Page last updated: 2024-09-05

atropine and terodiline

atropine has been researched along with terodiline in 10 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(terodiline)
Trials
(terodiline)
Recent Studies (post-2010) (terodiline)
26,7111,2591,697138283

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)terodiline (IC50)
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)4.8
Catechol O-methyltransferaseRattus norvegicus (Norway rat)4.8
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)4.8
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.1272
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)4.8
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)4.8

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19901 (10.00)18.7374
1990's6 (60.00)18.2507
2000's2 (20.00)29.6817
2010's1 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Ekström, B1
Kura, H; Obara, K; Yabu, H1
Deguchi, Y; Kumada, S; Ohtsuka, M; Terai, T1
Kontani, H; Nakagawa, M; Sakai, T; Takeno, S1
Andersson, KE; Husted, S; Ostergaard, JR; Sommer, L1
Kaneko, S; Nakano, D; Nishimori, T; Ohara, M1
Hirota, T; Isogai, M; Kaneko, S; Nagao, M; Shimizu, H1

Other Studies

10 other study(ies) available for atropine and terodiline

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Intravesical instillation of drugs in patients with detrusor hyperactivity.
    Scandinavian journal of urology and nephrology. Supplementum, 1992, Volume: 149

    Topics: Administration, Intravesical; Animals; Atropine; Butylamines; Female; Humans; Parasympatholytics; Phentolamine; Rabbits; Urinary Bladder; Urinary Bladder, Neurogenic; Urodynamics; Verapamil

1992
Contractile responses to electrical field stimulation and ATP in guinea-pig urinary bladder.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1992, Volume: 102, Issue:1

    Topics: Adenosine Triphosphate; Animals; Atropine; Butylamines; Calcium; Calcium Channel Blockers; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Neurotransmitter Agents; Urinary Bladder

1992
Effects of the anticholinergic drug prifinium bromide on urinary bladder contractions in rat in vivo and in guinea-pig in vitro.
    Arzneimittel-Forschung, 1991, Volume: 41, Issue:4

    Topics: Animals; Atropine; Barium; Barium Compounds; Butylamines; Calcium Channel Blockers; Chlorides; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Mandelic Acids; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Parasympatholytics; Potassium Chloride; Pyrrolidines; Rats; Rats, Inbred Strains; Urinary Bladder

1991
Evaluation of drugs for treatment of urinary bladder dysfunction in conscious rats with intact pelvic nerve and after resection of the left pelvic nerve.
    Japanese journal of pharmacology, 1990, Volume: 53, Issue:4

    Topics: Animals; Atropine; Butylamines; Decerebrate State; Drug Evaluation; Male; Mandelic Acids; Nifedipine; Parasympatholytics; Physostigmine; Rats; Rats, Inbred Strains; Urinary Bladder; Urinary Bladder Diseases

1990
Anticholinergic and calcium antagonistic effects of terodiline in rabbit urinary bladder.
    Acta pharmacologica et toxicologica, 1980, Volume: 46 Suppl 1

    Topics: Animals; Atropine; Butylamines; Calcium; Carbachol; Dose-Response Relationship, Drug; Female; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Parasympatholytics; Potassium; Rabbits; Urinary Bladder

1980
[Effects of propiverine hydrochloride (propiverine) on isolated rat and dog urinary bladder].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 113, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Benzilates; Butylamines; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Female; In Vitro Techniques; Male; Mandelic Acids; Muscarinic Antagonists; Muscle Contraction; Parasympatholytics; Potassium Chloride; Propantheline; Rats; Rats, Wistar; Urinary Bladder; Urination; Urination Disorders; Vasodilator Agents; Verapamil

1999
[Effects of propiverine hydrochloride (propiverine) on the muscarinic receptor binding affinity in guinea pig tissues and on salivation in conscious dogs].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 113, Issue:3

    Topics: Animals; Atropine; Benzilates; Binding, Competitive; Butylamines; Cerebral Cortex; Dogs; Dose-Response Relationship, Drug; Female; Guinea Pigs; Heart; Ileum; Male; Mandelic Acids; Muscarinic Agonists; Muscarinic Antagonists; Parasympatholytics; Pilocarpine; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Salivary Glands; Salivation; Urinary Bladder; Urination Disorders

1999