Page last updated: 2024-09-04

b-ht 958 and idazoxan

b-ht 958 has been researched along with idazoxan in 2 studies

Compound Research Comparison

Studies
(b-ht 958)
Trials
(b-ht 958)
Recent Studies (post-2010)
(b-ht 958)
Studies
(idazoxan)
Trials
(idazoxan)
Recent Studies (post-2010) (idazoxan)
15031,49940123

Protein Interaction Comparison

ProteinTaxonomyb-ht 958 (IC50)idazoxan (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.0083
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0195
Alpha-2B adrenergic receptorHomo sapiens (human)0.0195
Alpha-2C adrenergic receptorHomo sapiens (human)0.0537
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.0195
Alpha-1A adrenergic receptorHomo sapiens (human)2.884
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0195

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cichini, G; Singer, EA1
Brown, MJ; Harland, D1

Other Studies

2 other study(ies) available for b-ht 958 and idazoxan

ArticleYear
B-HT 920, B-HT 933, and B-HT 958: presynaptic effects on electrically evoked 3H-noradrenaline release from slices of rat brain cortex and hypothalamus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Cerebral Cortex; Dioxanes; Electric Stimulation; Hypothalamus, Anterior; Idazoxan; In Vitro Techniques; Male; Norepinephrine; Rats; Rats, Inbred Strains; Sulpiride; Tritium

1987
B-HT 958 lowers blood pressure and heart rate in the rat through stimulation of dopamine receptors.
    British journal of pharmacology, 1986, Volume: 87, Issue:2

    Topics: Animals; Azepines; Blood Pressure; Dioxanes; Drug Interactions; Heart Rate; Idazoxan; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Sulpiride

1986