azepexole and methoxamine

azepexole has been researched along with methoxamine in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-199023 (71.88)18.7374
1990's5 (15.63)18.2507
2000's3 (9.38)29.6817
2010's1 (3.13)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Guth, BD; Heusch, G; Miyamoto, MI; Rockman, HA; Ross, J1
Armstrong, PW; Forster, C1
Armstead, WM; Hyman, AL; Kadowitz, PJ; Lippton, HL1
Graziadei, L; Pana-Race, G; Pedrinelli, R; Salvetti, A; Taddei, S1
Bellan, JA; Hyman, AL; Kadowitz, PJ; Lippton, HL1
Pedrinelli, R; Salvetti, A; Taddei, S1
Hyman, AL; Kadowitz, PJ1
Graziadei, L; Panarace, G; Pedrinelli, R; Salvetti, A; Taddei, S1
Rhodes, KF; Waterfall, JF1
Pang, CC; Tabrizchi, R1
Armstead, WM; Hyman, AL; Kadowitz, PJ; Lippton, HL; Roland, PY1
Flint, NS; Opie, LH; Thandroyen, FT; Worthington, MG1
Medgett, IC; Ruffolo, RR2
Kobinger, W1
Fujita, T; Ruffolo, RR; Shebuski, RJ1
Hyman, AL; Kadowitz, PJ; Lippton, HL1
Jie, K; Timmermans, PB; van Brummelen, P; van Zwieten, PA; Vermey, P2
Ohlstein, EH; Ruffolo, RR; Shebuski, RJ; Smith, JM1
Kobinger, W; Pichler, L1
Kobinger, W; Lillie, C; Pichler, L1
Boyer, JL; Cárdenas, C; García-Sáinz, JA; Posadas, C1
Paciorek, PM; Pierce, V; Shepperson, NB; Waterfall, JF1
Ishii, K; Kato, R; Yamamoto, S1
Baumgart, D; Ehring, T; Heusch, G; Hümmelgen, M; Kompa, S; Krajcar, M1
Burgess, RS; Choe, EU; Cork, RC; Ferrara, JJ; Flint, LM; Hoang, TV1
Baumgart, D; Erbel, R; Haude, M; Heusch, G; Naber, C; Oldenburg, O; Siffert, W1
Baumgart, D; Erbel, R; Heusch, G; Huesing, J; Naber, CK; Oldenburg, O; Siffert, W1
Castillo, C; Castillo, EF; López, RM; Ortíz, CS; Ruíz, A; Vélez, JM1
Centurión, D; Cobos-Puc, LE; Márquez-Conde, JA; Monroy-Ordoñez, EB; Sánchez-López, A; Villalón, CM1
Acosta-Cota, SJ; Centurión, D; Gómez-Viquez, NL; Molina-Muñoz, T; Sánchez-López, A1

Reviews

1 review(s) available for azepexole and methoxamine

ArticleYear
Rudolf Buchheim lecture. Drugs as tools in research on adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2

    Topics: Angiotensin II; Animals; Azepines; Blood Pressure; Clonidine; Guanabenz; Guanfacine; Guanidines; Heart Rate; Humans; Imidazoles; Methoxamine; Oxymetazoline; Phenylacetates; Prazosin; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiophenes; Xylazine; Yohimbine

1986

Trials

1 trial(s) available for azepexole and methoxamine

ArticleYear
Influence of calcium entry blockade on alpha 1- and alpha 2-adrenoceptor mediated vasoconstriction in the forearm of hypertensive patients.
    European journal of clinical pharmacology, 1987, Volume: 32, Issue:2

    Topics: Adult; Azepines; Calcium Channel Blockers; Female; Forearm; Hemodynamics; Humans; Hypertension; Isradipine; Male; Methoxamine; Middle Aged; Nifedipine; Oxadiazoles; Receptors, Adrenergic, alpha; Regional Blood Flow; Vascular Resistance; Vasoconstriction

1987

Other Studies

30 other study(ies) available for azepexole and methoxamine

ArticleYear
Effect of alpha-adrenergic stimulation on regional contractile function and myocardial blood flow with and without ischemia.
    Circulation, 1991, Volume: 84, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Coronary Circulation; Coronary Disease; Dogs; Methoxamine; Myocardial Contraction; Receptors, Adrenergic, alpha; Vasoconstriction

1991
Pacing-induced heart failure in the dog: evaluation of peripheral vascular alpha-adrenoceptor subtypes.
    Journal of cardiovascular pharmacology, 1990, Volume: 16, Issue:5

    Topics: Animals; Azepines; Blood Pressure; Cardiac Pacing, Artificial; Dogs; Dose-Response Relationship, Drug; Epinephrine; Heart Failure; Male; Methoxamine; Prazosin; Receptors, Adrenergic, alpha; Saphenous Vein; Vasoconstriction; Yohimbine

1990
Influence of nisoldipine on vascular resistance and vasoconstrictor responses in cats.
    The American journal of physiology, 1987, Volume: 252, Issue:4 Pt 2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Angiotensin II; Animals; Azepines; Blood Pressure; Brimonidine Tartrate; Cardiac Output; Cats; Dinoprost; Dioxanes; Electric Stimulation; Female; Idazoxan; Male; Methoxamine; Nifedipine; Nisoldipine; Norepinephrine; Phenylephrine; Prostaglandin Endoperoxides, Synthetic; Prostaglandins F; Quinoxalines; Splanchnic Circulation; Sulfonamides; Sympathetic Nervous System; Tyramine; Vascular Resistance; Vasoconstriction

1987
Verapamil and alpha-mediated vasoconstriction in human forearm: a comparison between norepinephrine and selective alpha 1- and alpha 2-adrenergic agonists.
    Journal of cardiovascular pharmacology, 1987, Volume: 10 Suppl 10

    Topics: Adrenergic alpha-Agonists; Adult; Azepines; Female; Forearm; Humans; Infusions, Intravenous; Male; Methoxamine; Middle Aged; Norepinephrine; Vasoconstriction; Vasoconstrictor Agents; Verapamil

1987
Nisoldipine inhibits vasoconstrictor responses in the cat pulmonary vascular bed.
    Journal of applied physiology (Bethesda, Md. : 1985), 1989, Volume: 66, Issue:6

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Agonists; Animals; Azepines; Calcium Channel Blockers; Cats; Female; Male; Methoxamine; Nifedipine; Nisoldipine; Prostaglandin Endoperoxides, Synthetic; Pulmonary Circulation; Vasoconstriction; Vasodilator Agents

1989
Further evidence for the existence of alpha 2-mediated adrenergic vasoconstriction in human vessels.
    European journal of clinical pharmacology, 1988, Volume: 34, Issue:4

    Topics: Adult; Azepines; Female; Humans; Indoramin; Male; Methoxamine; Receptors, Adrenergic, alpha; Vasoconstriction; Yohimbine

1988
Evidence for existence of postjunctional alpha 1- and alpha 2-adrenoceptors in cat pulmonary vascular bed.
    The American journal of physiology, 1985, Volume: 249, Issue:4 Pt 2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Brimonidine Tartrate; Cats; Female; Male; Methoxamine; Norepinephrine; Phenylephrine; Prazosin; Propranolol; Pulmonary Artery; Pulmonary Veins; Quinoxalines; Receptors, Adrenergic, alpha; Vasoconstriction; Yohimbine

1985
Verapamil antagonizes forearm vasoconstriction mediated by selective alpha 1- and alpha 2-agonists in hypertensive patients.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:5

    Topics: Adrenergic alpha-Agonists; Adult; Azepines; Female; Forearm; Humans; Hypertension; Male; Methoxamine; Middle Aged; Vasoconstriction; Verapamil

1986
The effects of some alpha-adrenoceptor antagonists on the responses of the canine saphenous vein to B-HT 933, UK-14304 and methoxamine.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Azepines; Brimonidine Tartrate; Dioxanes; Dogs; Idazoxan; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Potassium Chloride; Quinoxalines; Saphenous Vein

1987
Comparative effects of rauwolscine, prazosin, and phentolamine on blood pressure and cardiac output in anesthetized rats.
    Canadian journal of physiology and pharmacology, 1987, Volume: 65, Issue:7

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Blood Pressure; Cardiac Output; Epinephrine; Heart Rate; Methoxamine; Norepinephrine; Phentolamine; Prazosin; Rats; Rats, Inbred Strains; Regional Blood Flow; Vascular Resistance; Yohimbine

1987
Inhibitory effects of diltiazem on vasoconstrictor responses in the cat.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Brimonidine Tartrate; Cats; Diltiazem; Electric Stimulation; Female; Male; Methoxamine; Norepinephrine; Phenylephrine; Potassium Chloride; Quinoxalines; Tyramine; Vasoconstriction

1988
Arrhythmogenic action of alpha 1-adrenoceptor stimulation in normoxic rat ventricular myocardium: influence of nisoldipine, reduced extracellular Ca2+ and ryanodine.
    Journal of molecular and cellular cardiology, 1987, Volume: 19, Issue:9

    Topics: Adrenergic alpha-Agonists; Alkaloids; Animals; Arrhythmias, Cardiac; Azepines; Calcium; Calcium Channel Blockers; Heart; Male; Methoxamine; Nifedipine; Nisoldipine; Prazosin; Rats; Rats, Inbred Strains; Ryanodine

1987
Characterization of alpha-adrenoceptors mediating sympathetic vasoconstriction in rat autoperfused hindlimb: effects of SK&F 104078.
    European journal of pharmacology, 1987, Dec-15, Volume: 144, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Azepines; Benzazepines; Male; Methoxamine; Perfusion; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Sympathetic Nervous System; Synaptic Transmission; Vasoconstriction; Yohimbine

1987
Alpha adrenoceptor-mediated vasoconstriction in rat hindlimb: innervated alpha-2 adrenoceptors in the saphenous arterial bed.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Arteries; Azepines; Dose-Response Relationship, Drug; Hindlimb; Male; Methoxamine; Nifedipine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vasoconstriction

1988
Evaluation of alpha-1 and alpha-2 adrenoceptor-mediated vasoconstriction in the in situ, autoperfused, pulmonary circulation of the anesthetized dog.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: Animals; Azepines; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Female; Male; Methoxamine; Norepinephrine; Prazosin; Propranolol; Pulmonary Circulation; Receptors, Adrenergic, alpha; Tyramine; Vasoconstriction; Yohimbine

1986
Nature of alpha 1 and postjunctional alpha 2 adrenoceptors in the pulmonary vascular bed.
    Federation proceedings, 1986, Volume: 45, Issue:9

    Topics: Animals; Azepines; Blood Pressure; Brimonidine Tartrate; Cats; Hydroxydopamines; Methoxamine; Norepinephrine; Oxidopamine; Phenylephrine; Prazosin; Propranolol; Pulmonary Artery; Quinoxalines; Receptors, Adrenergic, alpha; Vasoconstriction; Yohimbine

1986
Enhanced pulmonary alpha-2 adrenoceptor responsiveness under conditions of elevated pulmonary vascular tone.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Azepines; Blood Pressure; Dinoprost; Dogs; Female; Lung; Male; Methoxamine; Prazosin; Prostaglandin Endoperoxides, Synthetic; Prostaglandins F; Receptors, Adrenergic, alpha; Serotonin; Vasoconstriction; Yohimbine

1987
alpha 1-adrenoceptor blockade by alpha 2-adrenoceptor agonists in the isolated perfused hindquarter of rats.
    European journal of pharmacology, 1981, Jun-10, Volume: 72, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Clonidine; In Vitro Techniques; Male; Methoxamine; Oxazoles; Perfusion; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiazoles; Vasoconstriction

1981
Central cardiovascular alpha-adrenoceptors. Relation to peripheral receptors.
    Circulation research, 1980, Volume: 46, Issue:6 Pt 2

    Topics: Animals; Azepines; Blood Pressure; Cardiovascular System; Clonidine; Dose-Response Relationship, Drug; Heart Rate; Male; Methoxamine; Norepinephrine; Oxazoles; Perfusion; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiazoles; Vagotomy

1980
"Pertussis toxin induces tachycardia and impairs the increase in blood pressure produced by alpha 2-adrenergic agonists".
    Life sciences, 1983, Dec-26, Volume: 33, Issue:26

    Topics: Animals; Azepines; Bacterial Toxins; Blood Pressure; Bordetella pertussis; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Male; Methoxamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tachycardia

1983
Identification of vascular postsynaptic alpha 1- and alpha 2-adrenoceptors in man.
    Circulation research, 1984, Volume: 54, Issue:4

    Topics: Adult; Azepines; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Doxazosin; Female; Guanfacine; Guanidines; Heart Rate; Humans; Male; Methoxamine; Muscle, Smooth, Vascular; Phenylacetates; Prazosin; Receptors, Adrenergic, alpha; Receptors, Neurotransmitter; Yohimbine

1984
An investigation into the selectivity of a novel series of benzoquinolizines for alpha 2-adrenoceptors in vivo.
    British journal of pharmacology, 1984, Volume: 82, Issue:1

    Topics: 2H-Benzo(a)quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy-; Action Potentials; Animals; Azepines; Chlorisondamine; Clonidine; Female; Indoramin; Methoxamine; Quinolizines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1984
Development of clonidine-tolerance in the rat vas deferens: cross tolerance to other presynaptic inhibitory agents.
    Life sciences, 1982, Jan-18, Volume: 30, Issue:3

    Topics: Adenosine; Animals; Azepines; Clonidine; Drug Tolerance; Endorphins; Evoked Potentials; Male; Methoxamine; Muscle Contraction; Norepinephrine; Rats; Rats, Inbred Strains; Sympathetic Nervous System; Sympathomimetics; Vas Deferens

1982
Cholinergic and alpha-adrenergic coronary vasomotion [corrected] with increasing ischemia-reperfusion injury.
    The American journal of physiology, 1995, Volume: 268, Issue:2 Pt 2

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Animals; Azepines; Cholinergic Agents; Coronary Circulation; Dogs; Hemodynamics; Methoxamine; Myocardial Ischemia; Myocardial Reperfusion Injury; Myocardium; Vasoconstriction

1995
Characterization of alpha-adrenoceptor activity in the preterm piglet mesentery.
    Journal of pediatric surgery, 1996, Volume: 31, Issue:12

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Azepines; Dioxanes; Female; Fetal Organ Maturity; Mesenteric Arteries; Methoxamine; Perfusion; Pregnancy; Pressure; Receptors, Adrenergic, alpha; Swine; Vasoconstriction

1996
G protein beta3 subunit 825T allele and enhanced coronary vasoconstriction on alpha(2)-adrenoceptor activation.
    Circulation research, 1999, Nov-12, Volume: 85, Issue:10

    Topics: Adrenergic alpha-Agonists; Alleles; Azepines; Coronary Vessels; Female; GTP-Binding Proteins; Humans; Male; Methoxamine; Middle Aged; Protein Isoforms; Receptors, Adrenergic, alpha; Vasoconstriction; Vasoconstrictor Agents

1999
Role of the eNOS Glu298Asp variant on the GNB3825T allele dependent determination of alpha-adrenergic coronary constriction.
    Pharmacogenetics, 2003, Volume: 13, Issue:5

    Topics: Adrenergic alpha-Agonists; Amino Acid Substitution; Aspartic Acid; Azepines; Blood Pressure; Coronary Circulation; Coronary Disease; Coronary Vessels; Genetic Variation; Genotype; Glutamic Acid; Heart Rate; Heterotrimeric GTP-Binding Proteins; Humans; Methoxamine; Mutation, Missense; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Receptors, Adrenergic, alpha; Vascular Resistance; Vasoconstriction

2003
Evidence against alpha-adrenoceptors mediating relaxation in rat thoracic aortae: alpha-agonists relaxation depends on interaction with alpha-adrenoceptors.
    Fundamental & clinical pharmacology, 2006, Volume: 20, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Azepines; Brimonidine Tartrate; Clonidine; Dinoprost; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Male; Methoxamine; Nitric Oxide; Phenylephrine; Piperazines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Serotonin; Vasoconstrictor Agents; Vasodilation; Yohimbine

2006
Evidence that some imidazoline derivatives inhibit peripherally the vasopressor sympathetic outflow in pithed rats.
    Autonomic neuroscience : basic & clinical, 2008, Dec-05, Volume: 143, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Agmatine; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Blood Vessels; Clonidine; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Heart Rate; Imidazoles; Imidazoline Receptors; Imidazolines; Injections, Intravenous; Male; Methoxamine; Rats; Rats, Wistar; Sympathetic Nervous System; Vasomotor System

2008
Evidence that chronic administration of 17β-oestradiol decreases the vasopressor responses to adrenergic system stimulation in streptozotocin-diabetic female rats.
    Steroids, 2014, Volume: 83

    Topics: Adrenergic Agents; Animals; Area Under Curve; Azepines; Blood Glucose; Blood Pressure; Body Weight; Diabetes Mellitus, Experimental; Diastole; Estradiol; Estrous Cycle; Female; Methoxamine; Norepinephrine; Ovariectomy; Rats; Rats, Wistar; Streptozocin; Vasoconstrictor Agents

2014