Page last updated: 2024-09-05

atropine and methoctramine

atropine has been researched along with methoctramine in 83 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(methoctramine)
Trials
(methoctramine)
Recent Studies (post-2010) (methoctramine)
26,7111,2591,69740015
26,7111,2591,697332132

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)methoctramine (IC50)
CholinesteraseHomo sapiens (human)0.9772
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.0407
AcetylcholinesteraseHomo sapiens (human)5.3703
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.138
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.138
Carboxylic ester hydrolase Rattus norvegicus (Norway rat)0.9772

Research

Studies (83)

TimeframeStudies, this research(%)All Research%
pre-19908 (9.64)18.7374
1990's39 (46.99)18.2507
2000's25 (30.12)29.6817
2010's10 (12.05)24.3611
2020's1 (1.20)2.80

Authors

AuthorsStudies
Bonner, TI; Brann, MR; Buckley, CM; Buckley, NJ1
Angeli, P; Brasili, L; Giardinà, D; Melchiorre, C; Picchio, MT; Quaglia, W1
Kovacs, I; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1
Bolognesi, ML; Budriesi, R; Chiarini, A; Ghelardini, C; Melchiorre, C; Minarini, A; Rosini, M; Tumiatti, V; Wade, EJ1
Challiss, RA; Nahorski, SR; Nelson, CP1
Bellucci, C; Buccioni, M; Ghelardini, C; Marucci, G; Melchiorre, C; Milelli, A; Minarini, A; Rosini, M; Tumiatti, V1
Bhattacharjee, AK; Evans, SA; Gordon, RK; Pervitsky, D; Pomponio, JW1
Cassinelli, A; Melchiorre, C; Quaglia, W1
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Sastry, BV; Stephan, CC1
Cost, M; Majewski, H1
Jaiswal, N; Lambrecht, G; Malik, KU; Mutschler, E; Tacke, R1
Angeli, P; Brasili, L; Cingolani, ML; Marucci, G; Pigini, P; Tonnini, MC1
Yang, CM1
McLeskey, SW; Wojcik, WJ1
Alonso, R; Didier, M; Soubrie, P1
el-Fakahany, EE; Lee, NH1
Kenimer, JG; Takashima, A1
el-Fakahany, EE; Forray, C; Lee, NH1
Angeli, P; Lambrecht, G; Melchiorre, C; Moser, U; Mutschler, E; Wess, J1
Ortegón, ME; Raffa, RB; Watson, M1
Angeli, P; Lambrecht, G; Melchiorre, C; Mutschler, E; Picchio, MT; Wess, J1
Nakamura, K; Okuma, Y; Osumi, Y; Yokotani, K1
Eglen, RM; Ford, AP; Reddy, H; Watson, N1
Howell, RE; Kovalsky, MP1
Imaizumi, Y; Tanaka, M; Watanabe, M; Yamahara, NS1
Ballabeni, V; Barocelli, E; Caretta, A; Chiavarini, M; Impicciatore, M; Molina, E1
Howell, RE; Kovalsky, MP; Laemont, KD1
Bissonnette, BM; Brasitus, TA; Khare, S; Sitrin, MD; Tien, XY; Wali, RK; Wilson, D1
Davenport, TA; Fukumoto, Y; Gousse, A; Kamai, T; Latifpour, J; Weiss, RM; Yoshida, M1
De Klippel, N; Ebinger, G; Michotte, Y; Sarre, S1
Eglen, RM; Harris, GC1
Osumi, Y; Yokotani, K1
Acs, Z; Makara, GB; Pintér, I1
Latifpour, J; Mutoh, S; Saito, M; Weiss, RM1
Janković, SM; Milovanović, DR1
Levin, RJ; Przyborski, SA1
Semba, K; White, TD1
Hoover, DB; Neely, DA1
Hendrix, PK; Robinson, EP1
Abdollahi, M; Dehpour, AR; Kebriaeezadeh, A; Mohammad, M; Samini, M; Sharifzadeh, M1
Baba, H; Goldstein, PA; Kohno, T; Okamoto, M; Shimoji, K; Yoshimura, M1
Harsing, LG; Zigmond, MJ1
Eguchi, T; Ishida, H; Ishikawa, Y; Skowronski, MT1
Tobin, G1
Brefel-Courbon, C; Freslon, JL; Lazartigues, E; Montastruc, JL; Pelat, M; Rascol, O; Tellioglu, T; Tran, MA1
Pagano, AP; Parkman, HP; Ryan, JP1
Belmonte, KE; Costello, RW; Evans, CM; Fryer, AD; Gleich, GJ; Jacoby, DB; Yost, BL1
Bernardi, G; Bonci, A; Grillner, P; Mercuri, NB; Svensson, TH1
Goldie, RG; Preuss, JM1
Gharib, C; Lazartigues, E; Montastruc, JL; Montastruc, P; Pelat, M; Rascol, O; Tran, MA1
Halayko, AJ; Kahraman, S; Mitchell, RW; Solway, J; Wylam, ME1
Chang, KC; Chen, CL; Chiu, TH; Yang, YR1
Daniels, DV; Eglen, RM; Ford, AP; Hegde, SS; Meloy, TD1
Dohi, S; Ishizawa, Y; Ma, HC; Wang, YF; Yanagidate, F1
Herzog, M; Liu, J; Scherer, EQ; Scofield, MA; Shimozono, M; Wangemann, P1
Avellar, MC; Guaze, EF; Maróstica, E; Porto, CS1
Grbović, L; Jovanović, A; Pesić, S2
Goodhead, LH; Mitchell, SN; Moss, S; Sharott, A1
Abe, K; Chikuma, T; Hojyo, H; Kato, M; Miyatake, T; Taguchi, K; Utsunomiya, I1
Aita, T; Ishihata, A; Katano, Y; Tezuka, A1
Jankovic, SM; Jankovic, SV; Protic, BA1
Ando, S; Harasawa, I; Honda, K; Kamiya, HO; Koga, K; Takano, Y1
Funakami, Y; Hata, T; Itoh, E1
Avellar, MC; Maróstica, E; Porto, CS; Siu, ER; Yasuhara, F1
Gobbi, MD; Hita, FJ; Pujol Lereis, VA; Rodriguez, MC; Rothlin, RP; Verdi, MG1
Eguchi, K; Ohtubo, Y; Yoshii, K1
Huang, TJ; Ko, WC; Lin, LH; Lin, YL; Wang, SH; Wu, SN1
Advenier, C; Chen, HZ; Cui, YY; Devillier, P; Wang, H; Zhu, L1
Djokic, J; Grbovic, L; Nikolic, V; Pesic, S; Stoiljkovic, M1
Bae, H; Choi, SM; Kim, HN; Kim, SK; Koo, S; Min, BI; Park, JH; Sun, B1
Dentcheva, E; Gautam, D; Potluri, S; Rich, MM; Son, YJ; Tessler, A; Wang, X; Wess, J; Wright, MC1
Besalduch, N; Garcia, N; Lanuza, MA; Santafé, MM; Tomàs, J; Tomàs, M1
Chess-Williams, R; Moro, C; Uchiyama, J1
Chancellor, MB; Hirao, Y; Kita, M; Matsumoto, Y; Miyazato, M; Yokoyama, H; Yoshimura, N1
Alves-Do-Prado, W; Ambiel, CR; Antônio, MB; Correia-de-Sá, P; de Paula Ramos, E1
Killi, UK; Kuca, K; Soukup, O; Tobin, G; Winder, M; Wsol, V1
Anglister, L; Cherniak, M; Etlin, A; Finkel, E; Lev-Tov, A; Mor, Y1
Deng, J; Li, L; Shi, C; Song, B; Wu, Y; Zhang, X1
Giglio, D; Mukanyangezi, MF; Nieto-Marín, P; Podmolíková, L1
Lenina, OA; Petrov, KA1

Reviews

1 review(s) available for atropine and methoctramine

ArticleYear
The role of receptor binding in drug discovery.
    Journal of natural products, 1993, Volume: 56, Issue:4

    Topics: Animals; Drug Design; Humans; Receptors, Drug

1993

Other Studies

82 other study(ies) available for atropine and methoctramine

ArticleYear
Antagonist binding properties of five cloned muscarinic receptors expressed in CHO-K1 cells.
    Molecular pharmacology, 1989, Volume: 35, Issue:4

    Topics: Animals; Cell Line; Cloning, Molecular; Cricetinae; Humans; Kinetics; N-Methylscopolamine; Parasympatholytics; Rats; Receptors, Muscarinic; Scopolamine Derivatives

1989
Structure-activity relationships among methoctramine-related polymethylene tetraamines. Chain-length and substituent effects on M-2 muscarinic receptor blocking activity.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:1

    Topics: Animals; Carbachol; Chemical Phenomena; Chemistry; Diamines; Guinea Pigs; In Vitro Techniques; Male; Parasympatholytics; Polyamines; Rats; Receptors, Muscarinic; Structure-Activity Relationship

1989
Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Amino Acid Sequence; Animals; Carbachol; Cloning, Molecular; Cyclic AMP; Humans; Mice; Molecular Sequence Data; Muscarinic Agonists; Muscarinic Antagonists; Phosphatidylinositols; Radioligand Assay; Rats; Receptors, Muscarinic; Sequence Alignment; Sequence Homology, Amino Acid; Signal Transduction; Species Specificity

1998
Design, synthesis, and biological activity of methoctramine-related polyamines as putative G(i) protein activators.
    Journal of medicinal chemistry, 2001, Nov-22, Volume: 44, Issue:24

    Topics: Animals; Atrial Function; CHO Cells; Cricetinae; Diamines; Drug Design; Electric Stimulation; GTP-Binding Protein alpha Subunits, Gi-Go; Guinea Pigs; Heart Atria; Humans; In Vitro Techniques; Muscarinic Agonists; Polyamines; Rats; Receptors, Muscarinic; Structure-Activity Relationship

2001
Constitutive activity and inverse agonism at the M2 muscarinic acetylcholine receptor.
    The Journal of pharmacology and experimental therapeutics, 2006, Volume: 316, Issue:1

    Topics: Animals; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Immunoblotting; Inositol Phosphates; Ligands; Muscarinic Agonists; Mutagenesis, Site-Directed; Radioligand Assay; Receptor, Muscarinic M2; Transfection

2006
Structure-activity relationships of methoctramine-related polyamines as muscarinic antagonist: effect of replacing the inner polymethylene chain with cyclic moieties.
    Bioorganic & medicinal chemistry, 2007, Mar-15, Volume: 15, Issue:6

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Butyrylcholinesterase; Cerebral Cortex; CHO Cells; Cholinesterase Inhibitors; Cricetinae; Cricetulus; Diamines; Drug Design; Drug Evaluation, Preclinical; Guinea Pigs; Heart Atria; Humans; Ileum; Male; Mice; Molecular Structure; Muscarinic Antagonists; Muscle, Skeletal; Parietal Lobe; Photoaffinity Labels; Polyamines; Rabbits; Radioligand Assay; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Vas Deferens

2007
Discovery of subtype selective muscarinic receptor antagonists as alternatives to atropine using in silico pharmacophore modeling and virtual screening methods.
    Bioorganic & medicinal chemistry, 2013, May-01, Volume: 21, Issue:9

    Topics: Atropine; Computer Simulation; Drug Discovery; Humans; Models, Molecular; Molecular Structure; Receptor, Muscarinic M1; Structure-Activity Relationship

2013
Differential blockade of muscarinic receptor subtypes by polymethylene tetraamines. Novel class of selective antagonists of cardiac M-2 muscarinic receptors.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Guinea Pigs; Ileum; Indicators and Reagents; Kinetics; Male; Muscle, Smooth; Muscles; Myocardium; Polyamines; Ranidae; Receptors, Muscarinic; Receptors, Nicotinic; Structure-Activity Relationship; Urinary Bladder; Vas Deferens

1987
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
Characterization of the subtype of muscarinic receptor coupled to the stimulation of phosphoinositide hydrolysis in 132-1N1 human astrocytoma cells.
    Cellular and molecular biology (Noisy-le-Grand, France), 1992, Volume: 38, Issue:7

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Astrocytoma; Atropine; Carbachol; Diamines; Humans; Hydrolysis; Parasympathomimetics; Phosphatidylinositols; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine; Tumor Cells, Cultured

1992
Evidence for facilitatory and inhibitory muscarinic receptors on postganglionic sympathetic nerves in mouse isolated atria.
    British journal of pharmacology, 1991, Volume: 102, Issue:4

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Carbachol; Cocaine; Diamines; Dicyclomine; Female; Heart; Hexamethonium Compounds; In Vitro Techniques; Mice; Myocardium; Nerve Endings; Neurons; Norepinephrine; Parasympatholytics; Pirenzepine; Receptors, Muscarinic; Sympathetic Nervous System; Synaptic Transmission

1991
Pharmacological characterization of the vascular muscarinic receptors mediating relaxation and contraction in rabbit aorta.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Antihypertensive Agents; Aorta, Abdominal; Arecoline; Atropine; Diamines; Endothelium, Vascular; Hexamethonium; Hexamethonium Compounds; Indomethacin; Male; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Norepinephrine; Parasympatholytics; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic

1991
Pharmacological characterization of muscarinic receptor subtypes in rabbit isolated tissue preparations.
    Journal of autonomic pharmacology, 1991, Volume: 11, Issue:5

    Topics: Animals; Aorta, Thoracic; Atropine; Diamines; Jejunum; Male; Muscarinic Antagonists; Muscle Contraction; Myocardium; Parasympatholytics; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Vas Deferens; Vasodilation

1991
Characterization of muscarinic receptors in dog tracheal smooth muscle cells.
    Journal of autonomic pharmacology, 1991, Volume: 11, Issue:1

    Topics: Animals; Atropine; Carbachol; Diamines; Dogs; In Vitro Techniques; Kinetics; Muscle, Smooth; N-Methylscopolamine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives; Trachea

1991
Identification of muscarinic receptor subtypes present in cerebellar granule cells: prevention of [3H]propylbenzilyl choline mustard binding with specific antagonists.
    Neuropharmacology, 1990, Volume: 29, Issue:9

    Topics: Adenylyl Cyclase Inhibitors; Animals; Atropine; Cell Membrane; Cells, Cultured; Cerebellum; Diamines; Electrophoresis, Polyacrylamide Gel; Parasympatholytics; Pirenzepine; Propylbenzilylcholine Mustard; Quinuclidines; Receptors, Muscarinic; Xanthenes

1990
[3H]N-methylscopolamine binding studies reveal M2 and M3 muscarinic receptor subtypes on cerebellar granule cells in primary culture.
    Journal of neurochemistry, 1990, Volume: 55, Issue:1

    Topics: Animals; Atropine; Binding, Competitive; Cell Survival; Cells, Cultured; Cerebellum; Diamines; Granulocytes; N-Methylscopolamine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives; Tritium

1990
The allosteric binding profile of himbacine: a comparison with other cardioselective muscarinic antagonists.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Alkaloids; Allosteric Regulation; Animals; Atropine; Binding, Competitive; Diamines; Dose-Response Relationship, Drug; Furans; Gallamine Triethiodide; Male; Myocardium; N-Methylscopolamine; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives

1990
Muscarinic-stimulated norepinephrine release and phosphoinositide hydrolysis in PC12 cells are independent events.
    The Journal of biological chemistry, 1989, Jun-25, Volume: 264, Issue:18

    Topics: Adrenal Gland Neoplasms; Animals; Atropine; Cell Line; Diamines; Hydrolysis; Kinetics; Methacholine Chloride; Methacholine Compounds; Norepinephrine; Parasympathomimetics; Pheochromocytoma; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Pirenzepine; Rats; Receptors, Muscarinic

1989
Methoctramine, a cardioselective muscarinic antagonist, stimulates phosphoinositide hydrolysis in rat cerebral cortex.
    European journal of pharmacology, 1989, Aug-22, Volume: 167, Issue:2

    Topics: Animals; Atropine; Carbachol; Cerebral Cortex; Diamines; Hydrolysis; In Vitro Techniques; Male; Parasympatholytics; Phosphatidylinositols; Rats; Rats, Inbred Strains

1989
Methoctramine selectively blocks cardiac muscarinic M2 receptors in vivo.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 338, Issue:3

    Topics: Animals; Atropine; Blood Pressure; Diamines; Heart Rate; Male; Methacholine Chloride; Methacholine Compounds; Muscarine; Myocardium; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1988
Reciprocal hindlimb scratching and putative subtype-selective muscarinic agents.
    European journal of pharmacology, 1988, Dec-13, Volume: 158, Issue:3

    Topics: Animals; Atropine; Binding Sites; Diamines; Dose-Response Relationship, Drug; Drug Antagonism; Hindlimb; Injections, Spinal; Male; Mice; Parasympathomimetics; Pilocarpine; Receptors, Muscarinic; Succinimides; Trihexyphenidyl

1988
Antimuscarinic action of methoctramine, a new cardioselective M-2 muscarinic receptor antagonist, alone and in combination with atropine and gallamine.
    European journal of pharmacology, 1987, Dec-01, Volume: 144, Issue:2

    Topics: Animals; Atropine; Carbachol; Diamines; Drug Interactions; Gallamine Triethiodide; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Muscle Contraction; Myocardial Contraction; Rats; Receptors, Muscarinic

1987
Release of endogenous acetylcholine from a vascularly perfused rat stomach in vitro; inhibition by M3 muscarinic autoreceptors and alpha-2 adrenoceptors.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Adrenergic alpha-Antagonists; Animals; Atropine; Calcium; Clonidine; Diamines; Drug Interactions; Electric Stimulation; Gastric Mucosa; Hexamethonium; Hexamethonium Compounds; Male; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Perfusion; Phenylephrine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Stomach; Sympathetic Nervous System; Tetrodotoxin; Vagus Nerve

1993
Characterization of the interaction between muscarinic M2 receptors and beta-adrenoceptor subtypes in guinea-pig isolated ileum.
    British journal of pharmacology, 1995, Volume: 114, Issue:1

    Topics: Adrenergic beta-Agonists; Animals; Atropine; Cyclic AMP; Diamines; Dioxolanes; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; Male; Muscle, Smooth; Parasympatholytics; Receptors, Muscarinic

1995
Hypotensive effect of an M2-selective muscarinic antagonist in anaesthetized guinea-pigs.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:1

    Topics: Animals; Atropine; Blood Pressure; Depression, Chemical; Diamines; Guinea Pigs; Heart Rate; Male; Muscarinic Antagonists; Norepinephrine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic

1995
Pertussis toxin-sensitive muscarinic relaxation in the rat iris dilator muscle.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Diamines; Dose-Response Relationship, Drug; Furans; GTP-Binding Proteins; In Vitro Techniques; Iris; Male; Microinjections; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; Parasympatholytics; Pertussis Toxin; Phentolamine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Virulence Factors, Bordetella

1995
Regional differences in motor responsiveness to antimuscarinic drugs in rabbit isolated small and large intestine.
    Pharmacological research, 1995, Volume: 31, Issue:1

    Topics: Animals; Atropine; Benzodiazepinones; Diamines; Dose-Response Relationship, Drug; Gastrointestinal Motility; Intestine, Large; Intestine, Small; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic

1995
Methoctramine induces nonspecific airway hyperresponsiveness in vivo.
    European journal of pharmacology, 1994, Nov-14, Volume: 265, Issue:1-2

    Topics: Aerosols; Albuterol; Animals; Arachidonic Acid; Atropine; Bronchial Hyperreactivity; Bronchoconstriction; Diamines; Drug Synergism; Gallamine Triethiodide; Guinea Pigs; Histamine; Male; Muscarinic Antagonists; Ovalbumin; Parasympatholytics; Piperazines; Piperidines; Platelet Activating Factor; Propranolol; Receptors, Muscarinic

1994
Vitamin D status modulates rat colonic M3 muscarinic receptor characteristics and coupling to guanylate cyclase.
    FEBS letters, 1994, Jun-20, Volume: 347, Issue:1

    Topics: Animals; Atropine; Colon; Diamines; Enzyme Activation; Guanylate Cyclase; Male; Muscarinic Antagonists; Nutritional Status; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Vitamin D

1994
Diabetes-induced alterations in the properties of muscarinic cholinergic receptors in rat vas deferens.
    The Journal of urology, 1994, Volume: 152, Issue:3

    Topics: Animals; Atropine; Binding, Competitive; Diabetes Mellitus, Experimental; Diamines; Insulin; Male; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Up-Regulation; Vas Deferens

1994
Effect of M1- and M2-muscarinic drugs on striatal dopamine release and metabolism: an in vivo microdialysis study comparing normal and 6-hydroxydopamine-lesioned rats.
    Brain research, 1993, Dec-10, Volume: 630, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Atropine; Carbachol; Corpus Striatum; Diamines; Dopamine; Homovanillic Acid; Male; Microdialysis; Oxidopamine; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Reference Values

1993
Selective inactivation of muscarinic M2 and M3 receptors in guinea-pig ileum and atria in vitro.
    British journal of pharmacology, 1993, Volume: 109, Issue:4

    Topics: Alkylating Agents; Animals; Atropine; Diamines; Dioxolanes; Diphenylacetic Acids; Guinea Pigs; Heart; Heart Atria; Ileum; In Vitro Techniques; Isometric Contraction; Male; Muscarinic Antagonists; Muscle, Smooth; Parasympatholytics; Phenoxybenzamine; Pilocarpine; Piperidines; Receptors, Muscarinic

1993
Cholinergic M2 muscarinic receptor-mediated inhibition of endogenous noradrenaline release from the isolated vascularly perfused rat stomach.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:1

    Topics: Animals; Arteries; Atrial Function; Atropine; Depression, Chemical; Diamines; Electric Stimulation; Ethylmaleimide; Heart Atria; Male; Myocardial Contraction; Nerve Endings; Norepinephrine; Oxotremorine; Parasympatholytics; Perfusion; Pertussis Toxin; Phentolamine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Stomach; Sympathetic Nervous System; Vagus Nerve; Virulence Factors, Bordetella

1993
Acetylcholine stimulates growth hormone secretion in the neonatal rat pituitary.
    Journal of neuroendocrinology, 1996, Volume: 8, Issue:12

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Age Factors; Animals; Animals, Newborn; Atropine; Diamines; Dose-Response Relationship, Drug; Female; Growth Hormone; Male; Muscarinic Agonists; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Pituitary Gland; Rats; Rats, Wistar

1996
Evidence for the presence of regional differences in the subtype specificity of muscarinic receptors in rabbit lower urinary tract.
    The Journal of urology, 1997, Volume: 157, Issue:2

    Topics: Animals; Atropine; Carbachol; Diamines; Female; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Pirenzepine; Rabbits; Receptors, Muscarinic; Species Specificity; Urethra; Urinary Bladder

1997
Pharmacologic characterization of muscarine receptor subtypes in rat gastric fundus mediating contractile responses.
    The Indian journal of medical research, 1997, Volume: 105

    Topics: Acetylcholine; Animals; Atropine; Diamines; Female; Gastric Fundus; Gastrointestinal Motility; Male; Muscarinic Antagonists; Piperazines; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic

1997
Cholinergic modulation of electrogenic ion transport in different regions of the rat small intestine.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:7

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analysis of Variance; Animals; Atropine; Bethanechol; Carbachol; Chlorides; Diamines; Duodenum; Ileum; Intestinal Mucosa; Ion Transport; Jejunum; Male; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship; Tetrodotoxin

1997
M3 muscarinic receptor-mediated enhancement of NMDA-evoked adenosine release in rat cortical slices in vitro.
    Journal of neurochemistry, 1997, Volume: 69, Issue:3

    Topics: Adenosine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Atropine; Carbachol; Cerebral Cortex; Diamines; Drug Synergism; In Vitro Techniques; Kinetics; Magnesium; Male; Muscarinic Agonists; Muscarinic Antagonists; N-Methylaspartate; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic

1997
Differentiation of muscarinic receptors mediating negative chronotropic and vasoconstrictor responses to acetylcholine in isolated rat hearts.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Coronary Vessels; Depression, Chemical; Diamines; Heart Rate; In Vitro Techniques; Male; Pertussis Toxin; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Vasoconstriction; Virulence Factors, Bordetella

1997
Effects of a selective and a nonselective muscarinic cholinergic antagonist on heart rate and intestinal motility in dogs.
    Journal of veterinary pharmacology and therapeutics, 1997, Volume: 20, Issue:5

    Topics: Animals; Atropine; Cross-Over Studies; Diamines; Dog Diseases; Dogs; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Heart Rate; Injections, Intramuscular; Injections, Intravenous; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Regression Analysis; Tachycardia

1997
Alterations of physostigmine-induced yawning by chronic lithium administration in rats.
    Pharmacology & toxicology, 1997, Volume: 81, Issue:4

    Topics: Animals; Antimanic Agents; Atropine; Diamines; Dose-Response Relationship, Drug; Drug Synergism; Injections, Intraperitoneal; Injections, Intraventricular; Lithium Chloride; Male; Muscarinic Antagonists; Parasympatholytics; Physostigmine; Pirenzepine; Rats; Yawning

1997
Muscarinic facilitation of GABA release in substantia gelatinosa of the rat spinal dorsal horn.
    The Journal of physiology, 1998, Apr-01, Volume: 508 ( Pt 1)

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Carbachol; Diamines; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Muscarinic Agonists; Neostigmine; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin

1998
Postsynaptic integration of cholinergic and dopaminergic signals on medium-sized GABAergic projection neurons in the neostriatum.
    Brain research bulletin, 1998, Volume: 45, Issue:6

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Diamines; Electric Stimulation; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Models, Neurological; Muscarinic Agonists; Muscarinic Antagonists; Neostriatum; Neurons; Oxotremorine; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptors, Dopamine; Receptors, Muscarinic; Signal Transduction; Sulpiride; Tetrodotoxin

1998
Acetylcholine acts on M3 muscarinic receptors and induces the translocation of aquaporin5 water channel via cytosolic Ca2+ elevation in rat parotid glands.
    Biochemical and biophysical research communications, 1998, Apr-28, Volume: 245, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetylcholine; Animals; Aquaporin 5; Aquaporins; Atropine; Calcimycin; Calcium; Calcium Channel Blockers; Cytosol; Diamines; Enzyme Inhibitors; Gallic Acid; Ion Channels; Ionophores; Male; Membrane Proteins; Parasympatholytics; Parotid Gland; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic; Staurosporine

1998
Presynaptic muscarinic M1 and M2 receptor modulation of auriculotemporal nerve transmission in the rat.
    Journal of the autonomic nervous system, 1998, Aug-06, Volume: 72, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Diamines; Ear; Electric Stimulation; Male; Muscarinic Antagonists; Parasympathetic Nervous System; Parasympatholytics; Parotid Gland; Pirenzepine; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Regional Blood Flow; Scalp; Synaptic Transmission

1998
Pressor and bradycardic effects of tacrine and other acetylcholinesterase inhibitors in the rat.
    European journal of pharmacology, 1998, Nov-13, Volume: 361, Issue:1

    Topics: Adrenergic Antagonists; Animals; Antidiuretic Hormone Receptor Antagonists; Atropine; Atropine Derivatives; Blood Pressure; Carbamates; Cardiovascular Agents; Chlorisondamine; Cholinergic Antagonists; Cholinesterase Inhibitors; Diamines; Diastole; Dose-Response Relationship, Drug; Heart Rate; Male; Phenylcarbamates; Physostigmine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Rivastigmine; Systole; Tacrine

1998
Subtypes of muscarinic receptors regulating gallbladder cholinergic contractions.
    The American journal of physiology, 1999, Volume: 276, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Diamines; Electric Stimulation; Gallbladder; Guinea Pigs; Hexamethonium; Muscarinic Antagonists; Muscle Contraction; Parasympatholytics; Piperidines; Pirenzepine; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Tetrodotoxin; Tropicamide

1999
Antigen-induced hyperreactivity to histamine: role of the vagus nerves and eosinophils.
    The American journal of physiology, 1999, Volume: 276, Issue:5

    Topics: Animals; Antibodies; Antigens; Atropine; Blood Proteins; Bronchoconstriction; Diamines; Eosinophil Granule Proteins; Eosinophils; Guinea Pigs; Histamine; Integrin alpha4beta1; Integrins; Muscarinic Agonists; Muscarinic Antagonists; Ovalbumin; Receptor, Muscarinic M2; Receptors, Lymphocyte Homing; Receptors, Muscarinic; Ribonucleases; Vagotomy; Vagus Nerve

1999
Presynaptic muscarinic (M3) receptors reduce excitatory transmission in dopamine neurons of the rat mesencephalon.
    Neuroscience, 1999, Volume: 91, Issue:2

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Atropine; Carbachol; Diamines; Dicyclomine; Dopamine; Electric Stimulation; Excitatory Postsynaptic Potentials; Mesencephalon; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Parasympatholytics; Physostigmine; Piperidines; Pirenzepine; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Rats, Wistar; Reaction Time; Receptor, Muscarinic M3; Receptors, Muscarinic; Synaptic Transmission; Tetrodotoxin

1999
Muscarinic cholinoceptor subtypes mediating tracheal smooth muscle contraction and inositol phosphate generation in guinea pig and rat.
    European journal of pharmacology, 1999, May-21, Volume: 372, Issue:3

    Topics: Animals; Atropine; Diamines; Guinea Pigs; In Vitro Techniques; Inositol Phosphates; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Trachea

1999
Characterization of the central muscarinic cholinoceptors involved in the cholinergic pressor response in anesthetized dogs.
    European journal of pharmacology, 1999, 08-27, Volume: 379, Issue:2-3

    Topics: Acetylcholine; Anesthesia; Animals; Atropine; Blood Pressure; Diamines; Dogs; Dose-Response Relationship, Drug; Male; Muscarinic Antagonists; Norepinephrine; Receptor, Muscarinic M1; Receptors, Muscarinic; Vasodilator Agents; Vasopressins

1999
Selective restoration of calcium coupling to muscarinic M(3) receptors in contractile cultured airway myocytes.
    American journal of physiology. Lung cellular and molecular physiology, 2000, Volume: 278, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Blood Proteins; Blotting, Western; Bradykinin; Calcium; Calcium Channels; Cells, Cultured; Diamines; Dogs; Dose-Response Relationship, Drug; Fluorescent Dyes; Fura-2; Inositol 1,4,5-Trisphosphate Receptors; Macrocyclic Compounds; Muscarinic Antagonists; Muscle, Smooth; Oxazoles; Parasympatholytics; Phenotype; Piperidines; Pirenzepine; Receptor, Muscarinic M3; Receptors, Bradykinin; Receptors, Cytoplasmic and Nuclear; Receptors, Muscarinic; Trachea; Vasodilator Agents

2000
Arecoline excites rat locus coeruleus neurons by activating the M2-muscarinic receptor.
    The Chinese journal of physiology, 2000, Mar-31, Volume: 43, Issue:1

    Topics: Alzheimer Disease; Animals; Arecoline; Atropine; Cholinergic Agonists; Diamines; Hexamethonium; Locus Coeruleus; Male; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptors, Muscarinic

2000
Functional characterization of rat submaxillary gland muscarinic receptors using microphysiometry.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: Alkaloids; Animals; Atropine; Benzhydryl Compounds; Benzodiazepinones; Binding, Competitive; Biosensing Techniques; Carbachol; Cholinergic Agonists; Cresols; Diamines; Dose-Response Relationship, Drug; Furans; Male; Mandelic Acids; Muscarinic Antagonists; Naphthalenes; Phenethylamines; Phenylpropanolamine; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Submandibular Gland; Tolterodine Tartrate

2001
The antinociceptive and sedative effects of carbachol and oxycodone administered into brainstem pontine reticular formation and spinal subarachnoid space in rats.
    Anesthesia and analgesia, 2001, Volume: 92, Issue:5

    Topics: Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Atropine; Behavior, Animal; Carbachol; Cholinergic Agonists; Conscious Sedation; Diamines; Injections, Spinal; Male; Microinjections; Motor Activity; Muscarinic Antagonists; Pain Threshold; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Reticular Formation; Subarachnoid Space

2001
Muscarinic receptors control K+ secretion in inner ear strial marginal cells.
    The Journal of membrane biology, 2001, Aug-01, Volume: 182, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Atropine; Calcium; Carbachol; Cholinergic Agonists; Cloning, Molecular; Cyclic AMP; Diamines; Dose-Response Relationship, Drug; Gerbillinae; Isoproterenol; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Potassium; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; Stria Vascularis

2001
Characterization of muscarinic acetylcholine receptors in the rat epididymis.
    Biology of reproduction, 2001, Volume: 65, Issue:4

    Topics: Animals; Atropine; Cell Membrane; Diamines; Epididymis; Male; Muscarinic Antagonists; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tritium

2001
Muscarinic receptor subtypes mediating vasorelaxation of the perforating branch of the human internal mammary artery.
    Pharmacology, 2001, Volume: 63, Issue:3

    Topics: Acetylcholine; Adult; Aged; Atropine; Diamines; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Humans; In Vitro Techniques; Mammary Arteries; Middle Aged; Muscarinic Antagonists; Piperidines; Pirenzepine; Receptors, Muscarinic; Vasodilation; Vasodilator Agents

2001
Acetylcholine-induced contractions in the perforating branch of the human internal mammary artery: protective role of the vascular endothelium.
    Pharmacology, 2002, Volume: 64, Issue:4

    Topics: Acetylcholine; Atropine; Diamines; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Female; Humans; In Vitro Techniques; Indomethacin; Mammary Arteries; Middle Aged; Muscarinic Antagonists; Nitric Oxide Synthase; omega-N-Methylarginine; Phenylephrine; Piperidines; Pirenzepine; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents

2002
Role of muscarinic receptors in the activation of the ventral subiculum and the consequences for dopamine release in the nucleus accumbens.
    European journal of pharmacology, 2003, Jan-24, Volume: 460, Issue:2-3

    Topics: Animals; Atropine; Bicuculline; Bridged-Ring Compounds; Carbachol; Cholinergic Agonists; Diamines; Dopamine; Hippocampus; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nucleus Accumbens; Oxotremorine; Pilocarpine; Pyridines; Rats; Receptors, Muscarinic; Spiro Compounds; Thiadiazoles; Tropanes

2003
Characterization of muscarinic receptor subtypes in the rostral ventrolateral medulla and effects on morphine-induced antinociception in rats.
    European journal of pharmacology, 2003, Apr-04, Volume: 465, Issue:3

    Topics: Analgesics, Opioid; Animals; Atropine; Diamines; Male; Mecamylamine; Medulla Oblongata; Microinjections; Morphine; Naloxone; Narcotic Antagonists; Pain Measurement; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Time Factors

2003
Aging-related alterations in the contractile responses to acetylcholine, muscarinic cholinoceptors and cholinesterase activities in jejunum and colon of the male Fischer 344 rats.
    Experimental gerontology, 2004, Volume: 39, Issue:1

    Topics: Acetylcholine; Aging; Animals; Atropine; Cholinesterases; Colon; Diamines; Dose-Response Relationship, Drug; Gastrointestinal Motility; In Vitro Techniques; Intestine, Large; Jejunum; Male; Muscarinic Antagonists; Muscle, Smooth; Piperidines; Pirenzepine; Rats; Rats, Inbred F344

2004
Contractile effect of acetylcholine on isolated isthmic segment of fallopian tubes.
    Methods and findings in experimental and clinical pharmacology, 2004, Volume: 26, Issue:2

    Topics: Acetylcholine; Adult; Aged; Atropine; Diamines; Dose-Response Relationship, Drug; Fallopian Tubes; Female; Follicular Phase; Humans; Lidocaine; Luteal Phase; Mecamylamine; Middle Aged; Muscle Contraction; Muscle, Smooth; Nifedipine; Piperidines; Pirenzepine; Postmenopause; Receptors, Muscarinic

2004
Intrathecal clonidine inhibits mechanical allodynia via activation of the spinal muscarinic M1 receptor in streptozotocin-induced diabetic mice.
    European journal of pharmacology, 2004, Nov-28, Volume: 505, Issue:1-3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analgesics; Animals; Atropine; Blood Glucose; Clonidine; Diabetes Mellitus, Experimental; Diamines; Injections, Spinal; Male; Mice; Motor Activity; Muscarinic Agonists; Muscarinic Antagonists; Pain; Pain Threshold; Piperidines; Pirenzepine; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Spinal Cord; Streptozocin; Stress, Mechanical; Time Factors

2004
Effects of AF-DX116 and other muscarinic receptor antagonists on orthostatic hypotension in autonomic imbalanced (SART-stressed) rats.
    Journal of pharmacological sciences, 2005, Volume: 97, Issue:3

    Topics: Animals; Atropine; Atropine Derivatives; Blood Pressure; Cold Temperature; Diamines; Heart Rate; Hypotension, Orthostatic; Male; Muscarinic Antagonists; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Stress, Physiological

2005
Expression and localization of muscarinic acetylcholine receptor subtypes in rat efferent ductules and epididymis.
    Cell and tissue research, 2006, Volume: 323, Issue:1

    Topics: Animals; Atropine; Carbachol; Cell Membrane; Diamines; Ejaculatory Ducts; Epididymis; Immunohistochemistry; In Vitro Techniques; Male; Muscarinic Antagonists; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic

2006
Pharmacological characterization of muscarinic receptor subtypes mediating vasoconstriction of human umbilical vein.
    British journal of pharmacology, 2006, Volume: 147, Issue:5

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Atropine; Diamines; Humans; In Vitro Techniques; Piperidines; Pirenzepine; Receptors, Muscarinic; Umbilical Veins; Vasoconstriction

2006
Functional expression of M3, a muscarinic acetylcholine receptor subtype, in taste bud cells of mouse fungiform papillae.
    Chemical senses, 2008, Volume: 33, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Calcium Signaling; Cells, Cultured; Diamines; Electrophysiology; Gene Expression; Inositol 1,4,5-Trisphosphate Receptors; Mice; Mice, Inbred Strains; Muscarinic Antagonists; Patch-Clamp Techniques; Phospholipase C beta; Piperidines; Pirenzepine; Receptor, Muscarinic M3; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; Synaptosomal-Associated Protein 25; Taste Buds; Tropicamide; Vesicular Acetylcholine Transport Proteins

2008
Bronchodilatory effects of S-isopetasin, an antimuscarinic sesquiterpene of Petasites formosanus, on obstructive airway hyperresponsiveness.
    European journal of pharmacology, 2008, Apr-28, Volume: 584, Issue:2-3

    Topics: Acetylcholine; Animals; Atropine; Binding, Competitive; Bronchial Hyperreactivity; Bronchoconstrictor Agents; Bronchodilator Agents; Cells, Cultured; Cholinesterase Inhibitors; Diamines; Dose-Response Relationship, Drug; Guinea Pigs; Humans; Ipratropium; Male; Muscarinic Antagonists; Muscle, Smooth; N-Methylscopolamine; Neostigmine; Petasites; Piperidines; Protein Binding; Receptor, Muscarinic M3; Sesquiterpenes; Time Factors; Trachea

2008
Muscarinic receptors involved in airway vascular leakage induced by experimental gastro-oesophageal reflux.
    Life sciences, 2008, Apr-23, Volume: 82, Issue:17-18

    Topics: Animals; Atropine; Capillary Permeability; Diamines; Female; Ganglionic Blockers; Gastroesophageal Reflux; Guinea Pigs; Hexamethonium; In Vitro Techniques; Male; Muscarinic Antagonists; Nicotinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Receptors, Nicotinic; Regional Blood Flow; Respiratory System

2008
Functional characterization of the muscarinic receptors involved in endothelium-dependent relaxation in isolated canine uterine artery.
    Journal of veterinary pharmacology and therapeutics, 2009, Volume: 32, Issue:2

    Topics: Acetylcholine; Animals; Arteries; Atropine; Cholinergic Agents; Diamines; Dogs; Endothelium, Vascular; Female; Hysterectomy; In Vitro Techniques; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Uterus

2009
Spinal cholinergic mechanism of the relieving effects of electroacupuncture on cold and warm allodynia in a rat model of neuropathic pain.
    The journal of physiological sciences : JPS, 2009, Volume: 59, Issue:4

    Topics: Animals; Atropine; Cholinergic Agents; Cholinergic Fibers; Cold Temperature; Diamines; Disease Models, Animal; Electroacupuncture; Hot Temperature; Hyperesthesia; Male; Mecamylamine; Neuralgia; Pain Threshold; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Spinal Nerves

2009
Distinct muscarinic acetylcholine receptor subtypes contribute to stability and growth, but not compensatory plasticity, of neuromuscular synapses.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, Nov-25, Volume: 29, Issue:47

    Topics: Animals; Atropine; Denervation; Diamines; Female; Growth Cones; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Neurons; Muscarinic Antagonists; Muscle Fibers, Skeletal; Muscle, Skeletal; Nerve Regeneration; Neuromuscular Junction; Neuronal Plasticity; Paralysis; Presynaptic Terminals; Protein Isoforms; Receptors, Muscarinic; Wallerian Degeneration

2009
The interaction between tropomyosin-related kinase B receptors and presynaptic muscarinic receptors modulates transmitter release in adult rodent motor nerve terminals.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Dec-08, Volume: 30, Issue:49

    Topics: Acetylcholine; Animals; Atropine; Brain-Derived Neurotrophic Factor; Bungarotoxins; Carbazoles; Diamines; Dose-Response Relationship, Drug; Enzyme Inhibitors; Indole Alkaloids; Male; Mice; Motor Neurons; Muscarinic Antagonists; Nerve Growth Factors; Neuromuscular Junction; Neurotransmitter Agents; Pirenzepine; Qa-SNARE Proteins; Receptor, Nerve Growth Factor; Receptor, trkB; Receptors, Muscarinic

2010
Urothelial/lamina propria spontaneous activity and the role of M3 muscarinic receptors in mediating rate responses to stretch and carbachol.
    Urology, 2011, Volume: 78, Issue:6

    Topics: Animals; Atropine; Benzhydryl Compounds; Benzofurans; Carbachol; Cresols; Diamines; Mandelic Acids; Mucous Membrane; Muscarinic Antagonists; Muscle Contraction; Phenylpropanolamine; Piperidines; Pirenzepine; Pyrrolidines; Quinuclidines; Receptor, Muscarinic M3; Solifenacin Succinate; Stress, Mechanical; Swine; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urothelium

2011
Role of M2 and M3 muscarinic acetylcholine receptor subtypes in activation of bladder afferent pathways in spinal cord injured rats.
    Urology, 2012, Volume: 79, Issue:5

    Topics: Afferent Pathways; Animals; Atropine; Benzofurans; Diamines; Female; Mucous Membrane; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Parasympatholytics; Pressure; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; RNA, Messenger; Spinal Cord Injuries; Thoracic Vertebrae; Urinary Bladder; Urinary Bladder, Overactive

2012
Paradoxical neostigmine-induced TOFfade: on the role of presynaptic cholinergic and adenosine receptors.
    European journal of pharmacology, 2014, Jan-15, Volume: 723

    Topics: Animals; Atropine; Cholinesterase Inhibitors; Diamines; Diaphragm; In Vitro Techniques; Male; Muscarinic Antagonists; Neostigmine; Phrenic Nerve; Pirenzepine; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Cholinergic; Receptors, Presynaptic; Receptors, Purinergic P1; Synaptic Transmission; Triazines; Triazoles

2014
In vitro functional interactions of acetylcholine esterase inhibitors and muscarinic receptor antagonists in the urinary bladder of the rat.
    Clinical and experimental pharmacology & physiology, 2014, Volume: 41, Issue:2

    Topics: Animals; Atropine; Cholinesterase Inhibitors; Diamines; Dose-Response Relationship, Drug; Heart Atria; In Vitro Techniques; Male; Methacholine Chloride; Muscarinic Antagonists; Muscle Contraction; Obidoxime Chloride; Physostigmine; Rats; Receptor Cross-Talk; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Urinary Bladder

2014
Neuroanatomical basis for cholinergic modulation of locomotor networks by sacral relay neurons with ascending lumbar projections.
    The Journal of comparative neurology, 2014, Oct-15, Volume: 522, Issue:15

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Animals, Newborn; Atropine; Cholinergic Neurons; Cholinesterase Inhibitors; Diamines; Edrophonium; Electric Stimulation; Locomotion; Lumbosacral Region; Muscarinic Antagonists; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Spinal Cord

2014
Expression and function of muscarinic subtype receptors in bladder interstitial cells of cajal in rats.
    Urology journal, 2014, Jul-08, Volume: 11, Issue:3

    Topics: Action Potentials; Animals; Atropine; Calcium Channels; Carbachol; Cholinergic Agonists; Diamines; Interstitial Cells of Cajal; Male; Muscarinic Antagonists; Patch-Clamp Techniques; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Urinary Bladder

2014
Cholinergic regulation of proliferation of the urothelium in response to E. coli lipopolysaccharide exposition.
    International immunopharmacology, 2018, Volume: 56

    Topics: Animals; Apoptosis; Atropine; Caspase 3; Cell Line; Cell Proliferation; Cholinergic Agents; Diamines; Escherichia coli; Female; Humans; Immunity, Innate; Lipopolysaccharides; Pirenzepine; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, Muscarinic; Toll-Like Receptor 4; Urothelium

2018
Balanced modulation of neuromuscular synaptic transmission via M1 and M2 muscarinic receptors during inhibition of cholinesterases.
    Scientific reports, 2022, 02-01, Volume: 12, Issue:1

    Topics: Animals; Antidotes; Atropine; Cholinesterase Inhibitors; Cholinesterases; Diamines; Diaphragm; Disease Models, Animal; Mice; Muscarinic Antagonists; Muscle Contraction; Muscle Weakness; Paraoxon; Parasympatholytics; Pirenzepine; Protective Agents; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Signal Transduction; Synaptic Transmission; Treatment Outcome

2022