azacitidine and fluorouracil

azacitidine has been researched along with fluorouracil in 68 studies

Research

Studies (68)

TimeframeStudies, this research(%)All Research%
pre-199020 (29.41)18.7374
1990's7 (10.29)18.2507
2000's14 (20.59)29.6817
2010's22 (32.35)24.3611
2020's5 (7.35)2.80

Authors

AuthorsStudies
Hansch, C; Khwaja, TA; Selassie, CD1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1
Borsos, T; Ohanian, SH; Segerling, M2
Kashmin, R; Maruyama, Y; Meeker, WR; Moses, B; Vider, M1
Duff, R; Haspel, MV; Rapp, F1
Faulkner, GP; Follett, EA; Pringle, CR; Shirodaria, PV1
Lenches, EM; Strauss, EG; Strauss, JH1
Chabner, BA; Myers, CE; Oliverio, VT1
Sviridenko, OP1
Bender, RA; Chabner, BA; Cohen, M; Doroshow, JH; Hande, KR; Locker, GY; Murinson, DS; Myers, CE; Zwelling, LA1
de la Torre, JC; Domingo, E; Holland, JJ; Steinhauer, DA1
Canivet, M; Dianoux, L; Lasneret, J; Lesser, J; Peries, J1
Allegra, CJ; Grem, JL1
Blair, CD; Eastman, PS1
Aiba, K; Allegra, CJ; Baram, J; Chabner, BA; Curt, GA; Yeh, GC1
Cohen, MB; Glazer, RI1
Gang, M; Kline, I; Sirica, AE; Venditti, JM; Woodman, RJ1
Cihák, A; Veselỳ, J1
Price, LA1
Pitot, HC; Weiss, JW1
Grignani, F; Martelli, M; Tonato, M1
Ellims, PH1
Brawner, TA; Fleming, TP; Hollingshead, PG1
Chabner, BA; Clendeninn, NJ; Curt, GA1
Jahan, N; Mitsuya, H; O'Brien, MC; Ueno, T; Zajac-Kaye, M1
Chanock, RM; Crowe, JE; Davis, AR; Hsu, KH; Hung, PP; Lubeck, MD; Murphy, BR1
Chernoff, N; Elstein, KH; Lau, C; Rogers, JM; Shuey, DL; Zucker, RM1
Dávila, M; Domingo, E; Lowenstein, PR; Sierra, S1
Arnold, CN; Boland, CR; Goel, A1
Cockerell, GL; Goodman, JI; McKim, JM; Watson, RE1
Domingo, E; Escarmís, C; Lázaro, E; Manrubia, SC1
Airaksinen, A; Pariente, N; Sierra, S1
Imazeki, F; Kanda, T; Nagao, K; Saisho, H; Tada, M; Yokosuka, O1
Engelbrecher, A; Häuser, R; Titz, B; Uetz, P1
Dou, KF; Zhao, QZ1
Iida, S; Kato, K; Morita, S; Sugihara, K; Takagi, Y; Uetake, H1
Cheetham, S; Kennecke, H; Mesak, F; Owen, D; Tai, IT; Tang, MJ1
Banerjee, D; Bertino, JR; Humeniuk, R; Mishra, PJ1
Mirza, S; Pandya, P; Ralhan, R; Sharma, G1
Kortsaris, A; Krupitza, G; Mader, RM; Mikulits, W; Schmidt, WM; Steger, GG; Tentes, IK1
Kucerova, L; Matuskova, M; Poturnajova, M; Tyciakova, S1
Chen, Y; Ding, J; Feng, JM; Huang, YR; Jiang, Y; Li, JX; Miao, ZH; Tong, LJ; Zhang, J1
Dong, Y; Guo, M; Hu, L; Jing, K; Li, Y; Wu, K; Yan, W; Yang, Y; Yuan, J; Zhu, H1
Ikehata, M; Iwakawa, S; Ogawa, M; Tanaka, S; Ueda, K; Yamada, Y1
Arroyo-Solera, I; Barnadas, A; Casanova, I; Céspedes, MV; Gallardo, A; León, X; López, M; López-Pousa, A; Mangues, MA; Mangues, R; Pavón, MA; Quer, M; Téllez-Gabriel, M1
Chen, BB; Chen, XB; Li, J; Lü, HF; Luo, SX; Ma, YJ; Wang, XF1
Flis, K; Flis, S; Gnyszka, A1
Hucho, T; Isensee, J; Kaehler, C; Krobitsch, S; Lehrach, H1
Lauring, AS; Pauly, MD1
Cui, FB; Ding, H; Li, RT; Liu, BR; Liu, Q; Qian, XP; Wang, HY; Wu, FL; Wu, PY; Yang, M; Yu, LX; Yue, GF1
Khatun, A; Kim, WI; Shabir, N; Yoon, KJ1
Brock, MV; Guo, M; Herman, JG; Li, X; Liang, P; Tao, Q; Yu, J1
Broggini, M; Cavalli, IJ; Chilà, R; Damia, G; de Lima, RS; de Oliveira, SF; Ganzinelli, M; Generali, D; Maciel, ME; Ribeiro, EM; Serino, L; Urban, Cde A1
Gao, D; Guo, M; Herman, JG1
Almqvist, H; Artursson, P; Axelsson, H; Dan, C; Haraldsson, M; Jafari, R; Larsson, A; Lundbäck, T; Martinez Molina, D; Mateus, A; Nordlund, P1
Hussain, S1
Asaro, G; De Luca, A; Delfini, M; Guglielmi, G; Iavicoli, S; Sciubba, F; Spagnoli, M1
Li, H; Li, Z; Lu, Y; Shan, S; Shi, J; Zhang, X1
Li, C; Li, F; Shang, J; Wang, F; Wang, Q; Yuan, B1
Chen, D; Deng, X; Feng, T; Wei, C; Wen, Z; Xu, J1

Reviews

9 review(s) available for azacitidine and fluorouracil

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Antineoplastic drugs: clinical pharmacology and therapeutic use.
    Drugs, 1978, Volume: 16, Issue:1

    Topics: Alkaloids; Alkylating Agents; Antibiotics, Antineoplastic; Antineoplastic Agents; Azacitidine; Bleomycin; Cisplatin; Cyclophosphamide; Cytarabine; Drug Interactions; Fluorouracil; Humans; Kinetics; Methotrexate; Podophyllotoxin

1978
Antimetabolites.
    Cancer chemotherapy and biological response modifiers, 1987, Volume: 9

    Topics: Animals; Antimetabolites, Antineoplastic; Azacitidine; Cytarabine; Floxuridine; Fluorouracil; Folic Acid Antagonists; Humans; Mercaptopurine; Methotrexate; Purines; Thioguanine

1987
Resistance of mammalian tumour cells toward pyrimidine analogues. A review.
    Oncology, 1973, Volume: 28, Issue:3

    Topics: Animals; Antimetabolites; Azacitidine; Azauridine; Bromouracil; Carcinoma, Ehrlich Tumor; Cell Line; Cricetinae; Cytarabine; Deoxycytidine; Drug Resistance; Fluorouracil; Genetic Code; Leukemia, Experimental; Leukemia, Lymphoid; Mast-Cell Sarcoma; Mice; Mutation; Neoplasms, Experimental; Oncogenic Viruses; Phosphotransferases; Pyrimidines; Sarcoma, Experimental; Selection, Genetic; Thymidine Kinase; Uracil; Virus Replication

1973
Thymidine as an anticancer agent, alone or in combination. A biochemical appraisal.
    Cancer chemotherapy and pharmacology, 1982, Volume: 10, Issue:1

    Topics: Animals; Antineoplastic Agents; Azacitidine; Cytarabine; Decitabine; Drug Therapy, Combination; Fluorouracil; Humans; Methotrexate; Neoplasms; Thymidine

1982
Quasispecies dynamics and RNA virus extinction.
    Virus research, 2005, Volume: 107, Issue:2

    Topics: Animals; Azacitidine; Biological Evolution; Fluorouracil; Foot-and-Mouth Disease Virus; Mutagens; Mutation

2005
Action of mutagenic agents and antiviral inhibitors on foot-and-mouth disease virus.
    Virus research, 2005, Volume: 107, Issue:2

    Topics: Animals; Antiviral Agents; Azacitidine; Cell Line; Cricetinae; Fluorouracil; Foot-and-Mouth Disease Virus; Mutagens; Ribavirin

2005
The clinical value of aberrant epigenetic changes of DNA damage repair genes in human cancer.
    Oncotarget, 2016, Jun-14, Volume: 7, Issue:24

    Topics: Antimetabolites, Antineoplastic; Azacitidine; Biomarkers, Tumor; Carcinogenesis; CpG Islands; Decitabine; DNA Damage; DNA Methylation; DNA Modification Methylases; DNA Repair; DNA Repair Enzymes; Drug Resistance, Neoplasm; Epigenesis, Genetic; Fluorouracil; Humans; Molecular Targeted Therapy; Neoplasms; Prognosis; Promoter Regions, Genetic; Tumor Suppressor Proteins

2016
Catalytic crosslinking-based methods for enzyme-specified profiling of RNA ribonucleotide modifications.
    Methods (San Diego, Calif.), 2019, 03-01, Volume: 156

    Topics: Animals; Azacitidine; Biocatalysis; Cross-Linking Reagents; Escherichia coli Proteins; Fluorouracil; Humans; Immunoprecipitation; Methylation; Methyltransferases; Multienzyme Complexes; Pseudouridine; RNA Processing, Post-Transcriptional; RNA, Messenger; Transcriptome; Uridine

2019

Other Studies

59 other study(ies) available for azacitidine and fluorouracil

ArticleYear
Structure-activity relationships of antineoplastic agents in multidrug resistance.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:7

    Topics: Animals; Antineoplastic Agents; Cell Line; Cell Survival; Cricetinae; Dactinomycin; Drug Resistance; Leukemia L1210; Mice; Regression Analysis; Structure-Activity Relationship; Tumor Cells, Cultured

1990
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023
Chemotherapeutic drugs increase killing of tumor cells by antibody and complement.
    Science (New York, N.Y.), 1975, Apr-04, Volume: 188, Issue:4183

    Topics: Animals; Antigen-Antibody Reactions; Antineoplastic Agents; Azacitidine; Carcinoma, Hepatocellular; Cell Line; Complement System Proteins; Cyclophosphamide; Cytarabine; Fluorouracil; Guinea Pigs; Liver Neoplasms; Methotrexate; Neoplasms, Experimental; Nitrosamines; Vincristine

1975
Carcinoembryonic antigen (CEA) monitoring in the management of radiotherapeutic and chemotherapeutic patients.
    The American journal of roentgenology, radium therapy, and nuclear medicine, 1975, Volume: 124, Issue:4

    Topics: Antigens, Neoplasm; Azacitidine; Carcinoembryonic Antigen; Dacarbazine; Fluorouracil; Humans; Monitoring, Physiologic; Neoplasms; Radioisotope Teletherapy

1975
Isolation and preliminary characterization of temperature-sensitive mutants of measles virus.
    Journal of virology, 1975, Volume: 16, Issue:4

    Topics: Antigens, Viral; Azacitidine; Cell Line; Fluorouracil; Genetic Complementation Test; Measles virus; Mutagens; Mutation; Proflavine; RNA, Viral; Temperature; Viral Proteins; Virus Replication

1975
Enhancing effect by metabolic inhibitors on the killing of tumor cells by antibody and complement.
    Cancer research, 1975, Volume: 35, Issue:11 Pt 1

    Topics: Animals; Antibodies, Neoplasm; Antigen-Antibody Reactions; Antineoplastic Agents; Azacitidine; Carcinoma, Hepatocellular; Cells, Cultured; Complement System Proteins; Cyclophosphamide; Cytarabine; Dactinomycin; Doxorubicin; Fluorouracil; Guinea Pigs; Hydroxyurea; Liver Neoplasms; Mercaptopurine; Methotrexate; Mitomycins; Neoplasms, Experimental; Puromycin; Vincristine

1975
Respiratory syncytial virus ts mutants and nuclear immunofluorescence.
    Journal of virology, 1976, Volume: 20, Issue:2

    Topics: Animals; Antigens, Viral; Azacitidine; Cell Line; Cell Nucleus; Cytopathogenic Effect, Viral; Ethyl Methanesulfonate; Fluorouracil; Genetic Complementation Test; Haplorhini; HeLa Cells; Methylnitronitrosoguanidine; Mutagens; Mutation; Respiratory Syncytial Viruses; Temperature; Virus Replication

1976
Mutants of sindbis virus. I. Isolation and partial characterization of 89 new temperature-sensitive mutants.
    Virology, 1976, Oct-01, Volume: 74, Issue:1

    Topics: Azacitidine; Fluorouracil; Genes; Genetic Complementation Test; Methylnitronitrosoguanidine; Mutagens; Mutation; Nitrites; RNA, Viral; Sindbis Virus; Temperature; Viral Proteins

1976
Clinical pharmacology of anticancer drugs.
    Seminars in oncology, 1977, Volume: 4, Issue:2

    Topics: Animals; Antineoplastic Agents; Azacitidine; Bleomycin; Cyclophosphamide; Cytarabine; Dacarbazine; Daunorubicin; Doxorubicin; Female; Fluorouracil; Heart; Humans; Leucovorin; Lung; Male; Methotrexate; Neoplasms; Nitrosourea Compounds; Procarbazine; Triazenes; Vinblastine; Vincristine

1977
[Uridine kinase, its structure, properties and biological function].
    Nauchnye doklady vysshei shkoly. Biologicheskie nauki, 1978, Issue:4

    Topics: Animals; Azacitidine; Brain; Carcinoma, Ehrlich Tumor; Chick Embryo; Drug Resistance; Fluorouracil; Isoenzymes; Kinetics; Liver; Phosphotransferases; Rats; RNA; Sarcoma, Experimental; Uracil; Uridine Kinase

1978
Mutation frequencies at defined single codon sites in vesicular stomatitis virus and poliovirus can be increased only slightly by chemical mutagenesis.
    Journal of virology, 1990, Volume: 64, Issue:8

    Topics: Animals; Azacitidine; Cell Line; Codon; Ethyl Methanesulfonate; Fluorouracil; Hydrogen-Ion Concentration; Mutagens; Mutation; Nitrous Acid; Poliovirus; RNA, Messenger; Vesicular stomatitis Indiana virus

1990
In vitro induction of early mouse embryo intracisternal particles (epsilon particles) in cultured cell lines.
    Biology of the cell, 1990, Volume: 69, Issue:3

    Topics: Animals; Azacitidine; Cell Line; Cell Line, Transformed; Cell Transformation, Viral; Cycloheximide; Dexamethasone; Endoplasmic Reticulum; Fibroblasts; Fluorouracil; Idoxuridine; Inclusion Bodies; Kirsten murine sarcoma virus; Mice; Mice, Inbred AKR; Mice, Inbred BALB C; Microscopy, Electron; Mink; Moloney murine sarcoma virus; Puromycin; Rats; Species Specificity; Tumor Cells, Cultured

1990
Sequence-dependent interaction of 5-fluorouracil and arabinosyl-5-azacytosine or 1-beta-D-arabinofuranosylcytosine.
    Biochemical pharmacology, 1991, Jul-05, Volume: 42, Issue:2

    Topics: Antineoplastic Combined Chemotherapy Protocols; Azacitidine; Cell Division; Cell Line; Cell Nucleus; Cell Survival; Colonic Neoplasms; Cytarabine; Cytidine; Deoxycytosine Nucleotides; DNA, Neoplasm; Drug Administration Schedule; Drug Interactions; Fluorouracil; Humans; Nucleic Acids; Thymine Nucleotides; Tumor Stem Cell Assay

1991
Temperature-sensitive mutants of Japanese encephalitis virus.
    Journal of virology, 1985, Volume: 55, Issue:3

    Topics: Azacitidine; Electrophoresis, Polyacrylamide Gel; Encephalitis Virus, Japanese; Fluorouracil; Genetic Complementation Test; Mutation; Phenotype; RNA, Viral; Temperature; Viral Proteins

1985
Cytotoxicity and the inhibition of ribosomal RNA processing in human colon carcinoma cells.
    Molecular pharmacology, 1985, Volume: 27, Issue:2

    Topics: Azacitidine; Azaguanine; Cell Survival; Cells, Cultured; Colonic Neoplasms; Fluorouracil; Humans; Protein Biosynthesis; Pyrimidine Nucleosides; RNA, Ribosomal; Toyocamycin; Tubercidin

1985
The enhanced therapeutic effect of cis-platinum (II) diamminodichloride against L1210 leukemia when combined with cyclophosphamide or 1,2-bis(3,5-dioxopiperazine-1-yl)propane or several other antitumor agents.
    Chemotherapy, 1973, Volume: 18, Issue:3

    Topics: Amines; Animals; Antineoplastic Agents; Azacitidine; Camptothecin; Carmustine; Chlorides; Cyclophosphamide; Cytarabine; Drug Synergism; Emetine; Fluorouracil; Ketones; Leukemia L1210; Male; Methotrexate; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Piperazines; Platinum; Propane; Time Factors

1973
Possible approaches to the chemotherapy of gut cancer.
    Proceedings of the Royal Society of Medicine, 1973, Volume: 66, Issue:12

    Topics: Animals; Azacitidine; Culture Techniques; Fluorouracil; Humans; Intestinal Neoplasms; Methods; Mice; Neoplasm Transplantation; Nitrosourea Compounds; Podophyllin

1973
Inhibition of ribosomal ribonucleic acid maturation by 5-azacytidine and 8-azaguanine in Novikoff hepatoma cells.
    Archives of biochemistry and biophysics, 1974, Volume: 160, Issue:1

    Topics: Animals; Azacitidine; Azaguanine; Carcinoma, Hepatocellular; Cells, Cultured; Cytidine; Dactinomycin; Electrophoresis, Polyacrylamide Gel; Fluorouracil; Guanosine; Isotope Labeling; Liver; Liver Neoplasms; Neoplasms, Experimental; Rats; RNA, Neoplasm; RNA, Ribosomal; Spectrophotometry, Ultraviolet; Time Factors; Tritium; Uridine

1974
[Antimetabolites in the treatment of acute human leukoses. Mechanism of action and conditioning factors in the cellular response to drugs. II].
    La Clinica terapeutica, 1974, Apr-30, Volume: 69, Issue:2

    Topics: Antimetabolites; Azacitidine; Azaguanine; Azauridine; Cell Membrane Permeability; Cytarabine; DNA, Neoplasm; Fluorouracil; Humans; Immunity, Cellular; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Mercaptopurine; Methotrexate; Purines; Pyrimidines

1974
St. Louis encephalitis virus temperature-sensitive mutants. I. Induction, isolation and preliminary characterization.
    Archives of virology, 1983, Volume: 75, Issue:3

    Topics: Azacitidine; Dactinomycin; Encephalitis Virus, St. Louis; Flavivirus; Fluorouracil; Genetic Complementation Test; Hot Temperature; Methylnitronitrosoguanidine; Mutation; Phenotype; RNA, Viral

1983
Drug resistance in cancer.
    Cancer treatment reports, 1984, Volume: 68, Issue:1

    Topics: Alkylating Agents; Antibiotics, Antineoplastic; Antineoplastic Agents; Azacitidine; Cisplatin; Cytarabine; Drug Resistance; Fluorouracil; Humans; Methotrexate; Neoplasms

1984
HIV-1 expression induced by anti-cancer agents in latently HIV-1-infected ACH2 cells.
    Biochemical and biophysical research communications, 1995, Feb-27, Volume: 207, Issue:3

    Topics: Antineoplastic Agents; Azacitidine; Base Sequence; CD4-Positive T-Lymphocytes; Cell Line; Cell Survival; Cytarabine; DNA; Fluorouracil; HIV-1; Methotrexate; Methylation; Molecular Sequence Data; NF-kappa B; Phytohemagglutinins; Tetradecanoylphorbol Acetate; Vinblastine

1995
Isolation and characterization of a highly attenuated respiratory syncytial virus (RSV) vaccine candidate by mutagenesis of the incompletely attenuated RSV A2 ts-1 NG-1 mutant virus.
    Vaccine, 1995, Volume: 13, Issue:5

    Topics: Animals; Azacitidine; Carcinoma, Squamous Cell; Chlorocebus aethiops; Female; Fluorouracil; Male; Mice; Mice, Inbred BALB C; Mutagenesis; Pan troglodytes; Phenotype; Respiratory Syncytial Virus Infections; Respiratory Syncytial Virus, Human; Temperature; Tumor Cells, Cultured; Vaccines, Attenuated; Vero Cells; Viral Vaccines; Virus Replication

1995
Utility of the murine erythroleukemic cell (MELC) in assessing mechanisms of action of DNA-active developmental toxicants: application to 5-fluorouracil.
    Teratology, 1993, Volume: 48, Issue:1

    Topics: Animals; Azacitidine; Cell Cycle; Cell Survival; Culture Techniques; Cyclophosphamide; Decitabine; DNA; Fetus; Fluorouracil; Leukemia, Erythroblastic, Acute; Mice; Teratogens; Thymidylate Synthase; Toxicology; Tumor Cells, Cultured

1993
Response of foot-and-mouth disease virus to increased mutagenesis: influence of viral load and fitness in loss of infectivity.
    Journal of virology, 2000, Volume: 74, Issue:18

    Topics: Amino Acid Substitution; Animals; Antigens, Viral; Aphthovirus; Azacitidine; Capsid; Capsid Proteins; Cell Line; Cell Survival; Cells, Cultured; Cricetinae; Fluorouracil; Mutagenesis; Mutagens; Reverse Transcriptase Polymerase Chain Reaction; Sequence Analysis, RNA; Viral Load; Viral Nonstructural Proteins

2000
Role of hMLH1 promoter hypermethylation in drug resistance to 5-fluorouracil in colorectal cancer cell lines.
    International journal of cancer, 2003, Aug-10, Volume: 106, Issue:1

    Topics: Adaptor Proteins, Signal Transducing; Antimetabolites, Antineoplastic; Azacitidine; Base Pair Mismatch; Blotting, Western; Carrier Proteins; Cloning, Molecular; Colorectal Neoplasms; Cyclin-Dependent Kinase Inhibitor p16; Decitabine; DNA Methylation; DNA Repair; Drug Resistance, Neoplasm; Enzyme Inhibitors; Fluorouracil; Humans; Immunoblotting; Kruppel-Like Transcription Factors; Microsatellite Repeats; MutL Protein Homolog 1; Neoplasm Proteins; Nuclear Proteins; Promoter Regions, Genetic; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors; Transcription Factors; Transcriptional Activation; Tumor Cells, Cultured

2003
The value of DNA methylation analysis in basic, initial toxicity assessments.
    Toxicological sciences : an official journal of the Society of Toxicology, 2004, Volume: 79, Issue:1

    Topics: Animals; Azacitidine; Base Composition; Cell Line, Tumor; Cytosine; DNA Methylation; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Fluorouracil; Gene Expression; Guanine; Mutagenicity Tests; Polymerase Chain Reaction; Rats; Rotenone; Staurosporine

2004
5-aza-2'-deoxycytidine sensitizes hepatoma and pancreatic cancer cell lines.
    Oncology reports, 2005, Volume: 14, Issue:4

    Topics: Antimetabolites, Antineoplastic; Antineoplastic Agents; Apoptosis; Azacitidine; Carcinoma, Hepatocellular; Cell Line, Tumor; Cell Survival; Decitabine; DNA; DNA Methylation; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Fluorouracil; HeLa Cells; Humans; Liver Neoplasms; Pancreatic Neoplasms; Prognosis; Time Factors; Treatment Outcome; Trypan Blue

2005
The Escherichia coli protein YjjG is a house-cleaning nucleotidase in vivo.
    FEMS microbiology letters, 2007, Volume: 270, Issue:1

    Topics: Azacitidine; Bromodeoxyuridine; Decitabine; Deoxyuridine; DNA Damage; Escherichia coli; Escherichia coli Proteins; Fluorouracil; Models, Biological; Molecular Structure; Mutation; N-Glycosyl Hydrolases; Nucleotidases; Orotic Acid; Substrate Specificity; Thymidine Monophosphate; Uridine

2007
Methylation of Ras association domain family protein 1, isoform A correlated with proliferation and drug resistance in hepatocellular carcinoma cell line SMMC-7721.
    Journal of gastroenterology and hepatology, 2007, Volume: 22, Issue:5

    Topics: Animals; Antineoplastic Agents; Azacitidine; Carcinoma, Hepatocellular; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cisplatin; Decitabine; DNA Methylation; DNA Modification Methylases; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Enzyme Inhibitors; Fluorouracil; Gene Expression Regulation, Neoplastic; Humans; Inhibitory Concentration 50; Liver Neoplasms; Mice; Mice, Inbred BALB C; Mice, Nude; Mitomycin; Neoplastic Stem Cells; Transfection; Tumor Suppressor Proteins

2007
The synergistic effect of 5-aza-2'-deoxycytidine and 5-fluorouracil on drug-resistant tumors.
    Oncology, 2006, Volume: 71, Issue:5-6

    Topics: Animals; Apoptosis; Apoptosis Regulatory Proteins; Azacitidine; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line, Tumor; Cell Proliferation; Colorectal Neoplasms; Cyclin-Dependent Kinase Inhibitor p16; Death-Associated Protein Kinases; Decitabine; DNA Methylation; Drug Resistance, Neoplasm; Drug Synergism; Fluorouracil; Humans; Mice; Mice, Nude; Reverse Transcriptase Polymerase Chain Reaction; Tumor Suppressor Protein p14ARF; Up-Regulation; Xenograft Model Antitumor Assays

2006
SPARC promoter hypermethylation in colorectal cancers can be reversed by 5-Aza-2'deoxycytidine to increase SPARC expression and improve therapy response.
    British journal of cancer, 2008, Jun-03, Volume: 98, Issue:11

    Topics: Antimetabolites, Antineoplastic; Azacitidine; Cell Line, Tumor; Cell Proliferation; Colorectal Neoplasms; CpG Islands; Decitabine; DNA Methylation; Fluorouracil; HT29 Cells; Humans; Osteonectin; Promoter Regions, Genetic

2008
Epigenetic reversal of acquired resistance to 5-fluorouracil treatment.
    Molecular cancer therapeutics, 2009, Volume: 8, Issue:5

    Topics: Animals; Antimetabolites, Antineoplastic; Azacitidine; Base Sequence; Cell Line, Tumor; Colorectal Neoplasms; CpG Islands; Decitabine; DNA Methylation; Drug Resistance, Neoplasm; Epigenomics; Fluorouracil; Gene Expression Regulation, Neoplastic; Gene Order; Humans; Mice; Mice, Nude; Molecular Sequence Data; Nucleoside-Phosphate Kinase; Promoter Regions, Genetic; RNA Stability; Uridine; Xenograft Model Antitumor Assays

2009
Demethylating agent 5-aza-2-deoxycytidine enhances susceptibility of breast cancer cells to anticancer agents.
    Molecular and cellular biochemistry, 2010, Volume: 342, Issue:1-2

    Topics: Antineoplastic Combined Chemotherapy Protocols; Azacitidine; Blotting, Western; Breast Neoplasms; Cell Proliferation; Decitabine; DNA Methylation; DNA Modification Methylases; Doxorubicin; Drug Synergism; Enzyme Inhibitors; Female; Flow Cytometry; Fluorouracil; Gene Expression Regulation, Neoplastic; Humans; Paclitaxel; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured

2010
Long-term persistence of acquired resistance to 5-fluorouracil in the colon cancer cell line SW620.
    Experimental cell research, 2010, Nov-15, Volume: 316, Issue:19

    Topics: AC133 Antigen; Antigens, CD; Azacitidine; beta Catenin; Cadherins; Cell Adhesion; Cell Death; Cell Line, Tumor; Cell Proliferation; Colonic Neoplasms; Culture Media, Serum-Free; DNA Methylation; Drug Resistance, Neoplasm; Epigenesis, Genetic; Epithelium; Fluorouracil; Glycoproteins; Humans; Hyaluronan Receptors; Inhibitory Concentration 50; Kinetics; Mesoderm; Peptides; Time Factors

2010
Increased proliferation and chemosensitivity of human mesenchymal stromal cells expressing fusion yeast cytosine deaminase.
    Stem cell research, 2012, Volume: 8, Issue:2

    Topics: Adipose Tissue; Apoptosis; Azacitidine; Breast Neoplasms; Cell Death; Cell Line, Tumor; Cell Proliferation; Cytarabine; Cytosine Deaminase; Drug Screening Assays, Antitumor; Female; Fluorouracil; Genetic Engineering; Green Fluorescent Proteins; Humans; Mesenchymal Stem Cells; Recombinant Fusion Proteins; Retroviridae; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Transduction, Genetic; Transgenes

2012
Characterization of the conversion between CD133+ and CD133- cells in colon cancer SW620 cell line.
    Cancer biology & therapy, 2012, Volume: 13, Issue:14

    Topics: AC133 Antigen; Animals; Antigens, CD; Azacitidine; Biomarkers, Tumor; Cell Line, Tumor; Colonic Neoplasms; Drug Resistance, Neoplasm; Flow Cytometry; Fluorouracil; Gene Expression Regulation, Neoplastic; Glycoproteins; Humans; Membrane Potential, Mitochondrial; Mice; Mice, Inbred BALB C; Mice, Nude; Neoplasm Transplantation; Neoplastic Stem Cells; Peptides; Reactive Oxygen Species; Transplantation, Heterologous

2012
Epigenetic silencing of DACH1 induces loss of transforming growth factor-β1 antiproliferative response in human hepatocellular carcinoma.
    Hepatology (Baltimore, Md.), 2013, Volume: 58, Issue:6

    Topics: Adolescent; Adult; Aged; Azacitidine; Carcinoma, Hepatocellular; DNA Methylation; Eye Proteins; Female; Fluorouracil; Gene Silencing; Humans; Liver Neoplasms; Male; Middle Aged; Signal Transduction; Transcription Factors; Transforming Growth Factor beta1; Tumor Suppressor Proteins

2013
Different effects of epigenetic modifiers on the cytotoxicity induced by 5-fluorouracil, irinotecan or oxaliplatin in colon cancer cells.
    Biological & pharmaceutical bulletin, 2014, Volume: 37, Issue:1

    Topics: Antimetabolites, Antineoplastic; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Azacitidine; Camptothecin; Cell Line, Tumor; Colonic Neoplasms; Decitabine; DNA; DNA Modification Methylases; Drug Synergism; Epigenesis, Genetic; Fluorouracil; HCT116 Cells; Histone Deacetylase Inhibitors; HT29 Cells; Humans; Irinotecan; Organoplatinum Compounds; Oxaliplatin

2014
High RAB25 expression is associated with good clinical outcome in patients with locally advanced head and neck squamous cell carcinoma.
    Cancer medicine, 2013, Volume: 2, Issue:6

    Topics: Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Azacitidine; Carcinoma, Squamous Cell; Cell Line; Cell Line, Tumor; Cell Movement; Cisplatin; Decitabine; Female; Fluorouracil; Head and Neck Neoplasms; Humans; Keratinocytes; Male; Middle Aged; Prognosis; rab GTP-Binding Proteins; RNA, Messenger; Squamous Cell Carcinoma of Head and Neck; Treatment Outcome

2013
[Effects of 5-Aza-dC on 5-Fu chemosensitivity by modulating TIP30 gene expression in human colorectal cancer cells].
    Zhonghua zhong liu za zhi [Chinese journal of oncology], 2013, Volume: 35, Issue:11

    Topics: Acetyltransferases; Antimetabolites, Antineoplastic; Azacitidine; Cell Proliferation; CpG Islands; Decitabine; DNA Methylation; Drug Resistance, Neoplasm; Fluorouracil; Gene Expression Regulation, Neoplastic; HCT116 Cells; Humans; Inhibitory Concentration 50; RNA, Messenger; Transcription Factors

2013
DNA methyltransferase inhibitors improve the effect of chemotherapeutic agents in SW48 and HT-29 colorectal cancer cells.
    PloS one, 2014, Volume: 9, Issue:3

    Topics: Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Azacitidine; Cell Cycle; Cell Line, Tumor; Colorectal Neoplasms; Cytidine; Decitabine; DNA Damage; DNA-Cytosine Methylases; Enzyme Inhibitors; Fluorouracil; Humans; Membrane Potential, Mitochondrial; Organoplatinum Compounds; Oxaliplatin

2014
5-Fluorouracil affects assembly of stress granules based on RNA incorporation.
    Nucleic acids research, 2014, Volume: 42, Issue:10

    Topics: Antimetabolites, Antineoplastic; Azacitidine; Cell Line; DNA; Eukaryotic Initiation Factor-2; Fluorouracil; GTP-Binding Proteins; HeLa Cells; Humans; Neoplasm Proteins; Oxidative Stress; Receptors for Activated C Kinase; Receptors, Cell Surface; Ribonucleoproteins; RNA; Stress, Physiological; Thioguanine

2014
Effective lethal mutagenesis of influenza virus by three nucleoside analogs.
    Journal of virology, 2015, Volume: 89, Issue:7

    Topics: Animals; Azacitidine; Cell Line; Dogs; Drug Resistance, Viral; Fluorouracil; Influenza A Virus, H1N1 Subtype; Influenza A Virus, H3N2 Subtype; Microbial Viability; Mutagenesis; Nucleosides; Ribavirin; Serial Passage; Virus Cultivation; Virus Replication

2015
Gelatinases-stimuli nanoparticles encapsulating 5-fluorouridine and 5-aza-2'-deoxycytidine enhance the sensitivity of gastric cancer cells to chemical therapeutics.
    Cancer letters, 2015, Jul-10, Volume: 363, Issue:1

    Topics: Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Azacitidine; Cell Line, Tumor; Cell Proliferation; Chemistry, Pharmaceutical; Decitabine; DNA Methylation; Dose-Response Relationship, Drug; Drug Stability; Enzyme Activation; Epigenesis, Genetic; Fluorouracil; Gene Expression Regulation, Neoplastic; Humans; Matrix Metalloproteinase 2; Matrix Metalloproteinase 9; Nanoparticles; Stomach Neoplasms; Time Factors; Transcription Factor AP-2

2015
Effects of ribavirin on the replication and genetic stability of porcine reproductive and respiratory syndrome virus.
    BMC veterinary research, 2015, Feb-07, Volume: 11

    Topics: Amiloride; Animals; Antiviral Agents; Azacitidine; Cell Line; Chlorocebus aethiops; Fluorouracil; Genome, Viral; Mutagenesis; Mutagens; Porcine respiratory and reproductive syndrome virus; Ribavirin; Virus Replication

2015
Epigenetic silencing of BCL6B inactivates p53 signaling and causes human hepatocellular carcinoma cell resist to 5-FU.
    Oncotarget, 2015, May-10, Volume: 6, Issue:13

    Topics: Aged; Antimetabolites, Antineoplastic; Apoptosis; Azacitidine; Carcinoma, Hepatocellular; Cell Proliferation; Decitabine; DNA Methylation; DNA Modification Methylases; Drug Resistance, Neoplasm; Early Growth Response Protein 1; Enzyme Inhibitors; Female; Fluorouracil; G1 Phase Cell Cycle Checkpoints; Gene Expression Regulation, Neoplastic; Gene Silencing; Hep G2 Cells; Humans; Liver Neoplasms; Male; Middle Aged; Promoter Regions, Genetic; Repressor Proteins; RNA Interference; Signal Transduction; Time Factors; Transfection; Tumor Suppressor Protein p53

2015
Characterization of MTAP Gene Expression in Breast Cancer Patients and Cell Lines.
    PloS one, 2016, Volume: 11, Issue:1

    Topics: Adenocarcinoma, Mucinous; Antineoplastic Agents; Azacitidine; Carcinoma, Ductal, Breast; Carcinoma, Lobular; Cell Line, Tumor; Cyclin-Dependent Kinase Inhibitor p16; DNA Methylation; Estrogen Receptor alpha; Female; Fluorouracil; Gene Expression Regulation, Neoplastic; Humans; Lymphatic Metastasis; Methotrexate; Organ Specificity; Promoter Regions, Genetic; Purine-Nucleoside Phosphorylase; Receptor, ErbB-2; Receptors, Progesterone; RNA, Small Interfering; Signal Transduction; Triple Negative Breast Neoplasms

2016
CETSA screening identifies known and novel thymidylate synthase inhibitors and slow intracellular activation of 5-fluorouracil.
    Nature communications, 2016, Mar-24, Volume: 7

    Topics: Activation, Metabolic; Azacitidine; Biological Assay; Deamination; Decitabine; Drug Evaluation, Preclinical; Enzyme Inhibitors; Fluorouracil; Humans; Intracellular Space; K562 Cells; Kinetics; Phosphorylation; Small Molecule Libraries; Thymidylate Synthase; Time Factors

2016
Efficacy of sodium hypochlorite in the degradation antineoplastic drugs by NMR spectroscopy.
    Giornale italiano di medicina del lavoro ed ergonomia, 2020, Volume: 42, Issue:2

    Topics: Antineoplastic Agents; Azacitidine; Carcinogens; Cytarabine; Decontamination; Drug Interactions; Ethanol; Fluorouracil; Humans; Hypochlorous Acid; Irinotecan; Magnetic Resonance Spectroscopy; Occupational Exposure; Preliminary Data; Sodium Chloride; Sodium Hypochlorite; Time Factors

2020
Inhibitory effect of bound polyphenol from foxtail millet bran on miR-149 methylation increases the chemosensitivity of human colorectal cancer HCT-8/Fu cells.
    Molecular and cellular biochemistry, 2021, Volume: 476, Issue:2

    Topics: Antimetabolites, Antineoplastic; Apoptosis; Azacitidine; Cell Proliferation; Colorectal Neoplasms; DNA Methylation; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluorouracil; Humans; MicroRNAs; Polyphenols; Setaria Plant

2021
Construction of an Enzyme-Free Initiator-Replicated Hybridization Chain Reaction Circuit for Amplified Methyltransferase Evaluation and Inhibitor Assay.
    Analytical chemistry, 2021, 02-02, Volume: 93, Issue:4

    Topics: Antimetabolites; Azacitidine; Escherichia coli; Fluorouracil; Methyltransferases; Nucleic Acid Amplification Techniques

2021
Epigenetic Manipulation Induced Production of Immunosuppressive Chromones and Cytochalasins from the Mangrove Endophytic Fungus
    Marine drugs, 2022, Sep-29, Volume: 20, Issue:10

    Topics: Animals; Azacitidine; Butyric Acid; Chromones; Concanavalin A; Cytochalasins; DNA; Doxorubicin; Epigenesis, Genetic; Fluorouracil; Fungi; Histone Deacetylases; Humans; Immunosuppressive Agents; Lipopolysaccharides; Methyltransferases; Mice; Molecular Structure

2022