injections, Intraventricular; Male; Mice; Morphine; Pain Measurement; Receptors, GABA-A; Receptors, GABA-B | 2013 |
GABAB receptors inhibit low-voltage activated and high-voltage activated Ca(2+) channels in sensory neurons via distinct mechanisms.
Topics: Animals; Baclofen; Calcium Channels, L-Type; Calcium Channels, N-Type; Calcium Channels, T-Type; Dithiothreitol; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Guanosine Diphosphate; HEK293 Cells; Humans; Nociception; Pain; Patch-Clamp Techniques; Pertussis Toxin; Primary Cell Culture; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Sensory Receptor Cells; Signal Transduction; Thionucleotides | 2015 |
Stimulation of mu opioid, but not GABAergic, receptors of the lateral habenula alters free feeding in rats.
Topics: Analgesics, Opioid; Animals; Baclofen; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Feeding Behavior; GABA Agonists; Habenula; Locomotion; Male; Motivation; Muscimol; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, Opioid, mu | 2022 |