Page last updated: 2024-09-05

atropine and sq-11725

atropine has been researched along with sq-11725 in 20 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(sq-11725)
Trials
(sq-11725)
Recent Studies (post-2010) (sq-11725)
26,7111,2591,697878223125

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19902 (10.00)18.7374
1990's5 (25.00)18.2507
2000's7 (35.00)29.6817
2010's6 (30.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Bard, B; Carrupt, PA; Martel, S1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Bellera, CL; Bruno-Blanch, LE; Castro, EA; Duchowicz, PR; Goodarzi, M; Ortiz, EV; Pesce, G; Talevi, A1
Bellman, K; Knegtel, RM; Settimo, L1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Finkielman, S; Finocchiaro, LM; Goldstein, DJ; Nahmod, VE1
Beccaria, E; Brun, S; Conti, M; Gaita, F; Giustetto, C1
Barg, AP; Bernstein, KN; O'Connor, DT1
Jones, DR; Signore, PE1
Bagheri, H; Berlan, M; Chale, JJ; Guyen, LN; Montastruc, JL; Tran, MA1
Liu, L; Nattel, S1
Hicks, KK; Kennedy, RH; Seifen, E; Stimers, JR1
Farrell, AP; Hicks, JM1

Trials

1 trial(s) available for atropine and sq-11725

ArticleYear
Nadolol: evidence for sympathetic nerve inhibition by a beta blocker in essential hypertension.
    Journal of hypertension, 1983, Volume: 1, Issue:3

    Topics: Adrenergic beta-Antagonists; Adult; Atropine; Blood Pressure; Humans; Hypertension; Male; Middle Aged; Nadolol; Nitrates; Pentanols; Phentolamine; Phenylephrine; Pressoreceptors; Propanolamines; Reflex; Sympathetic Nervous System

1983

Other Studies

19 other study(ies) available for atropine and sq-11725

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Lipophilicity of basic drugs measured by hydrophilic interaction chromatography.
    Journal of medicinal chemistry, 2009, May-28, Volume: 52, Issue:10

    Topics: Chemistry, Pharmaceutical; Chromatography; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Pharmaceutical Preparations; Solubility; Technology, Pharmaceutical

2009
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Prediction of drug intestinal absorption by new linear and non-linear QSPR.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:1

    Topics: Humans; Intestinal Absorption; Linear Models; Molecular Conformation; Nonlinear Dynamics; Permeability; Pharmaceutical Preparations; Probability; Quantitative Structure-Activity Relationship; Thermodynamics

2011
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
    Pharmaceutical research, 2014, Volume: 31, Issue:4

    Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation

2014
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Interaction of angiotensin II with the cholinergic and noradrenergic systems in the rat pineal gland: regulation of indole metabolism.
    The Journal of endocrinology, 1990, Volume: 126, Issue:1

    Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Animals; Atropine; Electric Stimulation; Indoles; Male; Melatonin; Nadolol; Norepinephrine; Pineal Gland; Rats; Rats, Inbred Strains; Serotonin; Tryptophan

1990
[Torsade de pointes during an atropine sulfate test in a patient with congenital long QT syndrome].
    Cardiologia (Rome, Italy), 1989, Volume: 34, Issue:12

    Topics: Arrhythmias, Cardiac; Atropine; Cardiac Pacing, Artificial; Humans; Long QT Syndrome; Male; Middle Aged; Nadolol; Propranolol; Tachycardia

1989
Effect of pharmacological blockade on cardiovascular responses to voluntary and forced diving in muskrats.
    The Journal of experimental biology, 1995, Volume: 198, Issue:Pt 11

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Arvicolinae; Atropine; Cardiovascular Physiological Phenomena; Cardiovascular System; Diving; Female; Heart Rate; Male; Muscarinic Antagonists; Nadolol; Phentolamine; Propranolol

1995
Evidence for activation of both adrenergic and cholinergic nervous pathways by yohimbine, an alpha 2-adrenoceptor antagonist.
    Fundamental & clinical pharmacology, 1995, Volume: 9, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Atropine; Autonomic Pathways; Dogs; Female; Insulin; Lipids; Male; Muscarinic Antagonists; Nadolol; Norepinephrine; Parasympathetic Nervous System; Salivation; Sympathetic Nervous System; Yohimbine

1995
Differing sympathetic and vagal effects on atrial fibrillation in dogs: role of refractoriness heterogeneity.
    The American journal of physiology, 1997, Volume: 273, Issue:2 Pt 2

    Topics: Animals; Anti-Arrhythmia Agents; Atrial Fibrillation; Atrial Function; Atropine; Dogs; Electric Stimulation; Female; Male; Nadolol; Refractory Period, Electrophysiological; Sympathetic Nervous System; Time Factors; Vagus Nerve

1997
Effects of streptozotocin-induced diabetes on heart rate, blood pressure and cardiac autonomic nervous control.
    Journal of the autonomic nervous system, 1998, Mar-03, Volume: 69, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Atropine; Autonomic Nervous System; Blood Glucose; Blood Pressure; Body Weight; Diabetes Mellitus, Experimental; Heart Conduction System; Heart Rate; Male; Nadolol; Parasympatholytics; Rats; Rats, Sprague-Dawley

1998
The cardiovascular responses of the red-eared slider (Trachemys scripta) acclimated to either 22 or 5 degrees C. II. Effects of anoxia on adrenergic and cholinergic control.
    The Journal of experimental biology, 2000, Volume: 203, Issue:Pt 24

    Topics: Acid-Base Equilibrium; Acidosis; Acute Disease; Adaptation, Physiological; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atropine; Blood Pressure; Body Weight; Cardiac Output; Cardiovascular Physiological Phenomena; Chronic Disease; Cold Temperature; Epinephrine; Heart Rate; Hematocrit; Hemoglobins; Hypoxia; Muscarinic Antagonists; Nadolol; Receptors, Adrenergic, beta; Receptors, Cholinergic; Tachycardia; Time Factors; Turtles

2000