Page last updated: 2024-09-05

atropine and diphenidol

atropine has been researched along with diphenidol in 3 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(diphenidol)
Trials
(diphenidol)
Recent Studies (post-2010) (diphenidol)
26,7111,2591,69760528

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)diphenidol (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.77
Muscarinic acetylcholine receptor M4Homo sapiens (human)0.271
Muscarinic acetylcholine receptor M5Homo sapiens (human)1.191
Cytochrome P450 2D6Homo sapiens (human)0.3263
Muscarinic acetylcholine receptor M1Homo sapiens (human)0.324
D(2) dopamine receptorHomo sapiens (human)3.29
Muscarinic acetylcholine receptor M3Homo sapiens (human)0.245
5-hydroxytryptamine receptor 2AHomo sapiens (human)2.586
D(3) dopamine receptorHomo sapiens (human)2.311
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.256

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19902 (66.67)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
Eltz, M; Gmelin, G; Lambrecht, G; Mutschler, E; Strohmann, C; Tacke, R; Wess, J1

Other Studies

3 other study(ies) available for atropine and diphenidol

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Presynaptic muscarinic receptors mediating inhibition of neurogenic contractions in rabbit vas deferens are of the ganglionic M1-type.
    European journal of pharmacology, 1988, Dec-13, Volume: 158, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Binding Sites; Blood Pressure; Electric Stimulation; Ganglia, Sympathetic; Male; Muscle Contraction; Piperazines; Piperidines; Pirenzepine; Rabbits; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Receptors, Neurotransmitter; Vas Deferens

1988