Page last updated: 2024-09-05

atropine and trifluoperazine

atropine has been researched along with trifluoperazine in 31 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(trifluoperazine)
Trials
(trifluoperazine)
Recent Studies (post-2010) (trifluoperazine)
26,7111,2591,6973,696157198

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)trifluoperazine (IC50)
Genome polyprotein 0.7
Ubiquitin carboxyl-terminal hydrolase 1Homo sapiens (human)8
Bile salt export pumpHomo sapiens (human)10
Lysozyme C-1Rattus norvegicus (Norway rat)9
Beta-glucuronidaseRattus norvegicus (Norway rat)7.8
ATP-dependent translocase ABCB1Homo sapiens (human)6.75
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)6.226
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.35
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.35
Pleiotropic ABC efflux transporter of multiple drugsSaccharomyces cerevisiae S288C1.4
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.35
D(2) dopamine receptorRattus norvegicus (Norway rat)0.016
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)6.226
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)6.226
WD repeat-containing protein 48Homo sapiens (human)8

Research

Studies (31)

TimeframeStudies, this research(%)All Research%
pre-199018 (58.06)18.7374
1990's4 (12.90)18.2507
2000's4 (12.90)29.6817
2010's5 (16.13)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baldy, WJ; Davis, CB; DiStefano, DL; Elgin, RJ; Fedde, CL; Kesslick, JM; Martin, GE; Mathiasen, JR; Scott, MK; Shank, RP1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Duffy, EM; Jorgensen, WL1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Chen, M; Fang, H; Liu, Z; Shi, Q; Tong, W; Vijay, V1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Vanderwolf, CH1
Biswas, PK; Paul, AK1
Nakagawa-Yagi, Y; Saito, Y; Takada, Y; Takayama, M1
Crevel, H; Marthan, R; Savineau, JP1
Harvey, GC; Leung, LW; Vanderwolf, CH1
Hiley, CR; Miller, RJ1
Kronberger, L1
Barkhatova, VP; Gotovtseva, EV; Ivanova-Smolenskaia, IA; Markova, ED; Tkachev, RA1
Morrison, AB; Webster, RA1
Burov, IuV; Kurochkin, IG2
Rao, HN; Tonapi, GT1
Gilev, AP; Temenchuk, EV1
Enyedi, P; Fredholm, BB1
Schoomaker, E; Tang, LC; Wiesmann, WP1
Pappas, BA; Vanderwolf, CH1
Barrington, M; Majewski, H1
Hirst, RA; Lambert, DG1
CLARKE, RS; DUNDEE, JW; LOVE, WJ; MOORE, J; NICHOLL, RM1
LAVERTY, R; SHARMAN, DF1
Borda, ES; Casanova, M; Furlán, C; Sterin-Borda, L1
Khuller, GK; Sharma, S; Singh, A1
Chang, LC; Huang, SC; Liu, CW; Liu, JK; Tsai, CC; Tsai, PJ; Tsai, TR; Wang, HC1

Reviews

1 review(s) available for atropine and trifluoperazine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

30 other study(ies) available for atropine and trifluoperazine

ArticleYear
Activity of aromatic substituted phenylpiperazines lacking affinity for dopamine binding sites in a preclinical test of antipsychotic efficacy.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:5

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Dose-Response Relationship, Drug; Piperazines; Rats; Receptors, Dopamine; Receptors, Serotonin; Structure-Activity Relationship

1989
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Prediction of drug solubility from Monte Carlo simulations.
    Bioorganic & medicinal chemistry letters, 2000, Jun-05, Volume: 10, Issue:11

    Topics: Monte Carlo Method; Pharmaceutical Preparations; Solubility

2000
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
FDA-approved drug labeling for the study of drug-induced liver injury.
    Drug discovery today, 2011, Volume: 16, Issue:15-16

    Topics: Animals; Benchmarking; Biomarkers, Pharmacological; Chemical and Drug Induced Liver Injury; Drug Design; Drug Labeling; Drug-Related Side Effects and Adverse Reactions; Humans; Pharmaceutical Preparations; Reproducibility of Results; United States; United States Food and Drug Administration

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Neocortical and hippocampal activation relation to behavior: effects of atropine, eserine, phenothiazines, and amphetamine.
    Journal of comparative and physiological psychology, 1975, Volume: 88, Issue:1

    Topics: Animals; Antipsychotic Agents; Atropine; Avoidance Learning; Behavior, Animal; Blood Pressure; Cerebral Cortex; Chlorpromazine; Dextroamphetamine; Electrodes, Implanted; Hippocampus; Male; Physostigmine; Rats; Respiration; Time Factors; Trifluoperazine

1975
Trifluoperazine in preanaesthetic medication.
    Journal of the Indian Medical Association, 1976, May-16, Volume: 66, Issue:10

    Topics: Adult; Atropine; Drug Therapy, Combination; Female; Humans; Male; Meperidine; Middle Aged; Preanesthetic Medication; Trifluoperazine

1976
Carbachol enhances forskolin-stimulated cyclic AMP accumulation via activation of calmodulin system in human neuroblastoma SH-SY5Y cells.
    Biochemical and biophysical research communications, 1991, Jul-15, Volume: 178, Issue:1

    Topics: Adenosine; Alprostadil; Atropine; Calmodulin; Carbachol; Cell Line; Colforsin; Cyclic AMP; Drug Synergism; Humans; Kinetics; Naphthalenes; Neuroblastoma; Pertussis Toxin; Polycyclic Compounds; Protein Kinase C; Trifluoperazine; Vasoactive Intestinal Peptide; Virulence Factors, Bordetella

1991
Contraction of vascular smooth muscle induced by phorbol 12,13 dibutyrate in human and rat pulmonary arteries.
    British journal of pharmacology, 1991, Volume: 104, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atropine; Calcium; Humans; In Vitro Techniques; Isometric Contraction; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Phentolamine; Phorbol 12,13-Dibutyrate; Potassium; Propranolol; Protein Kinase C; Pulmonary Artery; Rats; Tetrodotoxin; Trifluoperazine; Verapamil

1991
Transcallosal evoked potentials in relation to behavior in the rat: effects of atropine, p-chlorophenylalanine, reserpine, scopolamine and trifluoperazine.
    Behavioural brain research, 1987, Volume: 25, Issue:1

    Topics: Animals; Atropine; Behavior, Animal; Cerebral Cortex; Corpus Callosum; Evoked Potentials; Fenclonine; Male; Rats; Reserpine; Scopolamine; Trifluoperazine

1987
Anti-muscarinic properties of neuroleptics and drug-induced Parkinsonism.
    Nature, 1974, Apr-12, Volume: 248, Issue:449

    Topics: Adenylyl Cyclase Inhibitors; Animals; Atropine; Azirines; Benzoates; Benztropine; Cerebral Cortex; Corpus Striatum; Dibenzazepines; Ethanol; Extrapyramidal Tracts; In Vitro Techniques; Kinetics; Male; Parasympatholytics; Phenothiazines; Pimozide; Piperazines; Rats; Receptors, Drug; Spiro Compounds; Thioridazine; Thioxanthenes; Tranquilizing Agents; Trifluoperazine; Tritium

1974
[Use of a new oral anticholinergic agent in acute pancreatitis].
    Deutsches medizinisches Journal, 1970, Volume: 21, Issue:23

    Topics: Acute Disease; Administration, Oral; Adult; Aged; Atropine; Cholecystitis; Cholelithiasis; Female; Humans; Male; Middle Aged; Pancreatitis; Parasympatholytics; Quaternary Ammonium Compounds; Trifluoperazine

1970
[Principles of the pathogenetic therapy of congenital extrapyramidal diseases].
    Zhurnal nevropatologii i psikhiatrii imeni S.S. Korsakova (Moscow, Russia : 1952), 1973, Volume: 73, Issue:4

    Topics: Adolescent; Adult; Atropine; Basal Ganglia Diseases; Chelating Agents; Chronic Disease; Dihydroxyphenylalanine; Female; Hepatolenticular Degeneration; Humans; Hyperkinesis; Male; Pantothenate Kinase-Associated Neurodegeneration; Parkinson Disease; Penicillamine; Phenothiazines; Pyridoxine; Sulfhydryl Compounds; Trifluoperazine; Tropanes

1973
Drug-induced experimental Parkinsonism.
    Neuropharmacology, 1973, Volume: 12, Issue:8

    Topics: Animals; Atropine; Benztropine; Butyrophenones; Cats; Chlorpromazine; Dose-Response Relationship, Drug; Electromyography; Motor Neurons; Parkinson Disease; Parkinson Disease, Secondary; Phenothiazines; Rabbits; Rats; Reserpine; Tetanus; Time Factors; Tremorine; Trifluoperazine

1973
[Effect of psychotropic drugs on the emotional behavior of cats caused by the administration of acetylcholine into the central grey matter].
    Biulleten' eksperimental'noi biologii i meditsiny, 1971, Volume: 72, Issue:12

    Topics: Acetylcholine; Animals; Atropine; Behavior, Animal; Benactyzine; Cats; Chlordiazepoxide; Chlorpromazine; Haloperidol; Imipramine; Meprobamate; Morphine; Tranquilizing Agents; Trifluoperazine

1971
Effect of tranquillizers on the heart of Periplaneta americana (L.).
    Comparative and general pharmacology, 1971, Volume: 2, Issue:8

    Topics: Animals; Atropine; Chlorpromazine; Cockroaches; Depression, Chemical; Drug Interactions; Ethyl Ethers; Female; Heart; Heart Rate; Hydroxyzine; In Vitro Techniques; Thioridazine; Tranquilizing Agents; Trifluoperazine

1971
[Effect of psychotropic substances on the behavior of cats, induced by administration of acetylcholine into the hypothalamus].
    Farmakologiia i toksikologiia, 1971, Volume: 34, Issue:1

    Topics: Acetylcholine; Action Potentials; Amygdala; Animals; Atropine; Behavior, Animal; Benactyzine; Cats; Chlordiazepoxide; Chlorpromazine; Depression, Chemical; Electroencephalography; Haloperidol; Hostility; Hypothalamus; Imipramine; Meprobamate; Morphine; Reticular Formation; Stimulation, Chemical; Tranquilizing Agents; Trifluoperazine

1971
[Analysis of the serotonin-reactive structures of the glossomandibular reflex].
    Biulleten' eksperimental'noi biologii i meditsiny, 1968, Volume: 66, Issue:10

    Topics: Acetylcholine; Animals; Atropine; Blood-Brain Barrier; Brain; Cats; Chlorpromazine; Epinephrine; Ergotamine; Indoles; Isoproterenol; Lung; Morphine; Procaine; Proguanil; Receptors, Drug; Reflex; Serotonin; Serotonin Antagonists; Trifluoperazine; Tryptamines

1968
Calcium-dependent enhancement by carbachol of the VIP-induced cyclic AMP accumulation in cat submandibular gland.
    Acta physiologica Scandinavica, 1984, Volume: 120, Issue:4

    Topics: Animals; Atropine; Calcium; Carbachol; Cats; Cyclic AMP; Dose-Response Relationship, Drug; Egtazic Acid; Ethanol; Phospholipids; Receptors, Muscarinic; Submandibular Gland; Trifluoperazine; Vasoactive Intestinal Peptide

1984
Cholinergic agonists stimulate calcium uptake and cGMP formation in human erythrocytes.
    Biochimica et biophysica acta, 1984, May-16, Volume: 772, Issue:2

    Topics: Atropine; Biological Transport, Active; Calcimycin; Calcium; Carbachol; Cyclic GMP; Egtazic Acid; Erythrocyte Membrane; Erythrocytes; Humans; Kinetics; Receptors, Muscarinic; Trifluoperazine

1984
Reserpine abolishes movement-correlated atropine-resistant neocortical low voltage fast activity.
    Brain research, 1980, Nov-24, Volume: 202, Issue:1

    Topics: Animals; Atropine; Cerebral Cortex; Chlorpromazine; Evoked Potentials; Male; Motor Activity; Nialamide; Pimozide; Rats; Reserpine; Trifluoperazine

1980
Trifluoperazine and calmidazolium have multiple actions on the release of noradrenaline from sympathetic nerves of mouse atria.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 349, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Atropine; Calmodulin; Desipramine; Electric Stimulation; Enterochromaffin Cells; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Male; Mice; Myocardium; Norepinephrine; Phentolamine; Sympathetic Nervous System; Trifluoperazine

1994
Adenylyl cyclase in SH-SY5Y human neuroblastoma cells is regulated by intra- and extracellular calcium.
    Biochemical pharmacology, 1995, May-26, Volume: 49, Issue:11

    Topics: Adenylyl Cyclases; Atropine; Calcium; Carbachol; Cell Line; Cyclic AMP; Humans; Muscarine; Neuroblastoma; Potassium; Receptors, Muscarinic; Trifluoperazine

1995
STUDIES OF DRUGS GIVEN BEFORE ANAESTHESIA. VI. THE PHENOTHIAZINE DERIVATIVES.
    British journal of anaesthesia, 1965, Volume: 37

    Topics: Anesthesia; Anesthesia, General; Atropine; Chlorpromazine; Chlorprothixene; Fluphenazine; Humans; Meperidine; Methohexital; Methotrimeprazine; Nitrous Oxide; Oxygen; Perphenazine; Pharmacology; Phenothiazines; Preanesthetic Medication; Prochlorperazine; Promazine; Promethazine; Thiazines; Thiethylperazine; Toxicology; Tranquilizing Agents; Trifluoperazine; Triflupromazine; Trimeprazine

1965
MODIFICATION BY DRUGS OF THE METABOLISM OF 3,4-DIHYDROXYPHENYLETHYLAMINE, NORADRENALINE AND 5-HYDROXYTRYPTAMINE IN THE BRAIN.
    British journal of pharmacology and chemotherapy, 1965, Volume: 24

    Topics: Animals; Atropine; Behavior, Animal; Brain; Brain Chemistry; Cats; Caudate Nucleus; Cerebral Cortex; Chlorpromazine; Chromatography; Dextroamphetamine; Dihydroxyphenylalanine; Dogs; Dopamine; Ephedrine; Fluorometry; Guanethidine; Morphine; Norepinephrine; Parasympatholytics; Parkinsonian Disorders; Pharmacology; Phenobarbital; Proteins; Rabbits; Radiometry; Research; Reserpine; Serotonin; Thalamus; Thioridazine; Trifluoperazine; Tritium

1965
Muscarinic cholinoceptor activation modulates DNA synthesis and CD40 expression in fibroblast cells.
    Autonomic & autacoid pharmacology, 2006, Volume: 26, Issue:3

    Topics: Atropine; Calmodulin; Carbachol; CD40 Antigens; Cells, Cultured; DNA; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Fibroblasts; Flow Cytometry; Humans; Inositol Phosphates; Muscarinic Agonists; Muscarinic Antagonists; Pirenzepine; Pyrrolidinones; Quinuclidinyl Benzilate; Radioligand Assay; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Receptors, Muscarinic; Trifluoperazine; Type C Phospholipases

2006
cAMP regulates vegetative growth and cell cycle in Candida albicans.
    Molecular and cellular biochemistry, 2007, Volume: 304, Issue:1-2

    Topics: Aminophylline; Atropine; Candida albicans; Cell Cycle; Cell Proliferation; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Signal Transduction; Trifluoperazine

2007
Salvia miltiorrhiza causes tonic contraction in rat ileum through Ca²⁺-calmodulin pathway.
    Journal of ethnopharmacology, 2012, Aug-01, Volume: 142, Issue:3

    Topics: Abietanes; Animals; Atropine; Calcium; Calcium Channel Blockers; Calmodulin; Cell Line; Ileum; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Nifedipine; Plant Extracts; Plant Roots; Rats; Rats, Sprague-Dawley; Salvia miltiorrhiza; Sodium Channel Blockers; Tetrodotoxin; Trifluoperazine

2012