baclofen has been researched along with cgp 52432 in 29 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 6 (20.69) | 18.2507 |
| 2000's | 16 (55.17) | 29.6817 |
| 2010's | 7 (24.14) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Bonanno, G; Cavazzani, P; Fassio, A; Raiteri, M | 1 |
| Baumann, PA; Bittiger, H; Feldtrauer, JJ; Mickel, SJ; Waldmeier, PC; Wicki, P | 1 |
| Bonanno, G; Gemignani, A; Paudice, P; Raiteri, M | 1 |
| Bonanno, G; Fassio, A; Gemignani, A; Lanza, M; Raiteri, M | 1 |
| Bon, C; Galvan, M | 1 |
| Bowery, NG; Malcangio, M; Teoh, H | 1 |
| Giniatullin, R; Nistri, A; Sokolova, E | 1 |
| Ganter, P; López-Bendito, G; Luján, R; Molnár, Z; Paulsen, O; Shigemoto, R | 1 |
| Jackson, GL; Kuehl, D | 1 |
| Enna, SJ | 1 |
| Burger, RM; Lu, Y; Rubel, EW | 1 |
| Carter, LP; Chen, W; Coop, A; France, CP; Koek, W; Lamb, RJ; Wu, H | 1 |
| Cremers, TI; Rea, K; Westerink, BH | 1 |
| Chen, Q; Pan, HL | 1 |
| Balcar, VJ; Griffin, JL; Nasrallah, FA; Rae, C | 1 |
| Besseyrias, V; Bettler, B; Ulrich, D | 1 |
| Breese, GR; Criswell, HE; Kelm, MK | 1 |
| Baumann, O; Blenau, W; Rotte, C; Walz, B; Witte, J | 1 |
| Luccini, E; Raiteri, L; Raiteri, M; Romei, C | 1 |
| Bosch, MA; Kelly, MJ; Rønnekleiv, OK; Zhang, C | 1 |
| Dong, Y; Ito, W; Morozov, A; Pan, BX; Shigemoto, R; Yanagawa, Y | 1 |
| Ayajiki, K; Fujii, T; Kobuchi, S; Matsumura, Y; Ohkita, M; Shintani, T; Sugiura, T; Suzuki, R; Tanaka, R; Tsutsui, H | 1 |
| Ayajiki, K; Kobuchi, S; Matsumura, Y; Ohkita, M; Shintani, T; Suzuki, R; Tanaka, R; Tsutsui, H | 1 |
| Andresen, MC; Fawley, JA; Peters, JH | 1 |
| Ma, H; Yang, K | 1 |
| Di Prisco, S; Grilli, M; Marchi, M; Pittaluga, A; Summa, M; Usai, C | 1 |
| Cryan, JF; O'Leary, OF; Sweeney, FF | 1 |
| Borgland, SL; Pitman, KA; Puil, E | 1 |
| Bosch, D; Ehrlich, I | 1 |
1 review(s) available for baclofen and cgp 52432
| Article | Year |
|---|---|
A GABA(B) mystery: the search for pharmacologically distinct GABA(B) receptors.
Topics: Acetates; Amines; Animals; Anticonvulsants; Baclofen; Benzylamines; Cyclohexanecarboxylic Acids; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gabapentin; gamma-Aminobutyric Acid; Humans; Molecular Structure; Morpholines; Phosphinic Acids; Protein Isoforms; Receptors, GABA-B; RNA, Messenger | 2001 |
28 other study(ies) available for baclofen and cgp 52432
| Article | Year |
|---|---|
Characterization of the GABA autoreceptor in human neocortex as a pharmacological subtype of the GABAB receptor.
Topics: Adolescent; Adult; Aged; Animals; Baclofen; Benzylamines; Binding, Competitive; Brain Neoplasms; Cerebral Cortex; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Humans; Male; Middle Aged; Organophosphorus Compounds; Phosphinic Acids; Rats; Receptors, GABA-B | 1994 |
GABA and glutamate release affected by GABAB receptor antagonists with similar potency: no evidence for pharmacologically different presynaptic receptors.
Topics: Animals; Baclofen; Benzylamines; Cerebral Cortex; Electric Stimulation; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Male; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Inbred Strains; Receptors, GABA-B; Receptors, Presynaptic | 1994 |
Pharmacological discrimination between gamma-aminobutyric acid type B receptors regulating cholecystokinin and somatostatin release from rat neocortex synaptosomes.
Topics: Animals; Baclofen; Benzylamines; Cerebral Cortex; Cholecystokinin; GABA Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Ligands; Male; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Somatostatin; Synaptosomes | 1994 |
CGP 52432: a novel potent and selective GABAB autoreceptor antagonist in rat cerebral cortex.
Topics: Animals; Baclofen; Benzylamines; Cerebral Cortex; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Wistar; Somatostatin | 1993 |
Electrophysiological actions of GABAB agonists and antagonists in rat dorso-lateral septal neurones in vitro.
Topics: Analysis of Variance; Animals; Baclofen; Benzylamines; Dose-Response Relationship, Drug; Electrophysiology; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Male; Membrane Potentials; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Receptors, GABA-B; Septal Nuclei | 1996 |
GABA, glutamate and substance P-like immunoreactivity release: effects of novel GABAB antagonists.
Topics: Animals; Baclofen; Benzoates; Benzylamines; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Isonicotinic Acids; Male; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Nerve Roots; Stereoisomerism; Substance P | 1996 |
The ATP-mediated fast current of rat dorsal root ganglion neurons is a novel effector for GABA(B) receptor activation.
Topics: Adenosine Triphosphate; Animals; Baclofen; Benzylamines; Cells, Cultured; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Membrane Potentials; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Phosphinic Acids; Picrotoxin; Rats; Receptors, GABA-A; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X3 | 2003 |
Blockade of GABA(B) receptors alters the tangential migration of cortical neurons.
Topics: Animals; Baclofen; Benzylamines; Cell Movement; Cerebral Cortex; Cerebral Ventricles; Culture Techniques; Dose-Response Relationship, Drug; Electrophysiology; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; Immunohistochemistry; Neurons; Phosphinic Acids; Rats; Rats, Wistar; Receptors, GABA-B | 2003 |
Effects of applying gamma-aminobutyric acid(B) drugs into the medial basal hypothalamus on basal luteinizing hormone concentrations and on luteinizing hormone surges in the female sheep.
Topics: Animals; Baclofen; Benzylamines; Breeding; Estrogens; Female; GABA Agonists; GABA-B Receptor Agonists; Hypothalamus, Middle; Luteinizing Hormone; Organophosphorus Compounds; Ovariectomy; Phosphinic Acids; Pituitary Gland, Anterior; Seasons; Sheep | 2004 |
GABA(B) receptor activation modulates GABA(A) receptor-mediated inhibition in chicken nucleus magnocellularis neurons.
Topics: Analysis of Variance; Animals; Baclofen; Benzylamines; Calcium; Chick Embryo; Cochlear Nucleus; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Magnesium; Membrane Potentials; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission | 2005 |
Discriminative stimulus effects of gamma-hydroxybutyrate (GHB) in rats discriminating GHB from baclofen and diazepam.
Topics: 4-Butyrolactone; Anesthetics, Intravenous; Animals; Baclofen; Benzocycloheptenes; Benzylamines; Butylene Glycols; Diazepam; Discrimination, Psychological; Dithiothreitol; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA Modulators; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Sodium Oxybate | 2005 |
HPLC conditions are critical for the detection of GABA by microdialysis.
Topics: Anesthetics, Local; Animals; Baclofen; Benzylamines; Brain; Brain Chemistry; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microdialysis; Nipecotic Acids; Phosphinic Acids; Potassium; Rats; Rats, Wistar; Tetrodotoxin; Time Factors | 2005 |
Regulation of synaptic input to hypothalamic presympathetic neurons by GABA(B) receptors.
Topics: 4-Aminopyridine; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Benzylamines; Bicuculline; Cadmium Chloride; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Ethylmaleimide; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Phosphinic Acids; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Receptors, GABA-B | 2006 |
Understanding your inhibitions: modulation of brain cortical metabolism by GABA(B) receptors.
Topics: Animals; Baclofen; Benzylamines; Carbon Isotopes; Cerebral Cortex; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; Guinea Pigs; Molecular Structure; Morpholines; Nuclear Magnetic Resonance, Biomolecular; Organophosphorus Compounds; Phosphinic Acids; Principal Component Analysis; Receptors, GABA-B | 2007 |
Functional mapping of GABA(B)-receptor subtypes in the thalamus.
Topics: Animals; Baclofen; Benzylamines; Brain Mapping; Cerebral Cortex; Excitatory Postsynaptic Potentials; Female; GABA Agonists; GABA Antagonists; Male; Mice; Mice, Inbred BALB C; Mice, Knockout; Phosphinic Acids; Receptors, GABA-B; Thalamus | 2007 |
The role of protein kinase A in the ethanol-induced increase in spontaneous GABA release onto cerebellar Purkinje neurons.
Topics: Animals; Animals, Newborn; Baclofen; Benzoxazines; Benzylamines; Calcium; Central Nervous System Depressants; Cerebellum; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Ethanol; GABA Agents; gamma-Aminobutyric Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Membrane Potentials; Morpholines; Naphthalenes; Patch-Clamp Techniques; Phosphinic Acids; Protein Kinase C; Purkinje Cells; Rats; Rats, Sprague-Dawley; Sodium Channel Blockers; Tetrodotoxin | 2008 |
Source, topography and excitatory effects of GABAergic innervation in cockroach salivary glands.
Topics: Analysis of Variance; Animals; Baclofen; Benzylamines; Electrophysiology; Fluorescent Antibody Technique; GABA Agonists; gamma-Aminobutyric Acid; Neurons; Organophosphorus Compounds; Periplaneta; Phosphinic Acids; Salivary Glands | 2009 |
GABA(B) presynaptic receptors modulate glycine exocytosis from mouse spinal cord and hippocampus glycinergic nerve endings.
Topics: Animals; Baclofen; Benzylamines; Exocytosis; Glycine; Glycine Plasma Membrane Transport Proteins; Hippocampus; Mice; Nerve Endings; Organophosphorus Compounds; Phosphinic Acids; Receptors, GABA-B; Spinal Cord | 2009 |
Gamma-aminobutyric acid B receptor mediated inhibition of gonadotropin-releasing hormone neurons is suppressed by kisspeptin-G protein-coupled receptor 54 signaling.
Topics: Animals; Baclofen; Benzylamines; Down-Regulation; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; Gonadotropin-Releasing Hormone; Kisspeptins; Membrane Potentials; Mice; Neurons; Phosphinic Acids; Receptors, G-Protein-Coupled; Receptors, GABA-B; Receptors, Kisspeptin-1; Signal Transduction; Synaptic Transmission; Tumor Suppressor Proteins | 2009 |
Selective gating of glutamatergic inputs to excitatory neurons of amygdala by presynaptic GABAb receptor.
Topics: Amygdala; Animals; Baclofen; Benzylamines; Biophysics; Electric Stimulation; GABA Agents; Glutamate Decarboxylase; Glutamic Acid; Green Fluorescent Proteins; In Vitro Techniques; Long-Term Potentiation; Mice; Mice, Transgenic; Microscopy, Electron, Transmission; Neural Pathways; Neurons; Nipecotic Acids; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Receptors, GABA-B; Synaptic Potentials | 2009 |
Renoprotective effects of gamma-aminobutyric acid on ischemia/reperfusion-induced renal injury in rats.
Topics: Animals; Baclofen; Benzylamines; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Kidney; Kidney Diseases; Kidney Function Tests; Kidney Tubular Necrosis, Acute; Male; Neurons; Norepinephrine; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Sympathetic Nervous System; Time Factors | 2009 |
Mechanisms underlying the renoprotective effect of GABA against ischemia/reperfusion-induced renal injury in rats.
Topics: Acute Kidney Injury; Animals; Baclofen; Benzylamines; Bicuculline; Blood Urea Nitrogen; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Injections, Intravenous; Injections, Intraventricular; Kidney; Kidney Function Tests; Male; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Reperfusion Injury; Sympathetic Nervous System | 2011 |
GABA(B)-mediated inhibition of multiple modes of glutamate release in the nucleus of the solitary tract.
Topics: Action Potentials; Animals; Baclofen; Benzylamines; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA-B Receptor Antagonists; Glutamic Acid; Male; Patch-Clamp Techniques; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Solitary Nucleus; Synaptic Vesicles; TRPV Cation Channels | 2011 |
Blockade of GABA(B) receptors facilitates evoked neurotransmitter release at spinal dorsal horn synapse.
Topics: Amino Acids; Animals; Baclofen; Benzylamines; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Agonists; GABA-A Receptor Antagonists; In Vitro Techniques; Male; Neurotransmitter Agents; Nipecotic Acids; Patch-Clamp Techniques; Phosphinic Acids; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Spinal Cord; Synapses; Synaptic Potentials; Tiagabine; Xanthenes | 2011 |
Presynaptic mGlu7 receptors control GABA release in mouse hippocampus.
Topics: Adenylyl Cyclase Inhibitors; Aminobutyrates; Animals; Baclofen; Benzhydryl Compounds; Benzoates; Benzylamines; Colforsin; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Exocytosis; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; Imines; Mice; Phosphinic Acids; Potassium Chloride; Pyridones; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Synaptosomes; Syntaxin 1; Vesicular Inhibitory Amino Acid Transport Proteins | 2013 |
Activation but not blockade of GABAB receptors during early-life alters anxiety in adulthood in BALB/c mice.
Topics: Analysis of Variance; Animals; Animals, Newborn; Anxiety; Baclofen; Benzylamines; Defense Mechanisms; Disease Models, Animal; Fever; GABA Antagonists; GABA-B Receptor Agonists; Male; Maze Learning; Mice; Mice, Inbred BALB C; Phosphinic Acids; Receptors, GABA-B; Stress, Psychological; Swimming | 2014 |
GABA(B) modulation of dopamine release in the nucleus accumbens core.
Topics: Animals; Baclofen; Benzylamines; Central Nervous System Stimulants; Cocaine; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Mice, Inbred C57BL; Motor Activity; Neurons; Nicotinic Antagonists; Nucleus Accumbens; Phosphinic Acids; Quinpirole; Receptors, Dopamine D2; Receptors, GABA-B; Tissue Culture Techniques | 2014 |
Postnatal maturation of GABAergic modulation of sensory inputs onto lateral amygdala principal neurons.
Topics: Amygdala; Animals; Baclofen; Benzylamines; Excitatory Postsynaptic Potentials; GABA Agents; Inhibitory Postsynaptic Potentials; Male; Mice, Inbred C57BL; Neurons; Nipecotic Acids; Phosphinic Acids; Picrotoxin; Propanolamines | 2015 |