baclofen has been researched along with colforsin in 34 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (23.53) | 18.7374 |
1990's | 13 (38.24) | 18.2507 |
2000's | 12 (35.29) | 29.6817 |
2010's | 1 (2.94) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
de Koning, HP; Huchedé, B; Jenks, BG; Roubos, EW | 1 |
Kamatchi, GL; Ticku, MK | 1 |
Wojcik, WJ; Xu, J | 1 |
Dolphin, AC; McGuirk, SM; Scott, RH | 1 |
Costa, E; Paez, X; Ulivi, M; Wojcik, WJ | 1 |
Boar, BR; Cross, AJ; Green, AR; Robinson, TN; Toczek, JM | 1 |
Hill, DR | 1 |
Barbaccia, ML; Costa, E; Szekely, AM | 1 |
Enna, SJ; Ferkany, JW; Scherer, RW | 1 |
Desrues, L; Lamacz, M; Tonon, MC; Vaudry, H | 1 |
Fisone, G; Greengard, P; Snyder, GL | 1 |
Bowery, NG; Malcangio, M | 1 |
González, MP; Oset-Gasque, MJ; Parramón, M | 1 |
Andrade, R | 1 |
Bowery, NG; Knight, AR | 1 |
Itoh, Y; Kimura, K; Oka, M; Shimidzu, T; Ukai, Y; Yoshikuni, Y | 1 |
Hashimoto, T; Kuriyama, K | 1 |
Olianas, MC; Onali, P | 1 |
Barilà, B; Cupello, A; Robello, M | 1 |
Bao, GB; Ma, L; Pei, G; Pu, L | 1 |
Snead, OC | 1 |
Beltrán-Parrazal, L; Clapp, C; Martínez de la Escalera, G; Noris, G | 1 |
Becú-Villalobos, D; Bianchi, M; Chamson-Reig, A; Libertun, C; Lux-Lantos, V; Pignataro, O; Rey-Roldán, E | 1 |
Gómez-Villafuertes, R; Gualix, J; Miras-Portugal, MT; Pintor, J | 1 |
Mascia, FM; Olianas, MC; Onali, P | 1 |
Ballabio, M; Cavarretta, IT; Froestl, W; Lambert, JJ; Magnaghi, V; Melcangi, RC; Zucchi, I | 1 |
Harvey, VL; Stephens, GJ | 1 |
Novotny, J; Stöhr, J; Svoboda, P | 1 |
Ivenshitz, M; Segal, M | 1 |
Desrayaud, S; Gjoni, T; Imobersteg, S; Urwyler, S | 1 |
Fujita, T; Oka, M; Wada, M; Wu, Q; Yamamoto, A | 1 |
Di Prisco, S; Grilli, M; Marchi, M; Pittaluga, A; Summa, M; Usai, C | 1 |
34 other study(ies) available for baclofen and colforsin
Article | Year |
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[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Dynamics of cyclic-AMP efflux in relation to alpha-MSH secretion from melanotrope cells of Xenopus laevis.
Topics: 1-Methyl-3-isobutylxanthine; alpha-MSH; Amphibian Proteins; Animals; Baclofen; Calcium; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; Dopamine; In Vitro Techniques; Peptide Hormones; Peptides; Pituitary Gland; Xenopus laevis | 1992 |
GABAB receptor activation inhibits Ca2(+)-activated 86Rb-efflux in cultured spinal cord neurons via G-protein mechanism.
Topics: Adenylate Cyclase Toxin; Animals; Baclofen; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; GTP-Binding Proteins; Mice; Mice, Inbred C57BL; Pertussis Toxin; Receptors, GABA-A; Rubidium Radioisotopes; Spinal Cord; Virulence Factors, Bordetella | 1990 |
Gamma aminobutyric acid B receptor-mediated inhibition of adenylate cyclase in cultured cerebellar granule cells: blockade by islet-activating protein.
Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Animals; Autoradiography; Baclofen; Bicuculline; Cerebellum; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Pertussis Toxin; Rats; Receptors, GABA-A; Time Factors; Virulence Factors, Bordetella | 1986 |
An investigation into the mechanisms of inhibition of calcium channel currents in cultured sensory neurones of the rat by guanine nucleotide analogues and (-)-baclofen.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Baclofen; Calcium Channels; Cells, Cultured; Cholera Toxin; Colforsin; Culture Techniques; Electrophysiology; Enzyme Activation; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Neurons, Afferent; Protein Kinase C; Rats; Thionucleotides; Type C Phospholipases | 1989 |
Islet-activating protein inhibits the beta-adrenergic receptor facilitation elicited by gamma-aminobutyric acidB receptors.
Topics: Adenosine Diphosphate Ribose; Animals; Baclofen; Cerebral Cortex; Colforsin; Cyclic AMP; Drug Synergism; GTP-Binding Proteins; Hippocampus; Isoproterenol; Male; Pertussis Toxin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, GABA-A; Virulence Factors, Bordetella | 1989 |
Effects of the putative antagonists phaclofen and delta-aminovaleric acid on GABAB receptor biochemistry.
Topics: Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Cerebral Cortex; Colforsin; Cyclic AMP; In Vitro Techniques; Isoproterenol; Kinetics; Male; Proteins; Radioligand Assay; Rats; Receptors, GABA-A | 1989 |
GABAB receptor modulation of adenylate cyclase activity in rat brain slices.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Baclofen; Brain; Cerebral Cortex; Colforsin; Cyclic AMP; Diterpenes; gamma-Aminobutyric Acid; In Vitro Techniques; Nipecotic Acids; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Effect of a protracted antidepressant treatment on signal transduction and [3H](-)-baclofen binding at GABAB receptors.
Topics: Adenylyl Cyclases; Animals; Anthracenes; Baclofen; Cerebral Cortex; Colforsin; Desipramine; Drug Administration Schedule; Imipramine; Injections, Intraperitoneal; Kinetics; Male; Maprotiline; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
Evidence for pharmacologically distinct subsets of GABAB receptors.
Topics: Animals; Baclofen; Binding, Competitive; Colforsin; Cyclic AMP; In Vitro Techniques; Isoproterenol; Male; Propylamines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Mechanism of action of gamma-aminobutyric acid on frog melanotrophs.
Topics: Adenylyl Cyclases; Animals; Baclofen; Calcium; Calcium Channels; Colforsin; Cyclic AMP; GABA-A Receptor Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Inositol Phosphates; Male; Melanocyte-Stimulating Hormones; Models, Biological; Pituitary Gland, Posterior; Rana ridibunda; Receptors, GABA-A; Receptors, GABA-B; Signal Transduction; Taurine | 1995 |
Phosphorylation of DARPP-32 is regulated by GABA in rat striatum and substantia nigra.
Topics: Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine and cAMP-Regulated Phosphoprotein 32; GABA Antagonists; gamma-Aminobutyric Acid; Male; Nerve Tissue Proteins; Phosphoproteins; Phosphorylation; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Nigra | 1994 |
GABAB receptor-mediated inhibition of forskolin-stimulated cyclic AMP accumulation in rat spinal cord.
Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Capsaicin; Colforsin; Cyclic AMP; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Norepinephrine; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Cord | 1993 |
GABAB receptors modulate catecholamine secretion in chromaffin cells by a mechanism involving cyclic AMP formation.
Topics: Adenylate Cyclase Toxin; Animals; Baclofen; Calcium; Catecholamines; Cattle; Cells, Cultured; Cholera Toxin; Chromaffin Granules; Colforsin; Cyclic AMP; Organophosphorus Compounds; Pertussis Toxin; Receptors, GABA-B; Virulence Factors, Bordetella | 1993 |
Enhancement of beta-adrenergic responses by Gi-linked receptors in rat hippocampus.
Topics: Adenylyl Cyclases; Animals; Baclofen; Colforsin; Electric Conductivity; Electrophysiology; GTP-Binding Proteins; Hippocampus; Male; Norepinephrine; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, GABA-A; Receptors, Serotonin | 1993 |
The pharmacology of adenylyl cyclase modulation by GABAB receptors in rat brain slices.
Topics: Adenylyl Cyclases; Animals; Baclofen; Brain; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Male; Norepinephrine; Rats; Rats, Wistar; Receptors, GABA-B | 1996 |
Involvement of metabotropic glutamate receptors in Gi- and Gs-dependent modulation of adenylate cyclase activity induced by a novel cognition enhancer NS-105 in rat brain.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic alpha-Agonists; Alanine; Animals; Baclofen; Brimonidine Tartrate; Cell Membrane; Cerebral Cortex; Cholera Toxin; Cognition; Colforsin; Cyclic AMP; Cycloleucine; Excitatory Amino Acid Antagonists; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Isoproterenol; Kinetics; Male; Manganese; Pertussis Toxin; Piperidines; Proline; Quinoxalines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, Neurotransmitter; Virulence Factors, Bordetella; Yohimbine | 1997 |
In vivo evidence that GABA(B) receptors are negatively coupled to adenylate cyclase in rat striatum.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Isoproterenol; Locomotion; Male; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Signal Transduction | 1997 |
GABA(B) receptor-mediated stimulation of adenylyl cyclase activity in membranes of rat olfactory bulb.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Baclofen; Calcium; Calmodulin; Colforsin; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Indomethacin; Injections, Intraventricular; Male; Membranes; Neuropeptides; Neuroprotective Agents; Olfactory Bulb; Organophosphorus Compounds; Pertussis Toxin; Phosphinic Acids; Phospholipases A; Phospholipids; Pituitary Adenylate Cyclase-Activating Polypeptide; Propanolamines; Propylamines; Quinacrine; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Transducin; Virulence Factors, Bordetella | 1999 |
GABA(B) receptor activation protects GABA(A) receptor from cyclic AMP-dependent down-regulation in rat cerebellar granule cells.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Baclofen; Cerebellar Cortex; Chloride Channels; Colforsin; Cyclic AMP; Down-Regulation; Enzyme Activation; GABA Agonists; Ion Channel Gating; Ion Transport; Muscimol; Nerve Tissue Proteins; Patch-Clamp Techniques; Pertussis Toxin; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Signal Transduction; Virulence Factors, Bordetella | 1999 |
Acute desensitization of nociceptin/orphanin FQ inhibition of voltage-gated calcium channels in freshly dissociated hippocampal neurons.
Topics: Animals; Baclofen; Barium; Calcium; Calcium Channel Blockers; Calcium Channels, P-Type; Carcinogens; Cells, Cultured; Colforsin; Electrophysiology; Extracellular Space; GABA Agonists; Hippocampus; Ion Channel Gating; Membrane Potentials; Nociceptin; Opioid Peptides; Patch-Clamp Techniques; Peptide Fragments; Protein Kinase C; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate; Tetrodotoxin | 1999 |
Evidence for a G protein-coupled gamma-hydroxybutyric acid receptor.
Topics: Adenylyl Cyclases; Animals; Baclofen; Brain; Brain Chemistry; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Female; GABA Agonists; GTP Phosphohydrolases; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Male; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, Presynaptic; Sodium Oxybate; Subcellular Fractions | 2000 |
GABA inhibition of immortalized gonadotropin-releasing hormone neuronal excitability involves GABA(A) receptors negatively coupled to cyclic adenosine monophosphate formation.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Baclofen; Bicuculline; Calcium; Calcium Channels; Cell Line, Transformed; Cell Membrane; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Kinetics; Muscimol; Neurons; Potassium; Receptors, GABA-A | 2001 |
GABA(B) receptors in anterior pituitary cells. Mechanism of action coupled to endocrine effects.
Topics: Animals; Baclofen; Barium Compounds; Calcium; Calcium Channel Blockers; Cells, Cultured; Chlorides; Colforsin; Cyclic AMP; Dopamine; Female; Luteinizing Hormone; Pertussis Toxin; Pituitary Gland, Anterior; Potassium Channel Blockers; Potassium Chloride; Proestrus; Prolactin; Rats; Receptors, GABA-B; Tetraethylammonium; Thyrotropin-Releasing Hormone; Virulence Factors, Bordetella | 2001 |
GABAB receptor-mediated presynaptic potentiation of ATP ionotropic receptors in rat midbrain synaptosomes.
Topics: Adenosine Triphosphate; Animals; Baclofen; Calcium; Colforsin; Competitive Bidding; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Fura-2; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Immunohistochemistry; In Vitro Techniques; Mesencephalon; Muscimol; Nerve Tissue Proteins; Picrotoxin; Rats; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X; Synaptosomes; Time Factors | 2003 |
Positive regulation of GABA(B) receptors dually coupled to cyclic AMP by the allosteric agent CGP7930.
Topics: Adenylyl Cyclases; Allosteric Regulation; Animals; Baclofen; Calmodulin; Colforsin; Corpus Striatum; Corticotropin-Releasing Hormone; Cyclic AMP; Cytoplasmic Granules; Drug Synergism; Frontal Lobe; gamma-Aminobutyric Acid; Gene Expression; Male; Olfactory Bulb; Phenols; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-B; Signal Transduction | 2003 |
GABAB receptors in Schwann cells influence proliferation and myelin protein expression.
Topics: Animals; Baclofen; Blotting, Northern; Blotting, Western; Bromodeoxyuridine; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA Antagonists; Hypoxanthine Phosphoribosyltransferase; Immunohistochemistry; Indoles; Membrane Proteins; Myelin Proteins; Protein Isoforms; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Schwann Cells; Sciatic Nerve; Tetrazolium Salts; Time Factors | 2004 |
Mechanism of GABA receptor-mediated inhibition of spontaneous GABA release onto cerebellar Purkinje cells.
Topics: Action Potentials; Age Factors; Animals; Baclofen; Barium; Cadmium; Calcium; Cerebellum; Colforsin; Drug Interactions; Enzyme Inhibitors; Exotoxins; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Neural Inhibition; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Purkinje Cells; Receptors, GABA-A; Ruthenium Red; Synaptic Transmission; Tetrodotoxin | 2004 |
Characterization of [3H]-forskolin binding sites in young and adult rat brain cortex: identification of suramin as a competitive inhibitor of [3H]-forskolin binding.
Topics: Adrenergic beta-Agonists; Aging; Animals; Baclofen; Binding, Competitive; Cell Membrane; Cerebral Cortex; Colforsin; GABA Agonists; Guanylyl Imidodiphosphate; Isoproterenol; Magnesium; Male; Rats; Rats, Wistar; Receptors, Drug; Suramin | 2005 |
Simultaneous NMDA-dependent long-term potentiation of EPSCs and long-term depression of IPSCs in cultured rat hippocampal neurons.
Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Evoked Potentials; Hippocampus; Long-Term Potentiation; Long-Term Synaptic Depression; Neuronal Plasticity; Neurons; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Quinoxalines; Rats; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Tetrodotoxin; Thionucleotides; Time Factors | 2006 |
The positive allosteric modulator GS39783 enhances GABA(B) receptor-mediated inhibition of cyclic AMP formation in rat striatum in vivo.
Topics: Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; Cyclopentanes; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA Antagonists; Male; Microdialysis; Phosphinic Acids; Pyrimidines; Radioimmunoassay; Rats; Rats, Wistar; Receptors, GABA-A; Time Factors | 2006 |
Functional expression of metabotropic GABAB receptors in primary cultures of astrocytes from rat cerebral cortex.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Astrocytes; Baclofen; Cell Membrane; Cells, Cultured; Cerebral Cortex; Colforsin; Gene Expression Regulation; Guanosine Triphosphate; Rats; Receptors, GABA-B; RNA, Messenger | 2006 |
Presynaptic mGlu7 receptors control GABA release in mouse hippocampus.
Topics: Adenylyl Cyclase Inhibitors; Aminobutyrates; Animals; Baclofen; Benzhydryl Compounds; Benzoates; Benzylamines; Colforsin; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Exocytosis; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; Imines; Mice; Phosphinic Acids; Potassium Chloride; Pyridones; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Synaptosomes; Syntaxin 1; Vesicular Inhibitory Amino Acid Transport Proteins | 2013 |