Page last updated: 2024-09-05

atropine and devazepide

atropine has been researched along with devazepide in 36 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(devazepide)
Trials
(devazepide)
Recent Studies (post-2010) (devazepide)
26,7111,2591,697780542

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)devazepide (IC50)
Bile salt export pumpHomo sapiens (human)10
Cholecystokinin receptor type ARattus norvegicus (Norway rat)0.0009
Gastrin/cholecystokinin type B receptorRattus norvegicus (Norway rat)0.0008
Cholecystokinin receptor type AHomo sapiens (human)0.0002
Gastrin/cholecystokinin type B receptorHomo sapiens (human)0.245
Cholecystokinin receptor type ACavia porcellus (domestic guinea pig)0.27

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's28 (77.78)18.2507
2000's5 (13.89)29.6817
2010's3 (8.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Arimura, A; Fujimura, M; Fujino, M; Hayashi, N; Itoh, Z; Mizumoto, A; Ohtawa, M; Ueki, S1
Dodds, WJ; Hanyu, N; Hogan, WJ; Layman, RD1
Chariot, J; Hugonet, F; Nagain, C; Rozé, C; Tsocas, A1
Arruebo, MP; Bueno, L; Liberge, M1
Adrian, TE; Basson, MD; Modlin, IM1
Bielański, W; Konturek, SJ; Solomon, TE1
Bhat, ST; Gardner, JD; Pollo, DA; Talkad, VD1
Maouyo, D; Morisset, J2
Adelson, JW; Guan, D; Maouyo, D; Morisset, J; Rivard, N1
Li, Y; Owyang, C1
Brodish, RJ; Fink, AS; Kuvshinoff, BW; McFadden, DW1
Green, GM; Spannagel, AW2
Guan, D; Maouyo, D; Morisset, J; Rivard, N1
Joehl, RJ; Samuel, I1
Haga, N; Itoh, Z; Sakai, T; Satoh, M; Sonobe, K1
Hara, H; Kasai, T; Narakino, H; Nishi, T1
Bhatia, M; Dawra, R; Hofbauer, B; Lu, L; Rünzi, M; Saluja, AK; Steer, ML; Yamaguchi, Y1
Kato, S; Mineo, H; Onaga, T1
Itoh, Z; Mizumoto, A; Muramatsu, S; Sonobe, K; Yamada, T1
Akuzawa, S; Ito, H; Miyake, A; Miyata, K; Nishida, A; Takemoto, Y; Takinami, Y; Yuki, H1
Hao, Y; Li, Y; Owyang, C1
Debas, HT; He, X; Nelson, MT1
Cox, JE; Randich, A1
Chen, YL; Chiu, JH; Hong, CY; Lui, WY1
Giralt, M; Vergara, P2
Ballaz, S; Barber, A; Del Río, J; Fortuño, A1
Ahn, W; Case, RM; Kim, H; Kim, KH; Lee, MG; Lee, SI; Moon, SJ; Seo, JT1
Chariot, J; Mahé, S; Nagain-Domaine, C; Pedersen, NL; Rozé, C; Tomé, D1
Cowles, RA; Mulholland, MW; Segura, BJ1
Bozkurt, A; Deniz, M; Kurtel, H1
Flemström, G; Herzig, KH; Jedstedt, G; Mäkelä, K; Purhonen, AK; Sjöblom, M; Walkowiak, J1

Other Studies

36 other study(ies) available for atropine and devazepide

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Pituitary adenylate cyclase activating polypeptide stimulates gallbladder motility in conscious dogs.
    Regulatory peptides, 1992, Nov-20, Volume: 42, Issue:1-2

    Topics: Animals; Atropine; Benzodiazepinones; Cholecystokinin; Devazepide; Digestion; Dogs; Drug Interactions; Electric Stimulation; Gallbladder; Ganglionic Blockers; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Injections, Intravenous; Muscle Contraction; Muscle, Smooth; Neuropeptides; Pituitary Adenylate Cyclase-Activating Polypeptide; Sincalide

1992
Cholecystokinin-induced contraction of opossum sphincter of Oddi. Mechanism of action.
    Digestive diseases and sciences, 1990, Volume: 35, Issue:5

    Topics: Ampulla of Vater; Animals; Antihypertensive Agents; Atropine; Benzodiazepinones; Cholecystokinin; Devazepide; Electrodes, Implanted; Food; Hexamethonium; Hexamethonium Compounds; Infusions, Intravenous; Methysergide; Muscle Contraction; Opossums; Sphincter of Oddi

1990
Control of interdigestive and intraduodenal meal-stimulated pancreatic secretion in rats.
    The American journal of physiology, 1990, Volume: 259, Issue:2 Pt 1

    Topics: Animals; Atropine; Benzodiazepinones; Cholecystokinin; Devazepide; Digestion; Duodenum; Eating; Hexamethonium; Hexamethonium Compounds; Kinetics; Male; Muscle, Smooth; Pancreas; Pirenzepine; Proglumide; Rats; Rats, Inbred Strains; Reference Values; Vagotomy

1990
Role of hypothalamic cholecystokinin octapeptide in the colonic motor response to a meal in rats.
    Gastroenterology, 1991, Volume: 100, Issue:2

    Topics: Animals; Atropine; Benzodiazepinones; Cholecystokinin; Colon; Devazepide; Electromyography; Food; Gastrointestinal Motility; Hypothalamic Area, Lateral; Hypothalamus; Male; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Receptors, Muscarinic; Sincalide; Ventromedial Hypothalamic Nucleus

1991
Effects of cholecystokinin and cholinergic receptor blockade on guinea pig pepsinogen secretion.
    Scandinavian journal of gastroenterology, 1990, Volume: 25, Issue:8

    Topics: Animals; Atropine; Benzodiazepinones; Carbachol; Cholecystokinin; Cholinergic Antagonists; Devazepide; Gastric Mucosa; Gastrins; Guinea Pigs; Male; Pentagastrin; Pepsinogens; Receptors, Cholecystokinin; Receptors, Cholinergic

1990
Effects of an antral mucosectomy, L-364,718 and atropine on cephalic phase of gastric and pancreatic secretion in dogs.
    Gastroenterology, 1990, Volume: 98, Issue:1

    Topics: Animals; Atropine; Benzodiazepinones; Cholecystokinin; Deoxyglucose; Devazepide; Dogs; Food; Gastric Acid; Gastric Mucosa; Gastrins; Insulin; Pancreas; Pyloric Antrum; Vagus Nerve

1990
Characterization of a persistent inhibitory action of L-364,718 on cholecystokinin-stimulated enzyme secretion in pancreatic acini.
    Pancreas, 1994, Volume: 9, Issue:1

    Topics: Amylases; Animals; Atropine; Benzodiazepinones; Carbachol; Cholecystokinin; Devazepide; Kinetics; Male; Pancreas; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide

1994
Amazing pancreas: specific regulation of pancreatic secretion of individual digestive enzymes in rats.
    The American journal of physiology, 1995, Volume: 268, Issue:2 Pt 1

    Topics: Animals; Atropine; Benzodiazepinones; Carbachol; Ceruletide; Cholecystokinin; Devazepide; Digestion; Male; Octreotide; Pancreas; Rats; Rats, Wistar

1995
Stability of circadian and minor cycles of exocrine pancreatic secretion in atropine- and MK-329-infused rats.
    The American journal of physiology, 1995, Volume: 268, Issue:2 Pt 1

    Topics: Animals; Atropine; Benzodiazepinones; Cholecystokinin; Circadian Rhythm; Devazepide; Eating; Male; Pancreas; Photoperiod; Rats; Rats, Wistar

1995
Endogenous cholecystokinin stimulates pancreatic enzyme secretion via vagal afferent pathway in rats.
    Gastroenterology, 1994, Volume: 107, Issue:2

    Topics: Afferent Pathways; Animals; Atropine; Benzodiazepinones; Capsaicin; Caseins; Cholecystokinin; Devazepide; Male; Pancreas; Rats; Rats, Sprague-Dawley; Vagotomy; Vagus Nerve

1994
Extrapancreatic cholinergic nerves mediate cholecystokinin-stimulated pancreatic polypeptide release.
    The Journal of surgical research, 1994, Volume: 56, Issue:5

    Topics: Animals; Atropine; Benzodiazepinones; Cholecystokinin; Denervation; Devazepide; Dogs; Fistula; Kinetics; Pancreas; Pancreatic Ducts; Pancreatic Polypeptide; Sincalide; Stomach; Time Factors

1994
Role of intraluminal nutrients in feedback regulation of pancreatic enzyme secretion.
    Annals of the New York Academy of Sciences, 1994, Mar-23, Volume: 713

    Topics: Amino Acids; Animal Nutritional Physiological Phenomena; Animals; Atropine; Benzodiazepinones; Bile; Cholecystokinin; Devazepide; Dietary Proteins; Enzymes; Feedback; Jejunum; Pancreas; Pancreatic Juice; Rats; Receptors, Cholecystokinin

1994
Modulation of the relationship between amylase and chymotrypsinogen secretion in atropine- and MK329-infused rats.
    Pancreas, 1995, Volume: 11, Issue:4

    Topics: Amylases; Animals; Atropine; Benzodiazepinones; Cholecystokinin; Chymotrypsinogen; Devazepide; Male; Parasympatholytics; Proteins; Rats; Rats, Wistar; Receptors, Cholecystokinin

1995
Bile-pancreatic juice replacement not cholinergic- and cholecystokinin-receptor blockade reverses acinar cell hyperstimulation after bile-pancreatic duct ligation.
    American journal of surgery, 1996, Volume: 171, Issue:1

    Topics: Amylases; Animals; Atropine; Benzodiazepinones; Bile; Bile Ducts; Cholinergic Antagonists; Devazepide; Ligation; Pancreas; Pancreatic Ducts; Pancreatic Juice; Pancreatitis; Rats; Receptors, Cholecystokinin

1996
Control of gallbladder contractions by cholecystokinin through cholecystokinin-A receptors in the vagal pathway and gallbladder in the dog.
    Regulatory peptides, 1995, Dec-07, Volume: 60, Issue:1

    Topics: Animals; Atropine; Autoradiography; Benzodiazepinones; Binding, Competitive; Cholecystokinin; Devazepide; Dogs; Eating; Gallbladder; Hexamethonium; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Phenylurea Compounds; Receptors, Cholecystokinin; Sincalide; Tetrodotoxin; Vagus Nerve

1995
CK-independent increases in pancreatic secretion induced by dietary protein in chronic BPJ-diverted rats.
    The American journal of physiology, 1996, Volume: 271, Issue:3 Pt 1

    Topics: Animals; Atropine; Benzodiazepinones; Bile; Cholecystokinin; Devazepide; Diet; Hormone Antagonists; Indoles; Male; Pancreas; Pancreatic Juice; Proteins; Rats; Rats, Sprague-Dawley

1996
Modulation of pancreatic secretion of individual digestive enzymes in octreotide (SMS 201-995)-infused rats.
    Pancreas, 1997, Volume: 14, Issue:1

    Topics: Amylases; Animals; Atropine; Benzodiazepinones; Cholecystokinin; Devazepide; Lipase; Octreotide; Pancreas; Rats; Trypsinogen

1997
A cholecystokinin-releasing factor mediates ethanol-induced stimulation of rat pancreatic secretion.
    The Journal of clinical investigation, 1997, Feb-01, Volume: 99, Issue:3

    Topics: Alcoholism; Amylases; Animals; Atropine; Benzodiazepinones; Cholecystokinin; Devazepide; Digestive System; Duodenum; Enzymes; Ethanol; Growth Substances; Hormone Antagonists; Intercellular Signaling Peptides and Proteins; Male; Muscarinic Antagonists; Pancreatitis; Rats; Rats, Wistar; Trypsin; Trypsin Inhibitor, Kazal Pancreatic

1997
Effect of L364718 on interdigestive pancreatic exocrine secretion and gastroduodenal motility in conscious sheep.
    Regulatory peptides, 1997, Jan-29, Volume: 68, Issue:2

    Topics: Animals; Atropine; Benzodiazepinones; Devazepide; Electromyography; Gastrointestinal Motility; Hormone Antagonists; Male; Muscle Contraction; Myoelectric Complex, Migrating; Pancreas; Pancreatic Juice; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sheep; Sincalide

1997
Relationship between gallbladder bile concentration and motility in conscious dogs: role of cholecystokinin.
    Peptides, 1997, Volume: 18, Issue:1

    Topics: Animals; Atropine; Benzodiazepinones; Bile; Bilirubin; Cholecystokinin; Devazepide; Dogs; Duodenum; Food; Gallbladder; Gastrointestinal Motility; Hexamethonium; Hormone Antagonists; Pyloric Antrum; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide; Sodium

1997
YM022, a potent and selective gastrin/CCK-B receptor antagonist, inhibits peptone meal-induced gastric acid secretion in Heidenhain pouch dogs.
    Digestive diseases and sciences, 1997, Volume: 42, Issue:4

    Topics: Animals; Atropine; Benzodiazepines; Benzodiazepinones; Devazepide; Dogs; Dose-Response Relationship, Drug; Eating; Famotidine; Gastric Acid; Histamine; Histamine H2 Antagonists; Hormone Antagonists; Male; Methacholine Chloride; Muscarinic Antagonists; Pentagastrin; Peptones; Phenylurea Compounds; Receptors, Cholecystokinin; Sincalide; Stomach

1997
High-affinity CCK-A receptors on the vagus nerve mediate CCK-stimulated pancreatic secretion in rats.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 1

    Topics: Animals; Atropine; Benzodiazepinones; Capsaicin; Caseins; Devazepide; Duodenum; Hexamethonium; Hormone Antagonists; Infusions, Intravenous; Infusions, Parenteral; Kinetics; Male; Pancreas; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide; Vagotomy; Vagus Nerve

1997
Rat exocrine pancreatic secretion by vagal stimulation occurs via multiple mediators.
    Chinese medical sciences journal = Chung-kuo i hsueh k'o hsueh tsa chih, 1996, Volume: 11, Issue:2

    Topics: Amylases; Animals; Atropine; Benzodiazepinones; Devazepide; Electric Stimulation; Ganglionic Blockers; Hexamethonium; Male; Muscarinic Antagonists; Pancreas; Rats; Rats, Sprague-Dawley; Sincalide; Vagus Nerve

1996
CCK-8 activates hepatic vagal C-fiber afferents.
    Brain research, 1997, Nov-21, Volume: 776, Issue:1-2

    Topics: Animals; Atropine; Benzodiazepinones; Devazepide; Electrophysiology; Ganglionic Blockers; Hexamethonium; Hormone Antagonists; Liver; Male; Nerve Fibers; Neurons, Afferent; Parasympatholytics; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Satiation; Sincalide; Vagus Nerve

1997
Local somatothermal stimulation inhibits the motility of sphincter of Oddi in cats, rabbits and humans through nitrergic neural release of nitric oxide.
    Life sciences, 1998, Volume: 63, Issue:6

    Topics: Animals; Arginine; Atropine; Benzodiazepinones; Body Temperature; Cats; Devazepide; Female; Hormone Antagonists; Humans; Male; Manometry; Muscle Contraction; Muscle Relaxation; Neurons, Efferent; NG-Nitroarginine Methyl Ester; Nitric Oxide; Phentolamine; Propranolol; Rabbits; Sphincter of Oddi; Sympatholytics

1998
Pancreatic hypersecretion in the jejunal-bypass rat.
    Pancreas, 1999, Volume: 18, Issue:1

    Topics: Animals; Atropine; Bile; Devazepide; Jejunum; Male; Pancreas; Pancreatic Juice; Rats; Rats, Wistar; Receptors, Cholecystokinin

1999
Both afferent and efferent nerves are implicated in cholecytokinin motor actions in the small intestine of the rat.
    Regulatory peptides, 1999, May-31, Volume: 81, Issue:1-3

    Topics: Anesthetics, Local; Animals; Atropine; Benzodiazepinones; Cholecystokinin; Devazepide; Duodenum; Gastrins; Hexamethonium; Hormone Antagonists; Intestinal Mucosa; Intestine, Small; Jejunum; Lidocaine; Male; Neurons, Afferent; Neurons, Efferent; Nitroarginine; Oligopeptides; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide; Tetragastrin

1999
CCK-mediated response in the activation of 5-HT receptor types in the guinea-pig ileum.
    Journal of physiology and biochemistry, 1999, Volume: 55, Issue:2

    Topics: Animals; Atropine; Cholecystokinin; Devazepide; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Physalaemin; Receptors, Serotonin; Serotonin Receptor Agonists

1999
A novel effect of rebamipide: generation of [Ca(2+)](i) oscillations through activation of CCK(1) receptors in rat pancreatic acinar cells.
    European journal of pharmacology, 2000, Jan-24, Volume: 388, Issue:1

    Topics: Alanine; Animals; Anti-Ulcer Agents; Atropine; Benzodiazepinones; Calcium; Devazepide; Fluorescent Dyes; Fura-2; In Vitro Techniques; Male; Muscarinic Antagonists; Pancreas; Phenylurea Compounds; Quinolones; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin

2000
Inhibition by CCK of ascending contraction elicited by mucosal stimulation in the duodenum of the rat.
    Neurogastroenterology and motility, 2000, Volume: 12, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Atropine; Benzodiazepinones; Cholecystokinin; Depression, Chemical; Devazepide; Duodenum; Electric Stimulation; Enteric Nervous System; Enzyme Inhibitors; Gastrins; Hexamethonium; Intestinal Mucosa; Male; Muscle Contraction; Nicotinic Antagonists; Nitroarginine; Oligopeptides; Parasympatholytics; Peristalsis; Phentolamine; Phenylurea Compounds; Propranolol; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Receptors, Vasoactive Intestinal Peptide; Sincalide; Tetragastrin; Vasoactive Intestinal Peptide

2000
Caseinomacropeptide specifically stimulates exocrine pancreatic secretion in the anesthetized rat.
    Peptides, 2000, Volume: 21, Issue:10

    Topics: Anesthesia; Animals; Atropine; Capsaicin; Caseins; Devazepide; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Glutens; Hexamethonium; Male; Milk Proteins; Models, Biological; Pancreas; Pancreatic Juice; Peptide Fragments; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide; Sodium Chloride; Trypsin; Trypsin Inhibitors; Vagotomy; Whey Proteins

2000
Stimulation of rat pancreatic exocrine secretion by cocaine- and amphetamine-regulated transcript peptide.
    Regulatory peptides, 2001, May-05, Volume: 99, Issue:1

    Topics: Amylases; Animals; Atropine; Cells, Cultured; Devazepide; Hormone Antagonists; Male; Muscarinic Antagonists; Nerve Tissue Proteins; Neurotransmitter Agents; Pancreas; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Signal Transduction; Vagotomy; Vagus Nerve

2001
Mediators of glucagon-like peptide 2-induced blood flow: responses in different vascular sites.
    Regulatory peptides, 2007, Jul-05, Volume: 142, Issue:1-2

    Topics: Animals; Atropine; Benzodiazepinones; Blood Flow Velocity; Blood Vessels; Devazepide; Female; Glucagon-Like Peptide 2; Hormone Antagonists; Indomethacin; Infusions, Intravenous; Lidocaine; Male; Mesenteric Artery, Superior; NG-Nitroarginine Methyl Ester; Peptide Fragments; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Time Factors

2007
Apelin stimulation of duodenal bicarbonate secretion: feeding-dependent and mediated via apelin-induced release of enteric cholecystokinin.
    Acta physiologica (Oxford, England), 2011, Volume: 201, Issue:1

    Topics: Animals; Apelin Receptors; Atropine; Bicarbonates; Cell Line; Cholecystokinin; Devazepide; Dinoprostone; Duodenum; Eating; Food Deprivation; Humans; Infusions, Intra-Arterial; Intercellular Signaling Peptides and Proteins; Intestinal Mucosa; Male; Parasympatholytics; Rats; Rats, Inbred Lew; Receptors, G-Protein-Coupled; Tryptamines

2011