baclofen and cgp 55845a

baclofen has been researched along with cgp 55845a in 64 studies

Research

Studies (64)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's26 (40.63)18.2507
2000's30 (46.88)29.6817
2010's8 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Henderson, G; Hicks, GA; Watts, AE1
Behbehani, MM; Nickell, WT; Shipley, MT1
Feldtrauer, JJ; Waldmeier, PC; Wicki, P1
Blake, JF; Brugger, F; Cao, CQ; Collingridge, GL; Evans, RH; Headley, PM1
Lambert, NA; Wilson, WA1
Collingridge, GL; Davies, CH; Pozza, MF1
Bon, C; Galvan, M1
Bowery, NG; Malcangio, M; Teoh, H1
Clarac, F; Vinay, L1
Guyenet, PG; Li, YW1
Fricker, D; Le Feuvre, Y; Leresche, N1
Gellerman, D; Nordholm, AF; Ramirez, OA; Thompson, JK; Thompson, RF1
Batini, C; Vigot, R2
Cody, C; Jones, RS; Maubach, KA1
Ferreira, SA; Hileman, SM; Jackson, GL; Kuehl, DE1
Harayama, N; Kabashima, N; Shibuya, I; Tanaka, K; Ueta, Y; Yamashita, H1
Cui, JG; Linderoth, B; Meyerson, BA; Sollevi, A1
Curtis, DR; Lacey, G1
Durgam, VR; Mifflin, SW; Vitela, M1
Olianas, MC; Onali, P1
Celada, P; Paladini, CA; Tepper, JM1
Browning, DA; Ferreira, SA; Jackson, GL; Kuehl, DE; Scott, CJ1
Paladini, CA; Tepper, JM1
Barnbrock, A; Elsen, F; Richter, DW; Zhang, W1
Kiyohara, T; Konishi, S; Saitow, F; Satake, S; Yamada, J1
Kreitzer, AC; Regehr, WG1
Lambert, NA; Wang, X1
Bäurle, J; Jarolimek, W; Misgeld, U1
Enna, SJ; McCarson, KE; Moran, JM1
Bulters, DO; Cobb, SR; Davies, CH; Manuel, NA; Morton, RA1
Mann-Metzer, P; Yarom, Y1
Easter, A; Spruce, AE1
Chowdhury, SA; Rasmusson, DD1
Finger, TE; Sharp, AA1
Fearon, IM; Johnson, RP1
Bailey, SJ; Dhillon, A; Jones, RS; Woodhall, GL1
Harvey, VL; Stephens, GJ1
Chen, L; Yung, WH1
Ackerson, LC; Galvan, A; Maidment, NT; Smith, Y; Villalba, RM; West, SM; Wichmann, T1
Henderson, Z; Jones, GA1
Heyward, PM; McGann, JP; Puche, AC; Shao, Z; Shipley, MT; Wachowiak, M1
Bernardi, G; Berretta, N; Giustizieri, M; Mercuri, NB1
Linden, DJ; Shin, JH1
Ivenshitz, M; Segal, M1
Liu, X; Raggenbass, M; Tribollet, E1
Leung, LS; Shen, B1
Badiu, CI; Bessaïh, T; Bourgeais, L; Carter, DA; Crunelli, V; Lambolez, B; Leresche, N; Ruano, D; Toth, TI1
de Nanteuil, G; Herbelles, C; Mannoury la Cour, C; Millan, MJ; Pasteau, V1
Li, DP; Pan, HL; Pan, HM; Yang, Q1
Capogna, M; Price, CJ; Rusakov, DA; Scott, R1
Dvorzhak, A; Grantyn, R; Kirischuk, S; Kirmse, K1
Adams, DJ; Berecki, G; Callaghan, B; Clark, RJ; Craik, DJ; Haythornthwaite, A1
Chen, L; Cui, QL; Han, XH; Li, YL; Wang, HT; Xie, JX1
Bajova, H; Cho, J; Gruol, DL; Nelson, TE1
Deisz, RA; Lehmann, TN; Meencke, HJ; Nitsch, R; Teichgräber, LA; Weiss, T1
Cools, AR; Ikeda, H; Koshikawa, N; Kotani, A1
Khundakar, AA; Zetterström, TS1
Regehr, WG; Thanawala, MS1
Edeline, JM; Gaucher, Q; Gourévitch, B; Huetz, C1
Bai, HP; Guo, WY; Guo, YX; Liu, P; Wang, XL; Wu, YM1
Budefeld, T; Carbone, D; Eitel, C; Handa, RJ; Majdic, G; Nash, C; Searcy, BT; Staros, M; Stratton, MS; Tobet, SA1
Amakhin, DV; Popov, VA; Veselkin, NP1
Bosch, D; Ehrlich, I1

Other Studies

64 other study(ies) available for baclofen and cgp 55845a

ArticleYear
Putative pre- and postsynaptic ATP-sensitive potassium channels in the rat substantia nigra in vitro.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:4

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Barium Compounds; Bicuculline; Chlorides; Diazoxide; GABA-A Receptor Antagonists; Glucose; In Vitro Techniques; Kinetics; Male; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Potassium Channels; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-A; Substantia Nigra; Synapses; Synaptic Transmission; Time Factors; Tolbutamide

1995
Evidence for GABAB-mediated inhibition of transmission from the olfactory nerve to mitral cells in the rat olfactory bulb.
    Brain research bulletin, 1994, Volume: 35, Issue:2

    Topics: Animals; Axons; Baclofen; Electric Stimulation; Evoked Potentials; GABA-B Receptor Antagonists; In Vitro Techniques; Male; Neurons; Olfactory Bulb; Olfactory Nerve; Phosphinic Acids; Propanolamines; Ranidae; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Regression Analysis; Synaptic Transmission

1994
Release of endogenous glutamate from rat cortical slices in presence of the glutamate uptake inhibitor L-trans-pyrrolidine-2,4-dicarboxylic acid.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 348, Issue:5

    Topics: Animals; Baclofen; Calcium; Cerebral Cortex; Chromatography, High Pressure Liquid; Dicarboxylic Acids; Electric Stimulation; GABA-B Receptor Antagonists; Glutamates; Kainic Acid; Male; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Phosphinic Acids; Potassium; Propanolamines; Pyrrolidines; Rats; Rats, Inbred Strains; Synaptosomes; Tetrodotoxin

1993
Antagonism of baclofen-induced depression of whole-cell synaptic currents in spinal dorsal horn neurones by the potent GABAB antagonist CGP55845.
    Neuropharmacology, 1993, Volume: 32, Issue:12

    Topics: Action Potentials; Animals; Animals, Newborn; Baclofen; Dose-Response Relationship, Drug; GABA-B Receptor Antagonists; Ganglia, Spinal; In Vitro Techniques; Neurons; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Spinal Cord; Synapses

1993
Heterogeneity in presynaptic regulation of GABA release from hippocampal inhibitory neurons.
    Neuron, 1993, Volume: 11, Issue:6

    Topics: Analgesics; Animals; Baclofen; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Evoked Potentials; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Homeostasis; In Vitro Techniques; Male; Naloxone; Nerve Fibers; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Opioid, mu; Synapses

1993
CGP 55845A: a potent antagonist of GABAB receptors in the CA1 region of rat hippocampus.
    Neuropharmacology, 1993, Volume: 32, Issue:10

    Topics: Animals; Baclofen; Evoked Potentials; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Phosphinic Acids; Propanolamines; Rats; Receptors, GABA-B; Synapses

1993
Electrophysiological actions of GABAB agonists and antagonists in rat dorso-lateral septal neurones in vitro.
    British journal of pharmacology, 1996, Volume: 118, Issue:4

    Topics: Analysis of Variance; Animals; Baclofen; Benzylamines; Dose-Response Relationship, Drug; Electrophysiology; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Male; Membrane Potentials; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Receptors, GABA-B; Septal Nuclei

1996
GABA, glutamate and substance P-like immunoreactivity release: effects of novel GABAB antagonists.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Animals; Baclofen; Benzoates; Benzylamines; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Isonicotinic Acids; Male; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Nerve Roots; Stereoisomerism; Substance P

1996
CGP 35348 and CGP 55845A block the baclofen-induced depression of dorsal root evoked potentials in lumbar motoneurons of the neonatal rat.
    Neuroscience letters, 1996, Aug-23, Volume: 214, Issue:2-3

    Topics: Animals; Animals, Newborn; Baclofen; Decerebrate State; Depression, Chemical; Evoked Potentials; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Ganglia, Spinal; Motor Neurons; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Reflex, Monosynaptic; Spinal Cord; Synaptic Membranes

1996
Activation of GABAB receptors increases a potassium conductance in rat bulbospinal neurons of the C1 area.
    The American journal of physiology, 1996, Volume: 271, Issue:5 Pt 2

    Topics: Action Potentials; Animals; Baclofen; Barium Compounds; Chlorides; Electric Conductivity; GABA Antagonists; In Vitro Techniques; Medulla Oblongata; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Potassium; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Spinal Cord; Tyrosine 3-Monooxygenase

1996
GABAA receptor-mediated IPSCs in rat thalamic sensory nuclei: patterns of discharge and tonic modulation by GABAB autoreceptors.
    The Journal of physiology, 1997, Jul-01, Volume: 502 ( Pt 1)

    Topics: Animals; Autoreceptors; Baclofen; Cadmium; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Geniculate Bodies; Interneurons; Isonicotinic Acids; Male; Membrane Potentials; Organ Culture Techniques; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Tetrodotoxin; Thalamic Nuclei

1997
The conditioned eyeblink response: a role for the GABA-B receptor?
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:1

    Topics: Animals; Baclofen; Blinking; Cerebellum; Conditioning, Classical; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Infusions, Intravenous; Injections; Male; Phosphinic Acids; Propanolamines; Rabbits; Receptors, GABA-B

1997
GABA(B) receptor activation of Purkinje cells in cerebellar slices.
    Neuroscience research, 1997, Volume: 29, Issue:2

    Topics: Animals; Baclofen; Cerebellum; Dose-Response Relationship, Drug; Electric Conductivity; Female; GABA Agonists; GABA Antagonists; In Vitro Techniques; Male; Neural Inhibition; Phosphinic Acids; Potassium; Propanolamines; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Synapses

1997
Tachykinins may modify spontaneous epileptiform activity in the rat entorhinal cortex in vitro by activating GABAergic inhibition.
    Neuroscience, 1998, Volume: 83, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Entorhinal Cortex; Epilepsy; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Neurokinin A; Neurokinin B; Neurons; Peptide Fragments; Phosphinic Acids; Propanolamines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Substance P; Synapses; Tachykinins

1998
Effects of dialyzing gamma-aminobutyric acid receptor antagonists into the medial preoptic and arcuate ventromedial region on luteinizing hormone release in male sheep.
    Biology of reproduction, 1998, Volume: 58, Issue:4

    Topics: Animals; Arcuate Nucleus of Hypothalamus; Baclofen; Bicuculline; GABA Antagonists; Luteinizing Hormone; Male; Microdialysis; Orchiectomy; Phosphinic Acids; Preoptic Area; Propanolamines; Receptors, GABA; Sheep; Testosterone

1998
Inhibition of N- and P/Q-type calcium channels by postsynaptic GABAB receptor activation in rat supraoptic neurones.
    The Journal of physiology, 1998, Jun-01, Volume: 509 ( Pt 2)

    Topics: Animals; Baclofen; Calcium Channel Blockers; Calcium Channels; GABA Antagonists; Guanosine Diphosphate; In Vitro Techniques; Male; Membrane Potentials; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Pertussis Toxin; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Supraoptic Nucleus; Synapses; Synaptic Transmission; Thionucleotides; Virulence Factors, Bordetella

1998
Effect of spinal cord stimulation on tactile hypersensitivity in mononeuropathic rats is potentiated by simultaneous GABA(B) and adenosine receptor activation.
    Neuroscience letters, 1998, May-15, Volume: 247, Issue:2-3

    Topics: Adenosine; Animals; Baclofen; Electric Stimulation; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hindlimb; Hyperesthesia; Male; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Purinergic P1; Sciatic Nerve; Sensory Thresholds; Spinal Cord; Theophylline

1998
Prolonged GABA(B) receptor-mediated synaptic inhibition in the cat spinal cord: an in vivo study.
    Experimental brain research, 1998, Volume: 121, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Electrophysiology; Female; GABA Agonists; GABA Antagonists; GABA Modulators; Male; Membrane Potentials; Motor Neurons; Neural Inhibition; Pentobarbital; Phosphinic Acids; Propanolamines; Receptors, GABA-A; Receptors, GABA-B; Reflex; Spinal Cord; Synapses

1998
Enhanced gamma-aminobutyric acid-B receptor agonist responses and mRNA within the nucleus of the solitary tract in hypertension.
    Hypertension (Dallas, Tex. : 1979), 1999, Volume: 33, Issue:1 Pt 2

    Topics: Animals; Baclofen; Bicuculline; Blood Pressure; GABA Agonists; GABA Antagonists; Hypertension, Renovascular; Male; Muscimol; Nephrectomy; Nipecotic Acids; Phosphinic Acids; Proline; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Solitary Nucleus; Transcription, Genetic

1999
GABA(B) receptor-mediated stimulation of adenylyl cyclase activity in membranes of rat olfactory bulb.
    British journal of pharmacology, 1999, Volume: 126, Issue:3

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Baclofen; Calcium; Calmodulin; Colforsin; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Indomethacin; Injections, Intraventricular; Male; Membranes; Neuropeptides; Neuroprotective Agents; Olfactory Bulb; Organophosphorus Compounds; Pertussis Toxin; Phosphinic Acids; Phospholipases A; Phospholipids; Pituitary Adenylate Cyclase-Activating Polypeptide; Propanolamines; Propylamines; Quinacrine; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Transducin; Virulence Factors, Bordetella

1999
Striatal, pallidal, and pars reticulata evoked inhibition of nigrostriatal dopaminergic neurons is mediated by GABA(A) receptors in vivo.
    Neuroscience, 1999, Volume: 89, Issue:3

    Topics: Afferent Pathways; Animals; Baclofen; Bicuculline; Corpus Striatum; Dopamine; Electric Stimulation; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Nerve Degeneration; Neurons; Phosphinic Acids; Picrotoxin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Receptors, Presynaptic; Substantia Nigra

1999
Effect of infusing gamma-aminobutyric acid receptor agonists and antagonists into the medial preoptic area and ventromedial hypothalamus on prolactin secretion in male sheep.
    Endocrine, 1998, Volume: 9, Issue:3

    Topics: Animals; Baclofen; Bicuculline; GABA Agonists; GABA Antagonists; Male; Muscimol; Phosphinic Acids; Preoptic Area; Prolactin; Propanolamines; Sheep; Ventromedial Hypothalamic Nucleus

1998
GABA(A) and GABA(B) antagonists differentially affect the firing pattern of substantia nigra dopaminergic neurons in vivo.
    Synapse (New York, N.Y.), 1999, Jun-01, Volume: 32, Issue:3

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; Dopamine; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Kinetics; Male; Neurons; Phosphinic Acids; Picrotoxin; Propanolamines; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Substantia Nigra

1999
Postnatal development of GABAB receptor-mediated modulation of voltage-activated Ca2+ currents in mouse brain-stem neurons.
    The European journal of neuroscience, 1999, Volume: 11, Issue:7

    Topics: Aging; Animals; Animals, Newborn; Baclofen; Brain Stem; Calcium Channels; Calcium Channels, L-Type; Electric Conductivity; Electrophysiology; Female; GABA Agonists; GABA Antagonists; Male; Mice; Mice, Inbred Strains; Neurons; Phosphinic Acids; Propanolamines; Receptors, GABA-B

1999
Purkinje cell inhibitory responses to 3-APPA (3-aminopropylphosphinic acid) in RAT cerebellar slices.
    Neuroscience research, 1999, Volume: 34, Issue:3

    Topics: 4-Aminopyridine; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Cerebellum; Dose-Response Relationship, Drug; Female; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Purkinje Cells; Rats; Rats, Sprague-Dawley; Tetrodotoxin

1999
GABA(B) receptor-mediated presynaptic inhibition of glutamatergic and GABAergic transmission in the basolateral amygdala.
    Neuropharmacology, 1999, Volume: 38, Issue:11

    Topics: Amygdala; Animals; Baclofen; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Receptors, Presynaptic; Synaptic Transmission

1999
Modulation of transmission during trains at a cerebellar synapse.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Feb-15, Volume: 20, Issue:4

    Topics: Animals; Baclofen; Calcium; Cerebellum; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glycine; GTP-Binding Proteins; In Vitro Techniques; Nerve Fibers; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Purinergic P1 Receptor Antagonists; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, Purinergic P1; Synapses; Xanthines

2000
GABA(B) receptors couple to potassium and calcium channels on identified lateral perforant pathway projection neurons.
    Journal of neurophysiology, 2000, Volume: 83, Issue:2

    Topics: Adenosine; Analgesics; Animals; Baclofen; Calcium Channels; Electrophysiology; Entorhinal Cortex; GABA Agonists; GABA Antagonists; Membrane Potentials; Neural Inhibition; Neurons; Perforant Pathway; Phosphinic Acids; Potassium Channels; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Synapses; Synaptic Transmission

2000
Impaired inhibition of epileptiform activity by baclofen, but not by adenosine in the weaver hippocampus.
    Neuropharmacology, 2000, Jan-04, Volume: 39, Issue:2

    Topics: 4-Aminopyridine; Adenosine; Analgesics; Animals; Baclofen; Drug Interactions; Female; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; Hippocampus; Male; Mice; Mice, Inbred CBA; Mice, Neurologic Mutants; Phosphinic Acids; Propanolamines

2000
Developmental regulation of GABA(B) receptor function in rat spinal cord.
    Life sciences, 2001, Apr-06, Volume: 68, Issue:19-20

    Topics: Age Factors; Animals; Baclofen; Calcium; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Magnesium; Male; Muscarinic Antagonists; Oxotremorine; Phosphinic Acids; Propanolamines; Rats; Receptors, GABA-B; RNA, Messenger; Spinal Cord; Sulfur Radioisotopes

2001
Regulation of muscarinic acetylcholine receptor-mediated synaptic responses by GABA(B) receptors in the rat hippocampus.
    The Journal of physiology, 2001, Sep-15, Volume: 535, Issue:Pt 3

    Topics: Animals; Atropine; Baclofen; Excitatory Postsynaptic Potentials; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Muscarinic Antagonists; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Receptors, Muscarinic; Synapses; Synaptic Transmission

2001
Pre- and postsynaptic inhibition mediated by GABA(B) receptors in cerebellar inhibitory interneurons.
    Journal of neurophysiology, 2002, Volume: 87, Issue:1

    Topics: Animals; Baclofen; Cerebellum; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Guinea Pigs; In Vitro Techniques; Interneurons; Membrane Potentials; Neural Inhibition; Patch-Clamp Techniques; Phosphinic Acids; Potassium Channel Blockers; Propanolamines; Receptors, GABA-B; Sodium Channel Blockers; Synaptic Transmission

2002
Recombinant GABA(B) receptors formed from GABA(B1) and GABA(B2) subunits selectively inhibit N-type Ca(2+) channels in NG108-15 cells.
    European journal of pharmacology, 2002, Apr-05, Volume: 440, Issue:1

    Topics: Animals; Baclofen; Calcium Channels, T-Type; DNA, Antisense; DNA, Recombinant; GABA Agonists; GABA Antagonists; Membrane Potentials; Nifedipine; Norepinephrine; omega-Conotoxin GVIA; Phosphinic Acids; Plasmids; Propanolamines; Protein Subunits; Receptors, GABA-B; Transfection; Tumor Cells, Cultured

2002
Comparison of receptive field expansion produced by GABA(B) and GABA(A) receptor antagonists in raccoon primary somatosensory cortex.
    Experimental brain research, 2002, Volume: 144, Issue:1

    Topics: Afferent Pathways; Animals; Baclofen; Female; Fingers; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Mechanoreceptors; Neural Inhibition; Neuronal Plasticity; Neurons; Phosphinic Acids; Propanolamines; Raccoons; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Skin; Somatosensory Cortex; Synaptic Transmission; Touch

2002
GABAergic modulation of primary gustatory afferent synaptic efficacy.
    Journal of neurobiology, 2002, Volume: 52, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Carrier Proteins; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Goldfish; Membrane Proteins; Membrane Transport Proteins; Muscimol; Neurons, Afferent; Organic Anion Transporters; Phosphinic Acids; Propanolamines; Receptors, GABA-A; Receptors, GABA-B; Solitary Nucleus; Synapses; Taste

2002
GABA(B) receptor activation augments TASK-1 in MAH cells and mediates autoreceptor feedback during hypoxia.
    Biochemical and biophysical research communications, 2003, Dec-12, Volume: 312, Issue:2

    Topics: Adaptation, Physiological; Adrenal Medulla; Animals; Autoreceptors; Baclofen; Cell Hypoxia; Cell Line; Chromaffin Cells; Feedback; GABA-B Receptor Antagonists; Homeostasis; Ion Channel Gating; Membrane Potentials; Nerve Tissue Proteins; Phosphinic Acids; Potassium Channels; Potassium Channels, Tandem Pore Domain; Propanolamines; Rats; Receptors, GABA-B; Zinc

2003
Lamina-specific differences in GABA(B) autoreceptor-mediated regulation of spontaneous GABA release in rat entorhinal cortex.
    Neuropharmacology, 2004, Volume: 46, Issue:1

    Topics: Action Potentials; Animals; Autoreceptors; Baclofen; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Entorhinal Cortex; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Neural Inhibition; Phosphinic Acids; Propanolamines; Rats; Receptors, GABA-B

2004
Mechanism of GABA receptor-mediated inhibition of spontaneous GABA release onto cerebellar Purkinje cells.
    The European journal of neuroscience, 2004, Volume: 20, Issue:3

    Topics: Action Potentials; Age Factors; Animals; Baclofen; Barium; Cadmium; Calcium; Cerebellum; Colforsin; Drug Interactions; Enzyme Inhibitors; Exotoxins; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Neural Inhibition; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Purkinje Cells; Receptors, GABA-A; Ruthenium Red; Synaptic Transmission; Tetrodotoxin

2004
Tonic activation of presynaptic GABA(B) receptors on rat pallidosubthalamic terminals.
    Acta pharmacologica Sinica, 2005, Volume: 26, Issue:1

    Topics: Animals; Baclofen; GABA Agonists; GABA Antagonists; Membrane Potentials; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Subthalamic Nucleus

2005
GABAergic modulation of the activity of globus pallidus neurons in primates: in vivo analysis of the functions of GABA receptors and GABA transporters.
    Journal of neurophysiology, 2005, Volume: 94, Issue:2

    Topics: Action Potentials; Animals; Anisoles; Baclofen; Brain Mapping; Enzyme Inhibitors; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Globus Pallidus; Immunohistochemistry; Macaca mulatta; Membrane Transport Modulators; Membrane Transport Proteins; Microdialysis; Microscopy, Immunoelectron; Muscimol; Neurons; Nipecotic Acids; Phosphinic Acids; Propanolamines; Pyridazines; Receptors, GABA

2005
GABAB receptors in the medial septum/diagonal band slice from 16-25 day rat.
    Neuroscience, 2005, Volume: 132, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; In Vitro Techniques; Kainic Acid; Membrane Potentials; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-A; Septum Pellucidum; Sodium Channel Blockers; Tetrodotoxin; Time Factors; Valine

2005
Inhibition [corrected] of olfactory receptor neuron input to olfactory bulb glomeruli mediated by suppression of presynaptic calcium influx.
    Journal of neurophysiology, 2005, Volume: 94, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Fluorescent Dyes; GABA Agonists; GABA Antagonists; In Vitro Techniques; Mice; Mice, Transgenic; Nerve Tissue Proteins; Neural Inhibition; Olfactory Bulb; Olfactory Pathways; Olfactory Receptor Neurons; omega-Conotoxin GVIA; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Time Factors

2005
Distinct mechanisms of presynaptic inhibition at GABAergic synapses of the rat substantia nigra pars compacta.
    Journal of neurophysiology, 2005, Volume: 94, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aminobutyrates; Animals; Animals, Newborn; Baclofen; Cadmium Chloride; Dopamine; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Ionomycin; Ionophores; Membrane Potentials; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Rats; Sodium Channel Blockers; Spider Venoms; Substantia Nigra; Synapses; Tetrodotoxin

2005
An NMDA receptor/nitric oxide cascade is involved in cerebellar LTD but is not localized to the parallel fiber terminal.
    Journal of neurophysiology, 2005, Volume: 94, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Animals; Animals, Newborn; Baclofen; Benzoates; Cadmium Chloride; Cerebellum; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Imidazoles; In Vitro Techniques; Long-Term Potentiation; Magnesium; Models, Neurological; N-Methylaspartate; Nerve Fibers; Nerve Tissue Proteins; Nitric Oxide; Nitroarginine; Phosphinic Acids; Propanolamines; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses; Time Factors

2005
Simultaneous NMDA-dependent long-term potentiation of EPSCs and long-term depression of IPSCs in cultured rat hippocampal neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-25, Volume: 26, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Evoked Potentials; Hippocampus; Long-Term Potentiation; Long-Term Synaptic Depression; Neuronal Plasticity; Neurons; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Quinoxalines; Rats; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Tetrodotoxin; Thionucleotides; Time Factors

2006
GABA(B) receptor-activation inhibits GABAergic synaptic transmission in parvocellular neurones of rat hypothalamic paraventricular nucleus.
    Journal of neuroendocrinology, 2006, Volume: 18, Issue:3

    Topics: Animals; Baclofen; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Hypothalamus; Immunohistochemistry; In Vitro Techniques; Male; Neurons; Paraventricular Hypothalamic Nucleus; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Synaptic Transmission

2006
Hippocampal partial kindling decreased hippocampal GABAB receptor efficacy and wet dog shakes in rats.
    Behavioural brain research, 2006, Oct-16, Volume: 173, Issue:2

    Topics: Amphetamines; Animals; Baclofen; Behavior, Animal; Drug Interactions; Electric Stimulation; Electroencephalography; GABA Agonists; GABA Antagonists; Head Movements; Hippocampus; Kindling, Neurologic; Male; Phosphinic Acids; Propanolamines; Rats; Reaction Time; Receptors, GABA-B; Serotonin Receptor Agonists; Time Factors

2006
Nucleus-specific abnormalities of GABAergic synaptic transmission in a genetic model of absence seizures.
    Journal of neurophysiology, 2006, Volume: 96, Issue:6

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Epilepsy, Absence; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Immunohistochemistry; In Vitro Techniques; Intralaminar Thalamic Nuclei; Membrane Potentials; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Receptors, GABA-A; Somatosensory Cortex; Synapses; Synaptic Transmission; Ventral Thalamic Nuclei

2006
Influence of positive allosteric modulators on GABA(B) receptor coupling in rat brain: a scintillation proximity assay characterisation of G protein subtypes.
    Journal of neurochemistry, 2008, Volume: 105, Issue:2

    Topics: Allosteric Site; Animals; Baclofen; Brain; Cell Line, Transformed; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA Antagonists; GTP-Binding Protein alpha Subunits, G12-G13; GTP-Binding Protein alpha Subunits, Gi-Go; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Phenols; Phosphinic Acids; Propanolamines; Protein Binding; Radioligand Assay; Rats; Receptors, GABA-B; Signal Transduction

2008
Plasticity of pre- and postsynaptic GABAB receptor function in the paraventricular nucleus in spontaneously hypertensive rats.
    American journal of physiology. Heart and circulatory physiology, 2008, Volume: 295, Issue:2

    Topics: Animals; Baclofen; Disease Models, Animal; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; Glutamine; GTP-Binding Proteins; Guanosine Diphosphate; Hypertension; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Neuronal Plasticity; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, GABA-B; Staining and Labeling; Sympathetic Nervous System; Synaptic Transmission; Thionucleotides

2008
GABA(B) receptor modulation of feedforward inhibition through hippocampal neurogliaform cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2008, Jul-02, Volume: 28, Issue:27

    Topics: Action Potentials; Animals; Baclofen; Calcium; Calcium Signaling; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Inhibitory Postsynaptic Potentials; Interneurons; Neural Inhibition; Neural Pathways; Neuroglia; Organ Culture Techniques; Phosphinic Acids; Propanolamines; Pyramidal Cells; Rats; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission

2008
GABA transporter 1 tunes GABAergic synaptic transmission at output neurons of the mouse neostriatum.
    The Journal of physiology, 2008, Dec-01, Volume: 586, Issue:23

    Topics: Action Potentials; Animals; Animals, Newborn; Baclofen; Bicuculline; Electric Impedance; Electric Stimulation; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Mice; Mice, Inbred C57BL; Neostriatum; Neurons; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Pyridazines; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Tetrodotoxin

2008
Analgesic alpha-conotoxins Vc1.1 and Rg1A inhibit N-type calcium channels in rat sensory neurons via GABAB receptor activation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2008, Oct-22, Volume: 28, Issue:43

    Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Barium; Calcium Channel Blockers; Calcium Channels, N-Type; Cells, Cultured; Conotoxins; Dose-Response Relationship, Radiation; Electric Stimulation; GABA Antagonists; Ganglia, Spinal; Membrane Potentials; omega-Conotoxins; Patch-Clamp Techniques; Pertussis Toxin; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA; Sensory Receptor Cells

2008
Behavioral and electrophysiological effects of pallidal GABAB receptor activation and blockade on haloperidol-induced akinesia in rats.
    Brain research, 2008, Dec-09, Volume: 1244

    Topics: Animals; Baclofen; Behavior, Animal; Dopamine Antagonists; Dystonia; Electrophysiology; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Globus Pallidus; Haloperidol; Injections, Intraperitoneal; Male; Motor Activity; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B

2008
Chronic CXCL10 alters neuronal properties in rat hippocampal culture.
    Journal of neuroimmunology, 2009, Feb-15, Volume: 207, Issue:1-2

    Topics: Animals; Antibodies; Baclofen; Calcium; Cells, Cultured; Chemokine CXCL10; Dose-Response Relationship, Drug; Embryo, Mammalian; GABA Agonists; GABA Antagonists; Glial Fibrillary Acidic Protein; Glutamate Decarboxylase; Hippocampus; N-Methylaspartate; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, GABA; Receptors, N-Methyl-D-Aspartate; Synapsins; Time Factors

2009
Impaired function of GABA(B) receptors in tissues from pharmacoresistant epilepsy patients.
    Epilepsia, 2009, Volume: 50, Issue:7

    Topics: Animals; Anticonvulsants; Baclofen; Bicuculline; Cerebral Cortex; Drug Resistance; Epilepsy; Epilepsy, Temporal Lobe; Excitatory Postsynaptic Potentials; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Immunohistochemistry; Mice; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Synaptic Transmission

2009
Differential role of GABAA and GABAB receptors in two distinct output stations of the rat striatum: studies on the substantia nigra pars reticulata and the globus pallidus.
    Neuroscience, 2010, Apr-28, Volume: 167, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Corpus Striatum; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Globus Pallidus; Male; Motor Activity; Muscimol; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Substantia Nigra

2010
Effects of GABAB ligands alone and in combination with paroxetine on hippocampal BDNF gene expression.
    European journal of pharmacology, 2011, Dec-05, Volume: 671, Issue:1-3

    Topics: Animals; Antidepressive Agents; Baclofen; Brain-Derived Neurotrophic Factor; Down-Regulation; Drug Interactions; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gene Expression Regulation; Hippocampus; Ligands; Male; Paroxetine; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; RNA, Messenger

2011
Presynaptic calcium influx controls neurotransmitter release in part by regulating the effective size of the readily releasable pool.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Mar-13, Volume: 33, Issue:11

    Topics: Animals; Animals, Newborn; Baclofen; Biophysics; Calcium; Calcium Channel Blockers; Computer Simulation; Electric Stimulation; Excitatory Postsynaptic Potentials; Female; GABA Antagonists; GABA-B Receptor Agonists; Male; Mice; Mice, Inbred C57BL; Models, Neurological; Neurons; Neurotransmitter Agents; Nickel; omega-Agatoxin IVA; Patch-Clamp Techniques; Phosphinic Acids; Pons; Presynaptic Terminals; Propanolamines

2013
Cortical inhibition reduces information redundancy at presentation of communication sounds in the primary auditory cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Jun-26, Volume: 33, Issue:26

    Topics: Algorithms; Animal Communication; Animals; Auditory Cortex; Auditory Perception; Baclofen; Brain Mapping; Cerebral Cortex; Discrimination, Psychological; Electrophysiological Phenomena; Extracellular Space; Female; GABA Antagonists; Guinea Pigs; Male; Microinjections; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Pyridazines; Receptors, GABA-A; Receptors, GABA-B; Vocalization, Animal

2013
Activation of spinal GABAB receptors normalizes N-methyl-D-aspartate receptor in diabetic neuropathy.
    Journal of the neurological sciences, 2014, Jun-15, Volume: 341, Issue:1-2

    Topics: Analysis of Variance; Animals; Antibiotics, Antineoplastic; Baclofen; CREB-Binding Protein; Diabetic Neuropathies; Disease Models, Animal; GABA Antagonists; GABA-B Receptor Agonists; Gene Expression Regulation; Male; Pain Measurement; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Streptozocin; Time Factors

2014
Embryonic GABA(B) receptor blockade alters cell migration, adult hypothalamic structure, and anxiety- and depression-like behaviors sex specifically in mice.
    PloS one, 2014, Volume: 9, Issue:8

    Topics: Animals; Anxiety; Baclofen; Cell Movement; Depression; Embryo, Mammalian; Female; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression; Hypothalamo-Hypophyseal System; Immobilization; Male; Maze Learning; Mice; Mice, Transgenic; Paraventricular Hypothalamic Nucleus; Phosphinic Acids; Pituitary-Adrenal System; Pregnancy; Propanolamines; Protein Subunits; Psychomotor Agitation; Receptors, GABA-B; Sex Factors; Stress, Psychological; Tissue Culture Techniques

2014
[Modulation of GABA- and kainate-activated currents by metabotropic receptors in isolated rat cortical neurons].
    Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova, 2014, Volume: 100, Issue:10

    Topics: Animals; Baclofen; Cycloleucine; Excitatory Amino Acid Agonists; Female; GABA Antagonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Kainic Acid; Male; Neuroprotective Agents; Phosphinic Acids; Propanolamines; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Synaptic Transmission

2014
Postnatal maturation of GABAergic modulation of sensory inputs onto lateral amygdala principal neurons.
    The Journal of physiology, 2015, Oct-01, Volume: 593, Issue:19

    Topics: Amygdala; Animals; Baclofen; Benzylamines; Excitatory Postsynaptic Potentials; GABA Agents; Inhibitory Postsynaptic Potentials; Male; Mice, Inbred C57BL; Neurons; Nipecotic Acids; Phosphinic Acids; Picrotoxin; Propanolamines

2015