azetidine has been researched along with pyrrolidine in 4 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 3 (75.00) | 24.3611 |
| 2020's | 1 (25.00) | 2.80 |
| Authors | Studies |
|---|---|
| Fotsch, C; St Jean, DJ | 1 |
| Bellman, K; Knegtel, RM; Settimo, L | 1 |
| Aulabaugh, A; Balbo, P; Banker, ME; Bauman, J; Casimiro-Garcia, A; Chrencik, J; Coe, JW; Czerwinski, R; Dowty, M; Juba, B; Knafels, JD; Kwon, S; Leung, L; Liang, S; Robinson, RP; Telliez, JB; Thorarensen, A; Trujillo, JI; Unwalla, R; Vajdos, F; Yang, X | 1 |
| Cocklin, S; Karadsheh, R; Meuser, ME | 1 |
1 review(s) available for azetidine and pyrrolidine
| Article | Year |
|---|---|
Mitigating heterocycle metabolism in drug discovery.
Topics: Animals; Biotransformation; Databases, Factual; Drug Discovery; Drug Interactions; Heterocyclic Compounds, 1-Ring; Heterocyclic Compounds, 4 or More Rings; Humans; Mice; Pharmaceutical Preparations; Rats | 2012 |
3 other study(ies) available for azetidine and pyrrolidine
| Article | Year |
|---|---|
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation | 2014 |
Identification of Cyanamide-Based Janus Kinase 3 (JAK3) Covalent Inhibitors.
Topics: Animals; Cyanamide; Drug Evaluation, Preclinical; Humans; Inhibitory Concentration 50; Janus Kinase 3; Male; Models, Molecular; Protein Conformation; Protein Kinase Inhibitors; Rats; Tissue Distribution | 2018 |
Composition and Orientation of the Core Region of Novel HIV-1 Entry Inhibitors Influences Metabolic Stability.
Topics: Anti-HIV Agents; Azabicyclo Compounds; Azetidines; Chromatography, Liquid; HEK293 Cells; HIV Core Protein p24; HIV Fusion Inhibitors; HIV Infections; HIV-1; Humans; Microsomes, Liver; Organophosphates; Piperazines; Protein Binding; Pyrrolidines; Tandem Mass Spectrometry; Triazoles | 2020 |