Page last updated: 2024-08-21

azetidine and urea

azetidine has been researched along with urea in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benwell, K; Brooks, T; D'Alessandro, J; Dokurno, P; Francis, G; Gibbons, B; Hart, T; Haymes, T; Kennett, G; Lightowler, S; Macias, AT; Mansell, H; Matassova, N; Misra, A; Padfield, A; Parsons, R; Pratt, R; Robertson, A; Roughley, S; Walls, S; Wong, M1
Beidler, D; Bowen, SJ; Madsen, HM; McDonald, J; Pelc, MJ; Schweitzer, BA; Tenbrink, RE; Thorarensen, A; Wang, JL1
Benwell, K; Brooks, T; Browne, H; D'Alessandro, J; Daniels, Z; Dugdale, S; Francis, G; Gibbons, B; Hart, T; Haymes, T; Kennett, G; Lightowler, S; Macias, AT; Mansell, H; Matassova, N; Merrett, A; Misra, A; Padfield, A; Parsons, R; Pratt, R; Robertson, A; Roughley, SD; Simmonite, H; Tan, K; Walls, SB; Wong, M1

Other Studies

3 other study(ies) available for azetidine and urea

ArticleYear
Fatty acid amide hydrolase inhibitors. Surprising selectivity of chiral azetidine ureas.
    Bioorganic & medicinal chemistry letters, 2009, Aug-01, Volume: 19, Issue:15

    Topics: Amidohydrolases; Animals; Azetidines; Catalysis; Chemistry, Pharmaceutical; Drug Design; Enzyme Inhibitors; Humans; Mice; Mice, Knockout; Models, Chemical; Piperidines; Rats; Receptor, Cannabinoid, CB1; Stereoisomerism; Urea

2009
Structure based design of novel irreversible FAAH inhibitors.
    Bioorganic & medicinal chemistry letters, 2009, Oct-15, Volume: 19, Issue:20

    Topics: Amidohydrolases; Analgesics; Animals; Azetidines; Binding Sites; Crystallography, X-Ray; Drug Design; Enzyme Inhibitors; Humans; Pyridazines; Rats; Structure-Activity Relationship; Urea

2009
Fatty acid amide hydrolase inhibitors. 3: tetra-substituted azetidine ureas with in vivo activity.
    Bioorganic & medicinal chemistry letters, 2012, Jan-15, Volume: 22, Issue:2

    Topics: Amidohydrolases; Animals; Azetidines; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Enzyme Inhibitors; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Models, Molecular; Molecular Structure; Rats; Stereoisomerism; Structure-Activity Relationship; Urea

2012