Page last updated: 2024-09-05

atropine and dexetimide

atropine has been researched along with dexetimide in 19 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(dexetimide)
Trials
(dexetimide)
Recent Studies (post-2010) (dexetimide)
26,7111,2591,69711744

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)dexetimide (IC50)
Muscarinic acetylcholine receptor M1Mus musculus (house mouse)0.0033
Muscarinic acetylcholine receptor M4Mus musculus (house mouse)0.0033
Muscarinic acetylcholine receptor M5Mus musculus (house mouse)0.0033
Muscarinic acetylcholine receptor M3Mus musculus (house mouse)0.0033
Muscarinic acetylcholine receptor M2Mus musculus (house mouse)0.0033

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-199011 (57.89)18.7374
1990's7 (36.84)18.2507
2000's1 (5.26)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kovacs, I; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1
Bertram, U; Kasten, A; Lüllmann, H; Ziegler, A1
Binenfeld, Z; Deljac, V; Fajdetić, A; Wilhelm, K1
Gianutsos, G; Lal, H1
Carson, S; Godwin, S; Kato, G; Massoulié, J1
Gianutsos, G; Hynes, MD; Lal, H1
Bottlaender, M; Brouillet, E; Cayla, J; Chavoix, C; Crouzel, C; Mazière, B; Mazière, M; Prenant, C; Stulzaft, O; Varastet, M1
Dannals, RF; Matsumura, K; Scheffel, U; Uno, Y; Wagner, HN; Wilson, AA1
Dannals, RF; Ravert, HT; Scheffel, UA; Stathis, M; Wagner, HN; Wilson, AA1
Delhaye, M; Larose, L; Longnecker, DS; Morisset, J; Poirier, GG; Swillens, S; Taton, G1
Domino, EF; Head, R; Pohorecki, R1
Gorissen, H; Laduron, PM; Leysen, JE1
Cepeda, C; Collard, P; Comar, D; Godot, JM; Mazière, M; Naquet, R1
Lüllmann, H; Schmaus, H; Staemmler, C; Ziegler, A1
Dorff, RJ; Gaginella, TS; O'Dorisio, TM; Rimele, TJ1
Dannals, RF; Guilarte, TR; Lever, JR; Müller-Gärtner, HW; Ravert, HT; Sasaki, M; Wagner, HN1
Bosman, IJ; de Zeeuw, RA; Ensing, K1
Fixmann, A; Holschbach, M; Müller-Gärtner, HW; Weckesser, M1
Christopoulos, A; Lanzafame, A; Mitchelson, F1

Other Studies

19 other study(ies) available for atropine and dexetimide

ArticleYear
Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Amino Acid Sequence; Animals; Carbachol; Cloning, Molecular; Cyclic AMP; Humans; Mice; Molecular Sequence Data; Muscarinic Agonists; Muscarinic Antagonists; Phosphatidylinositols; Radioligand Assay; Rats; Receptors, Muscarinic; Sequence Alignment; Sequence Homology, Amino Acid; Signal Transduction; Species Specificity

1998
Improved treatment of organophosphate intoxication by use of scopolamine or dexetimide.
    Experientia, 1977, Sep-15, Volume: 33, Issue:9

    Topics: Animals; Atropine; Dexetimide; Drug Therapy, Combination; Isoflurophate; Mice; Obidoxime Chloride; Organophosphorus Compounds; Oximes; Piperidines; Rabbits; Scopolamine

1977
Protective effect of dexetimide and HI-6 in poisoning with highly toxic organophosphorus compounds.
    Arhiv za higijenu rada i toksikologiju, 1979, Volume: 30, Issue:2

    Topics: Animals; Antidotes; Atropine; Dexetimide; Male; Mice; Organophosphate Poisoning; Piperidines; Pyridinium Compounds; Rats

1979
Modification of apomorphine induced aggression by changing central cholinergic activity in rats.
    Neuropharmacology, 1977, Volume: 16, Issue:1

    Topics: Aggression; Animals; Apomorphine; Atropine; Dexetimide; Humans; Iodides; Male; Parasympathetic Nervous System; Pilocarpine; Rats; Vocalization, Animal

1977
Biochemical studies on muscarinic receptors.
    Biomedicine / [publiee pour l'A.A.I.C.I.G.], 1977, Volume: 26, Issue:4

    Topics: Acetylcholine; Alkylating Agents; Animals; Atropine; Binding, Competitive; Brain; Carbachol; Cattle; Choline; Dexetimide; Kinetics; Ligands; Muscle Contraction; Muscle, Smooth; Quinuclidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Solubility; Subcellular Fractions

1977
Effects of cholinergic agonists and antagonists on morphine-withdrawal syndrome.
    Psychopharmacology, 1976, Sep-17, Volume: 49, Issue:2

    Topics: Animals; Atropine; Dexetimide; Humans; Male; Morphine Dependence; Pilocarpine; Rats; Scopolamine Derivatives; Substance Withdrawal Syndrome

1976
In vivo visualization of central muscarinic receptors using [11C]quinuclidinyl benzilate and positron emission tomography in baboons.
    European journal of pharmacology, 1992, Mar-24, Volume: 213, Issue:2

    Topics: Animals; Atropine; Cerebral Cortex; Dexetimide; Electroencephalography; Male; Papio; Quinuclidinyl Benzilate; Radioligand Assay; Receptors, Muscarinic; Tomography, Emission-Computed

1992
Effects of atropine treatment on in vitro and in vivo binding of 4-[125I]-dexetimide to central and myocardial muscarinic receptors.
    European journal of nuclear medicine, 1991, Volume: 18, Issue:7

    Topics: Animals; Atropine; Central Nervous System; Dexetimide; In Vitro Techniques; Iodine Radioisotopes; Male; Myocardium; Protein Binding; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Up-Regulation

1991
In vivo biodistribution of two [18F]-labelled muscarinic cholinergic receptor ligands: 2-[18F]- and 4-[18F]-fluorodexetimide.
    Life sciences, 1991, Volume: 48, Issue:14

    Topics: Animals; Atropine; Cerebellum; Cerebral Cortex; Corpus Striatum; Dexetimide; Male; Mice; Mice, Inbred Strains; Receptors, Muscarinic; Tomography, Emission-Computed

1991
Muscarinic cholinergic receptors in pancreatic acinar carcinoma of rat.
    International journal of cancer, 1985, Apr-15, Volume: 35, Issue:4

    Topics: Adenocarcinoma; Amylases; Animals; Atropine; Binding, Competitive; Carbachol; Carcinoma; Dexetimide; DNA; Kinetics; Pancreatic Neoplasms; Proteins; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Stereoisomerism

1985
Effects of selected muscarinic cholinergic antagonists on [3H]acetylcholine release from rat hippocampal slices.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Atropine Derivatives; Benactyzine; Carbachol; Dexetimide; Dose-Response Relationship, Drug; Electric Stimulation; Hemicholinium 3; Hippocampus; Male; Nicotine; Phenylpropionates; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1988
Muscarinic receptor: multiple sites or unitary concept?
    Archives internationales de pharmacodynamie et de therapie, 1981, Volume: 249, Issue:2

    Topics: Animals; Atropine; Benzodiazepinones; Brain; Dexetimide; Dogs; Gastric Mucosa; In Vitro Techniques; Microsomes; Piperazines; Piperidines; Pirenzepine; Receptors, Cholinergic; Receptors, Muscarinic

1981
In vivo characterization of myocardium muscarinic receptors by positron emission tomography.
    Life sciences, 1981, Dec-07, Volume: 29, Issue:23

    Topics: Animals; Atropine; Carbon Radioisotopes; Dexetimide; Dose-Response Relationship, Drug; Heart; Heart Rate; Liver; Male; Myocardium; Papio; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Tomography, Emission-Computed

1981
Comparison of atropine and dexetimide in treatment of intoxications by selected organophosphates.
    Acta pharmacologica et toxicologica, 1982, Volume: 50, Issue:3

    Topics: Animals; Atropine; Dexetimide; Diet; Guinea Pigs; Insecticides; Isoflurophate; Lethal Dose 50; Mice; Obidoxime Chloride; Organophosphate Poisoning; Organophosphorus Compounds; Paraoxon; Piperidines

1982
Pharmacologic identification of muscarinic receptors in the pylorus of the cat by binding of [3H]-quinuclidinyl benzilate.
    Life sciences, 1980, May-12, Volume: 26, Issue:19

    Topics: Animals; Atropine; Bethanechol Compounds; Cats; Dexetimide; Female; Kinetics; Male; Propantheline; Pylorus; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Stereoisomerism; Tropicamide

1980
Assessment of brain muscarinic acetylcholinergic receptors in living mice using a simple probe, [125I]-4-iododexetimide and [125I]-4-iodolevetimide.
    Neuropharmacology, 1993, Volume: 32, Issue:12

    Topics: Animals; Atropine; Binding, Competitive; Brain; Dexetimide; Iodine Radioisotopes; Kinetics; Male; Mice; Mice, Inbred Strains; Radioligand Assay; Receptors, Muscarinic; Time Factors

1993
Unusual reduction of the in vitro skin permeation of [3H]dexetimide by atropine.
    Pharmaceutical research, 1998, Volume: 15, Issue:1

    Topics: Adjuvants, Anesthesia; Administration, Cutaneous; Animals; Antiparkinson Agents; Atropine; Cell Membrane Permeability; Deuterium; Dexetimide; Drug Interactions; Membranes; Radiopharmaceuticals; Skin; Swine

1998
Influence of acetylcholine on binding of 4-[125I]iododexetimide to muscarinic brain receptors.
    Nuclear medicine and biology, 1998, Volume: 25, Issue:8

    Topics: Acetylcholine; Animals; Atropine; Binding Sites; Brain; Dexetimide; In Vitro Techniques; Iodine Radioisotopes; Receptors, Muscarinic; Swine; Synaptosomes; Tomography, Emission-Computed, Single-Photon

1998
The allosteric interaction of otenzepad (AF-DX 116) at muscarinic M2 receptors in guinea pig atria.
    European journal of pharmacology, 2001, Mar-30, Volume: 416, Issue:3

    Topics: Acetylcholine; Allosteric Regulation; Animals; Atropine; Carbachol; Cardiotonic Agents; Dexetimide; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Heart Atria; In Vitro Techniques; Kinetics; Male; Muscarinic Antagonists; N-Methylscopolamine; Nicotinic Antagonists; Parasympatholytics; Phthalimides; Pirenzepine; Quaternary Ammonium Compounds; Radioligand Assay; Receptor, Muscarinic M2; Receptors, Muscarinic

2001