Page last updated: 2024-09-05

atropine and tamsulosin

atropine has been researched along with tamsulosin in 16 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(tamsulosin)
Trials
(tamsulosin)
Recent Studies (post-2010) (tamsulosin)
26,7111,2591,6971,460468693

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)tamsulosin (IC50)
Alpha-1D adrenergic receptorHomo sapiens (human)0.0008
Alpha-1A adrenergic receptorHomo sapiens (human)0.0013
Alpha-1B adrenergic receptorHomo sapiens (human)0.0045
Alpha-1D adrenergic receptorMus musculus (house mouse)0.0018
Alpha-1B adrenergic receptorMus musculus (house mouse)0.0018
Alpha-1A adrenergic receptorMus musculus (house mouse)0.0018

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's8 (50.00)29.6817
2010's7 (43.75)24.3611
2020's1 (6.25)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Chen, M; Fang, H; Liu, Z; Shi, Q; Tong, W; Vijay, V1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Jones, LH; Nadanaciva, S; Rana, P; Will, Y1
Bendel, RE; Phillips, MB1
Osher, RH1
Belani, S; Masket, S1
Chang, DF; Koch, DD; Osher, RH; Wang, L1
Shugar, JK1
Akino, H; Aoki, Y; Ito, H; Miwa, Y; Oyama, N; Yokoyama, O1
Al-Ahmar, B; Haridas, A; Hingorani, M; Syrimi, M1
Ahmed, RO; Ajomale, K; Mustapha, A; Oladejo, RO; Owoyele, BV1
Bulut, AE; Esen, F; Toker, E1
Assia, EI; Atar Vardi, M; Eremenko, R; Hecht, I; Pras, E; Safir, M; Sharon, T1

Reviews

1 review(s) available for atropine and tamsulosin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

15 other study(ies) available for atropine and tamsulosin

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
FDA-approved drug labeling for the study of drug-induced liver injury.
    Drug discovery today, 2011, Volume: 16, Issue:15-16

    Topics: Animals; Benchmarking; Biomarkers, Pharmacological; Chemical and Drug Induced Liver Injury; Drug Design; Drug Labeling; Drug-Related Side Effects and Adverse Reactions; Humans; Pharmaceutical Preparations; Reproducibility of Results; United States; United States Food and Drug Administration

2011
Development of a cell viability assay to assess drug metabolite structure-toxicity relationships.
    Bioorganic & medicinal chemistry letters, 2016, 08-15, Volume: 26, Issue:16

    Topics: Adenosine Triphosphate; Benzbromarone; Cell Line; Cell Survival; Chromans; Cytochrome P-450 CYP2C9; Cytochrome P-450 CYP2D6; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Humans; Pharmaceutical Preparations; Thiazolidinediones; Troglitazone

2016
Preoperative use of atropine to prevent intraoperative floppy-iris syndrome in patients taking tamsulosin.
    Journal of cataract and refractive surgery, 2006, Volume: 32, Issue:10

    Topics: Adrenergic alpha-Antagonists; Atropine; Humans; Intraoperative Complications; Iris; Iris Diseases; Male; Mydriatics; Ophthalmic Solutions; Phacoemulsification; Preoperative Care; Prostatic Hyperplasia; Sulfonamides; Syndrome; Tamsulosin

2006
Preoperative atropine in IFIS.
    Journal of cataract and refractive surgery, 2007, Volume: 33, Issue:3

    Topics: Adrenergic alpha-Antagonists; Antineoplastic Agents; Atropine; Humans; Intraoperative Complications; Iris; Iris Diseases; Male; Mydriatics; Ophthalmic Solutions; Phacoemulsification; Preoperative Care; Prostatic Hyperplasia; Sulfonamides; Syndrome; Tamsulosin

2007
Combined preoperative topical atropine sulfate 1% and intracameral nonpreserved epinephrine hydrochloride 1:4000 [corrected] for management of intraoperative floppy-iris syndrome.
    Journal of cataract and refractive surgery, 2007, Volume: 33, Issue:4

    Topics: Administration, Topical; Adrenergic alpha-Antagonists; Atropine; Drug Therapy, Combination; Epinephrine; Humans; Intraoperative Complications; Iris; Iris Diseases; Male; Mydriatics; Preservatives, Pharmaceutical; Pupil; Sulfonamides; Syndrome; Tamsulosin

2007
Prospective multicenter evaluation of cataract surgery in patients taking tamsulosin (Flomax).
    Ophthalmology, 2007, Volume: 114, Issue:5

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Atropine; Eye Color; Humans; Incidence; Intraoperative Complications; Iris Diseases; Lens Implantation, Intraocular; Male; Phacoemulsification; Postoperative Complications; Prospective Studies; Sulfonamides; Syndrome; Tamsulosin; Treatment Outcome; Visual Acuity

2007
Prophylaxis for IFIS.
    Journal of cataract and refractive surgery, 2007, Volume: 33, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Atropine; Cataract Extraction; Drug Therapy, Combination; Epinephrine; Humans; Intraoperative Complications; Iris; Iris Diseases; Male; Mydriatics; Preservatives, Pharmaceutical; Prostatic Hyperplasia; Pupil; Sulfonamides; Syndrome; Tamsulosin

2007
Antimuscarinic drug inhibits detrusor overactivity induced by topical application of prostaglandin E2 to the urethra with a decrease in urethral pressure.
    The Journal of urology, 2007, Volume: 178, Issue:5

    Topics: Administration, Intravesical; Administration, Topical; Adrenergic alpha-Antagonists; Animals; Atropine; Benzilates; Calcium Channel Blockers; Cholinergic Antagonists; Dinoprostone; Disease Models, Animal; Female; Injections, Intra-Arterial; Muscarinic Antagonists; Muscle Contraction; omega-Conotoxins; Oxytocics; Pressure; Rats; Rats, Sprague-Dawley; Sulfonamides; Tamsulosin; Treatment Outcome; Urethra; Urinary Bladder; Urinary Bladder, Overactive; Verapamil

2007
Intraoperative floppy iris syndrome (IFIS) in patients receiving tamsulosin or doxazosin-a UK-based comparison of incidence and complication rates.
    Graefe's archive for clinical and experimental ophthalmology = Albrecht von Graefes Archiv fur klinische und experimentelle Ophthalmologie, 2013, Volume: 251, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Atropine; Doxazosin; Drug Therapy, Combination; Female; Humans; Incidence; Intraoperative Complications; Iris Diseases; Male; Muscle, Smooth; Mydriatics; Phacoemulsification; Phenylephrine; Prostatic Hyperplasia; Pupil; Retrospective Studies; Sulfonamides; Syndrome; Tamsulosin; United Kingdom

2013
Analgesic and anti-inflammatory effects of honey: the involvement of autonomic receptors.
    Metabolic brain disease, 2014, Volume: 29, Issue:1

    Topics: Adrenergic Antagonists; Analgesics, Non-Narcotic; Animals; Anti-Inflammatory Agents, Non-Steroidal; Atropine; Autonomic Nervous System; Carrageenan; Cholinergic Antagonists; Drug Evaluation, Preclinical; Drug Therapy, Combination; Edema; Formaldehyde; Hexamethonium; Honey; Hot Temperature; Indomethacin; Male; Pain Perception; Propranolol; Rats; Sulfonamides; Tamsulosin

2014
Efficacy and safety of low-concentration, bisulphite-containing, intracameral epinephrine and topical atropine treatments for the prevention of intraoperative floppy iris syndrome.
    Cutaneous and ocular toxicology, 2018, Volume: 37, Issue:3

    Topics: Administration, Ophthalmic; Adrenergic alpha-1 Receptor Antagonists; Aged; Aged, 80 and over; Atropine; Epinephrine; Follow-Up Studies; Humans; Incidence; Injections, Intraocular; Intraoperative Complications; Iris Diseases; Male; Middle Aged; Phacoemulsification; Preoperative Care; Preservatives, Pharmaceutical; Prostatic Hyperplasia; Pupil; Retrospective Studies; Sulfites; Sulfonamides; Tamsulosin; Treatment Outcome

2018
Preoperative atropine and non-steroidal anti-inflammatory drugs for the prevention of intraoperative floppy iris syndrome.
    Graefe's archive for clinical and experimental ophthalmology = Albrecht von Graefes Archiv fur klinische und experimentelle Ophthalmologie, 2022, Volume: 260, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Aged; Aged, 80 and over; Anti-Inflammatory Agents; Anti-Inflammatory Agents, Non-Steroidal; Atropine; Humans; Incidence; Intraoperative Complications; Iris; Iris Diseases; Male; Phacoemulsification; Pharmaceutical Preparations; Retrospective Studies; Sulfonamides; Tamsulosin

2022