Page last updated: 2024-09-03

b 4162 and bradykinin

b 4162 has been researched along with bradykinin in 49 studies

Compound Research Comparison

Studies
(b 4162)
Trials
(b 4162)
Recent Studies (post-2010)
(b 4162)
Studies
(bradykinin)
Trials
(bradykinin)
Recent Studies (post-2010) (bradykinin)
501014,1953551,520

Protein Interaction Comparison

ProteinTaxonomyb 4162 (IC50)bradykinin (IC50)
B2 bradykinin receptorHomo sapiens (human)0.0018

Research

Studies (49)

TimeframeStudies, this research(%)All Research%
pre-199016 (32.65)18.7374
1990's31 (63.27)18.2507
2000's2 (4.08)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Borkowski, JA; Fraher, J; Hess, JF; Macneil, T; Ransom, RW; Stonesifer, GY; Strader, CD1
Brunner, HR; Nussberger, J; Pellacani, A1
Ichihara, A; Kageyama, Y; Murakami, M; Naitoh, M; Nakamoto, H; Ohishi, A; Saruta, T; Suzuki, H1
Farmer, SG; Meeker, SA; Page, CP; Seeds, EA; Wilkins, DE1
Kindgen-Milles, D; Klement, W1
Carretero, O; Fenoy, FJ; Roman, RJ; Scicli, G1
Harik, SI; Homayoun, P1
Barnes, PJ; Mak, JC1
Lerner, UH; Ljunggren, O; Stewart, JM; Vavrek, R1
Kumazawa, T; Minagawa, M; Mizumura, K; Tsujii, Y1
Brunner, HR; Gavras, H; Niederberger, M; Nussberger, J; Waeber, B1
Genden, EM; Molineaux, CJ1
Jarvis, WD; Judd, AM; Kuan, SI; Login, IS; MacLeod, RM1
McGraw, DE; Smits, GJ; Trapani, AJ1
Raich, PC; Stewart, JM; Vavrek, RJ; Zimmerman, BG1
Glorioso, N; Grazia Melis, M; Madeddu, P; Manunta, P; Pazzola, A; Soro, A; Tonolo, G; Troffa, C1
Barnes, PJ; Ichinose, M1
Aubert, JF; Brunner, HR; Nussberger, J; Stewart, JM; Vavrek, R; Waeber, B3
Dickenson, AH; Haley, JE; Schachter, M1
Beierwaltes, WH; Carretero, OA1
Jin, LS; Page, CP; Schachter, M; Seeds, E1
Franco, R; Gavras, H; Gavras, I; Mulinari, R1
Barton, S; Karpinski, E; Schachter, M2
Akahoshi, M; Carretero, OA; Scicli, AG; Yang, XP1
Berg, T; Carretero, OA; Scicli, AG; Stewart, JM; Tilley, B1
Carretero, OA; Kaldunski, ML; Roman, RJ; Scicli, AG1
Carbonell, LF; Carretero, OA; Scicli, AG; Stewart, JM1
Carbonell, LF; Carretero, OA; Madeddu, P; Scicli, AG1
Beierwaltes, WH; Carretero, OA; Scicli, AG1
DeHaas, CJ; Enna, SJ; Snyder, SH; Steranka, LR; Stewart, JM; Vavrek, RJ1
Gebhart, GF; Gutterman, DD; McDermott, DA; Meller, ST1
Chung, HY; Kim, JS; Oura, H; Yokozawa, T1
Fu, T; Gu, ZL; Xu, YH1
Chong, CK; Honrath, U; Sonnenberg, H; Veress, AT1
Bender, N; Brett, SE; Chowienczyk, PJ; Cockcroft, JR; Ritter, JM1
Chou, SP; Hsia, HC; Hsieh, JT; Luo, SF; Ong, R; Yang, CM1
Berezin, M; Prior, T; Rangachari, PK1
Fukuo, K; Momose, N; Morimoto, S; Ogihara, T1
Bergelson, BA; Gavras, H; Gavras, I; Ruocco, NA; Yu, TK1
Kato, M; Kobayashi, I; Saito, Y; Tatemoto, K1
Bellini, C; De Mattia, G; Desideri, G; Ferri, C; Santucci, A1
Anderson, S; Oyama, TT; Thompson, MM; Vora, JP1
Andoh, T; Kuraishi, Y1
Chiu, CT; Huang, SC; Lee, YS; Lin, CC; Pan, SL; Tsai, YJ; Wang, CC; Wu, WB; Yang, CM1
Asghar, AU; Bountra, C; Coleman, RA; McQueen, DS; Wheeldon, A1
Borovickova, L; Katarzyńska, J; Kwiatkowska, A; Prahl, A; Slaninová, J; Sleszyńska, M; Sobolewski, D; Wierzba, TH; Zabrocki, J1

Reviews

1 review(s) available for b 4162 and bradykinin

ArticleYear
Antagonizing and measurement: approaches to understanding of hemodynamic effects of kinins.
    Journal of cardiovascular pharmacology, 1992, Volume: 20 Suppl 9

    Topics: Amino Acid Sequence; Animals; Blood Pressure; Bradykinin; Hemodynamics; Humans; Kallikrein-Kinin System; Kallikreins; Kinins; Molecular Sequence Data; Rats; Vasoconstriction

1992

Trials

1 trial(s) available for b 4162 and bradykinin

ArticleYear
Inhibition of bradykinin-induced vasodilation in human forearm vasculature by icatibant, a potent B2-receptor antagonist.
    British journal of clinical pharmacology, 1994, Volume: 38, Issue:4

    Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Adult; Analysis of Variance; Blood Pressure; Brachial Artery; Bradykinin; Bradykinin Receptor Antagonists; Dose-Response Relationship, Drug; Double-Blind Method; Forearm; Half-Life; Humans; Infusions, Intra-Arterial; Infusions, Intravenous; Linear Models; Male; Radioimmunoassay; Regional Blood Flow; Vascular Resistance; Vasodilation

1994

Other Studies

47 other study(ies) available for b 4162 and bradykinin

ArticleYear
Differential pharmacology of cloned human and mouse B2 bradykinin receptors.
    Molecular pharmacology, 1994, Volume: 45, Issue:1

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; DNA, Complementary; Humans; Mice; Molecular Sequence Data; Receptors, Bradykinin; Species Specificity

1994
Depressor systems contribute to hypertension induced by glucocorticoid excess in dogs.
    Journal of hypertension, 1992, Volume: 10, Issue:6

    Topics: Animals; Blood Pressure; Bradykinin; Dexamethasone; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Glucocorticoids; Hypertension; Indomethacin; Kallikrein-Kinin System; Male; Prostaglandins; Time Factors

1992
Effects of bradykinin receptor antagonists on antigen-induced respiratory distress, airway hyperresponsiveness and eosinophilia in guinea-pigs.
    British journal of pharmacology, 1992, Volume: 107, Issue:3

    Topics: Acetylcholine; Animals; Bradykinin; Bronchial Hyperreactivity; Dose-Response Relationship, Drug; Female; Guinea Pigs; Humans; Infant, Newborn; Male; Ovalbumin; Pulmonary Eosinophilia; Receptors, Bradykinin; Receptors, Neurotransmitter; Respiratory Distress Syndrome, Newborn

1992
Pain and inflammation evoked in human skin by bradykinin receptor antagonists.
    European journal of pharmacology, 1992, Jul-21, Volume: 218, Issue:1

    Topics: Bradykinin; Dose-Response Relationship, Drug; Histamine Release; Humans; Inflammation; Male; Pain; Receptors, Bradykinin; Receptors, Neurotransmitter; Skin

1992
Effect of an angiotensin II and a kinin receptor antagonist on the renal hemodynamic response to captopril.
    Hypertension (Dallas, Tex. : 1979), 1991, Volume: 17, Issue:6 Pt 2

    Topics: Angiotensin II; Animals; Bradykinin; Captopril; Hemodynamics; Imidazoles; Kinins; Lasers; Losartan; Punctures; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter; Renal Circulation; Tetrazoles; Ultrasonography

1991
Bradykinin receptors of cerebral microvessels stimulate phosphoinositide turnover.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1991, Volume: 11, Issue:4

    Topics: Animals; Binding, Competitive; Bradykinin; Brain; Hydrolysis; Inositol Phosphates; Male; Microcirculation; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter; Swine

1991
Autoradiographic visualization of bradykinin receptors in human and guinea pig lung.
    European journal of pharmacology, 1991, Feb-26, Volume: 194, Issue:1

    Topics: Adult; Aged; Animals; Autoradiography; Bradykinin; Guinea Pigs; Humans; In Vitro Techniques; Kinetics; Lung; Male; Middle Aged; Receptors, Bradykinin; Receptors, Neurotransmitter; Species Specificity

1991
Bradykinin-induced burst of prostaglandin formation in osteoblasts is mediated via B2 bradykinin receptors.
    Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 1991, Volume: 6, Issue:8

    Topics: Amino Acid Sequence; Animals; Binding Sites; Bradykinin; Dinoprostone; Epoprostenol; Mice; Molecular Sequence Data; Osteoblasts; Receptors, Bradykinin; Receptors, Neurotransmitter

1991
Sensitizing effects of bradykinin on the heat responses of the visceral nociceptor.
    Journal of neurophysiology, 1991, Volume: 66, Issue:6

    Topics: Analgesics; Animals; Bradykinin; Dogs; Epididymis; Hot Temperature; Male; Nociceptors; Pain; Peripheral Nerves; Receptors, Bradykinin; Receptors, Neurotransmitter; Testis

1991
Hemodynamic effects of a kinin antagonist.
    Journal of cardiovascular pharmacology, 1990, Volume: 15 Suppl 6

    Topics: Amino Acid Sequence; Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Body Weight; Bradykinin; Heart Rate; Hemodynamics; Kinins; Male; Molecular Sequence Data; Rats; Rats, Inbred Strains; Splanchnic Nerves

1990
Inhibition of endopeptidase-24.15 decreases blood pressure in normotensive rats.
    Hypertension (Dallas, Tex. : 1979), 1991, Volume: 18, Issue:3

    Topics: Animals; Blood Pressure; Bradykinin; Male; Metalloendopeptidases; Oligopeptides; Rats; Rats, Inbred Strains; Reference Values

1991
Physiological and biochemical effects of bradykinin and lys-bradykinin in pituitary cells.
    Molecular and cellular endocrinology, 1990, Sep-10, Volume: 72, Issue:3

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Bradykinin; Calcium; Cells, Cultured; Dopamine; Female; Growth Hormone; Inositol Phosphates; Kallidin; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter; Secretory Rate; Stimulation, Chemical

1990
Interaction of ANP and bradykinin during endopeptidase 24.11 inhibition: renal effects.
    The American journal of physiology, 1990, Volume: 258, Issue:5 Pt 2

    Topics: Animals; Atrial Natriuretic Factor; Bradykinin; Captopril; Diuretics; Drug Synergism; Kidney; Male; Natriuresis; Neprilysin; Peptide Fragments; Rats; Rats, Inbred Strains; Thiorphan

1990
Bradykinin contribution to renal blood flow effect of angiotensin converting enzyme inhibitor in the conscious sodium-restricted dog.
    Circulation research, 1990, Volume: 66, Issue:1

    Topics: Acetylcholine; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Bradykinin; Consciousness; Diet, Sodium-Restricted; Dogs; Enalaprilat; Female; Male; Renal Circulation; Renin-Angiotensin System; Saralasin

1990
Effect of a kinin antagonist on renal function and haemodynamics during alterations in sodium balance in conscious normotensive rats.
    Clinical science (London, England : 1979), 1990, Volume: 78, Issue:2

    Topics: Animals; Blood Pressure; Bradykinin; Diet; Hemodynamics; Kidney; Male; Rats; Rats, Inbred Strains; Renal Circulation; Sodium

1990
Bradykinin-induced airway microvascular leakage and bronchoconstriction are mediated via a bradykinin B2 receptor.
    The American review of respiratory disease, 1990, Volume: 142, Issue:5

    Topics: Animals; Bradykinin; Bronchoconstriction; Capillary Permeability; Guinea Pigs; Male; Receptors, Bradykinin; Receptors, Neurotransmitter; Respiratory System

1990
Influence of endogenous bradykinin on acute blood pressure response to vasopressors in normotensive rats assessed with a bradykinin antagonist.
    Journal of cardiovascular pharmacology, 1988, Volume: 11, Issue:1

    Topics: Angiotensin II; Animals; Blood Pressure; Bradykinin; Heart Rate; Kallikreins; Kinins; Male; Methoxamine; Oligopeptides; Rats; Rats, Inbred Strains; Vasoconstrictor Agents; Vasopressins

1988
Electrophysiological evidence for a role of bradykinin in chemical nociception in the rat.
    Neuroscience letters, 1989, Feb-13, Volume: 97, Issue:1-2

    Topics: Action Potentials; Animals; Bradykinin; Male; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter; Spinal Cord

1989
Kinin antagonist reverses converting enzyme inhibitor-stimulated vascular prostaglandin I2 synthesis.
    Hypertension (Dallas, Tex. : 1979), 1989, Volume: 13, Issue:6 Pt 2

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Aorta; Bradykinin; Captopril; Enalapril; Enalaprilat; Epoprostenol; In Vitro Techniques; Kidney Cortex; Kinins; Male; Prostaglandins; Rats; Rats, Inbred Strains

1989
Inhibition of bradykinin-induced bronchoconstriction in the guinea-pig by a synthetic B2 receptor antagonist.
    British journal of pharmacology, 1989, Volume: 97, Issue:2

    Topics: Acetylcholine; Animals; Blood Pressure; Bombesin; Bradykinin; Bronchodilator Agents; Electric Stimulation; Guinea Pigs; Histamine; In Vitro Techniques; Male; Platelet Activating Factor; Receptors, Bradykinin; Receptors, Neurotransmitter; Respiration; Time Factors

1989
Bradykinin antagonism and prostaglandins in blood pressure regulation.
    Hypertension (Dallas, Tex. : 1979), 1989, Volume: 13, Issue:6 Pt 2

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Bradykinin; Cyclooxygenase Inhibitors; Heart Rate; Indomethacin; Male; Prazosin; Prostaglandins; Rats; Rats, Inbred Strains

1989
The effect of a bradykinin antagonist on vasodilatation in the cat and rabbit.
    Advances in experimental medicine and biology, 1989, Volume: 247A

    Topics: Animals; Blood Pressure; Bradykinin; Cats; Dose-Response Relationship, Drug; Electric Stimulation; Male; Parasympathetic Nervous System; Rabbits; Regional Blood Flow; Submandibular Gland; Vasodilation

1989
Effects on blood pressure of intracerebroventricular administration of a kinin antagonist.
    Advances in experimental medicine and biology, 1989, Volume: 247A

    Topics: Animals; Blood Pressure; Bradykinin; Cerebral Ventricles; Injections, Intraventricular; Male; Rats; Rats, Inbred Strains; Reference Values

1989
Role of kinin in regulation of rat submandibular gland blood flow.
    Hypertension (Dallas, Tex. : 1979), 1989, Volume: 14, Issue:1

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Bradykinin; Kinins; Male; Rats; Rats, Inbred Strains; Regional Blood Flow; Submandibular Gland; Sympathetic Nervous System; Vasodilation

1989
Influence of kinins and angiotensin II on the regulation of papillary blood flow.
    The American journal of physiology, 1988, Volume: 255, Issue:4 Pt 2

    Topics: Angiotensin II; Animals; Bicarbonates; Bradykinin; Enalapril; Glomerular Filtration Rate; Glycopeptides; Kidney Cortex; Kidney Medulla; Kinins; Male; Rats; Rats, Inbred Strains; Reference Values; Regional Blood Flow; Saralasin; Sodium; Sodium Bicarbonate

1988
Effect of a kinin antagonist on the acute antihypertensive activity of enalaprilat in severe hypertension.
    Hypertension (Dallas, Tex. : 1979), 1988, Volume: 11, Issue:3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Bradykinin; Enalapril; Enalaprilat; Hypertension; Kinins; Male; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter

1988
[Attenuation of the vasopressor effect of angiotensin II, vasopressin and alpha 1-adrenergic stimulation by bradykinin].
    Archives des maladies du coeur et des vaisseaux, 1987, Volume: 80, Issue:6

    Topics: Angiotensin II; Animals; Blood Pressure; Bradykinin; Lypressin; Male; Methoxamine; Oligopeptides; Rats; Rats, Inbred Strains

1987
The effect of a bradykinin antagonist on vasodilator responses with particular reference to the submandibular gland of the cat.
    Experientia, 1988, Oct-15, Volume: 44, Issue:10

    Topics: Animals; Blood Pressure; Bradykinin; Cats; Electric Stimulation; Female; Male; Parasympathetic Nervous System; Submandibular Gland; Vasodilation

1988
Effects of a kinin antagonist on mean blood pressure.
    Hypertension (Dallas, Tex. : 1979), 1988, Volume: 11, Issue:2 Pt 2

    Topics: Adrenal Glands; Animals; Blood Pressure; Bradykinin; Consciousness; Kidney; Kinins; Oligopeptides; Pressoreceptors; Rats

1988
Renal hemodynamics in response to a kinin analogue antagonist.
    The American journal of physiology, 1988, Volume: 255, Issue:3 Pt 2

    Topics: Animals; Bradykinin; Diet, Sodium-Restricted; Diuresis; Dogs; Female; Glomerular Filtration Rate; Reference Values; Regional Blood Flow; Renal Circulation; Sodium; Vascular Resistance

1988
Influence of bradykinin on blood pressure regulation of spontaneously hypertensive rats maintained on different sodium intakes.
    Clinical and experimental pharmacology & physiology, 1987, Volume: 14, Issue:8

    Topics: Animals; Blood Pressure; Bradykinin; Hypertension; In Vitro Techniques; Male; Oligopeptides; Rats; Rats, Inbred SHR; Sodium, Dietary

1987
Antinociceptive effects of bradykinin antagonists.
    European journal of pharmacology, 1987, Apr-14, Volume: 136, Issue:2

    Topics: Analgesics; Animals; Bradykinin; Mice; Uric Acid

1987
Use of an indwelling catheter for examining cardiovascular responses to pericardial administration of bradykinin in rat.
    Cardiovascular research, 1995, Volume: 30, Issue:1

    Topics: Animals; Blood Pressure; Bradykinin; Bradykinin Receptor Antagonists; Catheters, Indwelling; Chloralose; Dose-Response Relationship, Drug; Heart Rate; Male; Models, Biological; Pentobarbital; Pericardium; Rats; Rats, Sprague-Dawley; Time Factors

1995
The promoting action of magnesium lithospermate B on the kinin-prostaglandin E2 system in the kidney.
    Pharmacology & toxicology, 1995, Volume: 76, Issue:4

    Topics: Animals; Arachidonic Acid; Benzofurans; Bradykinin; Dinoprostone; Drugs, Chinese Herbal; Kidney; Male; Microsomes; Oxygen; Rats; Rats, Wistar; Receptors, Bradykinin; Thiobarbituric Acid Reactive Substances

1995
Modulation of bradykinin-induced intracellular Ca2+ oscillations in v-Ki-ras-transformed fibroblasts.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1994, Volume: 15, Issue:6

    Topics: 3T3 Cells; Animals; Bradykinin; Bradykinin Receptor Antagonists; Calcium Channels; Calcium-Transporting ATPases; Genes, ras; Mice; Terpenes; Thapsigargin

1994
Effect of bradykinin B2 receptor antagonist and indomethacin on natriuretic and hypotensive responses to atrial natriuretic factor.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:12

    Topics: Animals; Atrial Natriuretic Factor; Blood Pressure; Bradykinin; Bradykinin Receptor Antagonists; Indomethacin; Male; Natriuresis; Prostaglandins; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B2

1994
Bradykinin-stimulated phosphoinositide metabolism in cultured canine tracheal smooth muscle cells.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: Animals; Bradykinin; Calcium; Cells, Cultured; Dogs; Down-Regulation; Female; GTP-Binding Proteins; Hydrolysis; Kallidin; Male; Muscle, Smooth; Phosphatidylinositols; Protein Kinase C; Receptors, Bradykinin; Tetradecanoylphorbol Acetate; Trachea

1994
Effects of bradykinin on the canine proximal colon.
    Regulatory peptides, 1993, Jul-23, Volume: 46, Issue:3

    Topics: Amino Acid Sequence; Animals; Bradykinin; Colon; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Electrophysiology; Epithelium; Female; In Vitro Techniques; Indomethacin; Intestinal Mucosa; Male; Molecular Sequence Data; Tetrodotoxin

1993
Captopril inhibits endothelin-1 secretion from endothelial cells through bradykinin.
    Hypertension (Dallas, Tex. : 1979), 1993, Volume: 21, Issue:6 Pt 2

    Topics: Arginine; Bradykinin; Captopril; Cells, Cultured; Endothelins; Endothelium, Vascular; Humans; Nitric Oxide; Nitroarginine; Receptors, Bradykinin; Receptors, Neurotransmitter

1993
Augmentation of coronary blood flow by ACE inhibition: role of angiotensin and bradykinin.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 1995, Volume: 17, Issue:7

    Topics: Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Biphenyl Compounds; Blood Flow Velocity; Blood Pressure; Bradykinin; Captopril; Coronary Vessels; Imidazoles; Losartan; Perfusion; Swine; Tetrazoles

1995
Effects of bradykinin on the intracellular calcium concentration of pancreatic acinar AR42J cells.
    Life sciences, 1996, Volume: 58, Issue:18

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Calcium; Cell Line; Dexamethasone; Dose-Response Relationship, Drug; Intracellular Fluid; Neomycin; Pancreas; Rats

1996
Effects of ACE inhibition on spontaneous and insulin-stimulated endothelin-1 secretion: in vitro and in vivo studies.
    Diabetes, 1997, Volume: 46, Issue:1

    Topics: Adult; Amnion; Angiotensin-Converting Enzyme Inhibitors; Blood Glucose; Bradykinin; Captopril; Cell Membrane Permeability; Cells, Cultured; Cholesterol; Cholesterol, HDL; Cholesterol, LDL; Cholesterol, VLDL; Endothelin-1; Endothelium, Vascular; Glucose Tolerance Test; Humans; Hypertension; Insulin; Male; Nitric Oxide; Reference Values; Umbilical Veins

1997
Interactions of the kallikrein-kinin and renin-angiotensin systems in experimental diabetes.
    Diabetes, 1997, Volume: 46, Issue:1

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Glucose; Body Weight; Bradykinin; Bradykinin Receptor Antagonists; Diabetes Mellitus, Experimental; Glomerular Filtration Rate; Hemodynamics; Hyperglycemia; Kallikreins; Kidney; Kinins; Male; Organ Size; Ramipril; Rats; Rats, Wistar; Receptor, Bradykinin B2; Renal Circulation; Renin-Angiotensin System

1997
Quantitative determination of endogenous nitric oxide in the mouse skin in vivo by microdialysis.
    European journal of pharmacology, 1997, Aug-13, Volume: 332, Issue:3

    Topics: Animals; Benzoates; Bradykinin; Bradykinin Receptor Antagonists; Enzyme Inhibitors; Imidazoles; Male; Mice; Mice, Inbred ICR; Microdialysis; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Receptor, Bradykinin B2; Skin

1997
Pharmacological and functional characterization of bradykinin receptors in rat cultured vascular smooth muscle cells.
    Cellular signalling, 1999, Volume: 11, Issue:12

    Topics: Animals; Aorta; Bradykinin; Calcium; Calcium Channel Blockers; Calcium Signaling; Cells, Cultured; Enzyme Activation; Inositol Phosphates; Kallidin; Muscle Contraction; Muscle Proteins; Muscle, Smooth, Vascular; Nifedipine; Pertussis Toxin; Phosphatidylinositol Diacylglycerol-Lyase; Phosphatidylinositols; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Type C Phospholipases; Verapamil; Virulence Factors, Bordetella

1999
Hoe 140 and pseudo-irreversible antagonism in the rat vas deferens in vitro.
    European journal of pharmacology, 2000, Jun-09, Volume: 398, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Angiotensin II; Animals; Bradykinin; Bradykinin Receptor Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Rats; Rats, Wistar; Vas Deferens

2000
New bradykinin B(2) receptor antagonists - influence of C-terminal segment modifications on their pharmacological properties.
    Acta biochimica Polonica, 2009, Volume: 56, Issue:4

    Topics: Amino Acid Sequence; Animals; Blood Pressure; Bradykinin; Bradykinin B2 Receptor Antagonists; Female; Rats; Rats, Wistar; Structure-Activity Relationship; Uterine Contraction

2009