Page last updated: 2024-09-04

b-ht 958 and clonidine

b-ht 958 has been researched along with clonidine in 2 studies

Compound Research Comparison

Studies
(b-ht 958)
Trials
(b-ht 958)
Recent Studies (post-2010)
(b-ht 958)
Studies
(clonidine)
Trials
(clonidine)
Recent Studies (post-2010) (clonidine)
150313,6922,0441,394

Protein Interaction Comparison

ProteinTaxonomyb-ht 958 (IC50)clonidine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.101
Alpha-2B adrenergic receptorHomo sapiens (human)0.0353
Alpha-2C adrenergic receptorHomo sapiens (human)0.0115
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)5.365
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-1D adrenergic receptorHomo sapiens (human)1.21
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)5.365
Alpha-2A adrenergic receptorBos taurus (cattle)0.002
NischarinRattus norvegicus (Norway rat)0.3662

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Eskinder, H; Gross, GJ1
Andén, NE; Grabowska-Andén, M1

Other Studies

2 other study(ies) available for b-ht 958 and clonidine

ArticleYear
Sensitivity of alpha-adrenoceptor agonists to the calcium channel activator, Bay K 8644, in canine saphenous vein.
    Pharmacology, 1987, Volume: 35, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Dogs; Female; In Vitro Techniques; Ion Channels; Male; Muscle, Smooth, Vascular; Saphenous Vein

1987
B-HT 958 stimulates dopamine autoreceptors but blocks noradrenaline autoreceptors in the brain.
    The Journal of pharmacy and pharmacology, 1984, Volume: 36, Issue:11

    Topics: Adrenergic alpha-Agonists; alpha-Methyltyrosine; Animals; Apomorphine; Azepines; Brain Chemistry; Clonidine; Dihydroxyphenylalanine; Dopamine; Haloperidol; Male; Methyltyrosines; Mice; Motor Activity; Norepinephrine; Receptors, Adrenergic; Receptors, Dopamine; Reserpine; Synapses

1984