Page last updated: 2024-08-24

azauracil and ce 224,535

azauracil has been researched along with ce 224,535 in 1 studies

Research

Studies (1)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	0 (0.00)	18.2507
2000's	0 (0.00)	29.6817
2010's	1 (100.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Beaulieu, AM; Chang, SP; Dombroski, MA; Duplantier, AJ; Gabel, CA; Jordan, C; Kalgutkar, AS; Kraus, KG; Labasi, JM; Mussari, C; Perregaux, DG; Shepard, R; Subramanyam, C; Taylor, TJ; Trevena, KA; Whitney-Pickett, C; Yoon, K	1

Other Studies

1 other study(ies) available for azauracil and ce 224,535

Article	Year
Optimization of the physicochemical and pharmacokinetic attributes in a 6-azauracil series of P2X7 receptor antagonists leading to the discovery of the clinical candidate CE-224,535. Bioorganic & medicinal chemistry letters, 2011, Jun-15, Volume: 21, Issue:12 Topics: Administration, Oral; Animals; Antirheumatic Agents; Benzamides; Drug Discovery; Humans; Inhibitory Concentration 50; Molecular Structure; Protein Binding; Purinergic P2 Receptor Antagonists; Rats; Receptors, Purinergic P2X7; Structure-Activity Relationship; Uracil	2011

Article

Year

Optimization of the physicochemical and pharmacokinetic attributes in a 6-azauracil series of P2X7 receptor antagonists leading to the discovery of the clinical candidate CE-224,535.

Bioorganic & medicinal chemistry letters, 2011, Jun-15, Volume: 21, Issue:12

Topics: Administration, Oral; Animals; Antirheumatic Agents; Benzamides; Drug Discovery; Humans; Inhibitory Concentration 50; Molecular Structure; Protein Binding; Purinergic P2 Receptor Antagonists; Rats; Receptors, Purinergic P2X7; Structure-Activity Relationship; Uracil

2011