azasetron and granisetron

azasetron has been researched along with granisetron in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (53.85)18.2507
2000's3 (23.08)29.6817
2010's3 (23.08)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Sakamori, M; Setoguchi, M; Takehara, S1
Enomoto, H; Furukawa, M; Ikema, Y; Kawai, S; Kohno, H; Matsuda, H; Mochimatsu, I; Tsukuda, M; Yago, T; Zhou, L1
Fukuda, T; Haga, K; Inaba, K; Morimoto, Y; Setoguchi, M; Shoji, H1
Kobayashi, S; Kumai, T; Nakura, H; Tanaka, M; Tateishi, T; Watanabe, M1
Funakoshi, A; Masuda, M; Miyasaka, K1
Asano, K; Fukuda, T; Haga, K; Katayama, K1
Ozaki, A; Sukamoto, T1
Akamatsu, H; Mikawa, K; Nishina, K; Niwa, Y; Shiga, M1
Iwase, O; Okuyama, K; Ozeki, T; Yamada, Y; Yoshimoto, K1
Ayuhara, H; Okuyama, K; Ozeki, T; Takayanagi, R; Yamada, Y; Yokoyama, H; Yoshimoto, K1
Endo, J; Funaguchi, N; Iihara, H; Ito, F; Itoh, Y; Kamiya, F; Minatoguchi, S; Ohno, Y; Yamada, M; Yanase, K1
Iwase, O; Nakajima, A; Nakamura, H; Okuyama, K; Takayanagi, R; Yamada, Y; Yokoyama, H; Yoshimoto, K1
Hashizume, J; Higuchi, N; Kitahara, T; Kodama, Y; Matsunaga, N; Nakamura, T; Sakamoto, T; Sasaki, H; Sato, K; Yamaguchi, K1

Trials

2 trial(s) available for azasetron and granisetron

ArticleYear
[A randomized crossover comparison of azasetron and granisetron in the prophylaxis of emesis induced by chemotherapy including cisplatin].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1995, Volume: 22, Issue:13

    Topics: Aged; Antiemetics; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Female; Granisetron; Head and Neck Neoplasms; Humans; Male; Middle Aged; Oxazines; Serotonin Antagonists; Vomiting

1995
A randomized controlled non-inferiority study comparing the antiemetic effect between intravenous granisetron and oral azasetron based on estimated 5-HT3 receptor occupancy.
    Anticancer research, 2012, Volume: 32, Issue:9

    Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Bridged Bicyclo Compounds, Heterocyclic; Carboplatin; Female; Granisetron; Humans; Injections, Intravenous; Lung Neoplasms; Male; Middle Aged; Oxazines; Receptors, Serotonin, 5-HT3; Serotonin Antagonists

2012

Other Studies

11 other study(ies) available for azasetron and granisetron

ArticleYear
[High affinity binding of Y-25130 for serotonin 3 receptor].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1992, Volume: 100, Issue:2

    Topics: Animals; Antiemetics; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Granisetron; In Vitro Techniques; Indazoles; Male; Ondansetron; Oxazines; Rats; Rats, Wistar; Receptors, Serotonin; Synaptic Membranes

1992
The effects of orally administered Y-25130, a selective serotonin3-receptor antagonist, on chemotherapeutic agent-induced emesis.
    Japanese journal of pharmacology, 1993, Volume: 63, Issue:3

    Topics: Administration, Oral; Animals; Antiemetics; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Cyclophosphamide; Dogs; Domperidone; Dose-Response Relationship, Drug; Doxorubicin; Female; Ferrets; Granisetron; Male; Metoclopramide; Ondansetron; Oxazines; Serotonin Antagonists; Vomiting

1993
The activity of dihydropyrimidine dehydrogenase from rat liver was not affected by any of five 5-hydroxytryptamine antagonists.
    Cancer letters, 1996, Nov-12, Volume: 108, Issue:1

    Topics: Animals; Antiemetics; Antimetabolites, Antineoplastic; Biotransformation; Bridged Bicyclo Compounds, Heterocyclic; Cytosol; Dihydrouracil Dehydrogenase (NADP); Fluorouracil; Granisetron; Indoles; Liver; Male; Ondansetron; Oxazines; Oxidoreductases; Quinolizines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Tropisetron

1996
Involvement of 5-hydroxytryptamine (5-HT)3 receptor mechanisms in regulation of basal pancreatic secretion in conscious rats.
    Journal of the autonomic nervous system, 1997, Jan-12, Volume: 62, Issue:1-2

    Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Granisetron; Male; Oxazines; Pancreas; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists

1997
High affinity binding of azasetron hydrochloride to 5-hydroxytryptamine3 receptors in the small intestine of rats.
    Japanese journal of pharmacology, 1997, Volume: 73, Issue:4

    Topics: Animals; Antiemetics; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Intestine, Small; Isotope Labeling; Male; Oxazines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Tritium; Vomiting

1997
Improvement of cisplatin-induced emesis and delayed gastric emptying by KB-R6933, a novel 5-HT3 receptor antagonist.
    General pharmacology, 1999, Volume: 33, Issue:3

    Topics: Animals; Antiemetics; Antineoplastic Agents; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Dose-Response Relationship, Drug; Ferrets; Gastric Emptying; Granisetron; Male; Ondansetron; Oxazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Vomiting

1999
Effects of ondansetron, granisetron, ramosetron, and azasetron on human neutrophil functions.
    Gynecologic and obstetric investigation, 2002, Volume: 53, Issue:2

    Topics: Antiemetics; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Chemotaxis, Leukocyte; Granisetron; Humans; Neutrophils; Ondansetron; Oxazines

2002
[Clinical evaluation of antiemetic effects of 5-hydroxytryptamine receptor type 3 (5HT3 receptor) antagonists based on changes in eating condition in cancer patients receiving chemotherapy].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 2008, Volume: 128, Issue:4

    Topics: Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Eating; Female; Granisetron; Humans; Male; Middle Aged; Nausea; Neoplasms; Oxazines; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Treatment Outcome; Vomiting

2008
Receptor occupancy theory-based analysis of interindividual differences in antiemetic effects of 5-HT3 receptor antagonists.
    International journal of clinical oncology, 2009, Volume: 14, Issue:6

    Topics: Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Drug Administration Schedule; Granisetron; Humans; Indoles; Models, Theoretical; Ondansetron; Oxazines; Serotonin 5-HT3 Receptor Antagonists; Treatment Outcome; Tropisetron; Vomiting

2009
Theoretical evaluation of antiemetic effects of 5-HT3 receptor antagonists for prevention of vomiting induced by cisplatin.
    European journal of drug metabolism and pharmacokinetics, 2015, Volume: 40, Issue:1

    Topics: Antineoplastic Agents; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Constipation; Creatinine; Granisetron; Humans; Hydroxyindoleacetic Acid; Intestine, Small; Isoquinolines; Models, Biological; Nausea; Oxazines; Palonosetron; Quinuclidines; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin 5-HT3 Receptor Antagonists; Vomiting

2015
Evaluation of Antiemetic Therapy for Hepatic Transcatheter Arterial Infusion Chemotherapy with Cisplatin.
    Biological & pharmaceutical bulletin, 2016, Volume: 39, Issue:4

    Topics: Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Agents; Aprepitant; Bridged Bicyclo Compounds, Heterocyclic; Catheterization, Peripheral; Cisplatin; Dexamethasone; Drug Therapy, Combination; Female; Granisetron; Humans; Isoquinolines; Liver; Liver Neoplasms; Male; Middle Aged; Morpholines; Nausea; Oxazines; Palonosetron; Quinuclidines; Serotonin 5-HT3 Receptor Antagonists; Vomiting

2016