Page last updated: 2024-09-03

azaprophen and physostigmine

azaprophen has been researched along with physostigmine in 4 studies

Compound Research Comparison

Studies
(azaprophen)
Trials
(azaprophen)
Recent Studies (post-2010)
(azaprophen)
Studies
(physostigmine)
Trials
(physostigmine)
Recent Studies (post-2010) (physostigmine)
11006,230252331

Protein Interaction Comparison

ProteinTaxonomyazaprophen (IC50)physostigmine (IC50)
AcetylcholinesteraseElectrophorus electricus (electric eel)0.1666
AcetylcholinesteraseTetronarce californica (Pacific electric ray)0.3023
CholinesteraseHomo sapiens (human)0.3055
Cytochrome P450 2D6Homo sapiens (human)0.2
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.857
AcetylcholinesteraseMus musculus (house mouse)0.0269
AcetylcholinesteraseHomo sapiens (human)0.0853
Acetylcholinesterase Bos taurus (cattle)0.7197
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.857
Delta-type opioid receptorMus musculus (house mouse)1.1821
AcetylcholinesteraseGallus gallus (chicken)0.02
AcetylcholinesteraseRattus norvegicus (Norway rat)0.0416
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.857
CholinesteraseEquus caballus (horse)0.4081
CholinesteraseMus musculus (house mouse)0.28
Acyl-CoA:cholesterol acyltransferase Oryctolagus cuniculus (rabbit)0.0189
Carboxylic ester hydrolase Rattus norvegicus (Norway rat)0.018
Carboxylic ester hydrolase Equus caballus (horse)1.263

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Anderson, DR; Harris, LW; Lennox, WJ; Murrow, ML; Solana, RP; Wade, JV1
Carchman, RA; Carter, WH; Gennings, C; Harris, LW; Solana, RP; Talbot, BG1
Boyle, RM; Campbell, ED; Carchman, RA; Carter, WH; Gennings, C; Harris, LW; Solana, RP; Talbot, BG1
Genovese, RF1

Other Studies

4 other study(ies) available for azaprophen and physostigmine

ArticleYear
Successful pretreatment/therapy of soman, sarin and VX intoxication.
    Drug and chemical toxicology, 1992, Volume: 15, Issue:4

    Topics: Animals; Cholinesterase Inhibitors; Female; Guinea Pigs; Lethal Dose 50; Male; Organothiophosphorus Compounds; Phenylpropionates; Physostigmine; Poisoning; Sarin; Soman; Trihexyphenidyl; Tropanes

1992
Evaluation of a two-drug combination pretreatment against organophosphorus exposure.
    Toxicology and applied pharmacology, 1990, Mar-01, Volume: 102, Issue:3

    Topics: Animals; Cholinesterase Inhibitors; Drug Therapy, Combination; Erythrocytes; Female; Guinea Pigs; Lethal Dose 50; Male; Phenylpropionates; Physostigmine; Soman; Tropanes

1990
Assessing the efficacy of azaprophen and physostigmine as a pretreatment for soman-induced incapacitation in guinea pigs by response-surface modeling.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1990, Volume: 14, Issue:2

    Topics: Animals; Confidence Intervals; Drug Therapy, Combination; Female; Guinea Pigs; Male; Models, Biological; Parasympatholytics; Phenylpropionates; Physostigmine; Soman; Tropanes

1990
Effects of azaprophen, scopolamine and trihexyphenidyl on schedule-controlled behavior, before and after chronic physostigmine.
    European journal of pharmacology, 1990, Feb-13, Volume: 176, Issue:3

    Topics: Acetylcholine; Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Tolerance; Male; Phenylpropionates; Physostigmine; Rats; Rats, Inbred Strains; Reinforcement Schedule; Scopolamine; Trihexyphenidyl; Tropanes

1990