Page last updated: 2024-09-05

atropine and himbacine

atropine has been researched along with himbacine in 13 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(himbacine)
Trials
(himbacine)
Recent Studies (post-2010) (himbacine)
26,7111,2591,6977309

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)himbacine (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.0175
Muscarinic acetylcholine receptor M4Homo sapiens (human)0.1144
Muscarinic acetylcholine receptor M5Homo sapiens (human)1.016
Muscarinic acetylcholine receptor M1Homo sapiens (human)0.5482
Muscarinic acetylcholine receptor M3Homo sapiens (human)0.3336

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19901 (7.69)18.7374
1990's8 (61.54)18.2507
2000's4 (30.77)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kovacs, I; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1
el-Fakahany, EE; Lee, NH1
Gilani, AU1
Anwar-ul, S; Cobbin, LB; Gilani, H1
Imaizumi, Y; Tanaka, M; Watanabe, M; Yamahara, NS1
Gillman, TA; Mitchelson, F; Pennefather, JN1
Shiraishi, K; Takayanagi, I1
Garland, CJ; Hillier, K; Kerr, PM; Wallis, RM1
De Neef, P; Domenach, V; Vandermeers, A; Vandermeers-Piret, MC; Waelbroeck, M1
Fitzgerald, ME; Reiner, A; Zagvazdin, Y1
Iannazzo, L; Majewski, H1
Daniels, DV; Eglen, RM; Ford, AP; Hegde, SS; Meloy, TD1
Bitzer, M; Feldkaemper, M; Kovacs, B; Schaeffel, F1

Other Studies

13 other study(ies) available for atropine and himbacine

ArticleYear
Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Amino Acid Sequence; Animals; Carbachol; Cloning, Molecular; Cyclic AMP; Humans; Mice; Molecular Sequence Data; Muscarinic Agonists; Muscarinic Antagonists; Phosphatidylinositols; Radioligand Assay; Rats; Receptors, Muscarinic; Sequence Alignment; Sequence Homology, Amino Acid; Signal Transduction; Species Specificity

1998
The allosteric binding profile of himbacine: a comparison with other cardioselective muscarinic antagonists.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Alkaloids; Allosteric Regulation; Animals; Atropine; Binding, Competitive; Diamines; Dose-Response Relationship, Drug; Furans; Gallamine Triethiodide; Male; Myocardium; N-Methylscopolamine; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives

1990
Comparison of the rate of occupancy of receptors by anti-cholinergic drugs.
    Biochemical Society transactions, 1990, Volume: 18, Issue:2

    Topics: Alkaloids; Animals; Atropine; Carbachol; Furans; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Naphthalenes; Parasympatholytics; Piperidines; Receptors, Cholinergic

1990
The cardio-selectivity of himbacine: a muscarine receptor antagonist.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:1

    Topics: Alkaloids; Animals; Atropine; Diethylstilbestrol; Female; Furans; Guinea Pigs; Heart; Ileum; In Vitro Techniques; Muscle, Smooth; Myocardial Contraction; Naphthalenes; Parasympatholytics; Piperidines; Rats; Trachea; Uterine Contraction

1986
Pertussis toxin-sensitive muscarinic relaxation in the rat iris dilator muscle.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Diamines; Dose-Response Relationship, Drug; Furans; GTP-Binding Proteins; In Vitro Techniques; Iris; Male; Microinjections; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; Parasympatholytics; Pertussis Toxin; Phentolamine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Virulence Factors, Bordetella

1995
Muscarinic receptors in rat uterus.
    European journal of pharmacology, 1994, Sep-12, Volume: 262, Issue:3

    Topics: Alkaloids; Animals; Atropine; Binding, Competitive; Computer Simulation; Female; Furans; In Vitro Techniques; Ligands; Muscarinic Antagonists; Naphthalenes; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Uterus

1994
Subtype of muscarinic receptors mediating relaxation and contraction in the rat iris dilator smooth muscle.
    General pharmacology, 1993, Volume: 24, Issue:1

    Topics: Alkaloids; Animals; Atropine; Carbachol; Furans; In Vitro Techniques; Iris; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic

1993
Characterization of muscarinic receptors mediating contractions of circular and longitudinal muscle of human isolated colon.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Alkaloids; Atropine; Carbachol; Carcinoma; Colon; Colonic Neoplasms; Dose-Response Relationship, Drug; Furans; Humans; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Naphthalenes; Piperidines; Pirenzepine

1995
Binding of the labelled muscarinic toxin 125I-MT1 to rat brain muscarinic M1 receptors.
    European journal of pharmacology, 1996, Jun-03, Volume: 305, Issue:1-3

    Topics: Alkaloids; Animals; Atropine; Binding, Competitive; Brain; Carbachol; Elapid Venoms; Furans; Gallamine Triethiodide; In Vitro Techniques; Iodine Radioisotopes; Isotope Labeling; Kinetics; Muscarinic Agonists; Muscarinic Antagonists; Naphthalenes; Oxotremorine; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Protein Binding; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Synaptic Membranes; Tubocurarine

1996
Role of muscarinic cholinergic transmission in Edinger-Westphal nucleus-induced choroidal vasodilation in pigeon.
    Experimental eye research, 2000, Volume: 70, Issue:3

    Topics: Alkaloids; Animals; Atropine; Blood Pressure; Choroid; Columbidae; Electric Stimulation; Furans; Heart Rate; Muscarinic Antagonists; Naphthalenes; Parasympatholytics; Piperidines; Receptors, Muscarinic; Regional Blood Flow; Vasodilation

2000
M(2)/M(4)-muscarinic receptors mediate automodulation of acetylcholine outflow from mouse cortex.
    Neuroscience letters, 2000, Jun-23, Volume: 287, Issue:2

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Autoreceptors; Binding, Competitive; Cerebral Cortex; Furans; Male; Mice; Muscarinic Antagonists; Naphthalenes; Neostigmine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic

2000
Functional characterization of rat submaxillary gland muscarinic receptors using microphysiometry.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: Alkaloids; Animals; Atropine; Benzhydryl Compounds; Benzodiazepinones; Binding, Competitive; Biosensing Techniques; Carbachol; Cholinergic Agonists; Cresols; Diamines; Dose-Response Relationship, Drug; Furans; Male; Mandelic Acids; Muscarinic Antagonists; Naphthalenes; Phenethylamines; Phenylpropanolamine; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Submandibular Gland; Tolterodine Tartrate

2001
Effects of muscarinic antagonists on ZENK expression in the chicken retina.
    Experimental eye research, 2006, Volume: 82, Issue:3

    Topics: Alkaloids; Animals; Atropine; Cell Count; Chickens; Excitatory Amino Acid Agonists; Furans; Gallamine Triethiodide; Glucagon; Immunohistochemistry; Intercellular Signaling Peptides and Proteins; Muscarinic Antagonists; Myopia; Naphthalenes; Peptides; Piperidines; Quisqualic Acid; Receptors, Cholinergic; Retina; Retinal Ganglion Cells

2006