azides has been researched along with gamma-aminobutyric acid in 64 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 15 (23.44) | 18.7374 |
1990's | 30 (46.88) | 18.2507 |
2000's | 15 (23.44) | 29.6817 |
2010's | 4 (6.25) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Plourde, G; Tremblay, JP | 1 |
Mattson, ME; O'Brien, RD | 1 |
Contreras, P; Sandoval, ME; Tapia, R | 1 |
Howard, BD; Vanker, AD; Wernicke, JF | 1 |
Skolnick, P; Wong, G | 2 |
Uusi-Oukari, M | 1 |
D'Amico, E; Koob, GF; Pulvirenti, L; Rassnick, S; Riley, E; Zieglgänsberger, W | 1 |
Mehta, AK; Mhatre, M; Ticku, MK | 1 |
Lanoir, J; Pinard, R; Segu, L | 1 |
Jones, EA | 1 |
Bottlaender, M; Brouillet, E; Chavoix, C; Dodd, RH; Fournier, D; Hantraye, P; Khalili-Varasteh, M; Mazière, M | 1 |
Chen, JP; Lal, H; Martin, MW; Prather, PL; Rezazadeh, SM | 1 |
Ewert, M; Kettenmann, H; Kleingoor, C; Seeburg, PH; von Blankenfeld, G | 1 |
Biggio, G; Concas, A; Sanna, E; Santoro, G; Serra, M | 1 |
Borden, LA; Gibbs, TT | 1 |
Kulkarni, SK; Ticku, MK | 1 |
Hoffer, BJ; Palmer, MR | 1 |
McIntyre, TD; Skolnick, P; Trullas, R | 1 |
Mehta, AK; Ticku, MK | 1 |
Collins, M; Zimmerman, EF | 1 |
Möhler, H; Richards, JG | 1 |
Harlan, JT; Moore, EA; Palmer, MR; van Horne, CG | 1 |
Celentano, JJ; Farb, DH; Gibbs, TT | 1 |
Gordon-Weeks, PR; Lockerbie, RO | 1 |
Henry, JP; Isambert, MF | 1 |
Askar, A; Knödgen, B; Seiler, N | 1 |
Boublik, M; Lin, FL; Ofengand, J | 1 |
Lloyd, HG; Stone, TW | 1 |
Beal, MF; Brouillet, E; Henshaw, DR; Hyman, BT; Jenkins, BG; Rosen, BR; Schulz, JB; Sodhi, P | 1 |
Chapin, JK; Lee, RS; Maddux, BN; Shimizu, N; Smith, SS; Waterhouse, BD; Woodward, DJ | 1 |
Chapin, JK; Lee, RS; Maddus, BN; Shimizu, N; Smith, SS; Waterhouse, BD; Woodward, DJ | 1 |
Alberts, GL; Binder, JA; Dillon, GH; Im, WB; Pregenzer, JF | 1 |
Baulieu, EE; Chesnoy-Marchais, D; Hauser, CA; Robel, P | 1 |
Kettenmann, H; Kleingoor, C; Korpi, ER; Seeburg, PH | 1 |
Korpi, ER; Seeburg, PH | 1 |
Casida, JE; Goeldner, MP; Hawkinson, JE; Kapfer, I | 1 |
D'Amico, E; Koob, GF; Rassnick, S; Riley, E | 1 |
File, SE; Hogg, S; Mills, AD | 1 |
Benke, D; Benson, JA; Carter, DB; Hamilton, BJ; Knoflach, F; Lüddens, H; Mohler, H; Scheurer, L; Wang, Y | 1 |
Berning, B; Gerner, FM; Hauser, CA; Rupprecht, R; Wetzel, CH | 1 |
Firestone, LL; Homanics, GE; Korpi, ER; Mäkelä, R; Quinlan, JJ; Uusi-Oukari, M; Wisden, W | 1 |
Acri, JB; Basile, AS; Lyon, T; Witkin, JM; Wong, G | 1 |
ffrench-Mullen, JM; Gong, QH; Hsu, FC; Li, X; Markowitz, RS; Smith, SS | 1 |
Benke, D; Fritschy, JM; Honer, M; Meskenaite, V; Mohler, H; Weinmann, O | 1 |
Korpi, ER; Lüddens, H; Panula, P; Särkioja, T; Sinkkonen, ST; Tiihonen, J; Tupala, E; Uusi-Oukari, M | 1 |
Hevers, W; Korpi, ER; Lüddens, H | 1 |
Paz, L; Peter, Y; Pick, CG; Weizman, R | 1 |
Atack, J; Banks, G; Kelly, MD; Maubach, KA; Seabrook, GR; Smith, A; Whiting, PW; Wingrove, P | 1 |
Hauer, B; Hevers, W; Homanics, GE; Korpi, ER; Lüddens, H; Mihalek, RM; Sieghart, W; Sinkkonen, ST | 1 |
Assandri, R; Crestani, F; Martin, JR; Rudolph, U; Täuber, M | 1 |
Bergman, RG; Duncan, AP | 1 |
Faber, DS; Hsu, FC; Smith, SS; Waldeck, R | 1 |
Chatelain, P; Fuks, B; Gillard, M; Massingham, R; Michel, P; Vertongen, P | 1 |
Igarashi, K; Kashiwagi, K; Tomonari, Y; Uemura, T | 1 |
Foster, AC; Grigoriadis, DE; Gross, RS; Petroski, RE; Sullivan, SK; Verge, G | 1 |
Hanchar, HJ; Olsen, RW; Wallner, M | 1 |
Paul, SM | 1 |
Marszalec, W; Narahashi, T; Yamashita, M; Yeh, JZ | 1 |
Beauvois, MC; Cheng-Xue, R; Gilon, P; Guiot, Y; Henquin, JC; Mattart, L; Quoix, N; Zeinoun, Z | 1 |
Cunningham, VJ; Erritzoe, D; Hammers, A; Kalk, NJ; Lingford-Hughes, AR; Myers, JF; Nutt, DJ; Riano Barros, D; Stokes, PR; Turkheimer, FE; Watson, BJ; Wilson, SJ | 1 |
De Santis, V; Lingford-Hughes, A; Myers, J; Nutt, D; Parker, C; Quelch, D; Strege, A; Tyacke, R; Wells, L | 1 |
Banks, ML; Shelton, KL; Tracy, ME | 1 |
Blicher, JU; Brooks, DJ; Hansen, KV; Lou, HC; Mouridsen, K; Møller, A; Rømer Thomsen, K | 1 |
2 review(s) available for azides and gamma-aminobutyric acid
Article | Year |
---|---|
GABAergic mechanisms in the electrophysiological actions of ethanol on cerebellar neurons.
Topics: Action Potentials; Animals; Azides; Benzodiazepines; Carbolines; Cerebellum; Dose-Response Relationship, Drug; Ethanol; gamma-Aminobutyric Acid; Male; Neural Inhibition; Rats; Rats, Inbred Strains | 1990 |
The benzodiazepine receptor: a pharmacological control element of brain function.
Topics: Animals; Azides; Benzodiazepines; Brain; Electrophysiology; gamma-Aminobutyric Acid; Midazolam; Models, Molecular; Receptors, GABA-A | 1988 |
1 trial(s) available for azides and gamma-aminobutyric acid
Article | Year |
---|---|
Acute increases in synaptic GABA detectable in the living human brain: a [¹¹C]Ro15-4513 PET study.
Topics: Adult; Azides; Benzodiazepines; Brain; Brain Chemistry; Dose-Response Relationship, Drug; Double-Blind Method; GABA Agonists; gamma-Aminobutyric Acid; Humans; Male; Memory; Middle Aged; Nipecotic Acids; Positron-Emission Tomography; Psychomotor Performance; Radiopharmaceuticals; Receptors, GABA-A; Synapses; Tiagabine | 2014 |
61 other study(ies) available for azides and gamma-aminobutyric acid
Article | Year |
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Presynaptic modulating effects of GABA on depression, facilitation, and posttetanic potentiation of a cholinergic synapse in Aplysia californica.
Topics: Acetylcholine; Aminobutyrates; Animals; Aplysia; Azides; Bicuculline; Chlorides; gamma-Aminobutyric Acid; Lithium; Membrane Potentials; Picrotoxin; Potassium; Sodium; Synapses | 1977 |
The binding of acetylcholine to synaptic vesicles from Torpedo californica electroplax.
Topics: Acetylcholine; Animals; Azides; Choline; Chromatography, Gel; Electric Organ; Fishes; Freezing; gamma-Aminobutyric Acid; Kinetics; Neuromuscular Blocking Agents; Ouabain; Parasympatholytics; Parasympathomimetics; Preservation, Biological; Synaptic Vesicles; Temperature | 1976 |
Evidence for a role of glutamate decarboxylase activity as a regulatory mechanism of cerebral excitability.
Topics: Aminobutyrates; Animals; Azides; Brain; Carboxy-Lyases; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Glutamates; Mice; Pyridoxal Phosphate; Seizures; Time Factors | 1975 |
The mechanism of action of beta-bungarotoxin.
Topics: Adenosine Triphosphate; Animals; Ascorbic Acid; Azides; Barium; Brain; Bungarotoxins; Calcium; Carbon Radioisotopes; Catalysis; Cell Membrane; Chromatography, Thin Layer; Deoxyglucose; Dinitrophenols; Erythrocytes; Fatty Acids; gamma-Aminobutyric Acid; Glucose; Glutamates; Iodoacetates; Mitochondria; Ouabain; Phospholipases; Phospholipids; Pyruvates; Rats; Strontium; Succinates; Synaptosomes | 1975 |
High affinity ligands for 'diazepam-insensitive' benzodiazepine receptors.
Topics: Animals; Azides; Benzodiazepines; Diazepam; gamma-Aminobutyric Acid; Male; Protein Conformation; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship | 1992 |
Effect of diethyl pyrocarbonate modification of benzodiazepine receptors on [3H]Ro 15-4513 binding.
Topics: Animals; Appetite Depressants; Azides; Benzodiazepines; Carbolines; Cerebellum; Cerebral Cortex; Diazepam; Diethyl Pyrocarbonate; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tritium | 1992 |
Ro 15-4513 binding to GABAA receptors: subunit composition determines ligand efficacy.
Topics: Animals; Azides; Benzodiazepines; Binding, Competitive; Brain; Cerebellum; Diazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Ligands; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1992 |
GABA and nucleus accumbens glutamate neurotransmission modulate ethanol self-administration in rats.
Topics: 2-Amino-5-phosphonovalerate; Acamprosate; Animals; Azides; Benzodiazepines; Choice Behavior; Convulsants; Ethanol; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Infusions, Parenteral; Male; Nucleus Accumbens; Organophosphorus Compounds; Rats; Receptors, GABA-A; Receptors, Glutamate; Receptors, Neurotransmitter; Self Administration; Taurine | 1992 |
Modulation of GABAergic transmission by ethanol.
Topics: Animals; Anticonvulsants; Azides; Benzodiazepines; Brain Chemistry; Ethanol; Female; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Mice; Mice, Inbred C57BL; Pentylenetetrazole; Rats; Rats, Inbred Strains; RNA, Messenger; Seizures; Synaptic Transmission | 1992 |
Transient increase in [3H]Ro 15-4513 specific binding in the superficial gray layer of the rat superior colliculus induced by visual deafferentation.
Topics: Animals; Autoradiography; Azides; Benzodiazepines; Bicuculline; Binding, Competitive; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mesencephalon; Neurons, Afferent; Ocular Physiological Phenomena; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Superior Colliculi; Vision, Ocular; Visual Cortex | 1991 |
Benzodiazepine receptor ligands and hepatic encephalopathy: further unfolding of the GABA story.
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Brain; Central Nervous System; Flumazenil; gamma-Aminobutyric Acid; Hepatic Encephalopathy; Humans; Ligands; Neurons; Receptors, GABA-A; Synaptic Transmission | 1991 |
In vivo bidirectional modulatory effect of benzodiazepine receptor ligands on GABAergic transmission evaluated by positron emission tomography in non-human primates.
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Carbolines; Cerebral Cortex; Diazepam; Electroencephalography; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Papio; Pentylenetetrazole; Receptors, GABA-A; Seizures; Synaptic Transmission; Tomography, Emission-Computed | 1991 |
Modulation of benzodiazepine agonist and inverse-agonist receptor binding by GABA during ethanol withdrawal.
Topics: Animals; Azides; Benzodiazepines; Binding, Competitive; Brain; Cerebellum; Cerebral Cortex; Ethanol; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Male; Rats; Receptors, GABA-A; Substance Withdrawal Syndrome; Synaptic Transmission | 1991 |
Inverse but not full benzodiazepine agonists modulate recombinant alpha 6 beta 2 gamma 2 GABAA receptors in transfected human embryonic kidney cells.
Topics: Action Potentials; Azides; Benzodiazepines; Carbolines; Cells, Cultured; Ethanol; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Kidney; Receptors, GABA-A; Recombinant Proteins; Transfection | 1991 |
Ex vivo binding of t-[35S )butylbicyclophosphorothionate: a biochemical tool to study the pharmacology of ethanol at the gamma-aminobutyric acid-coupled chloride channel.
Topics: Animals; Azides; Benzodiazepines; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Diazepam; Drug Interactions; Ethanol; gamma-Aminobutyric Acid; Ion Channels; Isoniazid; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes | 1991 |
Flunitrazepam photoaffinity labeling of the GABA(A) receptor reduces inhibition of [3H]Ro15-4513 binding by GABA.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Brain; Chick Embryo; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Membranes; Photochemistry; Receptors, GABA-A | 1990 |
Chronic benzodiazepine antagonist treatment and its withdrawal upregulates components of GABA-benzodiazepine receptor ionophore complex in cerebral cortex of rat.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Convulsants; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values; Up-Regulation | 1990 |
Differences in the biophysical properties of the benzodiazepine/gamma-aminobutyric acid receptor chloride channel complex in the long-sleep and short-sleep mouse lines.
Topics: Animals; Azides; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; Heart; Ion Channels; Male; Mice; Mice, Mutant Strains; Receptors, GABA-A; Sleep | 1988 |
Ethanol potentiation of GABAergic transmission in cultured spinal cord neurons involves gamma-aminobutyric acidA-gated chloride channels.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Cells, Cultured; Chlorine; Ethanol; Female; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Mice; Mice, Inbred C57BL; Neurons; Radioisotopes; Spinal Cord | 1988 |
Chloride transport in embryonic cells: effect of ethanol and GABA.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Azides; Benzodiazepines; Biological Transport, Active; Bumetanide; Cells, Cultured; Chlorides; Embryo, Mammalian; Ethanol; Extremities; Furosemide; gamma-Aminobutyric Acid; In Vitro Techniques; Mice; Mice, Inbred C57BL | 1989 |
Antagonism of ethanol effects on cerebellar Purkinje neurons by the benzodiazepine inverse agonists Ro 15-4513 and FG 7142: electrophysiological studies.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Ethanol; gamma-Aminobutyric Acid; Heart Conduction System; In Vitro Techniques; Male; Membrane Proteins; Purkinje Fibers; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Ethanol potentiates GABA- and glycine-induced chloride currents in chick spinal cord neurons.
Topics: Animals; Azides; Benzodiazepines; Cells, Cultured; Chick Embryo; Chlorides; Ethanol; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Glycine; Membrane Potentials; Receptors, GABA-A; Receptors, Glycine; Receptors, Neurotransmitter; Spinal Cord | 1988 |
gamma-Aminobutyric acidA (GABAA) receptors modulate [3H]GABA release from isolated neuronal growth cones in the rat.
Topics: Animals; Animals, Newborn; Axons; Azides; Baclofen; Benzamides; Bicuculline; Brain; Dendrites; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Homeostasis; Muscimol; Potassium; Rats; Receptors, GABA-A; Stimulation, Chemical; Subcellular Fractions; Tritium | 1985 |
Photoaffinity labeling of the tetrabenazine binding sites of bovine chromaffin granule membranes.
Topics: Adrenal Medulla; Affinity Labels; Animals; Azides; Binding Sites; Cattle; Cell Fractionation; Chromaffin Granules; Chromaffin System; gamma-Aminobutyric Acid; Hydrogen-Ion Concentration; Indicators and Reagents; Intracellular Membranes; Kinetics; Tetrabenazine | 1985 |
The formation of gamma-aminobutyrate in liver cell nuclei.
Topics: Aminobutyrates; Animals; Azides; Brain; Cell Nucleus; Centrifugation, Density Gradient; Chromatography, Thin Layer; Cyanides; Cytosol; Dansyl Compounds; gamma-Aminobutyric Acid; Liver; Mice; Microsomes, Liver; Mitochondria, Liver; Organ Specificity; Semicarbazides; Spectrometry, Fluorescence; Subcellular Fractions; Sulfhydryl Compounds; Time Factors; Ultracentrifugation | 1973 |
Immunoelectron microscopic localization of the S19 site on the 30 S ribosomal subunit which is crosslinked to A site bound transfer RNA.
Topics: Azides; Binding Sites; Epitopes; Escherichia coli; gamma-Aminobutyric Acid; Microscopy, Electron; Models, Biological; Ribosomal Proteins; Ribosomes; RNA, Transfer, Amino Acyl | 1984 |
Factors affecting the release of purines from mouse cerebral cortex: potassium removal and metabolic inhibitors.
Topics: Animals; Antimetabolites; Azides; Cerebral Cortex; Fluorides; gamma-Aminobutyric Acid; Hydroxymercuribenzoates; In Vitro Techniques; Male; Mice; Ouabain; Potassium; Purines | 1981 |
Systemic or local administration of azide produces striatal lesions by an energy impairment-induced excitotoxic mechanism.
Topics: 3,4-Dihydroxyphenylacetic Acid; Adenosine Triphosphate; Aging; Animals; Azides; Biogenic Amines; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Functional Laterality; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Homovanillic Acid; Injections, Intraperitoneal; Lactates; Magnetic Resonance Imaging; Male; Microinjections; NADPH Dehydrogenase; Neurons; Neuropeptide Y; Neuropeptides; Neurotoxins; Oxidative Phosphorylation; Oxidative Stress; Rats; Rats, Sprague-Dawley; Sodium Azide; Somatostatin; Substance P | 1994 |
Effects of systemic and local ethanol on responses of rat cerebellar Purkinje neurons to iontophoretically applied gamma-aminobutyric acid.
Topics: Action Potentials; Animals; Azides; Benzodiazepines; Central Nervous System Depressants; Cerebellum; Drug Synergism; Electrophysiology; Ethanol; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Iontophoresis; Purkinje Cells; Rats; Rats, Sprague-Dawley | 1995 |
Effects of systemic and local ethanol on responses of rat cerebellar Purkinje neurons to iontophoretically applied norepinephrine and gamma-aminobutyric acid.
Topics: Action Potentials; Animals; Azides; Benzodiazepines; Central Nervous System Depressants; Cerebellum; Drug Synergism; Electrophysiology; Ethanol; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Iontophoresis; Male; Norepinephrine; Purkinje Cells; Rats; Rats, Sprague-Dawley; Sympathomimetics | 1995 |
Chloride channel expression with the tandem construct of alpha 6-beta 2 GABAA receptor subunit requires a monomeric subunit of alpha 6 or gamma 2.
Topics: Affinity Labels; Azides; Base Sequence; Benzodiazepines; Binding Sites; Blotting, Northern; Cell Line; Chloride Channels; DNA, Complementary; gamma-Aminobutyric Acid; Gene Expression; Humans; Kidney; Kinetics; Macromolecular Substances; Membrane Potentials; Molecular Sequence Data; Muscimol; Oligodeoxyribonucleotides; Protein Multimerization; Receptors, GABA-A; Recombinant Proteins | 1995 |
Modulation of recombinant alpha 6 beta 2 gamma 2 GABAA receptors by neuroactive steroids.
Topics: Azides; Benzodiazepines; Binding, Competitive; Cell Line; Cells, Cultured; Electrophysiology; gamma-Aminobutyric Acid; Muscimol; Patch-Clamp Techniques; Receptors, GABA-A; Recombinant Proteins; Steroids | 1995 |
Benzodiazepine-induced motor impairment linked to point mutation in cerebellar GABAA receptor.
Topics: Affinity Labels; Amino Acid Sequence; Animals; Arginine; Autoradiography; Azides; Base Sequence; Benzodiazepines; Binding, Competitive; Cerebellum; Diazepam; Drug Tolerance; Ethanol; gamma-Aminobutyric Acid; Histidine; In Situ Hybridization; Kinetics; Macromolecular Substances; Models, Structural; Molecular Sequence Data; Motor Activity; Oligodeoxyribonucleotides; Point Mutation; Poly A; Protein Structure, Secondary; Rats; Rats, Mutant Strains; Receptors, GABA-A; RNA; RNA, Messenger; Tritium | 1993 |
Natural mutation of GABAA receptor alpha 6 subunit alters benzodiazepine affinity but not allosteric GABA effects.
Topics: Animals; Azides; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Cerebellum; Cloning, Molecular; Convulsants; Diazepam; gamma-Aminobutyric Acid; Granulocytes; Humans; Kidney; Muscimol; Mutation; Picrotoxin; Rats; Receptors, GABA-A; Recombinant Proteins; Transfection | 1993 |
Photoactivatable 2-(4'-azidotetrafluorophenyl)-5-tert-butyl-1,3-dithiane-bis- sulfone and related compounds as candidate irreversible probes for the GABA-gated chloride channels.
Topics: Affinity Labels; Animals; Azides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cell Membrane; Cerebral Cortex; Chloride Channels; Convulsants; gamma-Aminobutyric Acid; Ion Channel Gating; Light; Photochemistry; Sulfones | 1994 |
GABA antagonist and benzodiazepine partial inverse agonist reduce motivated responding for ethanol.
Topics: Alcohol Drinking; Animals; Appetitive Behavior; Arousal; Azides; Benzodiazepines; Brain; Chlordiazepoxide; Conditioning, Operant; Convulsants; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; Male; Motivation; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-A; Self Administration | 1993 |
Differences in benzodiazepine binding in quail selectively bred for differences in tonic immobility.
Topics: Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Brain; Chlorine; Coturnix; Diazepam; Ethanol; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Motor Activity; Radioisotopes; Receptors, GABA-A | 1996 |
Pharmacological modulation of the diazepam-insensitive recombinant gamma-aminobutyric acidA receptors alpha 4 beta 2 gamma 2 and alpha 6 beta 2 gamma 2.
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Binding Sites; Carbolines; Diazepam; Furosemide; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Imidazoles; Kinetics; Membrane Potentials; Radioligand Assay; Rats; Receptors, GABA-A; Recombinant Proteins; Sensitivity and Specificity; Zinc | 1996 |
Flunitrazepam has an inverse agonistic effect on recombinant alpha6beta2gamma2-GABAA receptors via a flunitrazepam-binding site.
Topics: Affinity Labels; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Cell Line; Chloride Channels; Flunitrazepam; GABA Agonists; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Kidney; Kinetics; Macromolecular Substances; Membrane Potentials; Receptors, GABA-A; Recombinant Proteins; Transfection | 1997 |
Cerebellar gamma-aminobutyric acid type A receptors: pharmacological subtypes revealed by mutant mouse lines.
Topics: Animals; Azides; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebellum; Convulsants; Diazepam; Diuretics; Furosemide; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Mice; Mice, Inbred C57BL; Mutation; Pregnanolone; Pyridazines; Receptors, GABA-A; Sulfur Radioisotopes; Tritium; Zinc | 1997 |
Localization and pharmacological characterization of pigeon diazepam-insensitive GABAA receptors.
Topics: Affinity Labels; Animals; Autoradiography; Azides; Benzodiazepines; Columbidae; Diazepam; GABA Modulators; gamma-Aminobutyric Acid; Ligands; Male; Radioligand Assay; Receptors, GABA-A | 1997 |
GABA(A) receptor alpha4 subunit suppression prevents withdrawal properties of an endogenous steroid.
Topics: Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Carbolines; Female; gamma-Aminobutyric Acid; Hippocampus; Indomethacin; Lorazepam; Oligonucleotides, Antisense; Patch-Clamp Techniques; Pregnanolone; Premenstrual Syndrome; Progesterone; Pyramidal Cells; Rats; Receptors, GABA-A; RNA, Messenger; Transcription, Genetic | 1998 |
GABAB-receptor splice variants GB1a and GB1b in rat brain: developmental regulation, cellular distribution and extrasynaptic localization.
Topics: Animals; Azides; Blotting, Western; Brain; Brain Chemistry; Cell Membrane; Dendrites; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Microscopy, Electron; Organophosphorus Compounds; Purkinje Cells; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; RNA Splicing; Synapses; Synaptic Transmission; Taurine | 1999 |
Characterization of gamma-aminobutyrate type A receptors with atypical coupling between agonist and convulsant binding sites in discrete brain regions.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Chickens; Convulsants; GABA Agonists; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Picrotoxin; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A; Sesterterpenes; Sulfur Radioisotopes; Thalamus; Tritium | 2001 |
Assembly of functional alpha6beta3gamma2delta GABA(A) receptors in vitro.
Topics: Affinity Labels; Anesthetics; Animals; Anticonvulsants; Azides; Benzodiazepines; Binding Sites; Cells, Cultured; Desoxycorticosterone; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Membrane Potentials; Muscimol; Protein Structure, Tertiary; Rats; Receptors, GABA-A; Transfection; Triazoles; Tritium | 2000 |
Mice performance on the staircase test following acute ethanol administration.
Topics: Animals; Azides; Benzodiazepines; Central Nervous System Depressants; Diazepam; Dose-Response Relationship, Drug; Ethanol; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Psychomotor Performance | 2001 |
Role of the histidine residue at position 105 in the human alpha 5 containing GABA(A) receptor on the affinity and efficacy of benzodiazepine site ligands.
Topics: Anticonvulsants; Arginine; Azides; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Cell Line; Cells, Cultured; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Histidine; Humans; Ligands; Mutation; Protein Subunits; Receptors, GABA-A | 2002 |
Altered receptor subtypes in the forebrain of GABA(A) receptor delta subunit-deficient mice: recruitment of gamma 2 subunits.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Binding Sites; Brain; Female; GABA Agonists; gamma-Aminobutyric Acid; Ion Channels; Male; Mice; Mice, Knockout; Muscimol; Mutation; Neural Inhibition; Neurons; Radioligand Assay; Receptors, GABA-A; Synaptic Transmission; Tritium | 2002 |
Contribution of the alpha1-GABA(A) receptor subtype to the pharmacological actions of benzodiazepine site inverse agonists.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Cell Line; Chloride Channels; Convulsants; Electrophysiology; GABA Agonists; gamma-Aminobutyric Acid; Humans; Mice; Mice, Transgenic; Motor Activity; Pentylenetetrazole; Point Mutation; Rats; Transfection | 2002 |
Selective transformations of organic compounds by imidozirconocene complexes.
Topics: Alkenes; Alkynes; Azides; Catalysis; gamma-Aminobutyric Acid; Imines; Molecular Conformation; Molecular Structure; Nitrogen; Organic Chemicals; Organometallic Compounds; Zirconium | 2002 |
Neurosteroid effects on GABAergic synaptic plasticity in hippocampus.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Female; gamma-Aminobutyric Acid; Hippocampus; Neural Inhibition; Neuronal Plasticity; Oligonucleotides, Antisense; Organ Culture Techniques; Pregnanolone; Rats; Rats, Long-Evans; Receptors, GABA; Synaptic Transmission | 2003 |
Binding characteristics of [3H]ucb 30889 to levetiracetam binding sites in rat brain.
Topics: Animals; Anticonvulsants; Azides; Binding, Competitive; Brain; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Levetiracetam; Male; Piracetam; Pyrrolidines; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tritium | 2003 |
Uptake of GABA and putrescine by UGA4 on the vacuolar membrane in Saccharomyces cerevisiae.
Topics: Azides; Biological Transport; Carrier Proteins; Cell Division; Enzyme Induction; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Intracellular Membranes; Macrolides; Nickel; Organic Anion Transporters; Ornithine Decarboxylase; Polyamines; Putrescine; Recombinant Proteins; RNA, Messenger; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Spermidine; Spermine; Subcellular Fractions; Vacuoles | 2004 |
Characterization of the interaction of indiplon, a novel pyrazolopyrimidine sedative-hypnotic, with the GABAA receptor.
Topics: Acetamides; Animals; Azides; Benzodiazepines; Binding Sites; Brain; Cell Membrane; Cerebellum; Cerebral Cortex; Chloride Channels; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Kinetics; Male; Pyridines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Thiophenes; Triazolam; Tritium; Zolpidem | 2004 |
Low-dose alcohol actions on alpha4beta3delta GABAA receptors are reversed by the behavioral alcohol antagonist Ro15-4513.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Electrophysiology; Esters; Ethanol; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Molecular Structure; Mutation; Oocytes; Patch-Clamp Techniques; Protein Subunits; Receptors, GABA-A; Xenopus laevis | 2006 |
Alcohol-sensitive GABA receptors and alcohol antagonists.
Topics: Alcohols; Animals; Azides; Benzodiazepines; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Receptors, GABA | 2006 |
Effects of ethanol on tonic GABA currents in cerebellar granule cells and mammalian cells recombinantly expressing GABA(A) receptors.
Topics: Animals; Azides; Benzodiazepines; Cells, Cultured; Cerebellum; CHO Cells; Cricetinae; Ethanol; Furosemide; gamma-Aminobutyric Acid; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Recombinant Proteins; Xenopus | 2006 |
Glucose and pharmacological modulators of ATP-sensitive K+ channels control [Ca2+]c by different mechanisms in isolated mouse alpha-cells.
Topics: Animals; Azides; Calcium; Diazoxide; gamma-Aminobutyric Acid; Glucagon-Secreting Cells; Glucose; Insulin-Secreting Cells; KATP Channels; Mice; Mice, Inbred Strains; NADP; Nimodipine; Tolbutamide | 2009 |
Influence of agonist induced internalization on [3H]Ro15-4513 binding-an application to imaging fluctuations in endogenous GABA with positron emission tomography.
Topics: Animals; Azides; Benzodiazepines; Binding, Competitive; Carbon Radioisotopes; Cell Membrane; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Male; Nipecotic Acids; Positron-Emission Tomography; Radiopharmaceuticals; Rats, Sprague-Dawley; Receptors, GABA-A; Tiagabine; Tritium | 2015 |
Negative allosteric modulation of GABAA receptors inhibits facilitation of brain stimulation reward by drugs of abuse in C57BL6/J mice.
Topics: Allosteric Regulation; Animals; Azides; Benzodiazepines; Brain; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Illicit Drugs; Male; Mice; Mice, Inbred C57BL; Microdialysis; Receptors, GABA-A; Reward; Self Stimulation | 2016 |
Attenuation of dopamine-induced GABA release in problem gamblers.
Topics: Adult; Azides; Benzodiazepines; Dopamine; Dopamine Agents; Double-Blind Method; Frontal Lobe; Gambling; gamma-Aminobutyric Acid; Humans; Levodopa; Male; Positron-Emission Tomography; Self-Control; Synaptic Transmission | 2019 |