Page last updated: 2024-09-04

b-ht 958 and apomorphine

b-ht 958 has been researched along with apomorphine in 2 studies

Compound Research Comparison

Studies
(b-ht 958)
Trials
(b-ht 958)
Recent Studies (post-2010)
(b-ht 958)
Studies
(apomorphine)
Trials
(apomorphine)
Recent Studies (post-2010) (apomorphine)
15039,205287780

Protein Interaction Comparison

ProteinTaxonomyb-ht 958 (IC50)apomorphine (IC50)
Tryptophan 5-hydroxylase 1Rattus norvegicus (Norway rat)0.22
D(2) dopamine receptorHomo sapiens (human)0.0146
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.75
DRattus norvegicus (Norway rat)0.4744
D(3) dopamine receptorRattus norvegicus (Norway rat)0.1432
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.063
D(2) dopamine receptorBos taurus (cattle)0.3385
D(1A) dopamine receptorHomo sapiens (human)0.025
D(4) dopamine receptorHomo sapiens (human)0.025
D(1B) dopamine receptorHomo sapiens (human)0.025
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.75
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(4) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(3) dopamine receptorHomo sapiens (human)0.025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.75
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0813
E3 ubiquitin-protein ligase Mdm2Homo sapiens (human)0.205
5-hydroxytryptamine receptor 4 Rattus norvegicus (Norway rat)1.35
DBos taurus (cattle)0.3385

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cichini, G; Placheta, P; Singer, EA1
Andén, NE; Grabowska-Andén, M1

Other Studies

2 other study(ies) available for b-ht 958 and apomorphine

ArticleYear
B-HT 920 and B-HT 958: presynaptic effects on electrically evoked 3H-dopamine release from slices of rat nucleus accumbens.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Apomorphine; Azepines; Dopamine; Electric Stimulation; In Vitro Techniques; Male; Nucleus Accumbens; Phentolamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Sulpiride; Synapses

1987
B-HT 958 stimulates dopamine autoreceptors but blocks noradrenaline autoreceptors in the brain.
    The Journal of pharmacy and pharmacology, 1984, Volume: 36, Issue:11

    Topics: Adrenergic alpha-Agonists; alpha-Methyltyrosine; Animals; Apomorphine; Azepines; Brain Chemistry; Clonidine; Dihydroxyphenylalanine; Dopamine; Haloperidol; Male; Methyltyrosines; Mice; Motor Activity; Norepinephrine; Receptors, Adrenergic; Receptors, Dopamine; Reserpine; Synapses

1984