Page last updated: 2024-09-05

atropine and vesamicol

atropine has been researched along with vesamicol in 10 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(vesamicol)
Trials
(vesamicol)
Recent Studies (post-2010) (vesamicol)
26,7111,2591,697248021

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)vesamicol (IC50)
Vesicular acetylcholine transporterTetronarce californica (Pacific electric ray)0.034
Vesicular acetylcholine transporterHomo sapiens (human)1.52

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (30.00)18.2507
2000's3 (30.00)29.6817
2010's4 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Marien, MR; Richard, JW1
Araujo, DM; Hefti, F; Lapchak, PA1
Robinson, NE; Zhang, XY; Zhu, FX1
Haghimoto, K; Lurie, KG; Sugiyama, A; Takahara, A; Takehana, S1
Favaron, GO; Ferreira, AJ; Gomez, MV; Gusmão, DR; Kalapothakis, E; Kushmerick, C; Pinto de Almeida, A1
Bewick, GS; Fong, SW; McIntyre, A; McLennan, IS; Reid, J; Shennan, KI1
Chávez, J; Cruz-Valderrama, JE; Montaño, LM; Vargas, MH1
Abramochkin, DV; Borodinova, AA; Rosenshtraukh, LV1

Other Studies

10 other study(ies) available for atropine and vesamicol

ArticleYear
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Drug effects on the release of endogenous acetylcholine in vivo: measurement by intracerebral dialysis and gas chromatography-mass spectrometry.
    Journal of neurochemistry, 1990, Volume: 54, Issue:6

    Topics: Acetylcholine; Animals; Atropine; Chromatography, Gas; Consciousness; Corpus Striatum; Dialysis; Haloperidol; Magnesium; Male; Mass Spectrometry; Phencyclidine; Physostigmine; Piperidines; Potassium; Rats; Rats, Inbred Strains; Tetrodotoxin

1990
Cholinergic regulation of hippocampal brain-derived neurotrophic factor mRNA expression: evidence from lesion and chronic cholinergic drug treatment studies.
    Neuroscience, 1993, Volume: 52, Issue:3

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Atropine; Blotting, Northern; Brain; Brain-Derived Neurotrophic Factor; Female; Gene Expression Regulation; Hippocampus; Nerve Growth Factors; Nerve Tissue Proteins; Neuromuscular Depolarizing Agents; Nicotine; Piperidines; Pyramidal Tracts; Rats; Rats, Wistar; RNA, Messenger; Stereotaxic Techniques

1993
Origin and modulation of ACh release from rat airway cholinergic nerves.
    The American journal of physiology, 1997, Volume: 272, Issue:1 Pt 1

    Topics: Acetylcholine; Animals; Atropine; Calcium; Electric Stimulation; Extracellular Space; Female; Neuromuscular Depolarizing Agents; Parasympathetic Nervous System; Piperidines; Prostaglandins; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Tissue Distribution; Trachea

1997
Effects of a novel vesamicol receptor ligand, m-(iodobenzyl)trozamicol, on the canine isolated, blood-perfused atrioventricular node preparation.
    Japanese journal of pharmacology, 2000, Volume: 82, Issue:2

    Topics: Animals; Atrioventricular Node; Atropine; Cholinergic Antagonists; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Iodobenzenes; Perfusion; Piperidines; Receptors, Cholinergic

2000
Effects of the venom of a Mygalomorph spider (Lasiodora sp.) on the isolated rat heart.
    Toxicon : official journal of the International Society on Toxinology, 2003, Volume: 41, Issue:1

    Topics: Animals; Atropine; Dose-Response Relationship, Drug; Heart Conduction System; Heart Rate; Male; Neostigmine; Piperidines; Rats; Rats, Wistar; Spider Venoms; Spiders

2003
TGF-beta2 alters the characteristics of the neuromuscular junction by regulating presynaptic quantal size.
    Proceedings of the National Academy of Sciences of the United States of America, 2010, Jul-27, Volume: 107, Issue:30

    Topics: Acetylcholine; Animals; Atropine; Dose-Response Relationship, Drug; Evoked Potentials; Macrolides; Male; Mice; Mice, Inbred C57BL; Miniature Postsynaptic Potentials; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Neurotransmitter Agents; Parasympatholytics; Piperidines; Presynaptic Terminals; Rats; Receptors, Transforming Growth Factor beta; Synaptic Transmission; Transforming Growth Factor beta2

2010
Non-quantal release of acetylcholine in guinea-pig airways: role of choline transporter.
    Experimental physiology, 2011, Volume: 96, Issue:4

    Topics: Acetylcholine; Animals; Atropine; Calcium; Cation Transport Proteins; Cholinesterase Inhibitors; Electric Stimulation; Guinea Pigs; Hemicholinium 3; Hexamethonium; Male; Membrane Transport Proteins; Muscle Contraction; Muscle, Smooth; Neurons; omega-Conotoxin GVIA; Organophosphates; Paraoxon; Piperidines; Tetrodotoxin; Trachea; Vesicular Acetylcholine Transport Proteins

2011
Effects of acetylcholinesterase inhibitor paraoxon denote the possibility of non-quantal acetylcholine release in myocardium of different vertebrates.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 2012, Volume: 182, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Cholinesterase Inhibitors; Gadus morhua; Heart; Heart Atria; Heart Ventricles; Hemicholinium 3; In Vitro Techniques; Male; Myocardium; Paraoxon; Piperidines; Rana temporaria; Rats; Rats, Wistar; Vertebrates

2012