b 4162 has been researched along with bradykinin in 49 studies
Studies (b 4162) | Trials (b 4162) | Recent Studies (post-2010) (b 4162) | Studies (bradykinin) | Trials (bradykinin) | Recent Studies (post-2010) (bradykinin) |
---|---|---|---|---|---|
50 | 1 | 0 | 14,195 | 355 | 1,520 |
Protein | Taxonomy | b 4162 (IC50) | bradykinin (IC50) |
---|---|---|---|
B2 bradykinin receptor | Homo sapiens (human) | 0.0018 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 16 (32.65) | 18.7374 |
1990's | 31 (63.27) | 18.2507 |
2000's | 2 (4.08) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Borkowski, JA; Fraher, J; Hess, JF; Macneil, T; Ransom, RW; Stonesifer, GY; Strader, CD | 1 |
Brunner, HR; Nussberger, J; Pellacani, A | 1 |
Ichihara, A; Kageyama, Y; Murakami, M; Naitoh, M; Nakamoto, H; Ohishi, A; Saruta, T; Suzuki, H | 1 |
Farmer, SG; Meeker, SA; Page, CP; Seeds, EA; Wilkins, DE | 1 |
Kindgen-Milles, D; Klement, W | 1 |
Carretero, O; Fenoy, FJ; Roman, RJ; Scicli, G | 1 |
Harik, SI; Homayoun, P | 1 |
Barnes, PJ; Mak, JC | 1 |
Lerner, UH; Ljunggren, O; Stewart, JM; Vavrek, R | 1 |
Kumazawa, T; Minagawa, M; Mizumura, K; Tsujii, Y | 1 |
Brunner, HR; Gavras, H; Niederberger, M; Nussberger, J; Waeber, B | 1 |
Genden, EM; Molineaux, CJ | 1 |
Jarvis, WD; Judd, AM; Kuan, SI; Login, IS; MacLeod, RM | 1 |
McGraw, DE; Smits, GJ; Trapani, AJ | 1 |
Raich, PC; Stewart, JM; Vavrek, RJ; Zimmerman, BG | 1 |
Glorioso, N; Grazia Melis, M; Madeddu, P; Manunta, P; Pazzola, A; Soro, A; Tonolo, G; Troffa, C | 1 |
Barnes, PJ; Ichinose, M | 1 |
Aubert, JF; Brunner, HR; Nussberger, J; Stewart, JM; Vavrek, R; Waeber, B | 3 |
Dickenson, AH; Haley, JE; Schachter, M | 1 |
Beierwaltes, WH; Carretero, OA | 1 |
Jin, LS; Page, CP; Schachter, M; Seeds, E | 1 |
Franco, R; Gavras, H; Gavras, I; Mulinari, R | 1 |
Barton, S; Karpinski, E; Schachter, M | 2 |
Akahoshi, M; Carretero, OA; Scicli, AG; Yang, XP | 1 |
Berg, T; Carretero, OA; Scicli, AG; Stewart, JM; Tilley, B | 1 |
Carretero, OA; Kaldunski, ML; Roman, RJ; Scicli, AG | 1 |
Carbonell, LF; Carretero, OA; Scicli, AG; Stewart, JM | 1 |
Carbonell, LF; Carretero, OA; Madeddu, P; Scicli, AG | 1 |
Beierwaltes, WH; Carretero, OA; Scicli, AG | 1 |
DeHaas, CJ; Enna, SJ; Snyder, SH; Steranka, LR; Stewart, JM; Vavrek, RJ | 1 |
Gebhart, GF; Gutterman, DD; McDermott, DA; Meller, ST | 1 |
Chung, HY; Kim, JS; Oura, H; Yokozawa, T | 1 |
Fu, T; Gu, ZL; Xu, YH | 1 |
Chong, CK; Honrath, U; Sonnenberg, H; Veress, AT | 1 |
Bender, N; Brett, SE; Chowienczyk, PJ; Cockcroft, JR; Ritter, JM | 1 |
Chou, SP; Hsia, HC; Hsieh, JT; Luo, SF; Ong, R; Yang, CM | 1 |
Berezin, M; Prior, T; Rangachari, PK | 1 |
Fukuo, K; Momose, N; Morimoto, S; Ogihara, T | 1 |
Bergelson, BA; Gavras, H; Gavras, I; Ruocco, NA; Yu, TK | 1 |
Kato, M; Kobayashi, I; Saito, Y; Tatemoto, K | 1 |
Bellini, C; De Mattia, G; Desideri, G; Ferri, C; Santucci, A | 1 |
Anderson, S; Oyama, TT; Thompson, MM; Vora, JP | 1 |
Andoh, T; Kuraishi, Y | 1 |
Chiu, CT; Huang, SC; Lee, YS; Lin, CC; Pan, SL; Tsai, YJ; Wang, CC; Wu, WB; Yang, CM | 1 |
Asghar, AU; Bountra, C; Coleman, RA; McQueen, DS; Wheeldon, A | 1 |
Borovickova, L; Katarzyńska, J; Kwiatkowska, A; Prahl, A; Slaninová, J; Sleszyńska, M; Sobolewski, D; Wierzba, TH; Zabrocki, J | 1 |
1 review(s) available for b 4162 and bradykinin
Article | Year |
---|---|
Antagonizing and measurement: approaches to understanding of hemodynamic effects of kinins.
Topics: Amino Acid Sequence; Animals; Blood Pressure; Bradykinin; Hemodynamics; Humans; Kallikrein-Kinin System; Kallikreins; Kinins; Molecular Sequence Data; Rats; Vasoconstriction | 1992 |
1 trial(s) available for b 4162 and bradykinin
Article | Year |
---|---|
Inhibition of bradykinin-induced vasodilation in human forearm vasculature by icatibant, a potent B2-receptor antagonist.
Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Adult; Analysis of Variance; Blood Pressure; Brachial Artery; Bradykinin; Bradykinin Receptor Antagonists; Dose-Response Relationship, Drug; Double-Blind Method; Forearm; Half-Life; Humans; Infusions, Intra-Arterial; Infusions, Intravenous; Linear Models; Male; Radioimmunoassay; Regional Blood Flow; Vascular Resistance; Vasodilation | 1994 |
47 other study(ies) available for b 4162 and bradykinin
Article | Year |
---|---|
Differential pharmacology of cloned human and mouse B2 bradykinin receptors.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; DNA, Complementary; Humans; Mice; Molecular Sequence Data; Receptors, Bradykinin; Species Specificity | 1994 |
Depressor systems contribute to hypertension induced by glucocorticoid excess in dogs.
Topics: Animals; Blood Pressure; Bradykinin; Dexamethasone; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Glucocorticoids; Hypertension; Indomethacin; Kallikrein-Kinin System; Male; Prostaglandins; Time Factors | 1992 |
Effects of bradykinin receptor antagonists on antigen-induced respiratory distress, airway hyperresponsiveness and eosinophilia in guinea-pigs.
Topics: Acetylcholine; Animals; Bradykinin; Bronchial Hyperreactivity; Dose-Response Relationship, Drug; Female; Guinea Pigs; Humans; Infant, Newborn; Male; Ovalbumin; Pulmonary Eosinophilia; Receptors, Bradykinin; Receptors, Neurotransmitter; Respiratory Distress Syndrome, Newborn | 1992 |
Pain and inflammation evoked in human skin by bradykinin receptor antagonists.
Topics: Bradykinin; Dose-Response Relationship, Drug; Histamine Release; Humans; Inflammation; Male; Pain; Receptors, Bradykinin; Receptors, Neurotransmitter; Skin | 1992 |
Effect of an angiotensin II and a kinin receptor antagonist on the renal hemodynamic response to captopril.
Topics: Angiotensin II; Animals; Bradykinin; Captopril; Hemodynamics; Imidazoles; Kinins; Lasers; Losartan; Punctures; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter; Renal Circulation; Tetrazoles; Ultrasonography | 1991 |
Bradykinin receptors of cerebral microvessels stimulate phosphoinositide turnover.
Topics: Animals; Binding, Competitive; Bradykinin; Brain; Hydrolysis; Inositol Phosphates; Male; Microcirculation; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter; Swine | 1991 |
Autoradiographic visualization of bradykinin receptors in human and guinea pig lung.
Topics: Adult; Aged; Animals; Autoradiography; Bradykinin; Guinea Pigs; Humans; In Vitro Techniques; Kinetics; Lung; Male; Middle Aged; Receptors, Bradykinin; Receptors, Neurotransmitter; Species Specificity | 1991 |
Bradykinin-induced burst of prostaglandin formation in osteoblasts is mediated via B2 bradykinin receptors.
Topics: Amino Acid Sequence; Animals; Binding Sites; Bradykinin; Dinoprostone; Epoprostenol; Mice; Molecular Sequence Data; Osteoblasts; Receptors, Bradykinin; Receptors, Neurotransmitter | 1991 |
Sensitizing effects of bradykinin on the heat responses of the visceral nociceptor.
Topics: Analgesics; Animals; Bradykinin; Dogs; Epididymis; Hot Temperature; Male; Nociceptors; Pain; Peripheral Nerves; Receptors, Bradykinin; Receptors, Neurotransmitter; Testis | 1991 |
Hemodynamic effects of a kinin antagonist.
Topics: Amino Acid Sequence; Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Body Weight; Bradykinin; Heart Rate; Hemodynamics; Kinins; Male; Molecular Sequence Data; Rats; Rats, Inbred Strains; Splanchnic Nerves | 1990 |
Inhibition of endopeptidase-24.15 decreases blood pressure in normotensive rats.
Topics: Animals; Blood Pressure; Bradykinin; Male; Metalloendopeptidases; Oligopeptides; Rats; Rats, Inbred Strains; Reference Values | 1991 |
Physiological and biochemical effects of bradykinin and lys-bradykinin in pituitary cells.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Bradykinin; Calcium; Cells, Cultured; Dopamine; Female; Growth Hormone; Inositol Phosphates; Kallidin; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter; Secretory Rate; Stimulation, Chemical | 1990 |
Interaction of ANP and bradykinin during endopeptidase 24.11 inhibition: renal effects.
Topics: Animals; Atrial Natriuretic Factor; Bradykinin; Captopril; Diuretics; Drug Synergism; Kidney; Male; Natriuresis; Neprilysin; Peptide Fragments; Rats; Rats, Inbred Strains; Thiorphan | 1990 |
Bradykinin contribution to renal blood flow effect of angiotensin converting enzyme inhibitor in the conscious sodium-restricted dog.
Topics: Acetylcholine; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Bradykinin; Consciousness; Diet, Sodium-Restricted; Dogs; Enalaprilat; Female; Male; Renal Circulation; Renin-Angiotensin System; Saralasin | 1990 |
Effect of a kinin antagonist on renal function and haemodynamics during alterations in sodium balance in conscious normotensive rats.
Topics: Animals; Blood Pressure; Bradykinin; Diet; Hemodynamics; Kidney; Male; Rats; Rats, Inbred Strains; Renal Circulation; Sodium | 1990 |
Bradykinin-induced airway microvascular leakage and bronchoconstriction are mediated via a bradykinin B2 receptor.
Topics: Animals; Bradykinin; Bronchoconstriction; Capillary Permeability; Guinea Pigs; Male; Receptors, Bradykinin; Receptors, Neurotransmitter; Respiratory System | 1990 |
Influence of endogenous bradykinin on acute blood pressure response to vasopressors in normotensive rats assessed with a bradykinin antagonist.
Topics: Angiotensin II; Animals; Blood Pressure; Bradykinin; Heart Rate; Kallikreins; Kinins; Male; Methoxamine; Oligopeptides; Rats; Rats, Inbred Strains; Vasoconstrictor Agents; Vasopressins | 1988 |
Electrophysiological evidence for a role of bradykinin in chemical nociception in the rat.
Topics: Action Potentials; Animals; Bradykinin; Male; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter; Spinal Cord | 1989 |
Kinin antagonist reverses converting enzyme inhibitor-stimulated vascular prostaglandin I2 synthesis.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Aorta; Bradykinin; Captopril; Enalapril; Enalaprilat; Epoprostenol; In Vitro Techniques; Kidney Cortex; Kinins; Male; Prostaglandins; Rats; Rats, Inbred Strains | 1989 |
Inhibition of bradykinin-induced bronchoconstriction in the guinea-pig by a synthetic B2 receptor antagonist.
Topics: Acetylcholine; Animals; Blood Pressure; Bombesin; Bradykinin; Bronchodilator Agents; Electric Stimulation; Guinea Pigs; Histamine; In Vitro Techniques; Male; Platelet Activating Factor; Receptors, Bradykinin; Receptors, Neurotransmitter; Respiration; Time Factors | 1989 |
Bradykinin antagonism and prostaglandins in blood pressure regulation.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Bradykinin; Cyclooxygenase Inhibitors; Heart Rate; Indomethacin; Male; Prazosin; Prostaglandins; Rats; Rats, Inbred Strains | 1989 |
The effect of a bradykinin antagonist on vasodilatation in the cat and rabbit.
Topics: Animals; Blood Pressure; Bradykinin; Cats; Dose-Response Relationship, Drug; Electric Stimulation; Male; Parasympathetic Nervous System; Rabbits; Regional Blood Flow; Submandibular Gland; Vasodilation | 1989 |
Effects on blood pressure of intracerebroventricular administration of a kinin antagonist.
Topics: Animals; Blood Pressure; Bradykinin; Cerebral Ventricles; Injections, Intraventricular; Male; Rats; Rats, Inbred Strains; Reference Values | 1989 |
Role of kinin in regulation of rat submandibular gland blood flow.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Bradykinin; Kinins; Male; Rats; Rats, Inbred Strains; Regional Blood Flow; Submandibular Gland; Sympathetic Nervous System; Vasodilation | 1989 |
Influence of kinins and angiotensin II on the regulation of papillary blood flow.
Topics: Angiotensin II; Animals; Bicarbonates; Bradykinin; Enalapril; Glomerular Filtration Rate; Glycopeptides; Kidney Cortex; Kidney Medulla; Kinins; Male; Rats; Rats, Inbred Strains; Reference Values; Regional Blood Flow; Saralasin; Sodium; Sodium Bicarbonate | 1988 |
Effect of a kinin antagonist on the acute antihypertensive activity of enalaprilat in severe hypertension.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Bradykinin; Enalapril; Enalaprilat; Hypertension; Kinins; Male; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter | 1988 |
[Attenuation of the vasopressor effect of angiotensin II, vasopressin and alpha 1-adrenergic stimulation by bradykinin].
Topics: Angiotensin II; Animals; Blood Pressure; Bradykinin; Lypressin; Male; Methoxamine; Oligopeptides; Rats; Rats, Inbred Strains | 1987 |
The effect of a bradykinin antagonist on vasodilator responses with particular reference to the submandibular gland of the cat.
Topics: Animals; Blood Pressure; Bradykinin; Cats; Electric Stimulation; Female; Male; Parasympathetic Nervous System; Submandibular Gland; Vasodilation | 1988 |
Effects of a kinin antagonist on mean blood pressure.
Topics: Adrenal Glands; Animals; Blood Pressure; Bradykinin; Consciousness; Kidney; Kinins; Oligopeptides; Pressoreceptors; Rats | 1988 |
Renal hemodynamics in response to a kinin analogue antagonist.
Topics: Animals; Bradykinin; Diet, Sodium-Restricted; Diuresis; Dogs; Female; Glomerular Filtration Rate; Reference Values; Regional Blood Flow; Renal Circulation; Sodium; Vascular Resistance | 1988 |
Influence of bradykinin on blood pressure regulation of spontaneously hypertensive rats maintained on different sodium intakes.
Topics: Animals; Blood Pressure; Bradykinin; Hypertension; In Vitro Techniques; Male; Oligopeptides; Rats; Rats, Inbred SHR; Sodium, Dietary | 1987 |
Antinociceptive effects of bradykinin antagonists.
Topics: Analgesics; Animals; Bradykinin; Mice; Uric Acid | 1987 |
Use of an indwelling catheter for examining cardiovascular responses to pericardial administration of bradykinin in rat.
Topics: Animals; Blood Pressure; Bradykinin; Bradykinin Receptor Antagonists; Catheters, Indwelling; Chloralose; Dose-Response Relationship, Drug; Heart Rate; Male; Models, Biological; Pentobarbital; Pericardium; Rats; Rats, Sprague-Dawley; Time Factors | 1995 |
The promoting action of magnesium lithospermate B on the kinin-prostaglandin E2 system in the kidney.
Topics: Animals; Arachidonic Acid; Benzofurans; Bradykinin; Dinoprostone; Drugs, Chinese Herbal; Kidney; Male; Microsomes; Oxygen; Rats; Rats, Wistar; Receptors, Bradykinin; Thiobarbituric Acid Reactive Substances | 1995 |
Modulation of bradykinin-induced intracellular Ca2+ oscillations in v-Ki-ras-transformed fibroblasts.
Topics: 3T3 Cells; Animals; Bradykinin; Bradykinin Receptor Antagonists; Calcium Channels; Calcium-Transporting ATPases; Genes, ras; Mice; Terpenes; Thapsigargin | 1994 |
Effect of bradykinin B2 receptor antagonist and indomethacin on natriuretic and hypotensive responses to atrial natriuretic factor.
Topics: Animals; Atrial Natriuretic Factor; Blood Pressure; Bradykinin; Bradykinin Receptor Antagonists; Indomethacin; Male; Natriuresis; Prostaglandins; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B2 | 1994 |
Bradykinin-stimulated phosphoinositide metabolism in cultured canine tracheal smooth muscle cells.
Topics: Animals; Bradykinin; Calcium; Cells, Cultured; Dogs; Down-Regulation; Female; GTP-Binding Proteins; Hydrolysis; Kallidin; Male; Muscle, Smooth; Phosphatidylinositols; Protein Kinase C; Receptors, Bradykinin; Tetradecanoylphorbol Acetate; Trachea | 1994 |
Effects of bradykinin on the canine proximal colon.
Topics: Amino Acid Sequence; Animals; Bradykinin; Colon; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Electrophysiology; Epithelium; Female; In Vitro Techniques; Indomethacin; Intestinal Mucosa; Male; Molecular Sequence Data; Tetrodotoxin | 1993 |
Captopril inhibits endothelin-1 secretion from endothelial cells through bradykinin.
Topics: Arginine; Bradykinin; Captopril; Cells, Cultured; Endothelins; Endothelium, Vascular; Humans; Nitric Oxide; Nitroarginine; Receptors, Bradykinin; Receptors, Neurotransmitter | 1993 |
Augmentation of coronary blood flow by ACE inhibition: role of angiotensin and bradykinin.
Topics: Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Biphenyl Compounds; Blood Flow Velocity; Blood Pressure; Bradykinin; Captopril; Coronary Vessels; Imidazoles; Losartan; Perfusion; Swine; Tetrazoles | 1995 |
Effects of bradykinin on the intracellular calcium concentration of pancreatic acinar AR42J cells.
Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Calcium; Cell Line; Dexamethasone; Dose-Response Relationship, Drug; Intracellular Fluid; Neomycin; Pancreas; Rats | 1996 |
Effects of ACE inhibition on spontaneous and insulin-stimulated endothelin-1 secretion: in vitro and in vivo studies.
Topics: Adult; Amnion; Angiotensin-Converting Enzyme Inhibitors; Blood Glucose; Bradykinin; Captopril; Cell Membrane Permeability; Cells, Cultured; Cholesterol; Cholesterol, HDL; Cholesterol, LDL; Cholesterol, VLDL; Endothelin-1; Endothelium, Vascular; Glucose Tolerance Test; Humans; Hypertension; Insulin; Male; Nitric Oxide; Reference Values; Umbilical Veins | 1997 |
Interactions of the kallikrein-kinin and renin-angiotensin systems in experimental diabetes.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Glucose; Body Weight; Bradykinin; Bradykinin Receptor Antagonists; Diabetes Mellitus, Experimental; Glomerular Filtration Rate; Hemodynamics; Hyperglycemia; Kallikreins; Kidney; Kinins; Male; Organ Size; Ramipril; Rats; Rats, Wistar; Receptor, Bradykinin B2; Renal Circulation; Renin-Angiotensin System | 1997 |
Quantitative determination of endogenous nitric oxide in the mouse skin in vivo by microdialysis.
Topics: Animals; Benzoates; Bradykinin; Bradykinin Receptor Antagonists; Enzyme Inhibitors; Imidazoles; Male; Mice; Mice, Inbred ICR; Microdialysis; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Receptor, Bradykinin B2; Skin | 1997 |
Pharmacological and functional characterization of bradykinin receptors in rat cultured vascular smooth muscle cells.
Topics: Animals; Aorta; Bradykinin; Calcium; Calcium Channel Blockers; Calcium Signaling; Cells, Cultured; Enzyme Activation; Inositol Phosphates; Kallidin; Muscle Contraction; Muscle Proteins; Muscle, Smooth, Vascular; Nifedipine; Pertussis Toxin; Phosphatidylinositol Diacylglycerol-Lyase; Phosphatidylinositols; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Type C Phospholipases; Verapamil; Virulence Factors, Bordetella | 1999 |
Hoe 140 and pseudo-irreversible antagonism in the rat vas deferens in vitro.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Angiotensin II; Animals; Bradykinin; Bradykinin Receptor Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Rats; Rats, Wistar; Vas Deferens | 2000 |
New bradykinin B(2) receptor antagonists - influence of C-terminal segment modifications on their pharmacological properties.
Topics: Amino Acid Sequence; Animals; Blood Pressure; Bradykinin; Bradykinin B2 Receptor Antagonists; Female; Rats; Rats, Wistar; Structure-Activity Relationship; Uterine Contraction | 2009 |