Page last updated: 2024-09-05

atropine and wb 4101

atropine has been researched along with wb 4101 in 10 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(wb 4101)
Trials
(wb 4101)
Recent Studies (post-2010) (wb 4101)
26,7111,2591,697477134

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)wb 4101 (IC50)
Alpha-1A adrenergic receptorHomo sapiens (human)0.001

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19903 (30.00)18.7374
1990's3 (30.00)18.2507
2000's1 (10.00)29.6817
2010's3 (30.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Kung, HF; Kung, MP; Zhuang, ZP1
Varma, DR; Yue, TL1
Eckelman, WC; Francis, B; Gibson, RE; Grissom, MP; Reba, RC1
Adachi, M; Manita, S; Matsuda, T; Shigenobu, K; Tanaka, H1
Hatano, A; Koizumi, T; Komeyama, T; Takahashi, H; Takeda, M; Tamaki, M; Tsutsui, T1
Corrêa, FM; Fernandes, KB; Resstel, LB1
Prado, WA; Silva, JR; Silva, ML1
Fujita, T; Kumamoto, E; Liu, T1
Blaes, F; Dubuis, E; Goebel, A; Greensmith, D; Kuttikat, A; Leite, MI; Leuwer, M; Maihöfner, C; Shenker, N; Thompson, V; Vincent, A1

Trials

1 trial(s) available for atropine and wb 4101

ArticleYear
Longstanding complex regional pain syndrome is associated with activating autoantibodies against alpha-1a adrenoceptors.
    Pain, 2014, Volume: 155, Issue:11

    Topics: Adult; Animals; Atropine; Autoantibodies; Calcium; Cells, Cultured; Complex Regional Pain Syndromes; Cross-Over Studies; Dioxanes; Female; Humans; Immunoglobulin G; Immunoglobulins, Intravenous; Male; Membrane Potentials; Middle Aged; Muscarinic Antagonists; Myocytes, Cardiac; Patch-Clamp Techniques; Protein Binding; Rats; Receptors, Adrenergic, alpha-1; Transfection; Young Adult

2014

Other Studies

9 other study(ies) available for atropine and wb 4101

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Synthesis of (R,S)-trans-8-hydroxy-2-[N-n-propyl-N-(3'-iodo-2'-propenyl)amino]tetral in (trans-8-OH-PIPAT): a new 5-HT1A receptor ligand.
    Journal of medicinal chemistry, 1993, Oct-15, Volume: 36, Issue:21

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Iodine Radioisotopes; Ligands; Rats; Receptors, Serotonin; Stereoisomerism; Tetrahydronaphthalenes; Tritium

1993
Adrenoceptor blocking properties of atropine-like agents anisodamine and anisodine on brain and cardiovascular tissues of rats.
    British journal of pharmacology, 1986, Volume: 87, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Atropine; Brain; Cardiovascular System; Clonidine; Dioxanes; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Phenylephrine; Rats; Rats, Inbred Strains; Scopolamine Derivatives; Solanaceous Alkaloids; Vasodilator Agents

1986
The use of tritium labeled compounds to develop gamma-emitting receptor-binding radiotracers.
    International journal of nuclear medicine and biology, 1982, Volume: 9, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Atropine; Dihydroalprenolol; Dioxanes; Dogs; Guinea Pigs; Heart; Humans; Male; N-Methylscopolamine; Parasympatholytics; Pindolol; Prazosin; Propanolamines; Quinuclidinyl Benzilate; Rabbits; Radionuclide Imaging; Rats; Scopolamine Derivatives; Tritium

1982
Sustained negative inotropism mediated by alpha-adrenoceptors in adult mouse myocardia: developmental conversion from positive response in the neonate.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Animals, Newborn; Atropine; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Mice; Myocardial Contraction; Myocardium; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha; Yohimbine

1995
Alpha 1-adrenoceptors in the human prostatic urethra are different from those of the human peripheral arteries.
    The Clinical investigator, 1993, Volume: 72, Issue:1

    Topics: Arteries; Atropine; Clonidine; Dioxanes; Humans; Iliac Artery; Isometric Contraction; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha-1; Urethra; Yohimbine

1993
alpha-Adrenergic and muscarinic cholinergic receptors are not involved in the modulation of the parasympathetic baroreflex by the medial prefrontal cortex in rats.
    Life sciences, 2005, Aug-12, Volume: 77, Issue:13

    Topics: Animals; Atropine; Baroreflex; Cobalt; Dioxanes; Idazoxan; Male; Parasympathetic Nervous System; Phenylephrine; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Muscarinic

2005
Analgesia induced by 2- or 100-Hz electroacupuncture in the rat tail-flick test depends on the activation of different descending pain inhibitory mechanisms.
    The journal of pain, 2011, Volume: 12, Issue:1

    Topics: Adjuvants, Anesthesia; Adrenergic alpha-Antagonists; Analgesia; Anesthetics, Intravenous; Animals; Atropine; Baclofen; Bicuculline; Biophysics; Dioxanes; Disease Models, Animal; Electroacupuncture; GABA Agents; Male; Methysergide; Models, Biological; Multivariate Analysis; Naloxone; Narcotic Antagonists; Pain; Pain Management; Pain Measurement; Rats; Rats, Wistar; Reaction Time; Serotonin Antagonists; Tail; Thiopental; Time Factors

2011
Acetylcholine and norepinephrine mediate GABAergic but not glycinergic transmission enhancement by melittin in adult rat substantia gelatinosa neurons.
    Journal of neurophysiology, 2011, Volume: 106, Issue:1

    Topics: Acetylcholine; Adrenergic alpha-Antagonists; Animals; Atropine; Carbachol; Dioxanes; gamma-Aminobutyric Acid; Glycine; Indoles; Inhibitory Postsynaptic Potentials; Male; Mecamylamine; Melitten; Muscarinic Antagonists; Neurons; Nicotine; Nicotinic Antagonists; Norepinephrine; Purinergic P2X Receptor Antagonists; Pyridoxal Phosphate; Rats; Serotonin Antagonists; Substantia Gelatinosa; Synaptic Transmission; Tropisetron

2011