Page last updated: 2024-09-05

azacrin and cgp 60474

azacrin has been researched along with cgp 60474 in 1 studies

Compound Research Comparison

Studies
(azacrin)
Trials
(azacrin)
Recent Studies (post-2010)
(azacrin)
Studies
(cgp 60474)
Trials
(cgp 60474)
Recent Studies (post-2010) (cgp 60474)
60019010

Protein Interaction Comparison

ProteinTaxonomyazacrin (IC50)cgp 60474 (IC50)
XBP1Homo sapiens (human)0.16
DNA damage-inducible transcript 3 proteinMus musculus (house mouse)0.16
Cyclin-T1Homo sapiens (human)0.013
Cyclin-dependent kinase 1Homo sapiens (human)0.0161
Cyclin-dependent kinase 4Homo sapiens (human)0.216
G2/mitotic-specific cyclin-B1Homo sapiens (human)0.026
Cyclin-A2Homo sapiens (human)0.004
G1/S-specific cyclin-D1Homo sapiens (human)0.216
G1/S-specific cyclin-E1Homo sapiens (human)0.003
Cyclin-dependent kinase 2Homo sapiens (human)0.0041
Serine/threonine-protein kinase mTORHomo sapiens (human)0.8
Cyclin-dependent kinase 7Homo sapiens (human)0.2
Cyclin-dependent kinase 9Homo sapiens (human)0.013
Cyclin-HHomo sapiens (human)0.2
CDK-activating kinase assembly factor MAT1Homo sapiens (human)0.2
Cyclin-dependent-like kinase 5 Homo sapiens (human)0.01
Cyclin-dependent kinase 5 activator 1Homo sapiens (human)0.01
Serine/threonine-protein kinase SMG1Homo sapiens (human)0.11

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adrián, F; Anderson, P; Brinker, A; Caldwell, JS; Chatterjee, A; Gray, NS; Henson, K; Janes, J; Kato, N; Kuhen, K; Matzen, JT; McNamara, C; Nagle, A; Nam, TG; Plouffe, D; Schultz, PG; Trager, R; Winzeler, EA; Yan, SF; Zhou, Y1

Other Studies

1 other study(ies) available for azacrin and cgp 60474

ArticleYear
In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Jul-01, Volume: 105, Issue:26

    Topics: Animals; Antimalarials; Cluster Analysis; Computational Biology; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Malaria; Models, Molecular; Parasites; Plasmodium falciparum; Reproducibility of Results; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase

2008